Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704) |
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01/07/1997 | US5591749 Imidazopyridines as serotonergic 5-HT3 -antagonists |
01/07/1997 | US5591748 Immunomodulatory azaspiranes |
01/01/1997 | CN1139122A Hydroxymethyl quenuclidine catalyst compositions for making polyurethane foams |
12/31/1996 | US5589477 Pyrimidine derivatives and drugs |
12/25/1996 | CN1138850A Novel high enantio-selective process for producing pure enantiomeric cyclopentane and cyclopentene-'beta'-amino acids |
12/24/1996 | US5587479 Basic derivatives of glutamic acid and aspartic acid as gastrin or cholecystokinin antagonists |
12/19/1996 | WO1996040641A1 Sulfonamide derivatives as cell adhesion modulators |
12/19/1996 | WO1996040100A1 ARYLSULFONYLAMINOBENZENE DERIVATIVES AND THE USE THEREOF AS FACTOR Xa INHIBITORS |
12/19/1996 | CA2223727A1 Arylsulfonylaminobenzene derivatives and the use thereof as factor xa inhibitors |
12/18/1996 | CN1033584C Benzo-fused lactams that promote release of growth hormone |
12/17/1996 | US5585357 Heteroaryloxymethyl ketones as interleukin-1βconverting enzyme inhibitors |
12/11/1996 | EP0747407A1 Hydroxymethyl quinuclidine catalyst compositions for making polyurethane foams |
12/11/1996 | EP0747355A1 Novel carbamate derivative and medicinal composition containing the same |
12/10/1996 | US5583140 Administering 2-azabicyclo(2.2.2)oct-5-ene derivatives to treat neurodegenerative disorders such as senile dementia of alzheimer's type |
12/10/1996 | US5583134 1-azoniabicyclo[2.2.2] octanes and pharmaceutical compositions in which they are present |
12/05/1996 | WO1996038430A1 Process for making heterocyclic compounds |
12/05/1996 | CA2222033A1 Process for making heterocyclic compounds |
12/04/1996 | EP0745602A1 Quinidine immunoassay and reagents |
12/04/1996 | EP0745601A1 Process for preparing 1,2,5-thiadiazole derivatives |
12/01/1996 | CA2176417A1 Quinidine immunoassay and reagents |
11/26/1996 | US5578602 Certain 1-azabicyclo[3.3.1]nonene derivatives and their pharmacological uses |
11/26/1996 | US5578601 Nonpeptide bradykinin antagonists |
11/21/1996 | WO1996036637A1 Pharmaceutical compositions for prevention and treatment of central nervous system disorders |
11/20/1996 | EP0743302A2 Sulfonamide fibrinogen receptor antagonists |
11/19/1996 | US5576434 5-ht3 receptor antagonist |
11/19/1996 | US5576323 Excitatory amino acid receptor antagonists |
11/19/1996 | US5576317 NK-1 receptor antagonists and 5HT3 receptor antagonists for the treatment of emesis |
11/19/1996 | CA2109613C Fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles |
11/12/1996 | US5574043 Certain [1,2,5-thiadiazol-4-yl]-1-azabicyclo [3.2.1]octane derivatives and their pharmaceutical uses |
11/07/1996 | WO1996034864A1 Piperazino derivatives as neurokinin antagonists |
11/05/1996 | US5571918 Reacting 3-hydroxy-3-mercaptomethylquinuclidine and a carbonyl compound in the presence of a catalyst |
10/30/1996 | EP0739204A1 Piperidines, pyrrolidines and hexahydro-1h-azepines promote release of growth hormone |
10/29/1996 | US5569662 Quinuclidine derivatives as substance P antagonists |
10/29/1996 | US5569447 Stannylated 3-quinuclidinyl benzilates and methods of preparing radiohalogenated derivatives |
10/24/1996 | WO1996033186A1 Substituted dihydrobenzofuran derivatives as 5-ht4 agonists |
10/24/1996 | WO1996033172A1 Arylsulfonyl hydroxamic acid derivatives as mmp and tnf inhibitors |
10/23/1996 | EP0738149A1 1-aminoindan derivatives and compositions thereof |
10/22/1996 | US5567818 Reduction; separation; dehydration |
10/17/1996 | WO1996032382A1 1-phenylpyrazole-3-carboxamides acting on neurotensin receptors |
10/17/1996 | CA2220827A1 1-phenylpyrazole-3-carboxamides acting on neurotensin receptors |
10/10/1996 | WO1996031498A1 Novel heterocyclic compounds |
10/10/1996 | CA2217197A1 Novel heterocyclic compounds |
10/09/1996 | EP0735869A1 A method of treating gastrointestinal motility disorders |
10/09/1996 | CN1133044A Antipsychotic method |
10/09/1996 | CN1132625A NK-1 receptor antagonits and 5HT3 receptor antagonists for treatment of emesis |
10/08/1996 | US5563148 Specific 5-HT3 antagonists |
10/03/1996 | WO1995027727A3 Process for peptide segment condensation |
10/02/1996 | CN1132072A NK-1 receptor antagonists for treatment of neuronal injury and stroke |
10/01/1996 | US5561149 For nasal administration |
09/24/1996 | US5559124 Depolarizing skeletal muscle relaxants |
09/17/1996 | US5556860 Quinazolinone derivatives possessing calcium uptake inhibiting activity |
