C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms

Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
01/1999
01/05/1999	US5856491 Reacting secondary amine with terminally unsaturated electrophilic compound in presence of n-methylpyrrolidinone solvent
01/05/1999	US5856353 Sulfonamide inhibitors of aspartyl protease
01/05/1999	US5856338 Sulfonamide-substituted compounds, processes for their preparation, their use as a medicament or diagnostic, and pharmaceutical preparation comprising them
01/05/1999	US5856326 Inhibitors of farnesyl-protein transferase
01/05/1999	US5856311 Derivatives of β-aminopropionic acid with a fungicidal activity
01/05/1999	US5855629 Alkoxy acetic acid derivatives
12/1998
12/30/1998	WO1998058919A1 Angiogenesis inhibiting 5-substituted-1,2,4-thiadiazolyl derivatives
12/30/1998	WO1998058902A1 INHIBITORS OF α4β1MEDIATED CELL ADHESION
12/30/1998	WO1998058901A1 3-anilino-2-cycloalkenone derivates
12/30/1998	EP0887340A1 Novel compounds and pharmaceutical use thereof
12/30/1998	EP0886636A1 Novel piperidines derived from 1-/(piperazin-1-yl)aryl(oxy/amino)carbonyl/-4-aryl-piperidine as selective 5-ht-1d.beta. receptor antagonists
12/30/1998	CN1203602A Acylated enol derivatives of 'alpha'-ketoesters and 'alpha'-ketoamides
12/29/1998	US5854277 Thiophenebutanoic acid derivatives as matrix metalloprotease inhibitors
12/29/1998	US5854250 N-benzoylamino acid derivatives, pharmaceutical compositions containing them and process of preparing same
12/29/1998	US5854249 Opioid diarylmethylpiperazines and piperidines
12/23/1998	WO1998057643A1 Use of draflazine-analogues for treating pain
12/23/1998	EP0885887A2 Sulfonamide inhibitors of HIV-Aspartyl protease
12/23/1998	EP0885213A1 Fibrinogen receptor antagonists
12/23/1998	EP0885205A1 Fibrinogen receptor antagonists
12/23/1998	EP0885204A1 Novel aryl glycinamide derivatives, method of producing said derivatives and pharmaceutical compositions containing these compounds
12/23/1998	EP0885199A1 Kappa agonist compounds and pharmaceutical formulations thereof
12/23/1998	EP0772588B1 Production of carbamic acid vinyl esters
12/23/1998	CN1202882A New LH-RH antigonists with improved effectiveness
12/23/1998	CN1202488A Monohydrates of aminobenzenesulfonic acid derivatives and method for preparing thereof
12/23/1998	CA2294011A1 Use of draflazine-analogues for treating pain
12/22/1998	US5852193 Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceuticals
12/22/1998	US5852160 Phosgenated oxime resins and their preparation
12/22/1998	US5852043 HIV protease inhibitors
12/22/1998	US5852007 Cysteine and serine protease inhibitors containing D-amino acid at the P2 position, methods of making same, and methods of using same
12/17/1998	WO1998056771A2 Piperazine derivatives and their use as anti-inflammatory agents
12/17/1998	WO1998056423A1 Novel lipid complexes for transferring at least a therapeutically active substance, in particular a polynucleotide into a target cell and use in gene therapy
12/17/1998	CA2263367A1 Novel lipid complexes for transferring at least a therapeutically active substance, in particular a polynucleotide into a target cell and use in gene therapy
12/16/1998	EP0883613A1 Sulfonamide derivatives as 5ht7 receptor antagonists
12/16/1998	EP0883405A1 Amidino protease inhibitors
12/16/1998	EP0883403A1 Method for treating sexual dysfunctions
12/16/1998	CN1202164A Diarylalkenylamine derivatives
12/16/1998	CN1202107A Selective 'beta'3 adrenergic agonists
12/16/1998	CN1202106A Selective 'beta'3 adrenergic agonists
12/16/1998	CN1201791A Antiallergic agent having anti-oxidant action
12/16/1998	CN1201782A Diaminoalkyl quaternary ammonium salts and method for their preparation and use
12/15/1998	US5849912 Biphenyl derivatives
12/15/1998	US5849801 4-amino-5-oxy-2,6,6-trimethyl-2-cycloheptene compounds
12/15/1998	US5849745 N-benzylpiperazine compounds
12/15/1998	US5849732 Phenol compound having antioxidative activity and the process for preparing the same
12/15/1998	US5849665 Synergistic composition and process for selective weed control
12/15/1998	US5849326 Method for treating neuronal diseases via administration of 2-acylaminopropanol derivatives
12/15/1998	CA1340191C Derivatives of p-substituted phenyl ester of pivalic acid
12/10/1998	WO1998055459A1 Process for producing piperazinesulfonamide derivatives and salts thereof
12/10/1998	WO1998055448A2 Fluoroalkene carboxylic acid derivatives, method for producing said derivatives, and insecticidal agents containing the same
12/10/1998	WO1998055153A1 Non-steroidal radiolabeled agonist/antagonist compounds and their use in prostate cancer imaging
12/10/1998	CA2291441A1 Fluoroalkene carboxylic acid derivatives, method for producing said derivatives, and insecticidal agents containing the same
12/09/1998	EP0882704A1 3,4-disubstituted phenylethanolaminotetralincarboxamide derivatives
