Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
08/1999
08/26/1999WO1999042445A1 Phtalimido arylpiperazines as alpha 1a receptor antagonists useful in the treatment of benign prostatic hyperplasia
08/26/1999WO1999042443A1 Sulfonylamino derivatives which inhibit matrix-degrading metalloproteinases
08/26/1999WO1999042436A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted-alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
08/26/1999WO1999042107A1 Piperazine derivatives for treating bone deficit conditions
08/26/1999WO1999029700A3 Cyclohexadiene-derivatives as pesticides
08/26/1999WO1998022435A9 Compounds useful for perhalogenoalkylation, reagent for implementing these compounds and synthesis method for obtaining these compounds
08/26/1999DE19844192A1 New substituted alkoxycarbonyl compounds
08/26/1999CA2321460A1 Substituted alxoxycarbonyl compounds
08/26/1999CA2320971A1 Cyclic amide compounds
08/26/1999CA2320469A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted-alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
08/26/1999CA2318836A1 Histamine h3 receptor ligands
08/26/1999CA2288178A1 Piperazine derivatives for treating bone deficit conditions
08/25/1999EP0937708A2 sulphonamide derivatives
08/25/1999EP0937696A1 Safety-catch linkers
08/25/1999EP0937065A1 Constrained somatostatin agonists and antagonists
08/25/1999EP0937064A1 Substituted oximes derivatives useful as neurokinin antagonists
08/25/1999EP0937054A1 4-(1-piperazinyl)benzoic acid derivatives, process for preparing them and their therapeutic applications
08/25/1999EP0937053A1 Sustained-release derivatives of hydroxylated analogs of substituted 1- 2 bis(aryl)methoxy]ethyl]-piperazines and -homopiperazines and their use as noncompetitive antagonists of dopamine reuptake
08/25/1999EP0937027A1 Alpha-branched fluoroalkylcarbonyl fluorides and their derivatives
08/25/1999EP0936909A1 Pharmaceutical composition for treating viral diseases
08/25/1999EP0805626B1 Crop protection products
08/25/1999CN1226892A Compounds and compositions for treating diseases associated with tryptase activity
08/25/1999CN1226886A Arylcycloalkane carboxylic esters, their use, pharmaceutical compositions and preparation
08/25/1999CN1226825A Use of amines to produce drugs for preventing tumour cell proliferation
08/24/1999US5942641 Fluorenone derivatives, process for preparing the same and central or peripheral nerve degeneration repair and protective agent
08/24/1999US5942544 Anticoagulants and treatment of thromboembolic disoeders
08/24/1999CA2166693C Difluoro statone analogs
08/19/1999WO1999041231A1 Amidino derivatives and drugs containing the same as the active ingredient
08/19/1999WO1999040919A1 Remedies for cardiac dilastolic disorders
08/19/1999WO1999029662A3 Urethanes, thio and dithio analogues, the salts thereof, medicaments containing said compounds, use and method for the production thereof
08/19/1999WO1999015894A3 Method of identification of leads or active compounds
08/19/1999WO1999001416A3 1-amino-alkylcyclohexane nmda receptor antagonists
08/18/1999EP0935597A2 Dihydropyrones with improved antiviral activity
08/18/1999EP0935486A1 Aqueous film-forming foam compositions
08/18/1999EP0620817B1 Piperazine derivatives as 5-ht receptors antagonists
08/18/1999CN1226230A Pesticidal composition
08/17/1999US5939587 N-protected/N-substituted-beta-amino hydroxy sulfonates
08/17/1999US5939563 Fungicides
08/17/1999US5939560 Inhibitors of DP-mediated processes, compositions and therapeutic methods thereof
08/17/1999US5939462 NPY5 receptor antagonists and methods for using same
08/17/1999US5939443 Selective β3 adrenergic agonists
08/17/1999US5939381 4-(4-(phenoxyacetyl)aminophenyl)butyric acid as a carrier for drug delivery
08/17/1999US5939332 Novel compounds optionally conjugated to reporter molecules aminofluorescein or aminomethylfluorescein capable of reacting with anti-phencyclidine(pcp) antibodies useful in immunoassays for selective detection of pcp in urine
08/17/1999CA2150610C Benzene derivatives and pharmaceutical composition
08/12/1999WO1999040083A2 Bifunctional tryptase inhibitors
08/12/1999WO1999040073A2 Tryptase inhibitors
08/12/1999WO1999039704A1 Antibacterial agents
