| Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704) |
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| 05/02/1989 | US4826663 Zirconium phosphate and method for its preparation |
| 04/26/1989 | EP0313393A2 Benzoxazine compounds and pharmaceutical use thereof |
| 04/19/1989 | EP0312283A2 Di-or tripeptide renin inhibitors containing lactam conformational restrictions in ACHPA |
| 04/19/1989 | EP0311724A1 Anxiolytic-R-N-(1-azabicyclo[2.2.2]oct-3-yl) benzamides and thiobenzamides |
| 04/12/1989 | EP0311313A2 Heterocyclic spiro compounds and their preparation |
| 04/11/1989 | US4820715 Anti-emetic quinuclidinyl benzamides |
| 04/04/1989 | US4818767 Quinate salts of antimalarial phenanthrenemethanol compounds |
| 04/04/1989 | CA1252101A1 2-azabicyclo ¬2.2.2| octane derivatives, process for their preparation and pharmaceutical compositions containing them |
| 03/29/1989 | EP0309423A2 New benzimidazoline-2-oxo-1-carboxylic acid derivatives useful as 5-ht receptor antagonists |
| 03/22/1989 | EP0308340A1 Process for the synthesis of N-alkylated alpha-amino acids and their esters, use in the synthesis of carboxyalkyl dipeptides |
| 03/22/1989 | CN1031841A Improvements in or relating to specific 5-ht3 antagonists |
| 03/15/1989 | EP0307172A2 Improvements in or relating to specific 5-HT3 antagonists |
| 03/15/1989 | EP0307142A1 Thiadiazoles useful in the treatment of senile dementia |
| 03/15/1989 | EP0307141A2 Oxazoles and thiazoles for the treatment of senile dementia |
| 03/15/1989 | CN1031701A Improvement relating to n-substituted benzamides |
| 03/14/1989 | CA1251211A1 Process for the preparation of triazole derivatives |
| 03/09/1989 | WO1989000571A3 Bicyclic compounds, their use as pharmaceuticals, their preparation, and intermediates useful in their preparation |
| 03/08/1989 | EP0306345A2 2-Alkoxy-n-(1-azabicyclo(2.2.2)-oct-3-yl) benzamides and thiobenzamides having an antischizophrenic activity |
| 03/08/1989 | EP0306148A2 Azabicyclic ethers |
| 03/01/1989 | EP0305297A1 Derivatives of aza-z-bicyclooctane-caboxylicacid-3, processes for their preparation and pharmaceutical compositions containing them |
| 02/28/1989 | US4808718 Fused polycyclic and bridged compounds useful as calcium channel blockers |
| 02/08/1989 | EP0302699A2 Improvements relating to n-substituted benzamides |
| 02/08/1989 | EP0302303A2 Bicyclic compounds, their use as pharmaceuticals, their preparation, and intermediates useful in their preparation |
| 02/07/1989 | US4803199 Pharmaceutically useful heterocyclic and carbocyclic acid esters and amides of alkylene bridged piperidines |
| 02/01/1989 | EP0301729A1 Pro-drugs for oxadiazole muscarinic agonists |
| 01/26/1989 | WO1989000571A2 Bicyclic compounds, their use as pharmaceuticals, their preparation, and intermediates useful in their preparation |
| 01/24/1989 | CA1249296A1 Salts of antimalarial phenanthrenemethanol |
| 01/18/1989 | EP0299352A2 Soluble magnesium hydrides, method of preparing them, and use thereof |
| 01/10/1989 | US4797406 Amides and esters containing bridged piperidines and use as serotonin M antagonists |
| 01/10/1989 | US4797387 Certain pharmaceutically useful ureas |
| 01/03/1989 | CA1248086A1 Fluorescence polarization immunoassay |
| 12/27/1988 | US4794116 Antiinflammatory agents, cytoprotective agents in treatment of hyperproliferative skin disease |
| 12/14/1988 | EP0294667A2 (2-cyano-2-oximinoacetyl)-amino acid derivatives |
| 12/08/1988 | DE3816799A1 Substituierte benzamide, verfahren zu ihrer herstellung und pharmazeutische mittel Substituted benzamides, methods for their preparation and pharmaceutical compositions |
| 12/06/1988 | US4789673 Antiserotonine agents |
| 11/08/1988 | US4783478 Treatment of emesis, nausea and vomiting |
