Patents
Patents for C07D 477 - Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula: , e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring (2,484)
07/2009
07/30/2009WO2009066917A3 2-arylmethylazetidine-carbapenem-3-carboxylic acid ester derivative or its salt, process for the preparation thereof and pharmaceutical composition comprising the same
07/29/2009EP1395587B1 Process for the preparation of imipenem
07/21/2009CA2379972C Prodrug of an ice inhibitor
06/2009
06/23/2009USRE40794 Antibiotic product for therapy of infections; purification for improved purity and stability
06/18/2009WO2009075323A1 Stable crystal of β-lactam compound
06/17/2009CN101456861A Carbapenem compound
06/10/2009CN101450948A Penem compounds with sulfhydryl pyrrolidine substituted by heterocycle formamido
06/10/2009CN100497338C 4-methyl-7-oxy-1-azabicyclo [3.2.0] hepta-2-olefin-2-carboxylic acid derivative preparation method
06/03/2009CN100494200C 2-arylmethylazetidine carbapenem derivatives and preparation thereof
05/2009
05/28/2009WO2009066917A2 2-arylmethylazetidine-carbapenem-3-carboxylic acid ester derivative or its salt, process for the preparation thereof and pharmaceutical composition comprising the same
05/27/2009CN101440094A Crystal crystal compound and manufacture method thereof
05/26/2009US7538212 Intermediate for carbapenem compound for oral administration and process for producing the same
05/22/2009WO2009064078A1 Method of preparing intermediates of penem antibiotics
05/19/2009US7534782 3-(2-Guanidinoacetylamino)pyrrolidin-1-ylcarbonyl]-1-methylpyrrolidin-4-ylthio]-6-[(1R)-1-hydroxyethyl]-1-methyl-1-carbapen-2-em-3-carboxylic acid ethanolate; viricide; antibiotic resistance; Staphylococcus aureus, Streptococcus pneumoniae, Escherichia coli and Pseudomonas aeruginosa; storage stability
05/13/2009EP2057989A1 Freeze-dried preparation of 1-methylcarbapenem
05/13/2009CN101432289A Improved method for the crystallization of intermediates of carbapenem antibiotics
05/07/2009WO2009038328A3 Acid addition salts of synthetic intermediates for carbapenem antibiotics and processes for preparing the same
04/2009
04/28/2009US7524952 Process for producing carbapenem compound for oral administration
04/28/2009CA2465336C Novel carbapenem compounds
04/22/2009CN101412720A Carbapenem compound containing mercapto nitrogen heterocyclic vinyl
04/22/2009CN101412719A Carbapenem derivatives
04/22/2009CN101412718A Carbapenem derivative containing sulfenyl heterocyclic amine formyl
04/22/2009CN101412717A Carbapenem derivative containing guanidyl alkanoylamino heterocycle
04/16/2009WO2009047604A1 Process for the preparation of carbapenem antibiotic
04/15/2009CN101410399A Process for production of intermediate for meropenem
04/15/2009CN101410398A Improved process for producing carbapenem compound
04/08/2009CN100475817C Crystal of 1-methyl carbapenem compound
04/07/2009US7514553 Dehalogenating a 6-halo- or 6,6-dihalo-carboxylic acid-protected penicillanic acid by reacting with a metal having a lower standard oxidation-reduction potential than bismuth (e.g., Al, Fe or Mg)) in the presence of bismuth metal or a bismuth compound and a reaction promoter
03/2009
03/26/2009WO2009038328A2 Acid addition salts of synthetic intermediates for carbapenem antibiotics and processes for preparing the same
03/26/2009US20090082327 Deuterium-enriched meropenem
03/24/2009US7507814 Process for preparation of imipenem
03/12/2009WO2009030107A1 Benzenesulfonamido methylene substituted mercapto pyrrolidine carbapenem derivatives
03/04/2009CN101376657A Penem derivative containing sulfhydryl piperidine formyl nitrogen heterocyclic ring
03/04/2009CN101376656A Penem derivative
03/04/2009CN101376643A Preparation of carbapenem penicillin ertapenem intermediate
03/04/2009CN101376641A Carbapenem penicillin ertapenem intermediate, and preparation and use thereof
03/04/2009CN101376636A Carbpenem penicillin ertapenem intermediate, and preparation and use thereof
02/2009
02/25/2009EP1692135A4 A new process for preparation of imipenem
02/25/2009CN101372490A Penem derivative containing sulfhydryl nitrogen heterocyclic ring and vinyl nitrogen heterocyclic ring
02/25/2009CN101372489A Carbapenem derivative containing sulfhydryl pyrrolidine formamide benzyl
02/25/2009CN101372488A Novel carbapenem compound
02/18/2009CN101367830A Synthesis of sulfomycin derivant
02/18/2009CN101367818A Penem compound containing amine vinyl substituted sulfhydryl aza ring
02/18/2009CN101367817A Carbpenem compound containing cyclohexenone formamido group
02/18/2009CN101367816A Carbpenem derivants
