Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
04/1999
04/29/1999WO1999020630A1 Photochromic compounds
04/28/1999EP0911350A1 Fabrication process for copolymers of controlled architecture via the use of functional radical initiators in a living radical polymerisation, and initiator compositions and corresponding copolymers
04/28/1999EP0911324A1 Process for the preparation of chiral succinic acid derivatives
04/28/1999EP0911320A2 1,2-Di-substituted benzenecarboxamide derivative, hair growth promoter and external composition for skin using the same
04/28/1999EP0911319A1 Malonic acid based matrix metalloproteinase inhibitors
04/28/1999EP0910565A1 Amide derivatives as selective neuropeptide y receptor antagonists
04/28/1999EP0910564A1 D-amino acid derived inhibitors of cysteine and serine proteases
04/28/1999EP0910415A1 Fluoro labelled anthracyclinone and anthracycline derivatives
04/28/1999EP0910370A1 Compositions comprising a nitrone compound for use in treating ocular inflammation
04/28/1999CN1215402A Compound containing nitroxyl
04/28/1999CN1215395A Novel substituted [2-(1-piperazinyl) ethoxy] methyl
04/28/1999CN1215393A Process to prepare oxazolidinones
04/28/1999CN1215054A Bychclic fibrinogen antagonists
04/22/1999WO1999019315A1 New process for producing aminopiperazine derivatives
04/22/1999WO1999019314A1 Process for preparing substituted pyrazine compounds
04/22/1999WO1999019301A1 Piperazine compounds and medicinal use thereof
04/22/1999WO1999019299A1 Heterocycles useful in the treatment of benign prostatic hyperplasia and intermediates thereof
04/22/1999WO1999019296A1 Aminobutanoic acid derivatives
04/22/1999WO1999019293A1 Novel aryloxy-alkyl-dialkylamines
04/22/1999WO1999018963A1 Use of flunarizine for the topical treatment of glaucoma
04/22/1999WO1999002146A8 Amino acid derivatives
04/22/1999CA2306811A1 Piperazine compounds and medicinal use thereof
04/22/1999CA2305770A1 Process for preparing substituted pyrazine compounds
04/22/1999CA2305353A1 Heterocycles useful in the treatment of benign prostatic hyperplasia and intermediates thereof
04/22/1999CA2304682A1 New process for producing aminopiperazine derivatives
04/21/1999EP0717731B1 Difluoro statone antiviral analogs
04/21/1999EP0712397B1 Amide derivatives as 5ht1d receptor antagonists
04/21/1999EP0695184B1 Hiv protease inhibitors
04/21/1999CN1214705A In Situ block copolymer formation during polymerization of vinyl axomatic monomer
04/21/1999CN1214677A Diphenyl stilbenes as prodrugs to cox-2 inhibitors
04/20/1999US5895816 Reactimg amines and aliphatic aldehydes on fixed bed catalyst, in presence of free pressurized hydrogen, by mixing reactants (only one of which has been preheated) in reactor, for use of comercially available aqueous formaldehyde solution
04/15/1999WO1999018066A1 Amidocarboxylic acid derivatives
04/15/1999WO1999017790A1 PEPTIDE-CONTAINING α-KETOAMIDE CYSTEINE AND SERINE PROTEASE INHIBITORS
04/15/1999DE19742951A1 Acylsulfamoylbenzoesäureamide, diese enthaltende nutzpflanzenschützende Mittel und Verfahren zu ihrer Herstellung Acylsulfamoylbenzamides, crop-protection agents containing them and methods for their preparation
04/15/1999CA2305808A1 Amidocarboxylic acid derivatives
04/15/1999CA2304116A1 Peptide-containing .alpha.-ketoamide cysteine and serine protease inhibitors
04/14/1999EP0907632A1 Inhibition of matrix metalloproteases by substituted phenethyl compounds
04/14/1999EP0810991B1 1-aryl-2-acylamino-ethane compounds and their use as neurokinin especially neurokinin 1 antagonists
04/14/1999CN1214047A Novel aromatic piperazines derived from substituted cycloazanes, method for prepairing same, pharmaceutical compsns, and use thereof as drugs
04/14/1999CN1214039A Carbamoyloxy derivatives of mutiline and their use as antibacterials
