Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
11/1998
11/24/1998US5840905 Reducing 4-oxo-2,2,6,6-tetramethylpiperidine, reacting formed 4-hydroxy-2,2,6,6-tetramethylpiperidine with formaldehyde and formic acid in water as solvent, separating aqueous phase, distilling product
11/24/1998US5840886 Silver halide photographic material and hydroxamic acid based compound used therefore
11/24/1998US5840761 Antiarrhythmia agents, inhibitors of the cellular na+/h+ antiporter
11/24/1998US5840735 Estrogen
11/24/1998US5840725 Substituted oximes, hydrazones and olefins as neurokinin antagonists
11/19/1998WO1998051298A1 Arylsubstituted piperazines useful in the treatement of benign prostatic hyperlasia
11/19/1998DE19720475A1 Preparation of N-alkyl-2,6-di:alkyl-morpholine derivatives e.g. fenpropimorph or dodimorph
11/18/1998EP0877737A1 Novel n-(arylsulphonyl)amino acid derivatives having bradykinin receptor affinity
11/18/1998EP0877612A1 Use of piperazine derivatives for the treatment of cognitive disorders
11/18/1998EP0757669B1 O-acyl-4-phenyl-cyclohexanols, their salts, medicaments containing such compounds and their use, as well as a method of preparing them
11/18/1998EP0724581B1 Crystalline anhydrous mycophenolate mofetil and intravenous formulation thereof
11/18/1998EP0688312B1 New derivatives of glutamic acid, a method of preparing them, and their use as drugs for enhancing memory and learning
11/18/1998CN1199398A 1-[2-(2,3-dihydro-1H-inden-1-yl) ethyl]-4-(naphthalen-1-yl) piperazine derivs, preparation thereof and therapeutical use thereof
11/18/1998CN1199394A Didepsipeptide-based endoparasiticides, new didepsipeptides and process for preparing same
11/18/1998CN1040751C Process for preparation of benzothiazepine derivs.
11/17/1998US5837873 Intermediates of retroviral protease inhibiting compounds
11/17/1998US5837870 Process to prepare oxazolidinones
11/17/1998US5837717 Hydroxamic acid anesthetic compounds
11/17/1998US5837710 Enzyme inhibitors for treatment of aids
11/17/1998US5837707 Dimeric piperidine, tetrahydropyridine and piperazine derivatives
11/17/1998US5837703 Amino-alcohol substituted cyclic compounds
11/17/1998US5837016 Fuel additive
11/12/1998WO1998050344A1 Substituted 3,3-diamino-2-propenenitriles, their preparation and use
11/12/1998WO1998050342A1 Protease inhibitors
11/12/1998WO1998050031A1 Inhibitors of protein isoprenyl transferases
11/12/1998WO1998050030A1 Inhibitors of protein isoprenyl transferases
11/12/1998WO1998050029A1 Inhibitors of protein isoprenyl transferases
11/12/1998WO1998035951A3 New aminopiperazine derivatives
11/12/1998CA2289602A1 Protease inhibitors
11/12/1998CA2289099A1 Substituted 3,3-diamino-2-propenenitriles, their preparation and use
11/12/1998CA2288330A1 Benzoyl amino acid derivatives useful as inhibitors of protein isoprenyl tranferases
11/11/1998EP0877019A1 Substituted diaminocarboxylic acid
11/11/1998EP0877018A1 Sulfonylaminocarboxylic acids
11/11/1998EP0877014A2 Diaminoalkylene quaternary ammonium salts, method for their preparation and use
11/11/1998EP0876359A1 (-) cis-6(s)-phenyl-5(r) 4-(2-pyrrolidin-1-ylethoxy)phenyl]-5,6,7,8-tetrahydronaphthalen-2-ol d-tartrate
11/11/1998EP0876338A1 Guanidine derivatives
11/11/1998EP0876337A2 New lh-rh antagonists with improved effectiveness
11/11/1998EP0876326A1 Process for producing amines from olefins on zeoliths of types ssz-26, ssz-33, cit-1 or mixtures thereof
11/11/1998EP0778832B1 Process for producing quaternary glycine nitriles
11/11/1998EP0641766B1 Alkoxyphenylalkylamine derivative
11/11/1998CN1198668A Naphthyl and dihydronaphthyl intermediates, compounds, compositions, and methods
11/10/1998US5834508 Ketone derivatives
11/10/1998US5834506 Treatment of hiv, aids; antiviral activity improved by judicious placement of polar substituents
11/10/1998US5834487 Inhibition of 26S and 20S proteasome by indanones
11/10/1998US5834471 Amide derivatives as 5HT1D receptor antagonists
11/10/1998US5834467 HIV protease inhibitors
11/09/1998CA2237052A1 Substituted diaminocarboxylic acids
11/05/1998WO1998049166A1 PYRAZOLOPYRIMIDINONES WHICH INHIBIT TYPE 5 CYCLIC GUANOSINE 3',5'-MONOPHOSPHATE PHOSPHODIESTERASE (cGMP PDE5) FOR THE TREATMENT OF SEXUAL DYSFUNCTION
11/05/1998WO1998049158A1 Peripherally selective kappa opioid agonists
11/05/1998WO1998049131A1 New benzylamine and phenylethylamine derivatives, processes for preparing the same and their use as medicaments
11/05/1998WO1998048806A1 Indene compounds having activity as serms
11/05/1998WO1998048773A1 Oxidation colorants
