Patents
Patents for C07D 489 - Heterocyclic compounds containing 4ah-8, 9 c- iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: (2,334)
05/2003
05/14/2003EP1310251A1 Antipruritic agent
05/13/2003US6562835 One morphinan selected from the group consisting of dextromethorphan, dextrorphan and at least one active agent selected from tricyclic antidepressants, antispasmodics, direct-acting bladder smooth muscle relaxants, and estrogens
05/07/2003EP0614898B1 Indole derivative, process for producing the same, and medicinal use thereof
05/01/2003US20030083499 Pyridomorphinans and use thereof
05/01/2003US20030083476 Morphine-6-glucuronide synthesis
04/2003
04/16/2003CN1105721C Process for preparing narcotic analgesics
04/09/2003CN1408714A Novel oripavine derivative and its medical use
04/02/2003EP0770081B1 Heterocycle-condensed morphinoid derivatives
04/02/2003CN1407884A Controlled release hydrocodone formulations
03/2003
03/27/2003WO2003024972A1 New oripavine derivatives and their uses as medicines
03/18/2003US6534514 Compound and selectively blocking the binding of a kappa opioid-receptor agonist to kappa opioid receptors in mammalian tissues
03/18/2003US6534092 Method for preparing microparticles having a selected polymer molecular weight
03/06/2003WO2003018588A2 Process for the preparation of a 14-hydroxynormorphinone derivative
03/06/2003US20030045720 Mixing the narcotic alkaloid with an acid in the presence of a catalyst in the substantial absence of hydrogen gas
02/2003
02/27/2003WO2003015783A1 Method of treating alcoholism or alcohol abuse
02/27/2003WO2002083135A3 Use of buprenorphine for the manufacture of a transdermal delivery device for the treatment of urinary incontinence, especially urge incontinence
02/26/2003EP1285902A1 Method for labeling with tritium
02/20/2003WO2003014122A1 Derivatives of morphine-like opioid compounds
02/20/2003WO2002098427A3 Sustained-release analgesic compounds
02/12/2003EP1282404A2 Method for preparing microparticles having a selected polymer molecular weight
02/11/2003CA2154620C Method of detecting surface contamination by an analyte
02/04/2003US6514773 Method of detecting surface contamination by an analyte
01/2003
01/30/2003WO2003007966A1 Active substance combination for medicamentous therapy of nicotine dependency
01/30/2003US20030023104 For prolonging or altering the activity of a compound which is a member of the chlorambucil family
01/30/2003US20030022876 Sustained-release analgesic compounds
01/28/2003US6512117 Method of preparing a ketone from a narcotic alkaloid having an allyl alcohol moiety comprising: mixing the narcotic alkaloid with an acid in the presence of a catalyst wherein the method is carried out in the substantial absence of
01/28/2003US6512115 Preparation of pigments
12/2002
12/19/2002US20020192277 Controlled release hydrocodone formulations
12/18/2002EP0880526B1 Heterocycle-condensed morphinoid derivatives (ii)
12/17/2002CA2095223C Topical compositions for transdermal delivery of prodrug derivatives of morphine
12/12/2002WO2002098427A2 Sustained-release analgesic compounds
12/12/2002CA2448665A1 Sustained-release analgesic compounds
11/2002
11/27/2002CN1382145A Remedies for neuropathic pain and model animals of neuropathic pain
11/14/2002WO2002089845A1 Remedies for sepsis
11/07/2002US20020165247 Use of morphine derivatives as medicaments for the treatment of neuropathic problems
11/07/2002US20020164373 Opioid sustained-released formulation
11/05/2002US6476044 Use of morphine derivatives as medicaments for the treatment of neuropathic problems
10/2002
10/31/2002WO2002043713A3 Use of weak opioids and mixed opioid agonists/antagonists for treating urinary incontinence
10/24/2002WO2002083135A2 Use of buprenorphine for the manufacture of a transdermal delivery device for the treatment of urinary incontinence, especially urge incontinence
10/22/2002US6469170 Method for preparing oxycodone
10/17/2002WO2002081477A1 7-substituted morphinane derivatives and medicinal use thereof
10/17/2002WO2002080918A1 Remedial or prophylactic agent for frequent urination or urinary incontinence
10/17/2002WO2002070524A3 N-but-3-enyl norbuprenorphine and its use as analgesic
10/16/2002CN1374963A Remedies or preventives for freqent urination or arinary incontinence
10/15/2002US6465479 Pyridomorphinans and use thereof
10/10/2002WO2002078744A1 Remedies for psychoneurosis
10/03/2002US20020143183 Producing a dienol organosilyl ether at position 6 of the C-ring of codeinone thereby forming dienol organosilyl ether congener of codeinone; oxidizing dienol organosilyl ether to form 14-hydroxycodeinone; hydrogenating to produce oxycodone
10/02/2002EP1244448A2 Novel methods for the treatment and prevention of ileus
10/02/2002EP1086114B1 Morphine-6-glucuronide synthesis
09/2002
