Patents
Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704)
09/2002
09/24/2002US6455523 Inhibitors of farnesyl protein transferase
09/19/2002WO2002014311A3 Urea compounds and methods of uses
09/18/2002EP1240167A1 Optically active isomers of quinine and quinidine and their respective biological action
09/18/2002CN1370048A Azabicyclo and azacyclo oxime and amine compounds as pesticides
09/12/2002WO2002070653A2 Peptide deformylase inhibitors
09/12/2002WO2002070494A1 Aryl and heteroaryl urea chk1 inhibitors for use as radiosensitizers and chamosensitizers
09/12/2002WO2002070479A1 N-4-piperidinyl compounds as ccr5 modulators
09/12/2002US20020128271 N-benzenesulfonyl l-proline compounds as bradykinin antagonists
09/11/2002CN1368848A Heterocyclic spiro compounds as pesticides
09/05/2002US20020123507 Bicyclic derivatives
09/04/2002EP1235826A1 Quinuclidine acrylamides
09/04/2002EP1235803A1 Urea compounds having muscarinic receptor antagonist activity
09/04/2002EP1235802A1 Carbamate derivatives having muscarinic receptor antagonist activity
09/03/2002US6444701 Compounds having reversible inhibiting activity of carnitine palmitoyl-transferase
08/2002
08/29/2002US20020119972 Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators for treating respiratory and non-respiratory diseases
08/29/2002DE10106971A1 Arzneimittelformulierung die einen muskarinischen Agonisten enthält Pharmaceutical formulation containing a muscarinic agonist
08/28/2002EP1233964A1 New use and novel n-azabicyclo-amide derivatives
08/28/2002CN1089764C Substituted heterocyclic compounds, preparation method thereof and pharmaceutical compositions containing same
08/22/2002WO2002064124A2 Medicament formulation containing a muscarinic agonist
08/22/2002US20020115678 Compounds, compositions and methods for treating antibiotic-resistant infections
08/22/2002CA2434976A1 Medicament formulation containing a muscarinic agonist
08/20/2002US6436386 Hydroxyapatite-targeting poly (ethylene glycol) and related polymers
08/14/2002EP1230243A1 Poycyloalkylpurines as adenosine receptor antagonists
08/14/2002EP0807111B1 Substituted heterocyclic compounds, preparation method therefor and pharmaceutical compositions containing same
08/14/2002EP0759920B1 Derivatives of quinuclidine n-oxide as muscarinic receptor ligands
08/13/2002US6433168 Chemical intermediate for mequitazine; antihistamines
08/13/2002US6432975 Aromatic alkylene azobicyclic compounds as nicotinic receptor antagonists; antidepressants; nervous system disorder treatment
08/08/2002US20020107392 Quinolinone derivatives
07/2002
07/31/2002EP1225955A1 Aryl olefinic azacyclic, and aryl acetylenic azacyclic compounds, pharmaceutical compositions containing them and their use as inhibitors of nicotinic cholinergic receptors
07/30/2002CA2078039C Process for the production of lactams
07/25/2002WO2002057254A1 Compositions for prevention or treatment of hepatopathy
07/25/2002CA2435141A1 Compositions for prevention or treatment of hepatopathy
07/24/2002EP0900218B1 Heterocyclic compounds
07/23/2002US6423713 Substituted pyrazoles as p38 kinase inhibitors
07/18/2002WO2002055515A1 Chemical derivatives and their use as anti-telomerase agent
07/18/2002WO2002016358A3 Quinuclidine-substituted aryl moieties for treatment of disease (nicotinic acetylcholine receptor ligands)
07/18/2002WO2002016355A3 Quinuclidine-substituted heteroaryl moieties for treatment of disease (nicotinic) acetylcholine receptor ligands
07/18/2002WO2002002556A3 AZA-BRIDGED-BICYCLIC AMINO ACID DERIVATIVES AS α4 INTEGRIN ANTAGONISTS
07/18/2002CA2433723A1 Chemical derivatives and their use as anti-telomerase agent
07/17/2002EP1223169A1 Agent for potentiating nerve growth factor activity containg 1,2-ethanediol derivate or salt thereof
07/17/2002EP0888340B1 4-(benzo-1,3-dioxolyl)-pyrrolidine-3-carboxylic acid derivatives as endothelin antagonists
07/17/2002EP0882044B1 1,4-dihydropyridine compounds as bradykinin antagonists
07/17/2002CN1087737C Dihygropyridine derivatives as bradykinin ant agonists
07/11/2002WO2002053564A2 Quinuclidine derivatives and their use as m3 antagonists
07/11/2002US20020091136 Pharmaceutical compositions containing cinchonine dichlorhydrate
07/11/2002US20020091135 Quinuclidine-substituted heteroaryl moieties for treatment of disease
07/11/2002US20020091115 Aza-bridged-bicyclic amino acid derivatives as alpha4 integrin antagonists
07/10/2002EP1220854A2 Novel tropane analogs
07/10/2002EP1220840A2 Bicyclic and tricyclic amines as modulators of chemokine receptor activity
07/10/2002CN1358188A Diphosphate salt of A4'-substituted-9-deoxo-9A-aza 9A-homoerythromycin derivative and its pharmaceutical composition
07/04/2002WO2002051841A1 Quinuclidine carbamate derivatives and their use as m3 antagonists
07/04/2002CA2441896A1 Quinuclidine carbamate derivatives and their use as m3 antagonists
07/03/2002EP1218349A2 Method for selectively dissociating cyclic carboxylic acid anhydrides
07/03/2002CN1356991A Quinoline and quinoxaline compounds as PDGF-R and/or LCD tyrosine kinase inhibitors