11/05/1998DE19718334A1 Neue Benzylaminderivate und Phenylethylaminderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel New benzylamine derivatives and phenylethylamine derivatives, processes for their preparation and their use as medicaments
11/05/1998DE19718187A1 Oxidationsfärbemittel An oxidation
11/05/1998CA2287244A1 Indene compounds having activity as serms
11/04/1998EP0875507A1 Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceuticals
11/04/1998EP0875501A2 Alkylenediamine derivative, anti-ulcer drug, and antibacterial drug
11/04/1998EP0874927A1 Process for preparation of an aqueous solution of n-methylmorpholin-n-oxide
11/04/1998EP0874836A1 Sulfonamide inhibitors of matrix metalloproteinases
11/04/1998EP0874834A1 Processes and intermediates for preparing 3-(1-piperazinyl)-1,2-benzisothiazole
11/04/1998EP0874830A1 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses, and methods and intermediates useful for their preparation
11/04/1998EP0874809A1 Carbamoyloxy derivatives of mutiline and their use as antibacterials
11/04/1998EP0874645A2 Perfluoroalkyl-containing metal complexes and their use in nmr diagnostics
11/04/1998EP0874625A1 Indane derivatives for antipsychotic compositions
11/04/1998EP0712838B1 Acylphenylglycine derivative and preventive and remedy for diseases caused by increased collagenase activity containing said compound as active ingredient
11/04/1998EP0705244B1 Nitrato amino acid disulphides for use in the therapy of disorders of the cardiovasculary system
11/04/1998EP0655992B1 Fluorenone derivatives, process for preparing the same and central or peripheral nerve degeneration repair and protective agent
11/04/1998EP0640069B1 Fluoroalkenyl compounds and their use as pest repellents
11/04/1998CN1198155A Process for preparation of piperidines
11/03/1998US5831094 Difluoro statone antiviral analogs
11/03/1998US5830896 Psychological disorders; antiepilepic agents; alzheimer'sand parkinson?s disease
11/03/1998CA1340113C Aryl-and heteroaryl piperazinyl carboxamides having central nervous system activity
10/1998
10/30/1998CA2231013A1 Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceuticals
10/29/1998WO1998047885A1 A bicyclic aryl or a bicyclic heterocyclic ring containing compounds having a combined 5ht1a, 5ht1b and 5ht1d receptor antagonistic activity
10/29/1998WO1998047863A1 Amino acid derivatives inhibiting extracellular matrix metalloproteinase and tnf alpha release
10/29/1998WO1998047859A1 Amphoteric surfactants having multiple hydrophobic and hydrophilic groups
10/29/1998WO1998047362A1 Use of hydroxylamine derivatives, and method and preparations for increasing the tolerance of field crops against weather stresses
10/29/1998CA2288172A1 A bicyclic aryl or a bicyclic heterocyclic ring containing compounds having a combined 5ht1a, 5ht1b and 5ht1d receptor antagonistic activity
10/29/1998CA2288075A1 Use of hydroxylamine derivatives, and method and preparations for increasing the tolerance of field crops against weather stresses
10/29/1998CA2287565A1 Amino acid derivatives inhibiting extracellular matrix metalloproteinase and tnf alpha release
10/28/1998EP0873992A1 Indene compounds having activity as SERMs
10/28/1998EP0873406A2 Protein induced by deprenyl
10/28/1998EP0873330A1 Diarylalkenylamine derivatives
10/28/1998EP0873329A1 Novel n-aminoalkylfluorenecarboxamides; a new class of dopamine receptor subtype specific ligands
10/28/1998EP0873308A1 O-carbamoyl-phenylalaninol compounds, their pharmaceutically useful salts and process for preparing the same
10/28/1998EP0873119A1 Use of the l-enantiomer of centchroman for the manufacture of a pharmaceutical composition for the treatment or prophylaxis of breast cancer
10/28/1998EP0656887B1 Hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
10/28/1998EP0627406B1 2-amino-1,3-propanediol compound and immunosuppressant
10/28/1998EP0476016B1 CNS active 8-heterocyclyl-2-aminotetralin derivatives
10/28/1998CN1197457A Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
10/28/1998CN1197062A Production of keto acids
10/27/1998US5827927 Rigid polymer rods and macromonomers with reactive end groups for reinforcement
10/27/1998US5827891 For treatment of aids, blocking replication of hiv virus
10/27/1998US5827881 Diesters of carbonic acid endowed with antiviral and anti-inflammatory activity
10/27/1998US5827877 Ketomethylene group-containing cysteine and serine protease inhibitors
10/27/1998US5827859 HIV protease inhibitors
10/27/1998US5827858 Administered to treat aids
10/27/1998US5827847 Treatment of cognitive disorders with piperazine derivatives
10/22/1998WO1998046591A1 SELECTIVE FACTOR Xa INHIBITORS
10/22/1998CA2285335A1 Selective factor xa inhibitors