| Patents for C07D 477 - Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula: , e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring (2,484) |
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| 05/30/2002 | CA2429675A1 Novel carbapenem derivatives |
| 05/28/2002 | US6395894 Process for the synthesis of carbapenem intermidiates, and compounds produced |
| 05/23/2002 | WO2002040483A1 1-methylcarbapenem derivatives |
| 05/23/2002 | WO2002040482A1 Process for producing carbapenem-type antibacterial |
| 05/23/2002 | CA2429346A1 1-methylcarbapenem derivatives |
| 05/23/2002 | CA2429071A1 Processes for the preparation of carbapenem-type antibacterial agents |
| 05/22/2002 | CN1085210C Process for synthesizing carbapehem antibiotics |
| 05/16/2002 | WO2002038564A1 NOVEL β-LACTAM COMPOUNDS AND PROECSS FOR PRODUCING THE SAME |
| 05/10/2002 | WO2002036594A1 Process for the preparation of crystalline n-formimidoyl thienamycin monohydrate (imipenem monohydrate) |
| 05/02/2002 | WO2002034750A1 Process for formulation of antibiotic compounds |
| 05/02/2002 | EP1201665A1 Process for the preparation of basic antibiotic-inorganic acid addition salts and intermediate oxalates |
| 04/16/2002 | US6372914 Intermediates useful for the manufacture of carbapenem and a stereoselective manufacturing method therefor |
| 04/11/2002 | US20020042523 Reacting an amino-protected aspartic anhydride with an aralkylamine, cyclodehydration to obtain a 1-aralkyl-3-(protected amino)pyrrolidine-2,5-dione, reducing carbonyl groups, then hydrogenolysis; carbapenems, drug intermediate |
| 04/11/2002 | US20020042408 Antibiotic compounds |
| 04/03/2002 | EP1193269A1 Crystalline 1-methylcarbapenem compounds |
| 03/27/2002 | CN1081641C Carbapenem derivatives and antimicrobials |
| 03/20/2002 | EP1188744A1 Process for producing 1H-3-aminopyrrolidine and derivatives thereof |
| 03/07/2002 | US20020028943 For lowering serum lipid, cholesterol and/or triglyceride levels; treating atherosclerosis |
| 03/06/2002 | EP0695295B1 3-(hetero)aryl carboxylic acid derivatives, methods of preparing them and intermediates used in their preparation |
| 02/27/2002 | EP1182204A1 Crystals of carbapenem derivatives and pharmaceutical preparations for injection |
| 02/21/2002 | WO2001090063A3 Prodrug of an ice inhibitor |
| 02/20/2002 | CN1336375A Spiro-and dicyclic diazine and carbozine oxazolidohne compound |
| 02/12/2002 | US6346617 Antibiotics formed by multistage reaction with catalytic oxidation and condensation |
| 02/12/2002 | US6346526 Carbapenicillin with 1,1-dioxo-2,3-dihydronaphtho(1,8-de)(1,2)thiazin-2-yl-substituent; treating staphylococcus infections resistant to methicillin; side effect reduction |
| 02/12/2002 | US6346525 Carbapenicillin with 1,1-dioxo-2h-1-thia-2,3-diaza-naphthalene substituent; treating staphylococcus infections resistant to methicillin; side effect reduction |
| 01/31/2002 | US20020013278 Using an interleukin-1 beta converting enzyme inhibitor pro-drug to treat apoptosis-, interferon-gamma inducing factor or interferon-gamma inducing diseases; antiinflammatory and -proliferative agents; autoimmune/degenerative disesesdiseases |
| 01/29/2002 | US6342494 Carbapenem compounds, use thereof, and intermediate compounds of the same |
| 01/24/2002 | WO2002006283A1 Improved preparation of (4r, 5s, 6s)-3-(((2r,3r)-2-((((s)-2-amino-3-methyl-1-oxobutyl)methyl)tetrahydro-3-furanyl)thio)-6-((r)-1-hydroxyethyl)-4-methyl-7-oxo-1-azabicyclo(3.2.0)hept-2-ene-2-carboxylic acid |
| 01/10/2002 | WO2002002561A1 NOVEL 1β-METHYLCARBAPENEM DERIVATIVES AND PROCESS OF PREPARATION THEREOF |
| 01/03/2002 | US20020002160 Process for formulation of antibiotic compounds |
| 01/01/2002 | CA2067741C 10(1-hydroxyethly)-11-oxo-1-azatricyclo[7.2.0.0.3.8]undec-2-ene-2-carboxylic acid esters and a process for preparing thereof |
| 12/12/2001 | EP0912576B1 Process for synthesizing carbapenem antibiotics |
| 11/29/2001 | WO2001090063A2 Prodrug of an ice inhibitor |
| 11/29/2001 | US20010047094 E.g., a 1-aza-10-(1-hydroxyethyl-11-oxo-4-(het-methylene)-tricyclo(7.2 .0.0(3,8))undec-2-ene-2-carboxylate; good activity against grampositive bacteria such as methicillin-resistant Staphylococcus aureus and epidermidis |
| 11/14/2001 | CN1074767C Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment |
| 10/31/2001 | EP0747381B1 Carbapenem derivative |
| 10/30/2001 | US6310055 Halophenoxy substituted carbapenem antibacterial compounds |
| 10/24/2001 | EP1097151A4 Improved process for synthesizing carbapenem intermediates |
| 10/18/2001 | US20010031749 Antibiotic |
| 10/17/2001 | EP1143991A2 Inhibitors of h+k+ -atpase |
| 10/04/2001 | EP0773222B1 Carbapenem derivative |
| 10/03/2001 | CN1315955A Novel carbapenem derivatives |
| 10/02/2001 | US6297231 Stabilized carbapenem antibiotic compositions and method of making |
| 09/27/2001 | US20010025103 Bactericides |
