| Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704) |
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| 04/19/2006 | EP0885215B1 Novel benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists |
| 04/12/2006 | EP1644370A2 Tetrahydroquinoline derivatives as cannabinoid receptor modulators |
| 04/12/2006 | EP1644335A1 Tetrahydroquinoline derivatives as cannabinoid receptor modulators |
| 04/12/2006 | EP1644325A2 Methods and compositions for treating amyloid-related diseases |
| 04/12/2006 | EP1005356B1 Novel antibacterial agents |
| 04/12/2006 | EP0903337B1 Process for the preparation of 1-alkoxycarbonyl-3-phenylpropyl derivatives |
| 04/12/2006 | CN1759108A Biphenyl derivatives |
| 04/12/2006 | CN1250545C Quinuclidine derivatives and medicine composition containing the derivatives |
| 04/06/2006 | US20060074110 Multicyclic compounds which inhibit leukocyte adhesion mediated by VLA-4 |
| 04/04/2006 | US7022259 include cyclic group chain structures similar to the liquid crystal to serve as the core structure, and multi-ring structures of natural alcohol with optical activity, such as alcoholates of terpenol, borneol, cinchonidine, quinine, or their derivatives; have a high helical twisting power |
| 04/04/2006 | CA2198266C Novel benzimidazole derivatives |
| 03/30/2006 | WO2005112644A3 Muscarinic acetylcholine receptor antagonists |
| 03/30/2006 | WO2005019211A3 Biaryl heterocyclic compounds and methods of making and using the same |
| 03/29/2006 | EP1638677A2 Catalytic asymmetric desymmetrization of prochiral and meso cyclic anhydrides |
| 03/29/2006 | EP1638560A1 3-aminopiperidines and 3-aminoquinuclidines as inhibitors of monoamine uptake |
| 03/29/2006 | CN1753891A Ccr-3 receptor antagonists |
| 03/28/2006 | US7019001 Substituted benzothiazole amide derivatives |
| 03/28/2006 | US7018987 Synthesis of combretastatin A-4 prodrugs and trans-isomers thereof |
| 03/28/2006 | CA2120374C 9-[(substituted glycyl) amido]-6-(substituted)-5-hydroxy-6-deoxytetracyclines |
| 03/23/2006 | WO2005000250A3 Imaging agents and methods of imaging alpha 7-nicotinic cholinergic receptor |
| 03/23/2006 | US20060063809 Tri-substituted heteroaryls and methods of making and using the same |
| 03/22/2006 | CN1751041A 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof |
| 03/16/2006 | WO2006027628A2 Naphthalimide derivatives as antiviral agents |
| 03/16/2006 | WO2005100349A3 Polycyclic pyridines as potassium ion channel modulators |
| 03/15/2006 | EP1633752A1 Isoquinoline-3-carboxylic acid amides and pharmaceutical uses thereof |
| 03/15/2006 | EP1633703A2 Isotopically labeled chemically stable reagents and process for the synthesis thereof |
| 03/15/2006 | EP1633349A1 4-bromo-5- (2-chloro-benzoylamino)-1h-pyrazole-3-carboxylic acid (1-(aminocarbonyl) eth-1-yl) amide derivatives and related compounds as bradykinin b1 receptor antagonists for the treatment of inflammatory diseases |
| 03/15/2006 | EP1633348A1 4- BROMO - 5 - (2- CHLORO - BENZOYLAMINO) - 1H - PYRAZOLE - 3 - CARBOXYLIC ACID AMIDE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ B sb 1 /sb RECEPTOR ANTAGONISTS FOR THE TREATMENT OF INFLAMMATORY DISEASES |
| 03/15/2006 | EP1309589B1 Urea compounds and methods of uses |
| 03/14/2006 | US7012078 For therapy and prophylaxis of migraine, inflammatory diseases, stroke, acute and chronic pain, hypovolemic shock, traumatic shock, reperfusion injury, Crohn's disease, ulcerative colitis, septic shock, multiple sclerosis, etc. |
| 03/14/2006 | CA2376748C Diphosphate salt of a 4''-substituted-9-deoxo-9a-aza-9a-homoerythromycin derivative and its pharmaceutical composition |
| 03/14/2006 | CA2180963C Novel high enantio-selective process for producing pure enantiomeric cyclopentane and cyclopentene-.beta.-amino acids |
| 03/09/2006 | CA2577964A1 Ligands for g-protein coupled receptors |
| 03/08/2006 | EP1631569A2 Quinuclidine derivatives binding to mucarinic m3 receptors |
