| Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005) |
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| 09/20/2000 | EP1036070A1 N-alkyl ammonium acetonitrile salts, methods therefor and compositions therewith |
| 09/20/2000 | EP1036060A2 Cyclohexadiene-derivatives as pesticides |
| 09/20/2000 | EP1036059A1 Adamantane derivatives |
| 09/20/2000 | EP1036058A1 Adamantane derivatives |
| 09/20/2000 | EP0707564B1 Difluoro statone analogs |
| 09/20/2000 | CN1267286A 2-{3-[4-(2-t-butyl-6-trifluoromethylpyridin-4-yl) piperazin-1-yl] propylmercapto} pyrimidin-4-ol-fumarate |
| 09/20/2000 | CN1267281A Glucagon antagonists/inverse agonists |
| 09/19/2000 | US6121322 Antiinflammatory agents |
| 09/19/2000 | US6121304 Pentafluorobenzenesulfonamides and analogs |
| 09/19/2000 | US6121281 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use |
| 09/19/2000 | US6121267 Substituted piperazines and piperidines as central nervous system agents |
| 09/19/2000 | US6121262 Neurokin (tachykinin) antagonists |
| 09/14/2000 | WO2000053663A1 A polymeric or oligomeric compound and its uses in absorption processes |
| 09/14/2000 | WO2000053583A1 Inhibitors of protein tyrosine phosphatase |
| 09/14/2000 | WO2000053572A1 Biphenyl derivatives as antagonists of the neurokinine-1 receptor |
| 09/14/2000 | WO2000004012A8 COMPOUNDS SPECIFIC FOR THE HUMAN α1d ADRENERGIC RECEPTOR AND USES THEREOF |
| 09/14/2000 | WO1999063999A8 H1-histamine receptor antagonists |
| 09/14/2000 | CA2366308A1 Inhibitors of protein tyrosine phosphatase |
| 09/13/2000 | EP1035110A1 Benzylaminodiacetamide derivatives, compositions containing the same, process for their preparation and uses |
| 09/13/2000 | EP1034171A1 Pseudopolymorphic forms of 2-[2-[4-[bis(4-fluorophenyl)methyl1]-1-piperazinyl]ethoxy]acetic acid dihydrochloride |
| 09/13/2000 | EP1034162A1 9,10-dihydro-9,10-ethanoanthracene derivatives as phospholipase inhibitors |
| 09/13/2000 | EP0763017B1 N-(3-amino-2-hydroxybutyl)sulphonamide derivatives as hiv protease inhibitors |
| 09/13/2000 | EP0691962B1 1-amino-3-phenoxy propane derivatives as modulators of multi-drug resistance |
| 09/13/2000 | CN1266423A 1-amino-alkylcyclohexane NMDA receptor antagonists |
| 09/12/2000 | US6117902 6,8-dimercaptooctanoic acid derivatives substituted at the 6-S and/or 8-S position with the (3-methylthiopropanoyl) radical and pharmaceutical compositions intended for the treatment of cancerous tumors |
| 09/12/2000 | US6117892 Crop protection products |
| 09/12/2000 | US6117887 Inhibition of 26S and 20S proteasome by indanones |
| 09/12/2000 | US6117870 Cyclic amide derivatives |
| 09/12/2000 | US6117841 Used to treat stroke, cerebral ischemia, pain, head trauma or epilepsy |
| 09/08/2000 | WO2000052002A1 N-substituted imide derivatives with serotonergic activity |
| 09/08/2000 | WO2000052001A1 Piperazine derivatives and process for the preparation thereof |
| 09/08/2000 | WO2000052000A1 A process for the preparation of 2-{2-[4-(diphenylmethyl)-1-piperazinyl]ethoxy}acetic acid compounds or salts thereof |
| 09/08/2000 | WO2000051998A1 Compounds useful as reversible inhibitors of cathepsin s |
| 09/08/2000 | WO2000051981A1 Aminocycloalkyl cinnamide compounds for arrhythmia and as analgesics and anesthetics |
