| Patents for C07D 453 - Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids (5,704) |
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| 05/02/2012 | EP1517905B1 Processes for preparing substituted pyrimidines and pyrimidine derivatives as inhibitors of protein kinases |
| 05/02/2012 | CN102438988A Resorcinol derivatives as hsp90 inhibitors |
| 05/01/2012 | US8168791 N-[(4r)-1-azatricyclo[3.3.1.13,7]dec-4-ylmethyl]-5-chloro-1H-indole-2-carboxamide; disorders or deficits modulated by an alpha 7 nicotinic acetylcholine receptor, an alpha 4 beta 2 nicotinic acetylcholine receptor or both; schizophrenia |
| 05/01/2012 | US8168656 Indoleacetic acid and indenacetic acid derivatives as therapeutic agents with reduced gastrointestinal toxicity |
| 05/01/2012 | US8168654 Quinuclidine derivatives binding to mucarinic M3 receptors |
| 04/26/2012 | WO2012052297A1 Carbonate derivatives for the treatment of cough |
| 04/26/2012 | US20120101094 Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof |
| 04/26/2012 | CA2815035A1 Carbonate derivatives for the treatment of cough |
| 04/25/2012 | EP2121137B1 Quinuclidinol derivatives as muscarinic receptor antagonists |
| 04/25/2012 | EP1719768B1 Novel benzothiazepine and benzothiepine compounds |
| 04/17/2012 | US8158784 Quinuclidine derivative useful in the preparation of mequitazine |
| 04/17/2012 | US8158649 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof |
| 04/17/2012 | US8158380 Imaging agents for protein misfolding |
| 04/12/2012 | US20120088917 New quinuclidine derivative useful in the preparation of mequitazine |
| 04/12/2012 | US20120088778 Azole derivatives and fused bicyclic azole derivatives as therapeutic agents |
| 04/11/2012 | EP1651612B1 3,4-disubstituted 1h-pyrazole compounds and their use as cyclin dependent kinases (cdk) and glycogen synthase kinase-3 (gsk-3) modulators |
| 04/10/2012 | US8153843 Antibacterial agents |
| 04/10/2012 | US8153799 Azabicyclic carbamates and their use as alpha-7 nicotinic acetylcholine receptor agonists |
| 04/04/2012 | CN102397793A 一类金鸡纳碱-方酰胺氢键催化剂、合成方法及其在不对称反应中的应用 A class of cinchona alkaloids - square amide hydrogen catalyst synthesis method and its application in asymmetric reactions |
| 03/28/2012 | EP2313404B1 Quinuclidine carbonate derivatives and medicinal composition thereof |
| 03/28/2012 | EP1432707B1 Azabicyclic-substituted fused-heteroaryl compounds for the treatment of disease |
| 03/27/2012 | US8143272 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof |
| 03/22/2012 | US20120073001 Methods and compositions for treating or preventing pruritis |
| 03/21/2012 | EP2431037A1 (2S,3R)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofuran-2-carboxamide, novel salt forms, and methods of use thereof |
| 03/20/2012 | US8138168 Renin inhibitors |
| 03/20/2012 | US8137582 Alkaloid monomers, liquid crystal compositions and polymer networks derived therefrom |
| 03/20/2012 | CA2472711C 2-acylaminothiazole derivative or salt thereof |
| 03/20/2012 | CA2405076C Dual molecules containing a peroxide derivative, synthesis and therapeutic applications thereof |
| 03/14/2012 | CN102372692A Dihydropyridine derivative |
| 03/13/2012 | US8134003 Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof |
| 03/07/2012 | EP2137180B1 Dibenzo [b,f][1,4] oxazapine compounds |
| 03/06/2012 | US8129405 Quinuclidine derivatives and medicinal compositions containing the same |
| 02/29/2012 | EP2423207A2 2-(cyclic amino)-pyrimidone derivatives as TPK1 inhibitors |
| 02/29/2012 | EP2421833A1 Resorcinol derivatives as hsp90 inhibitors |
| 02/28/2012 | US8124620 3-Substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof |
| 02/28/2012 | US8124619 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof |
| 02/28/2012 | US8124618 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof |
| 02/23/2012 | WO2012024397A2 2,5-methano-and 2,5-ethano-tetrahydrobenzazepine derivatives and use thereof to block reuptake of norepinephrine, dopamine, and serotonin |
| 02/23/2012 | US20120046468 Intermediates in the enantioselective synthesis of 3-(aminomethyl)-5-methyl-hexanoic acid |
| 02/23/2012 | US20120046266 Resorcinol derivatives as hsp90 inhibitors |
| 02/21/2012 | US8119808 Tetrahydroquinoline derivatives as cannabinoid receptor modulators |
| 02/21/2012 | US8119659 (2S,3R)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofuran-2-carboxamide, novel salt forms, and methods of use thereof |
| 02/07/2012 | CA2529269C Improved pharmaceutical drug candidates and methods for preparation thereof |
| 02/02/2012 | US20120029197 Method for Preparing Sulfur-Containing Compounds |
| 01/31/2012 | CA2514135C 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof |
| 01/26/2012 | US20120022100 Organic compounds |
| 01/26/2012 | US20120022099 Novel polymorphic forms of an azabicyclo-trifluoromethyl benzamide derivative |
| 01/25/2012 | EP2409703A1 Treatment with alpha7-selective ligands |
