C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms

Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
12/1999
12/02/1999	WO1999061431A1 New dipeptidyl peptidase iv effectors
12/02/1999	WO1999061416A1 Substituted dithio-bis-nitrobenzenes and their applications
12/02/1999	WO1999061413A1 Substituted 4-biarylbutyric and 5-biarylpentanoic acid derivatives as matrix metalloprotease inhibitors
12/02/1999	WO1999061410A1 2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia
12/02/1999	WO1999061409A1 Bioreductive cytotoxic agents
12/02/1999	DE19824470A1 Neue Neurokininantagonisten, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen New Neurokininantagonisten, processes for their preparation containing these compounds and pharmaceutical compositions
12/02/1999	DE19823831A1 Neue pharmazeutische Verwendung von Isoleucyl Thiazolidid und seinen Salzen New pharmaceutical use of isoleucyl thiazolidide and its salts
12/02/1999	CA2332806A1 Bioreductive cytotoxic agents
12/02/1999	CA2331056A1 2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia
12/01/1999	EP0960141A1 Cross-linked vinyl polymers with bile acid adsorbing effect
12/01/1999	EP0960108A1 Matrix metalloproteinase inhibitors
12/01/1999	EP0960106A1 1-phenyl-4-benzylpiperazines: dopamine receptor subtype specific ligands (d4)
12/01/1999	EP0960093A1 Method for hydrogenating compounds from the group of imines or enamines
12/01/1999	EP0655056B1 Azacyclyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
12/01/1999	CN1237161A New amino alcohol derivatives, process for production thereof and medicaments and reagents containing these compounds
11/1999
11/30/1999	US5994370 Indene compounds having activity as SERMS
11/30/1999	US5994369 Substituted piperidine or pyrrolidine compounds for treating sigma-receptor modulated disorders
11/30/1999	US5994356 Carboxylic acid derivatives, medicaments comprising these compounds, their use and processes for their production
11/30/1999	US5994351 Antiarthritic agents; anticancer agents; antiulcer agents; enzyme inhibitors
11/30/1999	US5994294 Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
11/30/1999	US5993777 Benzamide compounds for cancer imaging and therapy
11/25/1999	WO1999059960A1 Benzamide derivatives for the treatment of diseases mediated by cytokines
11/25/1999	WO1999059959A1 Benzamide derivatives for the treatment of diseases mediated by cytokines
11/25/1999	WO1999059957A1 Compounds having reversible inhibiting activity of carnitine palmitoyl-transferase
11/25/1999	WO1999059588A1 Medicinal composition reduced in bitterness
11/25/1999	WO1999059570A1 Protease inhibitors
11/25/1999	WO1999059568A1 Hydroxamic acid derivatives as antibacterials
11/25/1999	WO1999059527A2 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives
11/25/1999	WO1999059526A2 Protease inhibitors
11/25/1999	WO1999059499A2 Serotonergic 5ht7 receptor compounds for treating ocular and cns disorders
11/25/1999	WO1999059409A1 Compounds and uses thereof
11/25/1999	CA2332531A1 Protease inhibitors
11/25/1999	CA2332505A1 Serotonergic 5ht7 receptor compounds for treating ocular and cns disorders
11/25/1999	CA2332492A1 Protease inhibitors
11/25/1999	CA2328699A1 Benzamide derivatives for the treatment of diseases mediated by cytokines
11/24/1999	EP0958287A1 Sulfamide-metalloprotease inhibitors
11/24/1999	EP0958280A1 Arylpiperidinopropanol and arylpiperazinopropanol derivatives and pharmaceuticals containing the same
11/24/1999	CN1236313A Novel methods
11/24/1999	CN1236299A Method of treating post menopausal diseases, including osteoporosis
11/24/1999	CN1235826A 10, 11 methanodibenzosuberane derivatives used as chemosensitizing agents
11/24/1999	CN1046716C Novel intermediate for synthetic use and process for producing aminopiperazinoe derivatives
11/23/1999	US5990309 2-chloro-5-fluoro-4-morpholinonitrobenzene and 2-chloro-5-fluoro-4-morpholinoaniline
11/23/1999	US5990170 Possesses a profile of activity which is similar to, though less potent than .delta.9-thc (tetrahydrocannabinol) with a mimicking of the psychoactive effects; analgesics; side effect reduction; cardiovascular disorders
11/23/1999	US5990166 Compounds and compositions for delivering active agents
11/23/1999	US5990145 Antiinflammatory,-carcinogenic,-tumor,-metastasis agents; cardiovascular disorders, e.g., arteriosclerosis, restenosis; retinopaathies and nephropathies; osteoporosis
11/23/1999	US5990113 Monohydrate of 2-(1-piperazinyl)-5-methylbenzenesulfonic acid, free of anhydrous crystals; free from weight change due to moisture absorption and can be weighed accurately in manufacturing a pharmaceutical composition for heart diseases
11/23/1999	US5989539 Compounds and compositions for delivering active agents
11/23/1999	CA2207694C Process for preparing sildenafil
11/18/1999	WO1999058530A1 Water soluble azoles as broad-spectrum antifungals