| 09/25/2001 | US6294529 Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment |
| 09/25/2001 | US6294528 Antibiotics as bactericides |
| 09/18/2001 | US6291448 Carbapenem antibacterial compounds, compositions containing such compounds and method of treatment |
| 09/13/2001 | WO2001066547A1 Process for producing carbapenem derivatives |
| 09/11/2001 | US6288234 Fluorinated heterocyclic amido amine compounds as drugs |
| 09/11/2001 | US6288054 Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment |
| 09/06/2001 | US20010020018 Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment |
| 09/05/2001 | CN1311790A Novel C-2 5/O-and S/N formaldehyde acetal derivatives of carbapenem-3-carboxylic acids and their use as antibiotics and beta lactamase inhibitors |
| 09/04/2001 | US6284753 Grampositve bacteria |
| 08/29/2001 | EP0828741B1 Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones |
| 08/22/2001 | EP1124528A1 Multivalent macrolide antibiotics |
| 08/21/2001 | US6277843 Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment |
| 08/09/2001 | WO2001057041A1 1-methylcarbapenem compounds |
| 08/08/2001 | CN1307578A Carbapenem derivatives, utilization thereof and intermediate compounds of the same |
| 08/02/2001 | WO2001055155A1 Novel carbapenem derivatives of quaternary salt type |
| 08/02/2001 | WO2001055154A1 Novel carbapenem derivatives |
| 08/02/2001 | US20010011086 Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment |
| 08/02/2001 | CA2398481A1 Novel carbapenem derivatives |
| 08/02/2001 | CA2398478A1 Novel quaternary salt-type carbapenem derivatives |
| 07/24/2001 | US6265396 β-lactam compounds and process for preparing the same |
| 07/24/2001 | US6265395 Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment |
| 07/24/2001 | CA2111974C Carbapenem derivatives |
| 07/18/2001 | EP1115419A2 Carbapenem antibacterial compositions and methods of treatment |
| 07/18/2001 | EP1071685A4 Titanium catalyzed preparation of carbapenem intermediates |
| 07/11/2001 | EP1015452A4 Optionally protected 3-hydroxymethyl carbapenems and synthesis |
| 07/11/2001 | CN1068328C Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones |
| 07/04/2001 | EP1113016A1 Carbapenem compounds |
| 07/03/2001 | US6255300 Aminoacylase inhibitor; therapy for bacteria infections |
| 06/28/2001 | WO1999063937A9 Multivalent macrolide antibiotics |
| 06/26/2001 | US6251891 Carbapenem derivatives |
| 06/26/2001 | US6251890 Treating or preventing bacterial infections in mammalian patients |
| 06/19/2001 | CA2036163C Novel beta-lactam compounds and their production |
| 06/13/2001 | CN1298878A 1,3,4-thiadiazole carbapenem compound and its preparing process and usage |
| 06/13/2001 | CN1067074C Carbapenem antibiotic, composition and method of prepn. |
| 06/12/2001 | US6245811 Fatty acid esters as bioactive compounds |
| 06/07/2001 | WO2001040228A1 Carbapenem compounds, use of the same and intermediates thereof |
| 06/07/2001 | WO1999063940A3 INHIBITORS OF H+K+-ATPase |
| 06/06/2001 | EP1104424A1 Process for the synthesis of carbapenem intermediates, and compounds produced |
| 06/06/2001 | EP0741728B1 Improved process for synthesizing carbapenem intermediates |
| 06/05/2001 | US6242596 Preparation of betamethyl carbapenem intermediates |
| 05/30/2001 | CN1066438C Preparation of beta-methyl carbapenem intermediates |
| 05/23/2001 | EP1101766A1 Novel carbapenem derivatives |
| 05/23/2001 | EP1100800A1 Novel c-2 s/o- and s/n formaldehyde acetal derivatives of carbapenem-3-carboxylic acids and their use as antibiotics and beta-lactamase inhibitors |
| 05/23/2001 | CN1066141C 3-(hetero)aryl carboxylic acid derivatives, methods of preparing them and intermediates used in their preparation |
| 05/22/2001 | US6235898 Process for the synthesis of carbapenem intermediated and compounds produced |
| 05/15/2001 | CA2196539C Process for making quinolonyl lactam antimicrobials and novel intermediate compounds |
| 05/10/2001 | WO2001032172A1 Process for formulation of carbapenem antibiotic compositions |
| 05/09/2001 | EP1097151A1 Improved process for synthesizing carbapenem intermediates |
| 04/17/2001 | US6218550 Intermediates useful for the manufacture of carbapenem and a stereoselective manufacturing method therefor |
| 04/11/2001 | EP1090001A1 (heterocyclic)methyl substituted carbapenem antibacterials |
| 04/11/2001 | EP1090000A1 Naphtho 1,8-de]thiasin-2-yl methyl carbapenem antibacterials |
| 04/11/2001 | EP1089999A1 (heterocyclic) methyl substituted carbapenem antibacterials |
| 04/11/2001 | EP1089730A1 Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment |
| 04/11/2001 | EP1089729A1 Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment |
| 04/04/2001 | EP0808315B1 Carbapenem-3-carboxylic acid ester derivatives |
| 04/03/2001 | CA2102772C Azetidinone compound and process for preparation thereof |