| Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704) |
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| 06/14/2007 | CA2631037A1 Bradykinin 1 receptor antagonists |
| 06/13/2007 | CN1980923A Polycyclic pyridines as potassium ion channel modulators |
| 06/13/2007 | CN1980889A Adamantyl pyrrolidin-2-one derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors |
| 06/07/2007 | WO2007064861A2 Asymmetric friedel-crafts alkylations catalyzed by byfunctional cinchona alkaloids |
| 06/07/2007 | WO2007043653A9 Benzimidazole-5-carboxamide derivative |
| 06/07/2007 | US20070129398 3(R)-1-Phenethyl-(9[H]-xanthene-9-carbonyloxy)-1-azoniabicyclo[2.2.2] octane quaternary salt with a mono- or polyvalent anion; antimuscarinic agents used to treat chronic obstructive pulmonary disease, chronic bronchitis, bronchial hyperreactivity, asthma, or rhinitis |
| 06/06/2007 | CN1976706A Inhibition of FGFR3 and treatment of multiple myeloma |
| 06/06/2007 | CN1976701A 毒蕈碱性乙酰胆碱受体拮抗剂 Muscarinic acetylcholine receptor antagonist |
| 06/06/2007 | CN1319967C 2-acylaminothiazole derivative or salt thereof |
| 06/05/2007 | US7226918 DNA-PK inhibitors |
| 05/31/2007 | WO2007042660A3 Substituted 1-amino-phthalzine derivatives, preparation and therapeutic use thereof |
| 05/31/2007 | US20070123525 5-Substituted indole-2-carboxamide derivatives |
| 05/31/2007 | US20070123475 podophyllotoxin analogs such as 4-beta-[(4''-benzamido)-amino]-4'-demethyl-epipodophyllotoxins and their 4'-ester derivatives used in the chemotherapy for various types of cancer |
| 05/31/2007 | US20070122444 Medical devices employing triazine compounds and compositions thereof |
| 05/30/2007 | EP1790643A1 Quinuclidine compounds having quaternary ammonium group, it's preparation method and use as blocking agents of acetycholine |
| 05/30/2007 | CN1318031C Compositions containing benzoxazinone and nucleoside like materials |
| 05/24/2007 | WO2007028073A3 Synthetic methods and intermediates for stereoisomeric compounds useful for the treatment of gastrointestinal and central nervous system disorders |
| 05/24/2007 | WO2007018738A8 Fused bicycloheterocycle substituted quinuclidine derivatives |
| 05/24/2007 | US20070117817 Pyrimidine derivatives for treatment of hyperproliferative disorders |
| 05/24/2007 | US20070117796 Carbamate compounds as 5-HT4 receptor agonists |
| 05/24/2007 | US20070117795 Methods and compositions of novel triazine compounds |
| 05/23/2007 | EP1786810A1 Ligands for g-protein coupled receptors |
| 05/23/2007 | EP1786809A2 Aminopiperidine derivatives, preparation thereof and use thereof as melanocortin receptor agonists |
| 05/23/2007 | CN1968951A Novel 2-(1-aza-bicyclo[2.2.2]oct-3-yl)-2,3-dihydroisoindol-l-one/5,6-dihydro-furo[2,3-c]pyrrol-4one derivatives ligands for alpha 7 nicotinic acetylcholine receptor |
| 05/22/2007 | US7220856 Substituted quinoline CCR5 receptor antagonists |
| 05/22/2007 | US7220769 Azolylbenzamides and analogues and their use for treating osteoporosis |
| 05/22/2007 | CA2157579C Heterocyclic compounds, their use and preparation |
| 05/17/2007 | US20070112199 Asymmetric aldol additions using bifunctional cinchona-alkaloid-based catalysts |
| 05/17/2007 | US20070112023 (3R)-N-(4'-Aminobiphenyl-4-yl)quinuclidine-3-carboxamide dihydrochloride; nicotinic acetylcholine receptors of alpha7 subtype agonist; high permeability for calcium ions, increases glutamatergic neurotransmission, modulates neuronal plasticity; cognition activator, leaning and perception inhancement |
| 05/17/2007 | US20070111991 10,11-Dihydro-dibenzo[b,f]oxepine-10-carboxylic acid [(1S*,2S*,4R*)-4-butylcarbamoyl-2-hydroxy-1-(3-hydroxy-benzyl)-pentyl]-amide; treatment of neurological and vascular disorders related to beta-amyloid generation and/or aggregation |
| 05/10/2007 | WO2007051496A1 Process for the preparation of n-triazinylammonium salts |
