Patents
Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704)
07/1991
07/11/1991WO1991009593A2 5-ht3 antagonists for treatment of nausea, bradycardia of hypotension associated with myocardial instability
07/10/1991EP0436245A1 Substituted 3,4-annelated benzimidazol-2(1H)-ones
06/1991
06/28/1991CA2032885A1 Substituted 3,4-annelated benzimidazol-2(1h)-ones
06/27/1991WO1991009018A1 Dioscoretine and its use as a hypoglycemic agent
06/26/1991EP0434560A1 New derivatives of substituted aminoacids, process for their preparation and pharmaceutical compositions containing them
06/26/1991EP0434365A2 HIV protease inhibitors useful for the treatment of aids
06/26/1991EP0434202A1 Azabicyclo amides and esters as 5-HT3 receptor antagonists
06/25/1991US5026857 Cetnral nervous system disorders; antiserotonine agent
06/25/1991US5026710 Fungicides
06/22/1991CA2071994A1 Pharmaceuticals
06/21/1991CA2032735A1 Substituted amino-acid derivatives; process for preparing the same and pharmaceutical compositions containing them
06/19/1991EP0432975A1 Cyclic renin inhibitors
06/19/1991EP0432974A1 Cyclic renin inhibitors
06/19/1991EP0432751A2 Isomers of 1-azabicyclo[2.2.2]oct-3-yl 1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-5-nitropyridine-3-carboxylate
06/19/1991CA2032259A1 Hiv protease inhibitors useful for the treatment of aids
06/18/1991US5025022 Method of treating or preventing schizophrenia and/or psychosis using S-N-(1-azabicyclo[2.2.2]oct-3-yl)benzamides and thiobenzamides
06/18/1991CA1284953C 2-alkoxy-n-(1-azabicyclo[2.2.2] oct-3-yl) benzamides and thiobenzamides in amethod for alleviating emesis caused by non-platinum anticancer drugs
06/12/1991EP0431972A2 Macrocyclic lactones having renin inhibiting properties
06/09/1991CA2031755A1 Cyclic renin inhibitors
06/09/1991CA2031745A1 Cyclic renin inhibitors containing 2-substituted(3s, 4s)-4-amino-5-cyclohexyl-3-hydroxy pentanoic acid, 2-substituted (3s, 4s)-5-cyclohexyl-3,4-dihydroxy-pentanoic acid or 2 -substituted (4s, 5s)-5-amino-6- yclohexyl-4-hydroxyhexanoic acid or its analogs
06/09/1991CA2031735A1 Cyclic renin inhibitors containing 3(s)-amino-4-cyclohexyl-2(r)-hydroxy-butanoic acid or 4-cyclo-hexyl-(2r, 3s)-dihydroxybutanoic acid or related analogs
06/05/1991EP0430190A2 New tricyclic compounds
06/04/1991US5021425 Use of 2-azabicycloi[2.2.2]octane-3-carboxylic acid derivatives for the treatment of arteritis
05/1991
05/30/1991WO1991007402A1 Azabicyclo amides and esters as 5-ht3 receptor antagonists
05/28/1991US5019597 Bicycloalkyl tricycloalkyl, azabicycloalkyl and azatricycoalkyl amides
05/28/1991US5019580 Antidiabetic agents
05/21/1991US5017582 Method of inducing a serotonin M receptor antagonist effect with N-quinuclidinyl-benzamides
05/21/1991US5017580 Memory enhancing-R-N-(1-azabicyclo[2.2.2.]oct-3-yl)benzamides and thiobenzamides
05/15/1991EP0427390A2 Azabicyclic compounds, process and intermediates for their preparation and pharmaceutical compositions containing them
05/15/1991EP0247201B1 Propane-1,3-diol derivatives, a method for their production and a pharmaceutical composition
05/14/1991US5015655 1-azabicycloalkane derivatives, their preparation process and their use as medicaments
05/07/1991US5013733 Lactam derivatives
05/01/1991CN1051041A Antimuscarinic bronchodilators
04/1991
04/24/1991EP0424021A1 Antimuscarinic bronchodilators
04/23/1991CA1283412C Antidotes
04/20/1991CA2027896A1 Antimuscarinic bronchodilators
04/18/1991WO1991004738A1 Dibenzofurancarboxamides
04/15/1991WO1991005783A1 Heterocyclic compounds
04/08/1991CA2027093A1 Compounds
04/04/1991WO1991004253A1 Preparation of s-(-)- and r-(+)-n-(quinuclidinyl-3)-amide
03/1991
03/27/1991EP0419397A1 Substituted urea compounds and their preparation and use
03/19/1991US5001133 Benzoic acid derivatives
03/13/1991EP0416754A2 A novel substituted pyrazine, formulations thereof and use in medicine
03/13/1991EP0416373A2 Amino acid derivatives
03/09/1991WO1991003475A1 Substituted urea compounds and their preparation and use
03/09/1991CA2066696A1 Substituted urea compounds and their preparation and use
03/05/1991US4997956 Certain 2,3-dihydro-2;2-dimethyl-benzothiophene carboxylic acids which are intermediates
03/05/1991US4997839 2-quinolyl ethers
03/05/1991CA2023099A1 Amino acid derivatives