02/18/2009CN101367815A Six-membered ring methanamide substituted sulfhydryl pyrrolidine carbpenem compound
02/18/2009CN101367814A Sulfhydryl pyrrolidine formyl piperidine substituted penem derivant
02/18/2009CN101367813A Sulfhydryl pyrrolidine formyl arylamine heterocycle substituted penem derivant
02/18/2009CN101367812A Sulfhydryl pyrrolidine formamido cyclopentene acid substituted penem derivant
02/18/2009CN101367811A Carbon substituted penems antibiotics
02/18/2009CN101367810A Novel carbpenem antibiotic
02/18/2009CN101367809A Penem derivant containing sulfhydryl pyrrolidine formhydrazide
02/18/2009CN101367808A Carbpenem compound with heterocycle formyl substituted sulfhydryl pyrrolidine
02/18/2009CN101367807A Sulfhydryl pyrrolidine formamido pyridine substituted penem derivant
02/18/2009CN101367806A Formyl aniline substituted sulfhydryl pyrrolidine carbpenem compounds
02/18/2009CN101367805A Formyl guanidino substituted sulfhydryl pyrrolidine carbpenem compounds
02/18/2009CN101367804A Penem derivant containing adamantane
02/12/2009WO2009018723A1 Sulfonyl-substituted carbapenem compounds
02/12/2009US20090042819 Organic nitric oxide donor salts of antimicrobial compounds, compositions and methods of use
02/11/2009CN101362763A Carbapenem derivates containing sulfhydryl pyrrolidine
02/11/2009CN101362762A Penem compound containing sulfhydryl piperidine
02/11/2009CN101362761A Carbapenem antibiotic containing sulfhydryl piperidine
02/11/2009CN101362760A 1beta-methyl carbapenem compound
02/11/2009CN101362759A Dihydropyrrole methano substituted carbapenem derivates
02/11/2009CN101362758A Penem derivates containing sulfhydryl pyrrolidine vinyl heterocycle
02/11/2009CN101362757A Sulfonyl substituted carbpenems compounds
02/11/2009CN101362756A Carbapenem bicyclic nucleus preparation and purification method
02/11/2009CN100460389C Pentazane derivative intermediate, preparation and use thereof
02/04/2009CN101357920A Penem derivative containing sulfhydryl pyrrolidine formamido triazine
02/04/2009CN101357919A Penem derivative containing sulfhydryl formamide benzenesulfonyl pyrrolidine
02/04/2009CN101357918A Penem derivative containing isothioureido sulfhydryl pyrrolidine
02/04/2009CN101357917A Carbapenem compound containing formyl hydrazino
02/04/2009CN101357916A Penem compound containing dihydroimidazole formamido
01/2009
01/29/2009US20090029964 Novel carbapenem compound
01/21/2009CN101348486A Preparation of meropenem
01/21/2009CN101348485A Preparation of doripenem
01/14/2009EP2014666A1 Improved method for the crystallization of intermediates of carbapenem antibiotics
01/14/2009CN101343273A Penem compounds containing pyridine onium ion
01/14/2009CN101343272A Carbpenem compound containing cyclohexane
01/14/2009CN101343271A Penem derivant containing isoxazole alkyl ketone
01/08/2009US20090012149 Prodrug of an ice inhibitor
01/06/2009CA2457642C Crystalline forms of ertapenem sodium
12/2008
12/31/2008WO2009000210A1 Novel carbapenem derivatives
12/31/2008WO2005066173A3 Processes for the preparation of substituted azetidinone
12/31/2008CN101333219A Penem derivates with mercapto pyrrolidine formamide benzene alkyl heterocycle
12/31/2008CN101333218A Formamide alkylbenzene substituted mercapto pyrrolidine carbapenem compounds
12/31/2008CN101333217A 1-methyl carbapenem antibiotics
12/24/2008EP2006290A1 Improved process for producing carbapenem compound
12/24/2008CN101328181A Novel penem compounds
12/24/2008CN101328180A Sulfhydryl oxo heterocycle substituted penem derivates
12/24/2008CN101328179A Sulfhydryl pyrrolidine penem derivates containing oxo aza ring
12/24/2008CN101328178A Penem derivates containing thiophen substituted sulfhydryl pyrrolidine
12/24/2008CN101328177A Nitrogen heterocyclic ring vinyl substituted sulfhydryl heterocycle carbpenem compounds
12/24/2008CN101328176A Tetrahydrochysene pyrimidine vinyl substituted sulfhydryl heterocycle carbpenem compounds
12/24/2008CN100445284C Process for prepn. of crystalline N-forminidoyl thienamycin monohydrate (imipenem monohydrate)
12/23/2008US7468364 High oral absorption; gramnegative, grampositive bacteria and antibiotic resistant Staphlococcus pneumonia, Hemophilus influenza
12/17/2008CN101323616A Carbpenem derivates containing sulfhydryl thiazole
12/17/2008CN101323615A Pennem derivates containing formamide heterocycle sulfonic acid amide sulfhydryl pyrrolidine
12/09/2008US7462712 reacting keto ester corresponding compound with phosphorohalide in presence of basic catalyst
11/2008
11/26/2008CN101311178A Synthetic method of compound panipenan
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