| 05/10/2007 | US20070105897 Novel quinuclidine derivatives and medicinal compositions containing the same |
| 05/10/2007 | US20070105896 3-Imidazol-1-yl-1-azabicyclo[2.2.2]octane; agonist, partial agonist, or antagonist of the alpha 7 nicotinic acetylcholine receptor; antidepressant, anxiolytic agent, cognition activator, neuroprotectant; radiolabel |
| 05/09/2007 | EP1781651A1 Process for preparing quinuclidinium carbamate derivatives |
| 05/09/2007 | EP1781290A2 Anti-inflammatory agents |
| 05/08/2007 | US7214692 Medical use for tachykinin antagonists |
| 05/08/2007 | US7214688 Compounds |
| 05/08/2007 | US7214687 Quinuclidine derivatives and medicinal compositions containing the same |
| 05/08/2007 | US7214686 adjust release of neurotransmitters; Parkinson's disease; tourette Syndrome; attention deficit disorders; schizophrenia |
| 05/03/2007 | WO2006130437A3 Asymmetric carbon-carbon-bond-forming reactions catalyzed by bifunctional cinchona alkaloids |
| 05/03/2007 | US20070099953 3(R)-1-Phenethyl-(9[H]-xanthene-9-carbonyloxy)-1-azoniabicyclo[2.2.2] octane quaternary salt with a mono- or polyvalent anion; antimuscarinic agents used to treat chronic obstructive pulmonary disease, chronic bronchitis, bronchial hyperreactivity, asthma, or rhinitis |
| 05/03/2007 | US20070099874 Methods and compositions of novel triazine compounds |
| 05/02/2007 | EP1608645B1 Pyrazolidine-1,2-dicarboxyldiphenylamide derivatives as coagulation factor xa inhibitors for the treatment of thromboses |
| 05/02/2007 | CN1956964A Tetrahydro-indazole cannabinoid modulators |
| 05/02/2007 | CN1956943A Catalytic asymmetric desymmetrization of prochiral and meso cyclic anhydrides |
| 04/26/2007 | WO2007045478A1 Novel 1-aza bicycloalkyl derivatives for the treatment of psychotic and neurodegenerative disorders |
| 04/26/2007 | WO2007045151A1 Compounds and their pharmaceutical compositions for the treatment of nasal cavum hypersecretion and chronic obstructive pulmonary disease |
| 04/26/2007 | CA2622356A1 Novel 1-aza bicycloalkyl derivatives for the treatment of psychotic and neurodegenerative disorders |
| 04/25/2007 | EP1776360A1 3-(heteroaryl-oxy)-2-alkyl-1-aza-bicycloalkyl derivatives as alpha.7-nachr ligands for the treatment of cns diseases. |
| 04/25/2007 | EP1487834B1 Aza-bicyclic n-biarylamides with affinity for the alpha-7 nicotinic acetylcholine receptor |
| 04/25/2007 | CN1312131C Anti-acid-fast bacterial agents containing pyridonecarboxylic acids as the active ingredent |
| 04/24/2007 | US7208501 Potent and long lasting antimuscarinic agents; respiratory, urological or gastrointestinal disorders |
| 04/19/2007 | WO2007043653A1 Benzimidazole-5-carboxamide derivative |
| 04/19/2007 | US20070088054 Biphenyl derivatives |
| 04/18/2007 | EP1455792B1 Ureas of 2-aminobenzothiazoles as adenosine modulators |
| 04/18/2007 | CN1310914C Acid absorbing agent for preparing cinchona alkaloids ligand |
| 04/18/2007 | CN1310913C Recoverable repeatable use chirality cinchona alkaloid ligand and application |
| 04/17/2007 | US7205318 Inhibitors of trypsin-like serine protease enzymes; for use as anticoagulant agents for therapy of thromboembolic disorders |
| 04/17/2007 | CA2202775C Method for treating anxiety |
| 04/12/2007 | US20070083049 Asymmetric carbon-carbon-bond-forming reactions catalyzed by bifunctional cinchona alkaloids |
| 04/11/2007 | CN1946712A Pyrrolidine derivative |
| 04/11/2007 | CN1946699A Pyridazinone ureas as antagonists of alpha4 integrins |
| 04/05/2007 | WO2007038367A1 Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof |
| 04/05/2007 | US20070078265 Synthetic Methods and Intermediates for Stereoisomeric Compounds Useful for the Treatment of Gastrointestinal and Central Nervous System Disorders |
| 04/05/2007 | CA2622677A1 Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof |
| 04/04/2007 | CN1939307A 2,4,6-triamino-1,3,5-triazine derivative |
