Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
05/2000
05/30/2000CA1341011C Benzo-fused cycloalkane and oxa- and thia-, cycloalkane trans-1,2-diamine derivatives
05/25/2000WO2000028988A1 Nitrosated and nitrosylated h2 receptor antagonist compounds, compositions and methods of use
05/25/2000WO2000028983A1 Novel 4-dedimethy laminotetra cycline derivatives
05/25/2000CA2349575A1 Nitrosated and nitrosylated h2 receptor antagonist compounds, compositions and methods of use
05/24/2000EP1001777A1 Fibrinogen receptor antagonists
05/24/2000EP1001776A1 Aroylpiperazines for modulating sexual activity
05/24/2000EP1001766A1 Compounds and methods
05/24/2000CN1254337A N-hydroxy 4-sulfonyl butyramide compounds
05/23/2000US6066735 Treatment of erectile dysfunction
05/23/2000US6066730 Boronic ester and acid compounds, synthesis and uses
05/23/2000US6066656 2,5-diamino-3,4-disubstituted-1,6-diphenylhexane isosteres comprising benzamide, sulfonamide and anthranilamide subunits and methods of using same
05/23/2000CA2290249A1 Polysulfide solutions and hydroxyalkyl aminium ions for stabilizing elemental sulfur
05/18/2000WO2000027855A1 Chiral ligands for asymmetric catalysis
05/18/2000WO2000027843A1 Ccr-3 receptor antagonists
05/18/2000WO2000027833A1 Drug dependence remedies
05/18/2000WO2000027826A1 Novel pyrimidines, the production thereof and their use
05/18/2000WO2000027808A1 N-arylsulfonyl amino acid omega amides
05/18/2000WO2000027800A1 Ccr-3 receptor antagonists
05/18/2000WO2000027790A1 Mutilin compounds
05/18/2000WO2000027378A2 Cystine derivatives as therapeutic agents for matrix metalloprotease related diseases
05/18/2000WO2000010544A3 A method for preventing the onset of asthma
05/18/2000WO2000006140A3 Use of moclobemide for treating certain phsychiatric and medical disorders
05/18/2000CA2348946A1 Cystine derivatives as therapeutic agents for matrix metalloprotease related diseases
05/18/2000CA2347146A1 Chiral ligands for asymmetric catalysis
05/17/2000EP1000934A2 Pesticidal and parasiticidal use of 1-aryl-1-(substituted thio, sulfinyl and sulfonyl)-2-nitroethane compounds
05/17/2000EP1000090A1 Novel photoinitiators and applications therefor
05/17/2000EP1000048A1 Substituted 1,2,3,4-tetrahydronaphthalene derivatives
05/17/2000EP1000047A1 1-(n-phenylaminoalkyl)-piperazine derivatives substituted at position 2 of the phenyl ring
05/17/2000EP1000046A1 Piperazine derivatives active on the lower urinary tract
05/17/2000EP1000043A1 A crystalline dibenzothiazepine derivative and its use as an antipsychotic agent
05/17/2000EP1000023A2 Novel nitric oxide-releasing amidine- and enamine-derived diazeniumdiolates, compositions and uses thereof and method of making same
05/17/2000EP1000018A2 Urokinase inhibitors
05/17/2000EP1000016A1 Isocyanoalkyl carbonic acid derivatives, their conversion into secondary amidoalkyl carbonic acid derivatives by isocyanide-multicomponent reactions, as well as these secondary amidoalkyl carbonic acid derivatives.
