Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
12/1999
12/23/1999DE19827163A1 Verfahren zur katalytischen, unsymmetrischen Disubstitution von Carbonsäureamiden mit 2 unterschiedlichen Grignardreagenzien Process for the catalytic, asymmetric disubstitution of carboxamides with 2 different Grignard reagents
12/23/1999DE19827161A1 Verfahren zur katalytischen, symmetrischen Disubstitution von Carbonsäureamiden mit Grignardreagenzien Process for the catalytic symmetrical disubstitution of carboxamides with Grignard reagents
12/23/1999DE19822041A1 2,5-Diamino-1-phenylbenzol-Derivate enthaltende Oxidationshaarfärbemittel sowie neue 2,5-Diamino-1-phenylbenzol-Derivate 2,5-diamino-1-phenylbenzene derivatives containing oxidation hair as well as new 2,5-diamino-1-phenylbenzene derivatives
12/23/1999CA2335293A1 Inhibitors of transcription factor nf-.kappa.b
12/23/1999CA2335112A1 Therapeutic combinations for musculoskeletal frailty
12/23/1999CA2334797A1 Anthracene derivatives as anti-cancer agents
12/23/1999CA2334254A1 Cycloalkyl-substituted aryl-piperazines, piperidines and tetrahydropyridines as serotonergic agents
12/22/1999EP0965591A1 (s)-3-methyl-1-(2-piperidino-phenyl)-1-butylamine, its salts, synthesis and use in the long term therapy of diabetes mellitus
12/22/1999EP0964863A1 Oxazolidines as 5-ht2a-antagonists
12/22/1999EP0939628A4 Thiol sulfone metalloprotease inhibitors
12/22/1999EP0792261B1 O-benzyl oxime ether derivatives and their use as pesticides
12/22/1999EP0733033B1 Pharmaceutically active substituted aromatic compounds
12/22/1999EP0635018B1 4-(1H-2-METHYLIMIDAZO[4,5-c]PYRIDINYLMETHYL)PHENYLSULPHONAMIDE DERIVATIVES AS ANTAGONISTS OF PAF
12/22/1999CN1047594C Piperazinyl- and piperidinyl-cyclohexanols, its prepn. and application
12/21/1999US6005102 Aryloxy-alkyl-dialkylamines
12/21/1999US6004964 Administering amide or sulfonamide derivative; analgesics
12/21/1999US6004961 1,4-disubstituted piperazines
12/21/1999US6004959 Alkyloxyamino substituted fluorenones and their use as protein kinase-C inhibitors
12/21/1999US6004948 Derivatives of benzosulphonamides as inhibitors of the enzyme cyclooxygenase II
12/21/1999CA2006577C Hypoglycaemic phenylamidines and phenylguanidines
12/16/1999WO1999064595A1 THERAPEUTIC AND DIAGNOSTIC DOMAIN 1 β2GPI POLYPEPTIDES AND METHODS OF USING SAME
12/16/1999WO1999064407A1 α-(1-PIPERAZINYL)ACETAMIDO ARENECARBOXYLIC ACID DERIVATIVES AS ANTIDIABETIC AGENTS
12/16/1999WO1999064394A1 Neuropeptide y5 receptor antagonists
12/16/1999WO1999064393A1 Novel antiestrogens, a method for the production thereof, and their pharmaceutical application
12/16/1999WO1999064055A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht4 receptors
12/16/1999WO1999064053A1 β3-ADRENERGIC RECEPTOR AGONISTS
12/16/1999WO1999064052A1 Novel leukotriene receptor antagonists and their uses
12/16/1999WO1999064042A1 Novel therapeutic agents that modulate alpha-1a adrenergic receptors
12/16/1999WO1999064041A1 Multibinding agents that modulate nmda receptors
12/16/1999WO1999064038A1 Novel analgesic agents
12/16/1999WO1999064035A1 β2-ADRENERGIC RECEPTOR AGONISTS
12/16/1999WO1999064034A1 β2-ADRENERGIC RECEPTOR AGONISTS
12/16/1999WO1999064031A1 β2-ADRENERGIC RECEPTOR AGONISTS
12/16/1999WO1999064000A1 Novel therapeutic agents that modulate neurokinin receptors
12/16/1999WO1999063999A1 H1-histamine receptor antagonists
12/16/1999WO1999063996A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht2 receptors
12/16/1999WO1999063993A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the d1 receptors
12/16/1999WO1999063983A1 MULTIBINDING AGENTS THAT MODULATE PPARη AND RXR RECEPTORS
12/16/1999WO1999063944A2 Novel therapeutic agents that modulate estrogen receptors
12/16/1999WO1999063936A2 Novel therapeutic agents that modulate endothelin receptors
12/16/1999WO1999063933A2 Multivalent agonists, partial agonists and antagonists of the gaba receptors
12/16/1999WO1999063930A2 Novel angiotensin receptor modulators and their uses
12/16/1999DE19851300A1 Tryptase-Inhibitoren Tryptase inhibitors
12/16/1999DE19826396A1 Verfahren zur Herstellung von Aminen A process for preparing amines
12/16/1999DE19826213A1 Neue Antiestrogene, Verfahren zu ihrer Herstellung und ihre pharmazeutische Verwendung New antiestrogens, processes for their preparation and their pharmaceutical use
