| Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704) |
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| 08/06/1997 | EP0786988A1 Use of nk1 receptor antagonists for preparing cardio-regulatory drugs |
| 08/06/1997 | CN1156449A Dihygropyridine derivatives as bradykinin antagonists |
| 08/05/1997 | US5654315 Quinuclidine compounds useful in treating diseases |
| 07/30/1997 | EP0515537B1 Substituted urea compounds and their preparation and use |
| 07/23/1997 | EP0785198A1 Method for the preparation of optically active 3-hydroxyquinuclidine |
| 07/23/1997 | EP0784621A1 Quinidine conjugates and their use in immunoassays |
| 07/23/1997 | CN1155279A Neuroprotective 3-(piperidinyl-1)-chroman-4,7,-diol and 1-(4-hydrophenyl)-2-(piperidinyl-1)-alkane alcohol |
| 07/17/1997 | WO1997025317A1 4,5-dihydronaphth[1,2-c]isoxazoles and derivatives thereof having cns activity |
| 07/17/1997 | WO1997025309A1 Carbamoyloxy derivatives of mutiline and their use as antibacterials |
| 07/17/1997 | WO1997025043A1 A method of treating hypercholesterolemia and related disorders |
| 07/17/1997 | CA2240467A1 Carbamoyloxy derivatives of mutiline and their use as antibacterials |
| 07/15/1997 | US5648352 Piperazinylcamphorsulfonyl oxytocin antagonists |
| 07/08/1997 | US5646289 Reacting a 3-chloro-1,2,5-thiadiazole with alkali metal bis(trialkyl or arylsilyl)amide; dechlorination; treating nervous system disorders |
| 07/02/1997 | EP0781274A1 Improved process for r (+) 1,2,3,6-tetrahydro-4-phenyl-1-[(3-phenyl-3-cyclohexen-1-yl)methyl]pyridine, a central nervous system agent |
| 07/01/1997 | US5643923 Treatment of anxiety, cognition activators, senility or alzheimer's |
| 06/24/1997 | US5641791 Heterocyclic compounds and their preparation and use |
| 06/24/1997 | US5641786 Quinuclidine derivatives |
| 06/24/1997 | US5641777 Neurokinin receptor antagonist |
| 06/19/1997 | CA2239508A1 Naphthyl-substituted benzimidazole derivatives as anticoagulants |
| 06/18/1997 | CN1152313A Process for preparation of 2-(1-azabicyclo(2,2,2)oct-3-yl)-2,4,5,6-tetrahydro-1H-benz (DE)isoquinolin-1-1one and intermediate product |
| 06/18/1997 | CN1151893A Combination antiemetic therapy using NK-1 receptor antagonists |
| 06/17/1997 | US5639742 Antibiotic; bactericide |
| 06/12/1997 | WO1997020840A1 1,2,3-thiadiazole carboxylic acid (thio)esters and the use thereof as a pest control agent or as a microbicide |
| 06/12/1997 | WO1997020819A1 Composition for treating pain |
| 06/12/1997 | WO1997020556A1 Method for treating pain |
| 06/12/1997 | DE19545637A1 1,2,3-Thiadiazolcarbonsäure(thio)ester 1,2,3-thiadiazolecarboxylic (thio) ester |
| 06/12/1997 | CA2239732A1 Method for treating pain |
| 06/12/1997 | CA2239580A1 1,2,3-thiadiazole carboxylic acid (thio)esters and the use thereof as a pest control agent or as a microbicide |
| 06/12/1997 | CA2239301A1 Composition for treating pain |
| 06/11/1997 | EP0777671A1 Spiro-azabicyclic compounds useful in therapy |
| 06/11/1997 | EP0777653A1 Dihygropyridine derivatives as bradykinin antagonists |
| 06/11/1997 | EP0777652A1 Neuroprotective 3-(piperidinyl-1)-chroman-4,7-diol and 1-(4-hydrophenyl)-2-(piperidinyl-1)-alkanol derivatives |
| 06/11/1997 | CN1151743A Process for the preparation of azabicyclic derivatives |
| 06/10/1997 | US5637596 Reacting aminomethylindole derivative with a carbonyl containing cyclizing agent; 5-ht3 receptor atagonist; useful for treating anxiety, psychosis, gut motility disorder, emesis, migraine and drug addiction |
| 06/05/1997 | WO1997019944A1 Heterocyclic compounds and their use |
| 06/05/1997 | WO1997019669A2 Heterocyclic compounds and their use |
| 06/05/1997 | CA2238555A1 Heterocyclic compounds and their use |
| 06/04/1997 | EP0776897A1 Heterocyclic compounds and their use |
| 06/04/1997 | EP0776896A1 Heterocyclic compounds and their use |
| 06/03/1997 | US5635526 3-amidopyrazole derivatives, process for preparing these and pharmaceutical compositions containing them |
| 05/28/1997 | EP0468054B1 Benzenesulfonamide derivative |
| 05/22/1997 | WO1997017962A1 Method for treating anxiety |
| 05/22/1997 | WO1997017956A1 Method for treating anxiety |
| 05/22/1997 | WO1997017955A1 Method for treating anxiety |
| 05/22/1997 | CA2237311A1 Method for treating anxiety |
| 05/22/1997 | CA2237220A1 Method for treating anxiety |
| 05/22/1997 | CA2236594A1 Method for treating anxiety |
| 05/22/1997 | CA2235855A1 Morpholine derivatives and their use as therapeutic agents |
| 05/21/1997 | EP0774256A1 Use of azacyclic or azabicyclic thiadiazole compounds for treating anxiety |
| 05/14/1997 | EP0773027A1 Use of azacyclic or azabicyclic pyrazine compounds for treating anxiety |