07/02/2002US6413978 Basic derivatives of benz[e] isoindol-1-ones and pyrrolo[3,4-c] quinolin-1-ones with 5-HT3-antagonistic activity, their preparation and their therapeutic use
07/02/2002US6413947 Antiinflammatory agents; rheumatic diseases; anticholesterol agents
06/2002
06/26/2002EP1217001A1 Quinuclidine compounds and drugs containing the same as the active ingredient
06/20/2002WO2002048150A2 Agents useful for reducing amyloid precursor protein and treating demantia and methods of use thereof
06/13/2002WO2002018334A3 Sodium channel modulators
06/13/2002WO2002015662A3 Quinuclidine-substituted heteroaryl moieties for treatment of disease (nicotinic acetylcholine receptor antagonists
06/13/2002WO1999059957A9 Compounds having reversible inhibiting activity of carnitine palmitoyl-transferase
06/12/2002EP1213289A1 N-benzenesulfonyl L-proline compounds as bradykinin antagonists
06/12/2002EP1212301A1 Arylalkyloxyalkylamines and arylalkylthioalkylamines, pharmaceutical compositions containing them and their use as inhibitors of nicotinic cholinergic receptors
06/12/2002EP1211940A1 Azabicyclo and azacyclo oxime and amine compounds as pesticides
06/12/2002EP0984778B1 Neuropeptide-y ligands
06/12/2002EP0885221B1 Azabicyclic esters of carbamic acids useful in therapy
06/12/2002CN1353712A Polymorphs of crystalline (2-benzhydryl-2-azabicyclo [2.2.2] OCT-3-yl)-(5-isopropyl-2-methoxybenzyl)-amine citrate as NK-1 receptor antagonists
06/12/2002CN1353711A Polymorphs of crystalline azabicyclo (2,2,2) octan-3-amine citrate and their pharmaceutical compositions
06/12/2002CN1353702A Adamantane derivatives
06/11/2002US6403596 Substituted pyridones having cytokine inhibitory activity
06/11/2002CA2169838C Antipsychotic method
06/06/2002WO2002044176A1 3-substituted quinuclidines and their use as nicotinic agonists
06/06/2002WO2002044144A2 Nucleophilic approach for preparing radiolabeled imaging agents and associated compounds
05/2002
05/30/2002WO2002020526A3 Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents
05/30/2002WO2002017358A3 Quinuclidine-substituted heteroaryl moieties for treatment of disease (nicotinic acetylcholine receptor antagonists)
05/30/2002WO2002016357A3 Quinuclidine-substituted aryl moieties for treatment of disease (nicotinic acetylcholine receptor ligands)
05/29/2002EP1209157A1 Heteroarylamino and heteroarylsulfonamido substituted 3-benzylaminomethyl piperidines and related compounds
05/29/2002DE10028443C1 Production of optically active 3,3-diaryl-propylamine derivatives comprises six step process from 4-hydroxybenzoic acid or alkyl 4-hydroxybenzoate and cinnamic acid
05/29/2002CN1085529C Use of [R-(Z)]-alpha-(methoxyimino)-alpha-[1-azabicyclw[2.2.2.]oct-3-yl] acetonitrile to reduce amyloid beta A4 formation in Alzheimers disease
05/23/2002WO2002040058A2 Hydroxyapatite-targeting poly(ethylene glycol) and related polymers
05/21/2002US6392103 Using organometallic compound as catalyst
05/16/2002WO2002038528A1 Pleuromutilin derivatives with antimicrobial activity
05/16/2002WO2002016356A3 Quinuclidine-substituted aryl moieties for treatment of disease (nicotinic acetylcholine receptor ligands)
05/16/2002US20020058652 Pharmaceutical compositions and methods for use
05/15/2002CN1349527A Substituted benzolactam compounds
05/14/2002US6387925 Polymorphs of a crystalline azo-bicyclo (2.2.2) oct-3-yl amine citrate and their pharmaceutical compositions
05/14/2002US6387395 N-[1, (1-1) -dialkyloxy] - and N- [1, (1-1) -dialkenyloxy]- alk-1-yl-N,N,N-tetrasubstituted ammonium lipids and uses therefor
05/08/2002CN1347881A 法呢基蛋白转移酶抑制剂 Farnesyl protein transferase inhibitor
05/02/2002US20020052503 Substituted benzolactam compounds as substance p antagonists
05/02/2002US20020052389 Quinuclidine-substituted aryl compounds for treatment of disease
05/02/2002US20020052351 Novel medical use for tachykinin antagonists
05/02/2002US20020052348 Compounds having reversible inhibiting activity of carnitine palmitoyl-transferase
05/02/2002EP1200440A1 Quinuclidine derivatives for treatment of neurological disorders
05/02/2002EP1200431A2 Quinuclidine derivatives and their use as muscarinic m3 receptor ligands
05/02/2002EP0607164B1 Fused tricyclic nitrogen containing heterocycles as substance p receptor antagonists
04/2002
04/30/2002US6380396 Chemical intermediates for antiinflammatory agents
04/25/2002WO2002032863A1 2-, 3-, 4-, or 5-substituted-n1-(benzensulfonyl)indoles and their use in therapy
04/25/2002US20020049225 Quinuclidine-substituted aryl compounds for treatment of disease
04/25/2002US20020049195 Urea compounds that are muscarinic receptor antagonists and agonists, administering to the mammal the urea compound to treat urinary incontinence, chronic pulmonary obstructive disease, asthma, hyper salivation, blurred vision etc.
04/25/2002CA2422717A1 2-, 3-, 4-, or 5-substituted-n1-(benzensulfonyl)indoles and their use in therapy
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