02/1991
02/27/1991EP0414394A2 Azabicyclic Derivatives having muscarinic receptor affinity
02/26/1991US4996210 Cognition activators, nervous system disorders; muscarinic acetylcholine receptor agonists; 2,8-dimethyl-3-methylene-1-oxa-8-azaspiro[4.5]decane for example
02/26/1991CA1280749C Phenothiazine compounds
02/13/1991EP0412798A2 Substituted pyridines, their preparation, formulations and use in dementia
02/13/1991EP0412797A2 The therapeutic use of substituted benzenes, formulations thereof and novel substituted benzenes
02/09/1991CA2022887A1 Therapeutic use of substituted benzenes, formulations thereof and novel substituted benzenes
02/09/1991CA2022886A1 Substituted pyridines, their preparation, formulations and use in dementia
02/09/1991CA2022885A1 Substituted pyrazine, formulations thereof and use in medicine
02/06/1991CA2022633A1 Compounds
01/1991
01/29/1991US4988691 Analgesics, cardiovascular disorders, nervous system disorders
01/15/1991US4985437 Medicaments
01/15/1991US4985424 Certain substituted 1,7-annelated 1h-indazoles being selective antagonists of 5-ht-receptors
01/15/1991US4985420 1,7-annelated indolecarboxylic acid esters and -amides
01/09/1991EP0407137A2 Benzazine compounds and pharmaceutical uses thereof
01/08/1991US4983623 Prolyl endopeptidase inhibitors
01/08/1991US4983600 Heterocyclic compounds useful as 5-HT3 antagonists
01/04/1991CA2020315A1 Benzazine compounds and pharmaceutical uses thereof
01/02/1991EP0406119A1 New peptide derivatives, process of their preparation and pharmaceutical compositions containing them
01/02/1991EP0405617A2 Medicaments for the treatment of anxiety
01/01/1991US4981869 Xanthates as antitumor agents
12/1990
12/29/1990CA2019633A1 Peptide derivatives, process for their preparation and pharmaceutical compositions containing the same
12/27/1990EP0404737A2 New R(-) 3-quinuclidinol derivatives
12/20/1990CA2019251A1 R(-)3-quinuclidinol derivatives
12/18/1990CA1277917C Method of using 2-alkoxy-n-(1-azabicyclo ¬2.2.2|oct-3-yl)benzamide-n-oxides to control emesis caused by anticancer drugs
12/12/1990EP0402056A2 Azabicyclic compounds, process for their preparation and pharmaceutical compositions containing them
12/12/1990CN1010780B Process for preparation of berban derivatives
12/06/1990CA2018111A1 Compounds
12/04/1990US4975437 Isomers of 1-azabicyclo(2.2.2)oct-3-yl 1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-5-nitropyridine-3-carboxylate
11/1990
11/29/1990WO1990014347A1 Indole derivatives and medicine
11/22/1990EP0398617A2 Process for resolving 1-azabicyclo [2.2.1]heptane-3-carboxylates
11/20/1990US4971975 Novel compounds
11/15/1990CA2016707A1 Process for resolving 1-azabicyclo[2.2.1]heptane-3-carboxylates
11/13/1990US4970315 Thermochromic indicators for structural elements
11/07/1990EP0395729A1 Ligand-accelerated catalytic asymmetric dihydroxylation.
11/06/1990US4968691 Heterocyclo-substituted azabicyclo muscannic agonists
11/06/1990US4968341 Substituted aryloxyureas, processes for production thereof and uses thereof
10/1990
10/22/1990WO1990012569A1 Therapeutic use of 5-ht3 receptor antagonists
10/22/1990CA2031214A1 Therapeutic use of 5-ht receptor antagonists
10/17/1990EP0392803A1 Novel compounds
10/16/1990US4963548 Fungicides
10/03/1990EP0390215A2 Quinolone derivatives and salts thereof, preparation process es thereof, and antibacterial agents containing the same
09/1990
09/25/1990US4959485 5-ht3 antagonists
09/25/1990US4959372 Anti-hypertensive substituted 2-azabicyclooctane-3-carboxylic acids
09/25/1990US4959367 Analgesics, tranquilizers, gastrointestinal, cns
09/19/1990CN1045390A Pyrimidines and their pharmaceutical acceptable salts, and their use as medicines
09/05/1990EP0385722A2 Tricyclic lactam derivatives and pharmaceutical compositions containing them
09/05/1990EP0385517A2 Medicaments for the treatment of emesis
08/1990
08/28/1990US4952587 Physiologically active 1,2,4,-oxa- and thiadiazoles
08/28/1990CA1273297A1 Method of enhancing memory or correcting memory deficiency with arylamido (and arylthioamido) azabicycloalkanes
08/22/1990EP0383281A1 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
08/21/1990US4950759 Substituted 1,7-annelated 1H-indazoles
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