| 11/02/1988 | EP0289170A2 Azabicyclic compounds, process for their preparation and pharmaceutical compositions containing them |
| 11/01/1988 | US4782067 Anti-allergic composition containing zwitterionic bicyclic compounds |
| 10/19/1988 | EP0287356A2 Bridgehead substituted azabicyclic derivatives |
| 10/19/1988 | EP0287196A1 Indole derivatives, process for their preparation and pharmaceutical compositions containing them |
| 08/31/1988 | EP0280603A1 Absolute S confirmation enantiomers of amide derivatives of 3-aminoquinuclidine, process for their preparation and their therapeutical use |
| 08/31/1988 | EP0279990A2 Use of heterocyclic derivatives in the treatment of cognitive disorders |
| 08/24/1988 | EP0279512A2 Use of certain 5-HT3 receptor antagonists in the treatment of visceral pain |
| 08/24/1988 | EP0279149A2 Benzimidazole derivatives, process for their production and a pharmaceutical composition containing the same |
| 07/13/1988 | CN87107539A Substituted basic 2-aminotetralins |
| 06/22/1988 | EP0272052A1 Anxiolytic-N-(1-Azabicyclo[2.2.2]Oct-3-yl) Benzamides and Thobenzamides |
| 06/16/1988 | WO1988004172A1 Pharmaceutical compositions for treatment of hyperproliferate skin disease |
| 06/15/1988 | EP0270947A2 Substituted basic 2-aminotetralines |
| 06/15/1988 | EP0270683A1 Aryloxyureas, process for their preparation, and their use |
| 06/08/1988 | EP0269991A1 Process for the synthesis of 4-cyanoquinuclidine or a salt thereof |
| 06/02/1988 | WO1988003921A1 New benzimidazole derivatives a process for production thereof and a pharmaceutical composition containing the same |
| 03/30/1988 | EP0261964A2 Azabicyclic compounds and their use as 5-ht3 receptor antagonists |
| 03/30/1988 | EP0261763A1 Novel bridged bicyclic N-heterocycles |
| 02/18/1988 | DE3724059A1 Verwendung von mono- und bicyclischen carbocyclischen und heterocyclischen carbonsaeureestern und -amiden von stickstoffhaltigen alkoholen und aminen sowie deren saeureadditionssalzen und quaternaeren ammoniumsalzen sowie von imidazolyl-carbazolen zur behandlung von psychiatrischen stoerungen wie sozialen entzugserscheinungen, manisch-depressiven psychosen, psychosen und anderen in verbindung mit stress stehende krankheiten, stoerungen des wachheitszustandes wie geriatrischen krankheitsbildern, ferner zur behandlung der rhinitis, der lungenembolie und zur verbesserung der nasalen resorption anderer wirkstoffe .......... Use of mono- and bicyclic carbocyclic and heterocyclic carbonsaeureestern and amides of nitrogen-containing alcohols and amines and ammonium salts saeureadditionssalzen thereof and quaternary, as well as imidazolyl -carbazoles for the treatment of psychiatric disorders such as social withdrawal symptoms, manic-depressive psychosis, psychosis and others in connection with stress related diseases, disorders of the alertness state as geriatric disease images, and also for the treatment of rhinitis, pulmonary embolism and for the improvement of nasal resorption other ingredients .......... |
| 02/02/1988 | US4722834 Method of using 2-alkoxy-N-(1-azabicyclo[2.2.2]oct-3-yl)benzamide-N-oxides to control emesis caused by anticancer drugs |
| 01/26/1988 | US4721788 4-cyanopiperidine derivatives |
| 01/26/1988 | US4721783 Anti-spasmodic agents having a heterocyclic ring |
| 01/26/1988 | US4721720 Irritable bowel syndrome |
| 01/05/1988 | US4717563 2-alkoxy-N-(1-azabicyclo(2.2.2)oct-3-yl) benzamides and thiobenzamides in a method for alleviating emesis caused by non-platinum anticancer drugs |
| 12/29/1987 | US4716171 Antiarrhythmic quinidine derivatives |
| 12/08/1987 | US4711885 N-(N'-phenylpiperazine)-alkyl triazole compounds having anxiolytic and analgesic properties |
| 12/03/1987 | WO1987007269A1 Aryloxyureas, process for their preparation, and their use |
