Patents
Patents for C07D 477 - Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula: , e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring (2,484)
03/1996
03/21/1996WO1996008491A1 Novel carbapenem derivative
03/21/1996CA2199855A1 Novel carbapenem derivative
03/14/1996WO1996007655A1 Novel carbapenem derivative
03/13/1996EP0700382A1 Novel n-arylaliphatic-n-alkyl-functionalised amides, method for their prepation and pharmaceutical compositions containing same
03/05/1996US5496816 Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment
02/1996
02/27/1996US5495012 Process for preparing optically active 4-mercapto-2-pyrrolidone derivative and intermediate therefor
02/20/1996US5493018 Process for synthesizing carbapenem intermediates using a rhodium catalyst and lewis acid
02/15/1996WO1996004286A1 Process for making quinolonyl lactam antimicrobials and novel intermediate compounds
02/15/1996WO1996004282A1 Carbapenem compounds, compositions and methods of treatment
02/13/1996US5491139 Antimicrobial quinolonyl lactams
02/07/1996EP0695753A1 Carbapenem derivatives containing a bicyclic substituent, process for their preparation, and their use
02/07/1996EP0695295A1 3-(hetero)aryl carboxylic acid derivatives, methods of preparing them and intermediates used in their preparation
02/07/1996EP0669921A4 Preparation of 2-aryl carbapenems via a boronic acid coupling reaction.
02/07/1996CN1030918C Process for preparing 4-substituted alkyl carbapenem antibiotics
02/07/1996CN1030917C Process for preparing heterocyclic derivatives
01/1996
01/24/1996CN1030767C Method for preparing of 1-methylcarbapenem derivatives
01/18/1996WO1996001261A1 Novel carbapenem derivative
01/03/1996EP0689543A1 Process for the preparation of condensed carbapeneme derivatives
01/03/1996EP0689542A1 Process for the preparation of condensed carbapeneme derivatives
01/03/1996CN1030604C Methode for preparing of heterocyclic componds
01/02/1996US5480987 2-substituted alkyl-3-carboxy carbapenems as antibiotics and a method of producing them
01/02/1996US5480879 Quinolonecarboxylic acids
01/02/1996US5480720 Adhesive composition
12/1995
12/26/1995US5478820 Antibiotic compounds
12/13/1995CN1113233A A method for producing a pyrrolidire derivative
11/1995
11/23/1995WO1995031461A1 Preparation of 2-aryl carbapenems
11/22/1995EP0682667A1 2-phenanthridinyl carbapenem antibacterial agents
11/22/1995EP0682666A1 2-phenanthridinyl carbapenem antibacterial agents
11/09/1995WO1995029913A1 Crystal of pyrrolidylthiocarbapenem derivative, lyophilized preparation containing said crystal, and process for producing the same
11/02/1995EP0679652A1 Process for preparing carbapenem compounds
10/1995
10/31/1995US5463046 1-β-methyl-2-thiolic carbapenem derivatives
10/17/1995US5459260 In vivo stability
10/12/1995WO1995026966A1 Cephalosporin antibiotics
10/12/1995CA2186894A1 Cephalosporin antibiotics
10/05/1995WO1995026335A1 Novel n-arylaliphatic-n-alkyl-functionalised amides, method for their preparation and pharmaceutical compositions containing same
10/04/1995EP0674640A1 2-(2-substituted pyrrolidin-4-yl)thio-carbapenem derivatives
09/1995
09/30/1995CA2145800A1 Process for preparing carbapenem compound
09/21/1995WO1995025108A1 Carbapenem compounds, compositions and methods of treatment
09/21/1995CA2185458A1 Carbapenem compounds, compositions and methods of treatment
09/20/1995EP0672738A2 Adhesive composition
09/20/1995CN1108649A Noel 2-substituted alkyl-3-carboxy carbapenems as antibiotics and a method of producing them
09/20/1995CN1108648A Novel 2-substituted alkyl-3-carboxy carbapenems as antibiotics and a method of producing them
09/19/1995US5451579 1-β-methyl-carbapenem, compositions containing same and methods of use
09/12/1995US5449672 Bactericides
09/12/1995CA1336977C Azetidinone intermediates to carbacephalosporins and process
09/06/1995EP0669921A1 Preparation of 2-aryl carbapenems via a boronic acid coupling reaction
09/05/1995US5447925 Carbapenems with side-chain S; use to treat infections
09/02/1995CA2143170A1 Adhesive composition
08/1995