05/17/2000EP1000012A1 Process for converting propargylic amine-n-oxides to enaminones
05/17/2000EP0999840A1 Use of draflazine-analogues for treating pain
05/17/2000EP0726768B1 Use of nitric oxide releasing compounds for the manufacture of a medicament for protection in ischemia reperfusion injury
05/17/2000CN1253561A Pyrazolopyrimidinones which inhibit type 5 cyclic guanosine 3', 5'-monophosphate phosphodiesterase (cGMP PDE5) for treatment of sexual dysfunction
05/17/2000CN1253559A Sulfonyl divalent aryl alpha-hydroxamic acid compounds
05/17/2000CN1253555A Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and pharmaceutical compositions containing same
05/17/2000CN1253547A 1,4-substituted cyclic amine derivatives
05/17/2000CN1253545A Aryl sulfonamides and analogues thereof and their use in treatment of neurodegenerative diseases
05/17/2000CN1253474A Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
05/16/2000US6063792 Methods and compositions for treating urinary incontinence using enantiomerically enriched (S)-trihexyphenidyl
05/16/2000CA2289827A1 Pesticidal and parasiticidal use of 1-aryl-1-(substituted thio, sulfinyl and sulfonyl)-2-nitroethane
05/11/2000WO2000026189A1 Method for producing nitroxyl compounds of secondary amines
05/11/2000WO2000025776A1 Nitrosated and nitrosylated nonsteroidal antiinflammatory compounds, compositions and methods of use
05/11/2000DE19851421A1 Neue Pyrimidine, deren Herstellung und Verwendung New pyrimidines, their preparation and use
05/11/2000DE19851184A1 N-Arylsulfonyl-aminosäure-omega-amide N-arylsulfonyl-amino-omega-amides
05/10/2000EP0999220A2 Low molecular weight peptidomimetic growth hormone secretagogues
05/10/2000EP0999205A1 Aminocycloalkane compounds
05/10/2000EP0999204A1 Novel compound having effect of promoting neuron differentiation
05/10/2000EP0998469A1 Benzamide cycloalkyl stimulating high and low gastrointestinal motricity
05/10/2000EP0998451A1 Substituted 3,3-diamino-2-propenenitriles, their preparation and use
05/10/2000EP0998281A1 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith
05/10/2000EP0685234B1 Drug composition containing nucleic acid copolymer
05/10/2000CN1252790A N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
05/10/2000CN1252713A N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
05/10/2000CN1052231C 2-oxo-5-oxazolidone methyl compound their preparing method and medicinal composition containing them
05/10/2000CN1052228C Preparing method for n-formyl piperidine and homologs thereof
05/09/2000US6060513 Compounds and compositions for delivering active agents
05/09/2000US6060503 Antiestrogenic, anticarcinogenic stereospecific benzopyran derivative; breast cancer
05/09/2000US6060492 Side effect reduction
05/09/2000US6060476 α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
05/04/2000WO2000024710A1 N-(2-aryl-propionyl)-sulfonamides and pharmaceutical preparations containing them
05/04/2000WO2000024394A1 Antitumor chrysene derivatives
05/04/2000WO2000006254A3 Non-imidazole alkylamines as histamine h3-receptor ligands and their therapeutic applications
05/04/2000WO2000006139A3 Use of moclobemide and metabolites for treating and preventing substance abuse
05/04/2000WO1999064038A9 Novel analgesic agents
05/04/2000WO1999064031A9 β2-ADRENERGIC RECEPTOR AGONISTS
05/04/2000DE19850625A1 Verfahren zur Herstellung von Nitroxylverbindugen sekundärer Amine A process for preparing secondary amines Nitroxylverbindugen
05/04/2000CA2346873A1 Antitumor chrysene derivatives
05/03/2000EP0997459A1 Intermediates for preparing retroviral protease inhibiting compounds
05/03/2000EP0997147A1 Amino acid derivatives
05/03/2000EP0996614A1 Acrylonitrile compounds, process for their production and pesticides containing them
05/03/2000EP0996440A1 Method for treatment of glutamate related disorders
05/03/2000EP0996434A1 Kappa agonist anti-pruritic pharmaceutical formulations and method of treating pruritus therewith
05/03/2000EP0996433A1 Methods for treatment of conditions associated with lactosylceramide
05/03/2000EP0861233B1 N-protected/n-substituted-beta-amino hydroxy sulfonates
05/03/2000CN1252050A Hydrogenation of imine and enamine
05/02/2000US6057443 Dimorpholinodiethylether having improved isocyanate stability
05/02/2000US6057442 Preparation of amines
05/02/2000US6057419 Drugs and images
05/02/2000US6057371 Sigma receptor ligands and the use thereof
05/02/2000US6057362 Protease inhibitors
05/02/2000US6057358 Amine derivatives, processes for producing them and a use of them as antiarrhythmic drugs
05/02/2000US6057323 Kappa agonist compounds pharmaceutical formulations and method of prevention and treatment of pruritus therewith
04/2000
04/27/2000WO2000023420A1 Aromatic amine derivatives, process for the preparation thereof and agents containing the same
04/27/2000WO2000023419A1 Novel prodrugs of non-steroidal anti-inflammatory carboxylic acids, their preparation and use
04/27/2000WO2000023407A2 Ureido-thiobutyric acid derivatives as ppar-agonists
04/27/2000WO2000006137A3 Glucocorticoid-selective anti-inflammatory agents
04/27/2000WO1999063933A9 Multivalent agonists, partial agonists and antagonists of the gaba receptors
04/27/2000CA2348159A1 Aromatic amine derivatives, their production and use
04/26/2000EP0995741A1 Remedies/preventives for frequent urination/urinary incontinence and tropone derivatives
04/26/2000EP0994884A1 Diphosphonic acid salts for the treatment of osteoporosis
04/26/2000EP0994862A2 Sulphonamide derivatives being 5-ht6 receptor antagonists and process for their preparation
04/26/2000EP0994848A1 Glucagon antagonists/inverse agonists
04/26/2000EP0994712A1 Inhibitors of neutrophil mediated oxidant production
04/26/2000EP0994710A1 Pharmaceutical compositions for oral administration, comprising an active substance and a cyclodextrin
04/26/2000EP0973737A4 Efficient synthesis of a chiral mediator
04/26/2000EP0680469B1 Aminoacid derivates, medicaments containing these compounds and process for preparing the same