| 09/08/2000 | WO2000051975A1 Alkenyl- and alkynyl-containing metalloprotease inhibitors |
| 09/08/2000 | WO2000051974A1 Alpha-aminoacetic acid derivatives useful as alpha 4 beta 7 - receptor antagonists |
| 09/08/2000 | WO2000051973A1 Cyclobutene-3,4-dione derivatives, preparation method and therapeutic use |
| 09/08/2000 | WO2000051972A1 1,2,3,4-tetrahydro-1-naphthalenamine compounds useful in therapy |
| 09/08/2000 | WO2000051971A1 Oxamic acids and derivatives as thyroid receptor ligands |
| 09/08/2000 | WO1999064595A9 THERAPEUTIC AND DIAGNOSTIC DOMAIN 1 β2GPI POLYPEPTIDES AND METHODS OF USING SAME |
| 09/08/2000 | CA2365032A1 1,2,3,4-tetrahydro-1-naphthalenamine compounds useful in therapy |
| 09/08/2000 | CA2364897A1 A process for the preparation of 2-{2-[4-(diphenylmethyl)-1-piperazinyl]ethoxy}acetic acid compounds or salts thereof |
| 09/08/2000 | CA2364878A1 Alkenyl- and alkynyl-containing metalloprotease inhibitors |
| 09/08/2000 | CA2361182A1 N-substituted imide derivatives with serotonergic activity |
| 09/08/2000 | CA2361162A1 Alpha-aminoacetic acid derivatives useful as alpha 4 beta 7-receptor antagonists |
| 09/08/2000 | CA2360740A1 Compounds useful as reversible inhibitors of cathepsin s |
| 09/06/2000 | EP1033366A2 Amide derivatives useful as Neuropeptide Y (NPY) antagonists |
| 09/06/2000 | EP1032571A1 Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance p antagonists |
| 09/06/2000 | EP1032559A1 Aminoalkylphenol derivatives and related compounds |
| 09/06/2000 | EP1032401A2 Method for inhibiting cytokine production by cells |
| 09/06/2000 | CN1265654A 1-(N-phenylaminoalkyl)-piperazine derivatives substituted at position 2 of phenyl ring |
| 09/06/2000 | CN1265647A Acrylic metalloprotease inhibitor |
| 09/06/2000 | CN1265645A Urokinase inhibitors |
| 09/06/2000 | CN1056141C 哌嗪衍生物 Piperazine derivatives |
| 09/06/2000 | CN1056057C Pharmaceutical compositions permitting the prolonged release of trimetazidine after oral administraion |
| 09/05/2000 | US6114528 Fluorinated amide compounds |
| 09/05/2000 | US6114493 Contacting a compound to be phosgenated with an excess of a phosgene source in the form of a solid phase reagent; supports in combinatorial synthesis for the creation of libraries of compounds for lead identification |
| 09/05/2000 | US6114380 Antiviral agent; administering to treat hiv infection; n-(4-(n-benzyloxycarbonyl-l-valyl)amino-2,2-difluoro-1,3-dioxo-5-(4-(2-n -morpholyl)ethyloxy)phenyl-pentyl)-o-((2-pyridyl)methyl)-d-valinol, for example |
| 09/05/2000 | US6114335 Benzoylguanidine derivatives, process for their preparation their use in the preparation of medicines |
| 09/05/2000 | US6114325 1,2-di-substituted benzene-carboxamide derivative, hair growth promoter and external composition for skin using the same |
| 09/05/2000 | US6113799 Process for selective separation of morpholine |
| 09/05/2000 | CA2020340C Enantioselective synthesis of antifolates |
| 08/31/2000 | WO2000050470A2 Catalysts containing n-pyrrolyl substituted nitrogen donors |
| 08/31/2000 | WO2000050398A2 Phenyl- and pyridinyl derivatives as neurokinin 1 antagonists |