08/31/1995WO1995023150A1 Carbapenem derivative
08/31/1995WO1995023149A1 Phenylalkylamino derivatives of condensed carbapenemes
08/22/1995US5444057 For treating bacterial infections
08/17/1995WO1995021841A1 1-β-METHYL-CARBAPENEM, COMPOSITIONS CONTAINING SAME AND METHODS OF USE
08/15/1995US5442057 Preparation of 2-aryl carbapenems via a boronic acid coupling reaction
08/15/1995US5442056 Preparation of 2-aryl carbapenems
08/15/1995US5442055 Azetidinone compound and process for preparation thereof
08/15/1995US5441949 Therapy for bacteria infections
08/01/1995US5438054 Antibacterial agent
07/1995
07/27/1995WO1995019979A1 Improved process for synthesizing carbapenem intermediates
07/27/1995CA2178935A1 Improved process for synthesizing carbapenem intermediates
07/18/1995US5434147 Antimicrobial quinolonyl lactam esters
06/1995
06/28/1995CN1104214A Novel 2-thiosubstituted carbapenems
06/27/1995CA1336092C 2-(heterocyclylthio)carbapenem derivatives their preparation and their use as antibiotics
06/21/1995EP0658162A1 Carbapenem derivatives and processes for preparing the same
06/20/1995US5426104 Bactericides
06/14/1995EP0656900A1 Cationic-2-heteroarylphenyl-carbapenem antibacterial agents
06/14/1995EP0656899A1 Condensed carbapenem derivatives
06/13/1995US5424446 Process for preparing optically active 4-mercapto-2-pyrrolidone derivative and intermediate therefor
06/13/1995US5424422 Beta-lactams and their production
06/13/1995US5424306 Crystalline carbapenem derivative
06/13/1995US5424069 Production of crystalline penem
06/01/1995WO1995014692A1 Cabapenem derivatives and processes for preparing the same
05/1995
05/30/1995USRE34960 Carbapenem compounds, and compositions containing them
05/30/1995US5420122 3-pyrrolidinylthio-1-azabicyclo-[3.2.0]hept-2-ene-2-carboxylic acid compounds
05/30/1995US5420119 Carbapenem derivatives having antibiotic activity, their preparation and their use
05/18/1995WO1995013278A1 Urea derivatives
05/09/1995US5414081 Treating a 1-aza-3-thiabicycloalkane with base and phosphine or phosphite desulfurizing agent, and reacting the product with an active esterifying agent
05/04/1995WO1995011905A1 2-(pyrazol-3-yl)carbapenem derivatives
05/02/1995US5412103 Process for preparing (1R,5S,6S)-2-[(6,7-dihydro-5H-pyrazolo [1,2-A][1,2,4]triazolium-6-yl)]thio-6-[(R)-1-hydroxyethyl]-1-methyl-carbapenem-3-carboxylate and starting materials thereof
04/1995
04/25/1995US5409920 2-(3-pyridyl)-carbapenem antibacterial agents
04/20/1995WO1995010520A1 3-pyrrolidinylthio-carbapenem derivatives and their antimicrobal activity
04/18/1995US5407931 Bactericides
04/11/1995US5405844 Tetracyclic antibiotics and processes for their preparation
03/1995
03/28/1995US5401735 Bridged biphenyl carbapenem antibacterial compounds
03/15/1995CN1100100A 1-beta-methy1-2-thiolic carbapenem derivatives
03/08/1995EP0641795A1 Carbapenem derivative
03/07/1995US5395931 6-amido-1-methyl-2-(substituted-thio)carbapenems
02/1995
02/28/1995US5393751 Antibiotics
02/23/1995WO1995005380A1 Crystalline carbapenem derivatives
02/22/1995EP0639193A1 Esters of antibacterial condensed carbapeneme derivatives
02/09/1995WO1995003700A1 Bridged biphenyl carbapenem antibacterial compounds
02/09/1995WO1995003699A1 Bridged biphenyl carbapenem compounds and methods of use
02/07/1995US5387748 Antimicrobial dithiocarbamoyl quinolones
02/01/1995EP0636133A1 Substituted 3-pyrrolidinylthio-carbapenems as antimicrobial agents
02/01/1995CN1098104A Carbapenem derivatives and their salts
01/1995
01/25/1995EP0635488A2 Novel process for preparing azetidinone compound and novel starting compound therefor
01/24/1995US5384317 Bridged biphenyl carbapenem compounds, compositions containing such compounds and methods of use
01/18/1995CN1097424A Preparation of beta-lactam, compounds, and intermediates therefor
01/17/1995US5382575 (N-pyridiniumphenyl)-carbapenems
01/04/1995EP0632039A1 2-(1-(1,3-Thiazolin-2-yl)azetidin-3-yl)thio-carbapenem derivatives
12/1994
12/22/1994WO1994029313A1 NOVEL β-LACTAM COMPOUND AND PROCESS FOR PRODUCING THE SAME
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