| 05/14/1997 | EP0773026A2 NK-1 receptor antagonists for the treatment of cancer |
| 05/14/1997 | EP0773021A1 Use of azacyclic or azabicyclic oxadiazole compounds for treating anxiety |
| 05/07/1997 | EP0771199A1 Methods |
| 05/07/1997 | CA2189501A1 Nk-1 receptor antagonists for the treatment of cancer |
| 05/02/1997 | EP0770077A1 Process for the preparation of 2-(1-azabicyclo(2.2.2)oct-3-yl) -2,4,5,6-tetrahydro-1h-benz(de)isoquinolin-1-one and intermediate product |
| 04/30/1997 | CN1034732C Quinuclidine derivative for treatment of inflammatory and gastrointestinal disorders |
| 04/29/1997 | US5625066 Optically active hydroquinine (amino-3 phenyl)-1 ethanesulfonate, preparation and use thereof |
| 04/29/1997 | US5624941 Pyrazole derivatives, method of preparing them and pharmaceutical compositions in which they are present |
| 04/24/1997 | WO1997014417A1 Fibrinogen receptor antagonists |
| 04/24/1997 | CA2234967A1 Fibrinogen receptor antagonists |
| 04/23/1997 | EP0769300A2 Antiemetic composition containing an NK-1 receptor antagonists |
| 04/22/1997 | US5622976 Oxadiazole derivatives having acetylcholinesterase-inhibitory and muscarinic agonist activity |
| 04/22/1997 | US5622712 N-[ω, (ω-1)-dialkyloxy]- and N-[ω, (ω-1)-dialkenyloxy]-alk-1-yl-N, N, N-tetrasubstituted ammonium lipids and uses therefor |
| 04/17/1997 | WO1997013514A1 Nk-1 receptor antagonists for prevention of neurogenic inflammation in gene therapy |
| 04/15/1997 | US5621010 Urea derivatives and their use as ACAT inhibitors |
| 04/09/1997 | EP0766680A1 Substituted dihydrobenzofuran derivatives as 5-ht 4 agonists |
| 04/08/1997 | US5618812 Benzodiazepine derivatives |
| 04/01/1997 | US5616592 Useful for disorders of cardiovascular, gastrointestinal and psychological disorders |
| 03/27/1997 | WO1997011073A1 Novel substituted azacyclic or azabicyclic compounds |
| 03/27/1997 | WO1997011072A1 Novel substituted azacyclic or azabicyclic compounds |
| 03/26/1997 | EP0764165A1 Preparation of stereochemically pure oximes with muscarinic activity |
| 03/25/1997 | US5614629 Benzyl quaternary tropinium compound |
| 03/19/1997 | EP0763026A1 Gastrin and cck antagonists |
| 03/19/1997 | CN1145364A Heterocyclic compounds and their preparation and use |
| 03/18/1997 | US5612381 1,2-ethanediol derivative and salt thereof process for producing the same, and cerebral function-improving agent comprising the same |
| 03/18/1997 | US5612352 Inhibitors of squalene synthase and anticholesterol agents with biphenylquinuclidine derivatives |
| 03/18/1997 | US5612351 Azabicyclic derivatives of 1,2,3-oxa(or thia)diazole |
| 03/18/1997 | US5612336 Heterocyclic amide derivatives as tachykinin antagonists |
| 03/13/1997 | WO1997009308A1 Indolyl neuropeptide y receptor antagonists |
| 03/13/1997 | WO1997009046A1 Compounds and methods |
| 03/13/1997 | CA2203912A1 Indolyl neuropeptide y receptor antagonists |
| 03/06/1997 | WO1997008166A1 Piperazino derivatives as neurokinin antagonists |
| 03/05/1997 | EP0759921A1 Process for the preparation of azabicyclic derivatives |
| 03/05/1997 | EP0759920A1 Derivatives of quinuclidine n-oxide as muscarinic receptor ligands |
| 03/04/1997 | US5607958 Neurotensin receptor binders |
| 02/25/1997 | US5605908 Treating diseases of central nervous system caused by malfunctioning of muscarinic cholinergic system |
| 02/25/1997 | CA2049514C 3-amidopyrazole derivatives, process for preparing these and pharmaceutical compositions containing them |
| 02/20/1997 | WO1997006166A1 Quinidine conjugates and their use in immunoassays |
| 02/19/1997 | EP0758330A1 Biphenylcarboxamides useful as 5-ht1d antagonists |
| 02/18/1997 | US5604241 Substituted benzylaminoquinuclidines as substance P antagonists |
| 02/18/1997 | US5604239 Imidazopyridines as serotonergic 5-HT3 antagonists |
| 02/06/1997 | WO1997003984A1 Resolution of 1-azabicyclo[2.2.2]octan-3-amine, 2-(diphenylmethyl)-n-[[2-methoxy-5-(1-methylethyl)phenyl]methyl] |
| 02/04/1997 | US5599937 Heteroaromatic quinuclidinenes, their use and preparation |
| 01/30/1997 | WO1997003066A1 Substituted benzolactam compounds as substance p antagonists |
| 01/29/1997 | EP0755374A1 Process for peptide segment condensation |
| 01/21/1997 | CA2118704C Fused tricyclic nitrogen containing heterocycles as substance p receptor antagonists |
| 01/16/1997 | WO1997001558A1 Novel substituted azabicyclic compounds |
| 01/15/1997 | CN1140447A Novel carbamate deriv. and medicinal composition contg. the same |
| 01/15/1997 | CN1140165A Arylsulfonyl hydroxamic acid derivatives |
| 01/08/1997 | EP0668863B1 Quinuclidine derivative as substance p antagonist |