11/18/1999	WO1999058529A1 Water soluble azoles as broad-spectrum antifungals
11/18/1999	WO1999058517A2 Isocyanate derivatizing agent and methods of production and use
11/18/1999	WO1999058496A1 Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
11/18/1999	WO1999058495A1 Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
11/18/1999	WO1999058478A1 Novel derivatives of 3,3-diphenylpropylamines
11/18/1999	DE19821176A1 Reprocessing aqueous solutions of N-methyl-morpholine N-oxide, especially spent precipitation baths from cellulose spinning processes
11/18/1999	CA2331539A1 Isocyanate derivatizing agent and methods of production and use
11/17/1999	EP0957101A1 Water soluble azoles as broad-spectrum antifungals
11/17/1999	EP0957073A1 Novel derivatives of 3,3-diphenylpropylamines
11/17/1999	EP0956141A1 Amine heat stable salt neutralization having reduced solids
11/17/1999	EP0956050A1 Novel lipid complexes for transferring at least a therapeutically active substance, in particular a polynucleotide into a target cell and use in gene therapy
11/17/1999	EP0956031A1 Inhibition of 26s and 20s proteasome by indanones
11/17/1999	CN1046507C Heterocyclic compounds for treatment of CNS and cardiovasular disorders
11/16/1999	US5986102 Hydroxypropylamide peptidomimetics as inhibitors of aspartyl proteases
11/16/1999	US5985928 Bioactive bicyclic aromatic compounds and pharmaceutical/cosmetic compositions comprised thereof
11/16/1999	US5985917 Mercapto and seleno derivatives as inhibitors of nitric oxide synthase
11/16/1999	US5985899 Selective thrombin inhibitors
11/16/1999	US5985895 2-naphthamide derivatives and their therapeutic applications
11/16/1999	US5985881 Treatment and prevention of respiratory disorders, inflammatory eye diseases, inflammatory skin diseases, intestinal disorders, other inflammatory diseases
11/16/1999	US5985880 Compositions and methods for reducing respiratory depression and attendant side effects of mu opioid compounds
11/16/1999	US5985873 Useful in the diagnosis and treatment of feeding disorders such as obesity and bulimia and cardiovascular diseases such as essential hypertension and congestive heart failure due to the binding of these compounds to human neuropeptide y1
11/16/1999	US5985838 Peptide analogs as irreversible interleukin-1β protease inhibitors
11/16/1999	CA2137811C Dimeric piperidine, tetrahydropyridine and piperazine derivatives
11/16/1999	CA2088761C Benzimidazole derivatives, process for their preparation and application
11/11/1999	WO1999057099A1 Heterocyclic derivatives which inhibit factor xa
11/11/1999	WO1999057098A2 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
11/11/1999	WO1999042457A3 Substituted alxoxycarbonyl compounds
11/11/1999	WO1999040083A3 Bifunctional tryptase inhibitors
11/11/1999	WO1999040073A3 Tryptase inhibitors
11/11/1999	CA2329704A1 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
11/10/1999	EP0955372A2 Method for screening substance inhibiting activation of NF-kappa B
11/10/1999	EP0955296A2 Tertiary alkyl functionalized piperazine derivatives
11/10/1999	EP0955295A1 Therapeutically active levorotatory and dextrorotatory 1-((4-chlorophenyl)phenylmethyl) piperazines
11/10/1999	CN1234799A 1,4-disubstituted piperazines
11/10/1999	CN1234401A Synthesis of triethylene-diamide and diethylenediamine by using zeolite catalyst modified by silicon contained compound
11/10/1999	CN1046269C HIV protease inhibitors
11/09/1999	US5981585 Phenyl acetic acid derivatives as pesticides
11/09/1999	US5981531 For inhibiting platelet aggregation
11/09/1999	US5981530 Piperazine derivative
11/09/1999	US5981513 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith
11/09/1999	CA2106452C Amidinophenol derivatives
11/04/1999	WO1999055688A1 Substituted diarylalkyl amides as calcium channel antagonists
11/04/1999	WO1999055687A2 Hydroxypropylamide peptidomimetics as inhibitors of aspartyl proteases
11/04/1999	WO1999055661A1 Aminomethyl-benzoic ester derivatives as tryptase inhibitors
11/03/1999	EP0953567A2 Bicyclic substituted piperazine-, piperidine- and tetrahydropyridine derivatives, their preparation and their use as agents with central dopaminergic (dopamine D4 receptor) activity
11/03/1999	EP0953563A1 Process for producing depsipeptide derivatives and novel intermediates therefor
11/03/1999	EP0952842A2 A method of treating cancer
11/03/1999	EP0923544A4 Method for the synthesis of amines and amino acids with organoboron derivatives
11/03/1999	EP0784611B1 N-(ortho-substituted benzyloxy)imine derivatives and their use as fungicides, acaricides or insecticides
11/03/1999	CA2059786A1 Method of preparing heteroalicyclic n-nitro compounds
11/02/1999	US5977360 Process for producing cyclic hydrazine derivatives, tetra-hydropyridazine and hexahydropyridazine

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