12/09/1998	EP0882031A1 Novel benzoyl guanidine derivatives, process for their preparation and their use in the preparation of medicines
12/09/1998	EP0882016A1 Alkylated styrenes as prodrugs to cox-2 inhibitors
12/09/1998	EP0882015A1 Diphenyl stilbenes as prodrugs to cox-2 inhibitors
12/09/1998	EP0882010A1 Pharmaceutical agents containing perfluoroalkyl-containing metal complexes and the use thereof in tumour therapy and interventional radiology
12/09/1998	CN1201458A (-) cis-6(S)-phenyl-5(R)-[4-(2-pyrrolidin-1-ylethoxy) phenyl]-5,6,7,8-tetrahydronaphthalen-2-ol D-tartrate
12/09/1998	CN1201457A Process and intermediates for preparing 30(1-piperazinyl)-1,2-benzisothiazole
12/09/1998	CN1201454A Meta-guanidine, urea, thiourea or azacyclic amino benzoic acid derivatives as integrin antagonists
12/09/1998	CN1201033A Solid chemical compound, preparation method therefor and use in medicine
12/09/1998	CN1041087C Arylacetamides, preparation method and use thereof
12/08/1998	USRE35985 Fungicidal compositions
12/08/1998	US5847201 N-protected/N-substituted-beta-amino hydroxy sulfonates
12/08/1998	US5847159 1- ω-(3,4-dihydro-2-naphthalenyl)alkyl!-cyclic amine derivatives, process for preparing the same, and pharmaceutical composition containing the same
12/08/1998	US5847131 Preparation of N-substituted cyclic amines
12/08/1998	US5847130 Method for reducing the nitrosamine content of N-methylmorpholine-N-oxide
12/08/1998	US5847129 Process for the regeneration of an aqueous process liquid of the amine-oxide process
12/08/1998	US5847125 Amino acid derivatives with anticholecystokinin activity
12/08/1998	US5847117 Reagent and catalytic process useful for cleaving a protected functional group
12/08/1998	US5846987 Retroviral protease inhibiting compounds
12/08/1998	US5846959 Treatment for atherosclerosis and other cardiovascular and inflammatory diseases
12/08/1998	US5846941 Isosteric antiherpes peptide derivatives II
12/03/1998	WO1998054164A1 Sulfonamide derivatives, their production and use
12/03/1998	WO1998054123A1 Substituted peptidylamine calcium channel blockers
12/03/1998	WO1998054115A1 Use of a rhodium catalyst for hydroamination and/or oxidative amination of aryl-substituted olefins and method for producing a 2-aryl vinyl amine
12/03/1998	DE19722373A1 Verwendung eines Rhodiumkatalysators sowie ein neues Verfahren zur Herstellung von 2-arylsubstituierten Ethylen- und Ethylaminen The use of a rhodium catalyst and a novel process for preparing 2-aryl-substituted ethylene and ethylamines
12/03/1998	CA2287292A1 Sulfonamide derivatives, their production and use
12/02/1998	EP0881216A1 Solid methylphenidate, its preparation and use in medicine
12/02/1998	EP0880558A1 Combinatorial process for preparing substituted indane libraries
12/02/1998	EP0880512A1 Novel aromatic piperazines derived from substituted cycloazanes, method for preparing same, pharmaceutical compositions, and use thereof as drugs
12/02/1998	EP0880511A1 Integrin receptor antagonists
12/02/1998	CN1200373A Vitronectin receptor antagonists, their prepn. and use
12/02/1998	CN1040980C Second messenger cell signaling inhibitors
12/01/1998	US5844025 1,2-Bis-adducts of stable nitroxides with substituted ethylenes and stabilized compositions
12/01/1998	US5843948 Piperazinophenyl- and piperazinophenyloxycarboxylic acid derivatives, and processes and intermediates for their preparation and pharmaceutical compositions comprising them
12/01/1998	US5843946 α-and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
12/01/1998	US5843906 Meta-substituted phenylene sulphonamide derivatives
12/01/1998	CA2054213C Inclusion complexes of 3-morpholino-sydnonimine or its salts or its tautomer isomer, process for the preparation thereof and pharmaceutical compositions containing the same
11/1998
11/28/1998	CA2238554A1 Aryloxyalkylamines with serotonin receptor activity
11/26/1998	WO1998052929A1 Anti-inflammatory piperazinyl-benzyl-tetrazole derivatives and intermediates thereof
11/26/1998	WO1998052898A1 Pharmaceutical agents for the treatment of cerebral amyloidosis
11/26/1998	WO1998052553A1 Methods for treatment of conditions associated with lactosylceramide
11/26/1998	CA2290818A1 Pharmaceutical agents for the treatment of cerebral amyloidosis
11/25/1998	EP0879814A1 Triaromatic compounds, compositions containing them and uses thereof
11/25/1998	EP0800657B1 Polymers based on block copolymers
11/25/1998	EP0607252B1 Compositions for the treatment of hiv infection
11/25/1998	CN1200117A Phenylacetic acids, processes for their preparation and agents containing them
11/24/1998	US5840986 Reacting alkyne, carbonyl compound and amine using unsupported copper catalyst derived from malachite; intermediate for drugs, electroplating and corrosion inhibitors
11/24/1998	US5840974 Metalloproteinase inhibitors
11/24/1998	US5840918 Isoprenyl transferase inhibitors

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