09/26/2002WO2002028917A3 Resin and its use in converting morphine to codeine
09/26/2002US20020137760 Antipruritic
09/12/2002WO2002070567A1 Novel compound, process for producing the same, and use thereof as support for solid-phase reaction
09/12/2002WO2002070524A2 N-but-3-enyl norbuprenorphine and its use as analgesic
09/12/2002CA2439859A1 N-but-3-enyl norbuprenorphine and its use as analgesic
09/06/2002WO2002067916A2 Pharmaceutical salts
09/06/2002WO2002067651A2 Pharmaceutical salts
09/06/2002CA2725635A1 Pharmaceutical salts of 6-dimethylaminomethyl-1-phenylcyclohexane compounds
09/05/2002DE10109763A1 Pharmazeutische Salze Pharmaceutical Salts
09/04/2002CN1090190C Heterocycle-condensed morphinoid derivatives and its preparing method and use
09/04/2002CN1090189C Pyrazolopyrimidines type compound
08/2002
08/29/2002WO2002066031A1 Utilization of buprenorphine in urinary incontinence therapy
08/29/2002US20020119203 Preparing first phase comprising nucleophilic active agent, a polymer and solvent; combining with second phase in a static mixer to form emulsion; extracting solvent from the emulsion, thereby forming microparticles
08/28/2002EP1233966A1 Hydromorphinone and hydrocodeinone compositions and methods for their synthesis
08/27/2002US6440987 Antipruritic
08/08/2002US20020106761 Production of thebaine and oripavine
08/07/2002EP1227798A1 Controlled release hydrocodone formulations
07/2002
07/24/2002EP1224188A2 A salt of morphine
07/03/2002EP1219624A1 Remedies for neuropathic pain and model animals of neuropathic pain
06/2002
06/27/2002US20020082357 Resin comprising a solid support and at least one cationic methylated sulfonium, sulfoxonium, selenonium or phosphonium salt immobilized on the solid support for use as methylating agent
06/11/2002US6403798 Method for preparing oxycodone
06/11/2002US6403602 Morphine-6-sulfate analogues and their use for the treatment of pain
06/06/2002WO2002043713A2 Use of weak opioids and mixed opioid agonists/antagonists for treating urinary incontinence
06/06/2002DE10059415A1 Verwendung von schwachen Opioiden und gemischten Opioidagonisten/-antagonisten zur Therapie der Harninkontinenz Use of weak opioids and mixed opioid agonist / antagonist for the treatment of urinary incontinence
06/05/2002EP1210084A1 Pyridomorphinans, thienomoprhinans and use thereof
05/2002
05/28/2002US6395900 N-deprotection and/or o-demethylation of an opioid compound or of a nonpeptidic delta tert-amide agonist with a lithium trialkylborohydride
05/15/2002EP1204414A2 Use of morphinan derivates as medicines
05/15/2002EP1204406A2 Opioid sustained-released formulation
05/14/2002US6387917 Nasal administering
05/10/2002WO2002036573A2 8- substituted-2, 6-methano-3-benzazocines and 3-substituted morphinanes as opioid receptor binding agents
05/10/2002WO2002036099A1 Controlled release hydrocodone formulations
05/10/2002WO2001046198A3 Nonpeptide kappa opioid receptor antagonists
05/08/2002EP1203771A1 Remedies or preventives for frequent urination or urinary incontinence
05/02/2002WO2001042207A3 Novel methods for the treatment and prevention of ileus
05/02/2002EP1200089A1 Pyridomorphinans and use thereof
04/2002
04/30/2002US6379704 Method for preparing microparticles having a selected polymer molecular weight
04/23/2002US6376221 Harvesting poppy capsules of stably reproducing papaver somniferum to produce straw containing thebaine and oripavine in at least 50% by weight of alkaloid mixture formed, chemically extracting thebaine and/or oripavine
04/18/2002WO2002030936A1 Pyrrole-condensed morphinoid derivatives
04/18/2002WO2002030935A1 Morphinoid derivatives as delta-opioid agonists and antagonists
04/18/2002US20020045755 N-deprotection and/or O-demethylation of an opioid compound or of a nonpeptidic delta tert-amide agonist with a lithium trialkylborohydride
04/11/2002WO2002028917A2 Resin and its use in converting morphine to codeine
04/10/2002EP0915884B1 Preparation of narcotic analgesics
04/02/2002US6365742 Preparation of opiates, intermediates and uses of salts
04/02/2002US6365594 As opioid agonists and antagonists and are useful as i.a. analgesics
03/2002
03/20/2002EP1017696B1 Acidic addition salts of morphine alkaloids and the application thereof
03/19/2002US6359111 Useful in treating cancer, and in a method of imaging opioid receptors either inside or outside of the central nervous system
03/07/2002WO2001029047A3 Method for preparing oxycodone
03/06/2002EP1183027A1 Pharmaceutical formulations and methods comprising intranasal morphine
02/2002
02/28/2002WO2002016367A1 Chemical methods
02/21/2002WO2001089482A3 Method for preparing microparticles having a selected polymer molecular weight
02/13/2002EP0861250B1 Amidine and isothiourea derivatives as inhibitors of nitric oxide synthase
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