08/12/1999DE19851299A1 Tryptase-Inhibitoren Tryptase inhibitors
08/12/1999CA2320476A1 Antibacterial agents
08/11/1999EP0934920A2 Preparation of hydrogenated compounds using noble metal Raney catalysts
08/11/1999EP0934316A1 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
08/11/1999EP0934312A1 1,4-disubstituted piperazines
08/11/1999EP0934302A2 Aminophenol derivates
08/11/1999EP0934293A1 Novel compounds and compositions for treating diseases associated with tryptase activity
08/11/1999EP0934292A1 Metalloproteinase inhibitors
08/11/1999EP0934291A1 Protease inhibitors
08/11/1999EP0934273A1 New derivates from piperidine-keto acid, their preparation and use
08/11/1999EP0934256A1 Process for the production of cyanocinnamamides
08/11/1999EP0934068A1 Compounds and methods
08/11/1999EP0933993A1 Substituted cyclopentane compounds useful as neuraminidase inhibitors
08/11/1999EP0666741B1 Dithiocarbamates for the treatment of atherosclerosis and other cardiovascular and inflammatory diseases
08/11/1999EP0642509B1 Novel potent inducers of terminal differentiation and methods of use thereof
08/11/1999CN1225624A Inhibition of matrix metalloproteases by substituted phenethyl compounds
08/11/1999CN1225621A Inhibition of matrix metalloproteases by substituted biaryl oxobutyric acids
08/11/1999CN1044604C Method for preparing high purity N-(2-sulfatoethyl) piperazin
08/11/1999CN1044603C N-(2-sulfatoethyl) piperazin-sulfate and method for preparing same
08/11/1999CN1044600C N-arylhydrazine derivatives as insecticidal and acaricidal agents
08/11/1999CA2260472A1 Safety-catch linkers
08/10/1999US5935997 O-thiocarbamoyl-aminoalkanol compounds, their pharmaceutically useful salts and process for preparing the same
08/10/1999US5935976 Viricides, hiv
08/10/1999US5935958 Muscarinic antagonists
08/05/1999WO1999038844A1 Method for preparing an n-[(aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound
08/05/1999WO1999038843A1 Hydroxamic and carboxylic acid derivatives
08/05/1999WO1999038515A1 Optic papillary circulation improving agents
08/05/1999CA2318601A1 Method for preparing an n-[(aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound
08/04/1999EP0933346A1 NOVEL p-TERPHENYL COMPOUNDS
08/04/1999EP0932657A2 Asymmetrical bleach activators and compositions employing the same
08/04/1999CN1225009A Pentafluorobenzenesulfonamides and analogs
08/04/1999CN1224714A N-(4-carbamimido-phenyl)-phenylglycinamid derivatives
08/04/1999CN1224712A 1,2-Di-substituted benzene-carboxamide derivative, hair growth promoter and external composition for skin using the same
08/03/1999US5932745 Process for converting propargylic amine-N-oxides to enaminones
08/03/1999US5932734 N-aminoalkylfluorenecarboxamides
08/03/1999US5932616 Potent inducers of terminal differentiation and methods of use thereof
08/03/1999US5932586 Prostaglandin synthase inhibitors
08/03/1999US5932582 Fibrinogen receptor antagonist prodrugs
08/03/1999US5932575 Cardiac diseases improving agents
08/03/1999US5932538 Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
07/1999
07/29/1999WO1999037623A2 Sulphonamide derivatives for treatment of cns disorders
07/29/1999WO1999037307A1 Pharmaceutically active compounds and methods of use thereof
07/29/1999WO1999037306A1 Pharmaceutically active compounds and methods of use thereof
07/29/1999WO1999023587A3 Method of virtual retrieval of analogs of lead compounds
07/29/1999DE19801597A1 1-Aryl-4-arylethyl-piperazine derivative preparation in high yield from aryl-piperazine and aryl olefin, used as drug intermediate
07/29/1999CA2318580A1 Pharmaceutically active compounds and methods of use thereof
07/29/1999CA2317740A1 Sulphonamide derivatives for treatment of cns disorders
07/28/1999EP0931067A1 D4 receptor selectivity piperazine derivatives
07/28/1999EP0766665B1 Metalloproteinase inhibitors
07/28/1999EP0737189B1 Heterocyclic compounds for the treatment of cns and cardiovascular disorders
07/28/1999CN1044365C Alpha, omega-diarylalkane derivs., their preparation and their use in treatment and prevention of circulatory diseases and psychosis
07/27/1999US5929281 Process for producing heterocyclic aromatic amine or arylamine
07/27/1999US5929266 Chiral organometallic compounds