| 03/07/2006 | US7008951 Such as asthma or chronic obstructive pulmonary disease; mixture of a corticoid such as budesonide, fluticasone propionate or mometasone furoate and 5-(1-hydroxy-2-((5,6-diethylindan-2-yl)amino)ethyl)8-hydroxy-1,2-dihydroquinolin-2-one or its salt |
| 03/02/2006 | WO2006021656A2 Aminopiperidine derivatives, preparation thereof and use thereof as melanocortin receptor agonists |
| 03/02/2006 | WO2005072132A3 TRICYCLIC MODULATORS OF THE GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-κB ACTIVITY AND USE THEREOF |
| 03/02/2006 | US20060047122 Process for producing optically active-3-quinuclidinols |
| 03/02/2006 | CA2574454A1 Aminopiperidine derivatives, preparation thereof and use thereof as melanocortin receptor agonists |
| 03/01/2006 | EP1628974A2 Hydantoin derivatives as inhibitors of tumor necrosis factor-alpha converting enzyme (tace) |
| 02/23/2006 | WO2006018609A2 Anti-inflammatory agents |
| 02/23/2006 | CA2577274A1 Anti-inflammatory agents |
| 02/22/2006 | EP1626967A1 Substituted pyrazoles |
| 02/21/2006 | US7001914 Compounds |
| 02/21/2006 | US7001900 Central nervous system disorders |
| 02/15/2006 | CN1733762A Acid absorbing agent for preparing cinchona alkaloids ligand |
| 02/08/2006 | CN1732154A Alkyne compounds with MCH antagonistic activity and medicaments comprising these compounds |
| 02/02/2006 | WO2006010452A1 Process for preparing quinuclidinium carbamate derivatives |
| 02/02/2006 | WO2005092890A3 Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof |
| 02/01/2006 | CN1239502C Macromolecule immobilized cinchonine alkaloid ligand, synthesis method and use thereof |
| 01/31/2006 | CA2208839C Quinuclidine derivatives and medicinal composition thereof |
| 01/26/2006 | US20060019996 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto |
| 01/25/2006 | EP1618087A2 Antibacterial agents |
| 01/19/2006 | WO2006005608A1 3-(heteroaryl-oxy)-2-alkyl-1-aza-bicycloalkyl derivatives as alpha.7-nachr ligands for the treatment of cns diseases |
| 01/19/2006 | US20060014964 Bicyclic and tricyclic amines as modulators of chemokine receptor activity |
| 01/19/2006 | US20060014956 Asymmetric Michael and Aldol additions using bifunctional cinchona-alkaloid-based catalysts |
| 01/19/2006 | US20060014780 Nicotinamide derivatives useful as PDE4 inhibitors |
| 01/19/2006 | CA2570155A1 3-(heteroaryl-oxy)-2-alkyl-1-aza-bicycloalkyl derivatives as alpha.7-nachr ligands for the treatment of cns diseases |
| 01/18/2006 | EP1615889A2 Biphenyl derivatives having beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity |
| 01/18/2006 | EP1363612A4 Peptide deformylase inhibitors |
| 01/12/2006 | WO2005111033A3 Novel azabicyclic aryl derivatives |
| 01/10/2006 | CA2364178C N-benzenesulfonyl l-proline compounds as bradykinin antagonists |
| 01/05/2006 | DE69828607T2 CHINOLIN- UND CHINOXALIN-VERBINDUNGEN DIE DEN VON BLUTPLÄTTCHEN ABSTAMMMENDEN WACHSTUMSFAKTOR UND/ODER PDGF- UND P56lck-TYROSIN-KINASE HEMMEN Quinoline and quinoxaline THE COMPOUNDS OF THE PLATELET FACTOR ABSTAMMMENDEN GROWTH AND / OR PDGF-TYROSINE KINASE AND p56 HEMMEN |
| 01/04/2006 | CN1234679C Shortened synthesis of 3, 3-diaryl propylamine derivatives |
| 01/03/2006 | US6982271 selective norepinephrine and serotonin reuptake inhibitor (SSNRI); antidepressant; treating cocaine addiction; "N3 bridged" tropanes |
| 12/29/2005 | WO2005123671A1 Pyrrole derivative |
| 12/29/2005 | US20050288315 4-((7-chloroquinolin-4-yl)aminoalkyleneamino-)-spiro(cyclohexane-1.5'-1H-4,5,6-trioxaindene )dicitrate; malaria; paraciticides; antiprotozoa agents; Plasmodium; synergistic; chloroquine-resistant; cost efficiency; industrial scale; penetration and activity of artemisine |
| 12/28/2005 | EP1609790A2 Benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists |
| 12/28/2005 | EP1608645A1 Pyrazolidine-1,2-dicarboxyldiphenylamide derivatives as coagulation factor xa inhibitors for the treatment of thromboses |