| 03/29/2007 | WO2007018738A3 Fused bicycloheterocycle substituted quinuclidine derivatives |
| 03/29/2007 | WO2006108965A3 Npy antagonists, preparation and use |
| 03/29/2007 | US20070072887 Spirofuropyridine aryl derivatives |
| 03/29/2007 | US20070072812 Quaternary salt derivatives of 1,4-diphenylazetidin-2-ones |
| 03/28/2007 | EP1256581B1 Preventive or therapeutic agents for gastric or esophageal regurgitation |
| 03/28/2007 | CN1938283A Pyridazinones as antagonists of alpha4 integrins |
| 03/27/2007 | US7196104 (2-substituted-4-yl-thiazole)-urea-1-pyridine-2-yl derivative effective for prophylaxis and treatment of diseases, such as cell proliferation or apoptosis mediated diseases |
| 03/27/2007 | US7196098 Quinuclidine derivatives and medicinal compositions containing the same |
| 03/27/2007 | US7196095 anti-protoazoal; poultry feed; therapy for cytokine mediated disease i.e. osteoarthritis, cerebral malaria, chronic pulmonary inflammatory disease, silicosis, pulmonary sarcosis, bone resorption diseases, reperfusion injury, graft v. host rejection |
| 03/27/2007 | CA2180841C 1-aminoindan derivatives and compositions thereof |
| 03/22/2007 | US20070066663 disorders of the central and/or peripheral nervous system; minimal interaction with metabolic enzymes, improved selectivity, potentiation, acid resistance, bioavailibility; (3S) N-(2-Methylpropyl)-N-{[2-(trifluoromethyl)-phenyl]methyl}piperidin-3-amine; depression, urinary incontinence; pain |
| 03/22/2007 | US20070066592 5-{6-[(3R)-1-azabicyclo[2.2.2]oct-3-yloxy]pyridazin-3-yl}-1H-indole; attention deficit disorder, attention deficit hyperactivity disorder, Alzheimer's disease, senile dementia, AIDS dementia, Pick's Disease, dementia associated with Down's syndrome; alpha 7 nAChR ligands modulators |
| 03/21/2007 | CN1934109A Composition for solid pharmaceutical preparation of solifenacin or salt thereof |
| 03/21/2007 | CN1934090A Substituted n-cyclohexyl imidazolinones having an mch-modulatory effect |
| 03/15/2007 | US20070060588 Fused bicycloheterocycle substituted quinuclidine derivatives |
| 03/15/2007 | US20070060563 Quinuclidine derivatives binding to mucarinic m3 receptors |
| 03/14/2007 | EP1040103B1 Anilide derivative, production and use thereof |
| 03/14/2007 | CN1930158A New quaternized quinuclidine esters |
| 03/14/2007 | CN1304382C New p2X* receptor antagonists for use in the treatment of inflammatory immune or cardiovascular diseases |
| 03/08/2007 | WO2007028073A2 Synthetic methods and intermediates for stereoisomeric compounds useful for the treatment of gastrointestinal and central nervous system disorders |
| 03/07/2007 | EP1758899A1 Asymmetric michael and aldol addition using bifunctional cinchona-alkaloid-based catalysts |
| 03/07/2007 | EP1442025B1 Pyrimidinones as melanin concentrating hormone receptor 1 |
| 03/06/2007 | US7186731 2-cyanopyrrolidinecarboxamide compound |
| 03/06/2007 | CA2294990C Pharmaceutical compositions and methods for effecting dopamine release |
| 02/28/2007 | EP1757604A1 Process for producing solifenacin or its salt |
| 02/28/2007 | EP1461335B1 2-heteroarylcarboxylic acid amides |
| 02/28/2007 | CN1922176A Condensed bicycle heterocycle substituted quinuclidine derivant |
| 02/28/2007 | CN1922172A Substituted heterocyclic compounds and uses thereof |
| 02/27/2007 | US7183323 Sodium channel modulators |
| 02/27/2007 | US7183277 Alpha-((aryl or heteroaryl)ureido or carbamoyloxy)-N-heteroaryl amides; blood-coagulation factor Xa and VIIa inhibitors; synergistic mixtures with other antitumor agents or anticoagulants |
| 02/22/2007 | US20070043051 Methods and compositions of novel triazine compounds |
| 02/22/2007 | US20070043017 Ring-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use |
| 02/21/2007 | EP1651645B1 N-biarylamides |
| 02/21/2007 | CN1918157A Stereoisomeric compounds and methods for the treatment of gastrointestinal and central nervous system disorders |