| 12/02/1987 | EP0247266A1 Indole derivatives having an azabicyclic side chain, process for their preparation, intermediates, and pharmaceutical compositions |
| 11/18/1987 | CN87102972A Oxadiazoles useful in the treatment of senile dementia |
| 11/10/1987 | US4705854 Phenothiazine compounds |
| 10/07/1987 | EP0240180A1 2-alkoxy-N-(1-azabicyclo[2.2.2]-oct-3-yl) benzamides and thiobenzamides in the alleviation of emesis caused by non-platinum anticancer drugs |
| 09/30/1987 | EP0239309A2 Oxadiazoles useful in the treatment of senile dementia |
| 09/16/1987 | EP0237281A1 2-alkoxy-N-(1-azabicyclo[2.2.2]-oct-3-yl) benzamide-N-oxides in the control of emesis caused by anticancer drugs |
| 09/09/1987 | EP0235878A2 Novel compounds |
| 08/04/1987 | US4684727 Zwitterionic 1,8-naphthyridine and pyrazino[2,3-b]pyridine containing compounds useful as anti-allergic, anti-inflammatory and cycloprotective agents |
| 08/04/1987 | CA1225090A1 Dibenz ¬b,e| oxepin derivatives |
| 06/30/1987 | US4676880 Decarbonylation, detecting microquantitiles of toxic a,a-diar yglycolate esters, forming visible color |
| 06/23/1987 | US4675326 Bisquaternary antidotes |
| 06/09/1987 | US4672119 Chemical agents |
| 06/04/1987 | WO1987003281A1 Propane-1,3-diol derivatives, a method for their production and a pharmaceutical composition |
| 05/27/1987 | EP0223385A2 8-Azabicyclo[3,2,1]octane and 9-azabicyclo[3,3,1]nonane derivatives |
| 05/21/1987 | WO1987000752A3 Zwitterionic bicyclic compounds and their salts, solvates, hydrates and esters |
| 05/19/1987 | CA1221969A1 3-methylflavone-8-carboxylic acid esters |
| 05/13/1987 | EP0221702A2 Quinolidine derivatives |
| 05/13/1987 | EP0052645B1 Gamma-emitting receptor-binding quinuclidinyl benzilates methods of preparation thereof and imaging and assay methods utilizing same |
| 04/14/1987 | US4657911 3-amino quinuclidine derivatives and the application thereof as accelerators of gastro-intestinal motor function |
| 03/31/1987 | US4654337 Perfluoro-1-azatricyclic amine compounds useful as blood substitutes or in infusion fluids |
| 03/17/1987 | CA1219258A1 Perfluoro-1-azatricyclic amine compound |
| 03/11/1987 | EP0213337A1 4-cyanopiperidine derivatives, preparation and use thereof |
| 02/17/1987 | US4644003 3-quinuclidinol esters, useful as antagonists of muscarinic acetylcholine receptors |
| 02/17/1987 | US4643995 Analgesic pyridine-2-ethers or pyridine-2-thioethers having a nitrogen-containing cycloaliphatic ring |
| 02/12/1987 | WO1987000752A2 Zwitterionic bicyclic compounds and their salts, solvates, hydrates and esters |
| 01/06/1987 | US4634701 Furan derivatives having anti-ulcer activity |
| 12/17/1986 | EP0205247A2 Derivatives of quinuclidine |
| 12/03/1986 | CN86103519A Process for preparation of berban derivatives |
| 11/26/1986 | EP0202950A2 Berban derivatives and their preparation and pharmaceutical formulation |
| 11/26/1986 | EP0202710A2 Zirconium phosphate and method for its preparation |
| 11/20/1986 | EP0202062A2 Quinuclidine derivatives |
| 11/12/1986 | EP0201165A2 Medicaments for the treatment of emesis |
| 11/05/1986 | EP0200444A2 Azabicyclononyl-indazole-carboxamide having 5-HT antagonist activity |
| 10/29/1986 | EP0199641A1 Triazole derivatives, process for their preparation and pharmaceutical compositions containing them |
| 10/15/1986 | CN85101353A Process for the preparation of new pyridine-2-ethers or pyridine-2-thioethers having a nitrogen-containing cycloalkyl ring |
| 09/23/1986 | US4613605 Perfluoro-1-azatricyclic amines as blood substitutes |
| 08/13/1986 | EP0190920A2 Method of enhancing memory or correcting memory deficiency with arylamido (and arylthioamido)azabicycloalkanes |
| 08/13/1986 | EP0190915A2 Process for the preparation of 2-alkoxy-N-(1-azabicyclo[2.2.2]octan-3-yl) aminobenzamides |