C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms

Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
11/1999
11/02/1999	US5977357 Phenyl alkyl ketone substituted by cyclic amine and a process for the preparation thereof
11/02/1999	US5977182 O-benzyl oxime ether derivatives and their use as pesticides
11/02/1999	US5977154 Obesity, diabetes
11/02/1999	US5977141 Sulfonamide inhibitors of matrix metalloproteinases
11/02/1999	US5977115 Alpha 1a adrenergic receptor antagonists
11/02/1999	US5977114 Selective thrombin inhibitors
11/02/1999	US5977075 N-aroylamino acid amides as endothelin inhibitors
11/02/1999	US5977074 Inhibitors of β-amyloid protein production
11/02/1999	US5976858 (s)-(e)-3-(4-morpholine-carbonylleucyl)amino-5-phenyl-1-phenyl sulfonyl-1-pentene and others; antiarthritis/antitumor/ antiinflammatory/antimetastasis agents; treatment of muscular dystrophy, malaria, alzheimer's and autoimmune diseases
11/02/1999	US5976781 Diagnosing malaria by mixing blood with enzyme inhibitor, determining enzyme activity, comparing to control sample; plasmodium enzyme is more sensitive to inhibition so deactivation indicates disease
10/1999
10/28/1999	WO1999054337A1 Ancillary ligands and metal complexes thereof
10/28/1999	WO1999054321A1 Substituted diamines and their use as cell adhesion inhibitors
10/28/1999	WO1999054320A1 Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
10/28/1999	WO1999054310A2 New substituted amides, their production and their use
10/28/1999	WO1999054305A1 Heterocyclically substituted amides used as calpain inhibitors
10/28/1999	WO1999054293A1 Substituted benzamides, their production and their use as cysteine protease inhibitors
10/28/1999	WO1999053911A1 Antifungal agents
10/28/1999	WO1999024460B1 Dipeptide nitriles
10/28/1999	CA2328720A1 Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
10/28/1999	CA2328430A1 Substituted benzamides, their production and their use as cysteine protease inhibitors
10/28/1999	CA2290362A1 Ancillary ligands and metal complexes thereof
10/27/1999	EP0952154A2 N-acyl and N-aroyl aralkyl amides
10/27/1999	EP0952153A2 A process for the preparation of esters of [2-[4-[(4-chlorophenyl)phenylmethyl]-1-piperazinyl]-ethoxy]acetic acid
10/27/1999	EP0952152A2 Triethylenediamine and piperazine synthesis using zeolithe catalysts modified with a silicon-containing compound
10/27/1999	EP0951438A1 Granular n-alkyl ammonium acetonitrile compositions
10/26/1999	US5973075 Methods for preparing rigid-rod macromonomers with reactive end groups
10/26/1999	US5972977 Ophthalmic pharmaceutical compositions comprising a nitrone compound and methods for treating ocular inflammation using such compositions
10/26/1999	US5972964 Aminomethylindans, -benzofurans and -benzothiophenes
10/26/1999	US5972940 Arginine analogues having nitric oxide synthase inhibitor activity
10/26/1999	US5972939 Cyclopentene derivatives useful as antagonists of the motilin receptor
10/26/1999	US5972928 Administering an antigrowth agent
10/26/1999	US5972897 Acylated enol derivatives as prodrugs of elastase inhibitors
10/26/1999	US5972307 Administering to human or animal body an effective amount of a diagnostic agent comprises a metal chelate of a compound having two macrocyclic chelant groups linked by a bridge containing ester or amide bond
10/21/1999	WO1999053039A1 Treatment of parasitic diseases by inhibition of cysteine proteases of the papain superfamily
10/21/1999	WO1999052876A1 Azacycloalkane derivatives, preparation and therapeutic application
10/21/1999	WO1999052368A1 Plant growth regulator compositions
10/21/1999	WO1999037623A3 Sulphonamide derivatives for treatment of cns disorders
10/21/1999	WO1999033454A3 S-procyclidine for treating urinary incontinence
10/21/1999	DE19817461A1 New benzamide derivatives useful as cysteine protease inhibitors for treating neurodegenerative diseases, neuronal damage, stroke, cranial trauma, Alzheimer's disease, etc.
10/21/1999	DE19816929A1 New amino acid derivatives useful as neuropeptide Y agonists and/or antagonists for treating cardiovascular disorders, coronary, cerebral or renal vasospasms, obesity, bulimia and asthma
10/21/1999	DE19816889A1 New piperazine derivatives useful in treatment of e.g. cardiovascular, renal and central nervous system disorders, obesity and diabetes, in antibody production and as analytical and diagnostics aids
10/21/1999	CA2327282A1 Treatment of parasitic diseases by inhibition of cysteine proteases of the papain superfamily
10/20/1999	EP0950016A1 Liquid compositions containing n-alkyl ammonium acetonitrile salts
10/20/1999	CN1232462A Muscarinic antagonists
10/20/1999	CN1232447A Hydroxamic acid derivs.