| 12/28/2005 | EP1608374A1 2-phenoxy- and 2-phenylsulfomamide derivatives with ccr3 antagonistic activity for the treatment of asthma and other inflammatory or immunological disorders |
| 12/28/2005 | EP1389208B1 Substituted azabicyclic moieties for the treatment of disease (nicotinic acethylcholine receptor agonists) |
| 12/22/2005 | WO2005121137A1 Asymmetric michael and aldol addition using bifunctional cinchona-alkaloid-based catalysts |
| 12/22/2005 | WO2005120707A1 Clean osmium-catalyzed asymmetric dihydroxylation and aminohydroxylation of olefins in ionic liquids followed by supercritical co2 product recovery |
| 12/22/2005 | US20050283006 Heteroaryl-substituted pyrrole derivatives, their preparation and their therapeutic uses |
| 12/22/2005 | US20050282857 e.g. 1-(4-amino-3-chloro-5-trifluoromethyl-benzyl)-2-oxo-2-[4-(2-piperidin-1-yl-ethyl)-piperidin-1-yl]-ethyl 4-(2-oxo-1 ,2,4,5-tetrahydro-benzo[d][1,3]diazepin-3-yl)-piperidine-1-carboxylate; calcitonin gene related peptide antagonist; migraine or cluster headaches, non-insulin-dependent diabetes |
| 12/21/2005 | EP1606288A1 Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain |
| 12/21/2005 | CN1709891A Medicinal compound, its composition and use in pharmaceutical process |
| 12/15/2005 | WO2004098590A8 4-bromo-5- (2-chloro-benzoylamino)-1h-pyrazole-3-carboxylic acid (1-(aminocarbonyl) eth-1-yl) amide derivatives and related compounds as bradykinin b1 receptor antagonists for the treatment of inflammatory diseases |
| 12/15/2005 | US20050277640 Pyrimidine derivatives for treatment of hyperproliferative disorders |
| 12/14/2005 | CN1708493A Selected CGRP antagonists, method for production and use thereof as medicament |
| 12/14/2005 | CN1231480C 1,2,3-thiadiazole carboxylic acid (thio) esters and use thereof as pest control agent or as microbicide |
| 12/14/2005 | CN1231455C Continuously hydrogen adding method |
| 12/14/2005 | CN1231212C Multicyclic compounds which inhibit beukocyte adhesion mediated by VLA-4 |
| 12/08/2005 | WO2005116012A1 Pyrrolidine derivative |
| 12/08/2005 | WO2004098589A8 4- bromo - 5 - (2- chloro - benzoylamino) - 1h - pyrazole - 3 - carboxylic acid amide derivatives and related compounds as bradykinin b1 receptor antagonists for the treatment of inflammatory diseases |
| 12/08/2005 | US20050272763 antagonists of the Cannabinoid-1 (CB1) receptor; treating obesity |
| 12/08/2005 | US20050272753 signal transducer and activator of transcription-6 inhibitors; asthma, COPD, respiratory, inflammatory and allergic diseases; compounds have less suppressive effect on immunological functions; 4-[(2,5 -difluorobenzyl) amino]-2-[(4-morpholin-4-ylphenyl)amino]pyrimidine-5 -carboxamide |
| 12/08/2005 | US20050272739 N-aryl diazaspiracyclic compounds and methods of preparation and use thereof |
| 12/08/2005 | CA2564668A1 Pyrrolidine derivatives |
| 12/07/2005 | EP1601635A1 Process for producing optically active alcohol in the presence of rhodium, a chiral ferrocenyldiphosphine and an optically active diamine |
| 12/07/2005 | EP1217001B1 Quinuclidine compounds and drugs containing the same as the active ingredient |
| 12/07/2005 | CN1705664A Process for the preparation of (S,S)-cis-2-benzhydryl-3-benzylaminoquinuclidine |
| 12/01/2005 | WO2005112644A2 Muscarinic acetylcholine receptor antagonists |
| 12/01/2005 | WO2005077899A3 Amino-substituted tricyclic derivatives and methods of use |
| 12/01/2005 | US20050267111 Pharmaceutical compositions and methods for use |
| 11/30/2005 | EP1599472A1 Ccr-3 receptor antagonists |
| 11/30/2005 | CN1703403A Metabotropic glutamate receptor antagonists |
| 11/30/2005 | CN1229375C Nicotinic acetylcholine receptor inhibitor, its prepn. and application |
| 11/29/2005 | US6969726 can be used as anti-proliferative agents and/or anti-infective agents that can be used without limitation as anti-inflammatory agents |
| 11/24/2005 | WO2005111033A2 Novel azabicyclic aryl derivatives |