| 01/25/2012 | EP1988075B1 Pyrrole derivative or salt thereof |
| 01/25/2012 | CN102329314A Industrial preparation method of palonosetron hydrochloride |
| 01/25/2012 | CN102329313A Azasetron hydrochloride compound and preparation method thereof |
| 01/24/2012 | US8101640 Antibacterial agents |
| 01/19/2012 | WO2012008435A1 Biaryl amide derivative or pharmaceutically acceptable salt thereof |
| 01/19/2012 | US20120015925 Novel benzothiazepine and benzothiepine compounds |
| 01/18/2012 | EP2406257A1 A new method for the preparation of solifenacin and new intermediate thereof |
| 01/18/2012 | CN1976706B Inhibition of FGFR3 and treatment of multiple myeloma |
| 01/17/2012 | US8097750 Highly enantioselective, converting aromatic and aliphatic aldehydes into optically active aryl and alkyl beta -amino acids |
| 01/12/2012 | WO2012004264A1 Solifenacin salts |
| 01/12/2012 | US20120010200 Biaryl Heterocyclic Compounds And Methods Of Making And Using The Same |
| 01/12/2012 | CA2804107A1 Solifenacin salts |
| 01/10/2012 | CA2564742C Quaternary quinuclidine derivatives and their use as muscarinic receptor antagonists |
| 01/05/2012 | WO2012001481A1 Novel process for the preparation of solifenacin succinate |
| 01/05/2012 | WO2012000925A1 Preparation of n-(s)-1-azabicyclo[2.2.2]oct-3-yl-1h-indazole-3-carboxamide hydrochloride salt |
| 01/05/2012 | US20120004413 Isotopically labeled chemically stable reagents and process for the synthesis thereof |
| 01/05/2012 | US20120004258 Quinuclidine carbonate salts and medicinal composition thereof |
| 01/04/2012 | EP1735286B1 Tetrahydro-indazole cannabinoid modulators |
| 01/03/2012 | US8088794 Substituted amide derivatives and methods of use |
| 01/03/2012 | CA2456717C Phenyl derivatives as factor xa inhibitors |
| 12/29/2011 | WO2011161018A1 Alkaloid aminoester derivatives and medicinal compositions thereof |
| 12/29/2011 | WO2011160919A1 Alkaloid aminoester derivatives and medicinal composition thereof |
| 12/29/2011 | WO2011160918A1 Alkaloid aminoester derivatives and medicinal composition thereof |
| 12/29/2011 | WO2011160252A1 Organic acid salts of penehyclidine optical isomer |
| 12/29/2011 | US20110319621 Method for the preparation of solifenacin and intermediate thereof |
| 12/29/2011 | US20110319407 Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and use thereof |
| 12/29/2011 | US20110318688 Salt, acid generator and resist composition |
| 12/29/2011 | CA2803459A1 Alkaloid aminoester derivatives and medicinal compositions thereof |
| 12/29/2011 | CA2803433A1 Alkaloid aminoester derivatives and medicinal composition thereof |
| 12/29/2011 | CA2803416A1 Alkaloid aminoester derivatives and medicinal composition thereof |
| 12/28/2011 | EP1414456B1 Phenyl derivatives as factor xa inhibitors |
| 12/28/2011 | CN102293773A 含有苯并硫氮杂卓和苯并虑平化合物的药物 Benzothiazepine and benzo drugs containing compounds doxepin |
| 12/27/2011 | US8084615 Antibacterial agents |
| 12/27/2011 | US8084463 Quinuclidine derivatives and their use as muscarinic M3 receptor antagonists |
| 12/27/2011 | US8084462 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof |
| 12/22/2011 | US20110312994 Biphenyl derivatives |
| 12/22/2011 | US20110312903 Fluorination of organic compounds |
| 12/22/2011 | US20110311461 Alkaloid aminoester derivatives and medicinal composition thereof |
| 12/22/2011 | US20110311459 Alkaloid aminoester derivatives and medicinal composition thereof |
| 12/22/2011 | US20110311458 Alkaloid aminoester derivatives and medicinal compositions thereof |
| 12/21/2011 | EP2396300A1 New substituted tetrahydronapthalenes, method for the production thereof, and use thereof as drugs |
| 12/21/2011 | CN102292335A (2s,3r)-n-2-((3-吡啶基)甲基)-1-氮杂双环[2.2.2]辛-3-基)-3,5-二氟苯甲酰胺的制备和治疗应用 (2s, 3r) -n-2 - ((3- pyridinyl) methyl) -1-azabicyclo [2.2.2] oct-3-yl) -3,5-difluorophenyl-carboxamide and therapeutic use |
| 12/20/2011 | US8080666 3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators |
| 12/20/2011 | US8080663 Process for the preparation of 2-methylspiro(1,3-oxathiolane-5,3′)quiniclidine |
| 12/15/2011 | US20110306612 Quinazolinone, quinolone and related analogs as sirtuin modulators |
| 12/13/2011 | US8076355 2-heteroarylcarboxylic acid amides |
| 12/08/2011 | US20110301352 Process for the preparation of cis-2-methylspiro (1, 3-oxathiolane 5-3') quinuclidine |
| 12/07/2011 | EP1940832B1 Novel 1-aza bicycloalkyl derivatives for the treatment of psychotic and neurodegenerative disorders |
| 12/07/2011 | CN102267924A 抗菌剂 Antibacterial agents |
| 12/07/2011 | CN101797519B 氟代双苯磺酰亚胺作为氮杂Diels-Alder反应催化剂的应用 Application catalyst fluorinated double Benzenesulfonimide as aza-Diels-Alder reaction |
| 12/06/2011 | US8071601 Aminoquinoline derivatives and their use as adenosine A3 ligands |
| 12/06/2011 | CA2504160C Novel alkyne compounds having an mch antagonistic effect and medicaments containing these compounds |