10/20/1999	CN1232446A Process for producing depsipeptide derivs, and noval intermidiates therefor
10/20/1999	CN1232443A Novel p-terphenyl compounds
10/20/1999	CN1232388A Antimalarial and anti-babesiosis agent and pharmaceutical compositions contg. same
10/20/1999	CN1232035A Preparation of beta-methyl carbapenem intermediates
10/20/1999	CN1232022A [6-(substd. methyl)-3-cyclohexenyl] carboxamide derivs., and hair tonic and external use preparation for skin
10/19/1999	US5969133 Bioreductive cytotoxic agents
10/19/1999	US5969114 Azo compound
10/19/1999	US5968985 Benzoylguanidine derivatives as medicaments
10/19/1999	US5968977 Ketonitrile derivatives and antibacterial agent and drugs containing the same
10/19/1999	US5968968 Analgesic or antiinflammatory agents, also for treatment of strokes, asthma, parkinsonism, psoriasis, irritable bowel syndrome
10/19/1999	US5968962 Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
10/19/1999	US5968938 Treating preterm labor in mammals, treating dysmenorrhea, stopping labor prior to cesarean delivery
10/19/1999	US5968936 Methods for treating or preventing Alzheimer's Disease using substituted 1-aryl-3-morpholinopropanones
10/19/1999	US5968916 Agricultural insecticides, nematocides or miticides
10/16/1999	CA2269049A1 N-acyl and n-aroyl aralkyl amides
10/14/1999	WO1999051609A1 Method for producing grignard compounds
10/14/1999	WO1999051571A1 Benzamide and sulfonamide substituted aminoguanidines and alkoxyguanidines as protease inhibitors
10/14/1999	WO1999051564A1 Propanolamine derivatives
10/14/1999	WO1999027937A3 Method for inhibiting cytokine production by cells
10/14/1999	CA2326759A1 Benzamide and sulfonamide substituted aminoguanidines and alkoxyguanidines as protease inhibitors
10/13/1999	EP0948455A1 Mixed peroxygen activator compositions
10/13/1999	EP0783486B1 Novel prostaglandin synthase inhibitors
10/13/1999	EP0692977B1 Novel heterocycle based nitrogen-sulfur ligands useful in radiographic imaging agents
10/13/1999	CN1231665A Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
10/13/1999	CN1231612A Inhibition of 2,3-dihydrogen-indone to 26S and 20S prolease
10/13/1999	CN1045594C Nitrato amino acid disulphides for use in the therapy of disorders of the cardiovasculary system
10/13/1999	CN1045590C Hydrazine derivative and application of same
10/12/1999	US5965560 Substituted piperazines and piperidines as central nervous system agents
10/12/1999	US5965434 Compounds contain cationic groups whose positive charge increases with decreasing ph; cationic liposomes fuse at ph's in the low end of the physiologic range; use in drug delivery systems; efficiency, less toxicity
10/12/1999	US5965121 Compounds and compositions for delivering active agents
10/07/1999	WO1999050247A1 Compounds with activity on muscarinic receptors
10/07/1999	WO1999050238A1 Novel urea derivatives
10/07/1999	WO1999050237A1 Sulfonamide derivatives and drugs containing the same as the active ingredient
10/07/1999	WO1999050225A1 Aminocyclohexyl ether compounds and uses thereof
10/07/1999	WO1999050211A1 Reduction of carbonyl compounds by a silane in the presence of a zinc catalyst
10/07/1999	WO1999033453A3 R-procyclidine for treating urinary incontinence
10/07/1999	DE19812058C1 New 2-heterocyclyl-1,4-phenylenediamine derivatives
10/07/1999	CA2325997A1 Sulfonamide derivatives and drugs containing the same as the active ingredient
10/07/1999	CA2291486A1 Reduction of carbonyl compounds by a silane in the presence of a zinc catalyst
10/06/1999	EP0947503A1 6,8-Dimethylmercaptooctanoic acid derivatives substituted on 6-S and/or 8-S by the 3-methylthiopropanoyl radical and pharmaceutical compositions for the treatment of cancerous tumours
10/06/1999	EP0947496A1 Bicyclic aromatic compounds and their use in human and veterinary medicine as well as in cosmetology
10/06/1999	EP0946551A2 N-piperazin-1-ylphenyl-benzamide derivatives
10/06/1999	EP0946539A1 Sulphonamide derivatives, process for their preparation, and their use as medicaments
10/06/1999	EP0946526A1 Macrocyclic metal complex carboxylic acids, use and method for the production thereof
10/06/1999	EP0946519A1 Benzamide derivatives having a vasopressin antagonistic activity
10/06/1999	EP0946504A1 Compounds useful for perhalogenoalkylation, reagent for implementing these compounds and synthesis method for obtaining these compounds
10/06/1999	EP0946166A1 Use of matrix metalloproteinase inhibitors for treating neurological disorders and promoting wound healing
10/06/1999	CN1230884A Thiol sulfone metalloprotease inhibitors
10/06/1999	CN1230541A Preparation of N-formyl piperidine
10/05/1999	US5962682 Aryl- and hetaryl-sulfonamide derivatives, their preparation and their use as endothelin antagonists
10/05/1999	US5962531 5-aroylnaphthalene derivatives as anti-inflammatory agents
10/05/1999	US5962529 Metalloproteinase inhibitors
10/05/1999	US5962507 O-acyl-4-phenyl-cyclohexanols, their salts, medicaments containing such compounds, and their use, as well as a method of preparing them
10/05/1999	US5962456 Peptic ulcers
10/05/1999	US5962455 Eating disorders, cardiovascular disorders, hypotensive agents

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