12/16/1999CA2334780A1 Novel antiestrogens, a method for the production thereof, and their pharmaceutical application
12/16/1999CA2334558A1 .alpha.-(1-piperazinyl)acetamido arenecarboxylic acid derivatives as antidiabetic agents
12/16/1999CA2329942A1 Therapeutic and diagnostic domain 1 .beta.2gpi polypeptides and methods of using same
12/16/1999CA2321273A1 Novel analgesic agents
12/16/1999CA2321170A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the d1 receptors
12/16/1999CA2321152A1 Novel therapeutic agents that modulate endothelin receptors
12/16/1999CA2321120A1 .beta.3-adrenergic receptor agonists
12/16/1999CA2320926A1 Novel leukotriene receptor antagonists and their uses
12/16/1999CA2319756A1 Novel therapeutic agents that modulate alpha-1a adrenergic receptors
12/16/1999CA2319751A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht2 receptors
12/16/1999CA2319651A1 H1-histamine receptor antagonists
12/16/1999CA2319643A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht4 receptors
12/16/1999CA2319497A1 Novel therapeutic agents that modulate estrogen receptors
12/16/1999CA2319496A1 Multivalent agonists, partial agonists and antagonists of the gaba receptors
12/16/1999CA2319175A1 Multibinding agents that modulate nmda receptors
12/16/1999CA2319159A1 Novel therapeutic agents that modulate neurokinin receptors
12/16/1999CA2319068A1 Novel angiotensin receptor modulators and their uses
12/16/1999CA2318894A1 .beta.2-adrenergic receptor agonists
12/16/1999CA2318286A1 Multibinding agents that modulate ppar.gamma. and rxr receptors
12/16/1999CA2318055A1 .beta.2-adrenergic receptor agonists
12/15/1999EP0963982A2 New diaminobenzene derivatives and these componends containing colouring agents
12/15/1999EP0963975A1 Amines preparation process
12/15/1999EP0685457B1 Glycerol derivative, device and pharmaceutical composition
12/15/1999CN1238688A Thiol sulfonamide metalloprotease inhibitors
12/14/1999US6002002 Anti-ischaemic hydroxylamine derivatives and pharmaceutical compositions
12/14/1999US6001880 Disubstituted n-(2-dialkylaminoethyl)benzamide derivatives of given formula; antibacterial activity against helicobacter pyroli, administering for the prevention or cure of peptic ulcers
12/14/1999US6001877 Of given formula, which acts as an antagonist of leukotrienes; administering to treat leukotriene-b4 induced diseases, such as allergies and inflammation
12/14/1999US6001855 Thiazole derivatives
12/14/1999US6001347 Organic acid compound of given structure having an aromatic amide group, a methoxy group in the ortho position on the aromatic ring, and a lipophilic chain terminated with a carboxylic acid is useful as a nontoxic carrier
12/09/1999WO1999062962A1 Novel photoinitiators and applications therefor
12/09/1999WO1999062893A2 Novel neurokinin antagonists, method for the production thereof and pharmaceutical compositions containing said compounds
12/09/1999WO1999062873A1 Benzenesulphonamide derivatives as pyruvate dehydrogenase activators
12/09/1999WO1999062867A1 Indan derivatives
12/09/1999WO1999062520A1 Hiv integrase inhibitors
12/09/1999WO1999062506A1 Use of compounds for the elevation of pyruvate dehydrogenase activity
12/09/1999WO1999062505A2 Method for treating neurodegenerative disorders
12/09/1999WO1999043285A3 Sulphonamide derivatives
12/09/1999CA2334412A1 Indan derivatives
12/09/1999CA2333707A1 Hiv integrase inhibitors
12/09/1999CA2333689A1 New neurokinin antagonists, processes for preparing them and pharmaceutical compositions containing said compounds
12/09/1999CA2298468A1 Novel photoinitiators and applications therefor
12/08/1999EP0712387B1 2-aminoindans as selective dopamine d3 ligands
12/08/1999CN1237961A Aminoguanidines and alkoxyguanidines as protease inhibitors
12/08/1999CN1047196C Additive concentrate
12/08/1999CN1047195C 润滑油组合物 The lubricating oil composition
12/07/1999US5998615 Alzheimer's disease; nervous system disorders
12/07/1999US5998470 Osteoporosis; oral diseases; antiarthritic agents
12/07/1999US5998444 Antiasthma agents; neurokinin antagonist
12/07/1999US5998419 Bactericides
12/07/1999US5998414 Troponyl piperazines as dopamine D4 receptor ligands
12/07/1999US5998412 Sulfamide-metalloprotease inhibitors
12/07/1999US5998410 Sulfonamide derivatives
12/07/1999US5998401 Naphthyl compounds, intermediates, compositions, and methods
12/07/1999US5998399 Hypotensive agents
12/07/1999CA2013037C Aminobenzenesulfonic acid derivative