| 08/31/2000 | WO2000050389A1 Efficient carbamate synthesis |
| 08/31/2000 | WO2000050386A1 Compounds and compositions for delivering active agents |
| 08/31/2000 | WO2000050380A1 Monoamine reuptake inhibitors for treatment of cns disorders |
| 08/31/2000 | WO2000050377A1 Efficient synthesis of secondary amines by selective alkylation of primary amines |
| 08/31/2000 | WO2000050376A2 Efficient synthesis of alkyl carbonates |
| 08/31/2000 | WO2000040558A8 Aspartic protease inhibitors |
| 08/31/2000 | WO2000001375A3 Calcium channel blockers |
| 08/31/2000 | DE19907829A1 Verfahren zur Herstellung von cis-2,6-Dimethylpiperazin A process for preparing cis-2,6-dimethylpiperazine |
| 08/31/2000 | CA2364849A1 Compounds and compositions for delivering active agents |
| 08/31/2000 | CA2363628A1 Catalysts containing n-pyrrolyl substituted nitrogen donors |
| 08/30/2000 | EP1031626A1 Method for stabilising and/or isolating nucleic acids |
| 08/30/2000 | EP1031568A1 Process for the preparation of cis-Dimethylpiperazine |
| 08/30/2000 | EP1031563A1 Sulfonyl derivatives |
| 08/30/2000 | EP0787141B1 Cyclic depsipeptide sulfonylation, sulfenylation and phosphorylation process |
| 08/30/2000 | CN1265101A Crystalline dibentothiazepine derivatives and its use as antipsychotic agent |
| 08/30/2000 | CN1265096A Hydrazine derivatives |
| 08/30/2000 | CN1055920C Aklyl benzoylguanidines derivatives |
| 08/29/2000 | US6111132 Compounds and methods for synthesis and therapy |
| 08/29/2000 | US6111105 Chemical intermediates for ziprasidone, a neuroleptic agent; reacting a 2-(piperidino) or (1,2-benzisoxazol-3-yl) or (2-cyanophenyl)thio),3-cyanobenzene with piperazine at a temperature from 80-170 degrees c. |
| 08/29/2000 | US6111100 Preparation of bis(2-morpholinoethyl) ether |
| 08/29/2000 | US6110947 An analgesic agent for treating stroke, abdominal pain; as antiinflammatory, diuretic, anesthetic or neuroprotective agents |
| 08/29/2000 | US6110944 LTA4, hydrolase inhibitors |
| 08/29/2000 | US6110933 Amino acid derivatives and their use as phospholipase A2 inhibitor |
| 08/29/2000 | US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds |
| 08/24/2000 | WO2000049002A1 Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils |
| 08/24/2000 | WO2000048993A1 Arylaminoalkylamides |
| 08/24/2000 | WO2000048992A1 Acylated aminoacetonitriles as cysteine protease inhibitors |
| 08/24/2000 | WO2000048987A1 Novel substituted 3-phenoxy and 3-phenylalkyloxy-2-phenyl-propylamines |
| 08/24/2000 | WO2000002887B1 Ligands for metals and metal-catalyzed processes |
| 08/24/2000 | DE19907385A1 New 3-(phenoxy or phenylalkoxy)-2-phenyl-propylamines, useful for treating e.g. arrhythmia, spasms, pain or neurodegenerative diseases, are tension-dependent sodium channel blockers |
| 08/24/2000 | CA2364281A1 Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils |
| 08/23/2000 | EP1029861A1 Benzisothiazol-piperazinyl derivative and its use as neuroleptic |
| 08/23/2000 | EP1029851A1 Piperazine compounds and medicinal use thereof |
| 08/23/2000 | EP1029297A2 Method of virtual retrieval of analogs of lead compounds |
| 08/23/2000 | EP1028942A2 Dipeptide nitriles |
| 08/23/2000 | EP1028940A1 Process to produce oxazolidinones |