09/17/1996 | US5556856 Anitarrhythmia, analgesics |
09/17/1996 | US5556851 Treatment of nausea or emesis from anticancer drugs or x-ray treatment |
09/10/1996 | US5554763 1-azoniabicyclo[2.2.1] heptanes and pharmaceutical compositions in which they are present |
09/10/1996 | US5554753 Catalytic enantioselective synthesis of α-amino acid derivatives by phase-transfer catalysis |
09/10/1996 | US5554627 Tachykinin antagonists |
09/10/1996 | US5554613 Quinuclidine derivatives, qualene synthase inhibitors, treatment of hypercholesterolemia, atherosclerosis and fungus infections |
09/06/1996 | WO1996026938A1 Novel quinuclidine derivatives having tricyclic fused hereto ring |
09/06/1996 | CA2213706A1 Novel quinuclidine derivative having tricyclic hetereo condensed ring |
09/04/1996 | EP0589924B1 Fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles |
09/03/1996 | US5552408 Benzimidazoline-2-oxo-1-carboxylic acid derivatives useful as 5-ht receptor antagonists |
08/28/1996 | EP0727993A1 (non descriptive)-a method for delaying hiv individual aids by administration of substituted azaspirane compounds |
08/28/1996 | CN1129942A Aza spiro-compounds acting on the cholinergic system with muscarinic agonist activity |
08/28/1996 | CN1129934A Benzazepine derivative, pharmaceutical composition containing the same, and intermediate for the same |
08/27/1996 | US5550289 N-(1,(1-1)-dialkyloxy)-and N-(1,(1-1)-dialkenyloxy alk-1-yl-N-N,N-tetrasubstituted ammonium lipids and uses therefor |
08/22/1996 | WO1996025160A1 The use of heterocyclic compounds |
08/20/1996 | US5547964 Antiemetic during drug therapy |
08/14/1996 | CN1032534C Method for prepn. of diaminotrifluoromethylpyridine derivatives |
08/13/1996 | US5545740 Nitrosation process |
08/13/1996 | US5545412 Using lipophilic compounds to transfect dna and for drug delivery by forming complexes to penetrate cellular membranes |
08/08/1996 | WO1996023787A1 Substituted heterocyclic compounds, preparation method therefor and pharmaceutical compositions containing same |
08/06/1996 | US5543426 Use of certain 3,7-disubstituted indole compounds for treating depression or cognitive disorders |
08/06/1996 | US5543419 Treating chronic obstructive airways disease or asthma; antimuscarinic bronchodilator agents |
07/31/1996 | EP0723959A1 Heterocyclic compounds as tachykinin receptor antagonists, process for their preparation and pharmaceuticals containing them |
07/30/1996 | US5541194 Pharmaceutical compostion used to treat dementia |
07/23/1996 | US5538982 Medical use for tachykinin antagonists |
07/18/1996 | WO1996021644A1 Indole derivatives useful in the treatment of osteoporosis |
07/18/1996 | CA2209936A1 Indole derivatives useful in the treatment of osteoporosis |
07/17/1996 | EP0721778A2 NK-1 receptor antagonists for the treatment of neuronal injury and stroke |
07/10/1996 | EP0720601A1 Gastrin and cck receptor ligands |
07/09/1996 | US5534521 Serotonin antagonists |
07/09/1996 | US5534520 Spiro compounds containing five-membered rings |
07/04/1996 | WO1996020194A1 Novel quinuclidine derivatives and medicinal composition thereof |
07/03/1996 | EP0719266A1 Heteroarylamino and heteroarylsulfonamido substituted 3-benzylaminomethyl piperidines and related compounds |
06/27/1996 | WO1996019474A1 Quinazolines as inhibitors of endothelin converting enzyme |
06/27/1996 | WO1996019452A1 A process for the preparation of substituted 4-ethyl-piperidines and an intermediate for the preparation of same |
06/27/1996 | CA2206046A1 Quinazolines as inhibitors of endothelin converting enzyme |
06/26/1996 | EP0718297A1 Pyrazine derivatives as muscarinic receptor agonists |
06/25/1996 | US5530118 Phospholipase inhibitor |
06/22/1996 | CA2165751A1 Quinuclidine and azabicyclo¬2.2.1|heptane pyrazinyl ethers as muscarinic agonists |
06/18/1996 | US5527813 Heterocyclic compounds and their preparation and use |
06/18/1996 | US5527808 Fused tricyclic nitrogen containing heterocycles |
06/13/1996 | WO1996017630A1 Substituted benzamides and radioligand analogs and methods of use |
06/12/1996 | EP0716083A1 Benzazepine derivative, pharmaceutical composition containing the same, and intermediate for the same |
06/12/1996 | EP0715855A2 NK-1 receptor antagonists and 5HT3 receptor antagonists for the treatment of emesis |
06/05/1996 | EP0714880A1 Bis(methylidene)-phenylene-derivatives |
06/05/1996 | EP0714394A1 Antipsychotic method |
06/04/1996 | US5523299 Administering in treatment of psychotic disorders |
05/30/1996 | WO1996007410A3 Depolarizing skeletal muscle relaxants |
05/23/1996 | WO1996014846A1 Dihydropyrimidines and uses thereof |