04/14/1999CN1213663A Process for manufacture of chiral succinic acid derivatives of formula
04/14/1999CN1213586A Hexanolactam hydrogenation for preparing hexamethylene radical imine catalyst and its application
04/14/1999CN1042933C Benzoylguanidine, prepn. of same and application as pharmaceutical and pharmaceutical containing same
04/08/1999WO1999016809A1 Specific fluorinated ethers as reaction medium
04/08/1999WO1999016807A1 Bis(alkylamino)alkylether compounds and the use thereof
04/08/1999WO1999016751A1 Benzamidine derivatives as factor xa inhibitors
04/08/1999WO1999016747A1 Sulfonyl derivatives
04/08/1999WO1999016746A1 Aminoalkylphenol derivatives and related compounds
04/08/1999WO1999016744A1 Acylsulfamoyl benzoic acid amides, plant protection agents containing said acylsulfamoyl benzoic acid amides, and method for producing the same
04/08/1999DE19743435A1 Benzamidinderivate Benzamidine derivatives
04/08/1999CA2305568A1 Benzamidinderivates
04/08/1999CA2304285A1 Sulfonyl derivatives
04/07/1999EP0906268A1 Alkyloxyamino substituted fluorenones and their use as protein kinase c inhibitors
04/07/1999EP0758317B1 N-sulphonyl and n-sulphinyl amino acid amides as microbiocides
04/07/1999EP0659181B1 Sulfonamide inhibitors of hiv-aspartyl protease
04/06/1999US5892125 Reacting 1,3-butadiene with an amine; isomerization
04/06/1999US5892052 Process for making retroviral protease inhibiting compounds
04/06/1999US5892038 Hydroxy-amino acid amides
04/06/1999US5892030 Process for producing 5,6-dihydro-1,3-oxazines
04/06/1999US5891890 Benzamide derivatives, anti-ulcer drug, and antibacterial drug
04/06/1999US5891881 Propane 1,2,3-substituted with one of each: ether or sulfide group; hydroxy group; and aminoheterocyclic group; wound healing promoter for mammals
04/06/1999US5891200 Dye in vehicle for dyeing hair
04/06/1999CA2024700C Benzoylguanidines, a process for their preaparation, their use as medicaments and medicaments containing them
04/06/1999CA1340479C Indane derivatives, process for preparing the same, new intermediates produced, use thereof as therapeutic agents and pharmaceutical compositions containing them
04/03/1999CA2247580A1 Process for preparing chiral succinic acid derivatives
04/01/1999WO1999015894A2 Method of identification of leads or active compounds
04/01/1999WO1999015493A1 9,10-dihydro-9,10-ethanoanthracene derivatives as phospholipase inhibitors
04/01/1999WO1999015164A1 Amide derivatives for the treatment of diseases mediated by cytokines
04/01/1999WO1998055153A9 Non-steroidal radiolabeled agonist/antagonist compounds and their use in prostate cancer imaging
04/01/1999WO1998052898A9 Pharmaceutical agents for the treatment of cerebral amyloidosis
04/01/1999DE19831803A1 N-aralkyl-hydrazino or -hydrazono derivatives of oxalic acid
04/01/1999DE19742720A1 Bis(alkylamino)alkylether-Verbindungen und ihre Verwendung Bis (alkylamino) alkylether compounds and their use
04/01/1999CA2304879A1 New tetracycles, process for their production and pharmaceutical preparations containing these compounds
04/01/1999CA2304783A1 Method of identification of leads or active compounds
04/01/1999CA2300051A1 Amide derivatives for the treatment of diseases mediated by cytokines
03/1999
03/31/1999EP0905512A1 Method of identification of leads or active compounds
03/31/1999EP0905122A2 Process for the preparation of amines
03/31/1999EP0904265A1 Preparation of bis(fluoroalkylenesulfonyl)imides and (fluoroalkylsulfonyl) (fluorosulfonyl)imides
03/31/1999EP0904262A1 Conformationally restricted aromatic inhibitors of microsomal triglyceride transfer protein and method
03/31/1999EP0733035B1 Tricyclic derivatives, pharmaceutical compositions containing them
03/31/1999EP0637298B1 Substituted cyclohexene-1,2-bicarboxylic acid derivatives and raw materials for producing them
03/31/1999CN1212690A Novel piperidines derived from 1-(piperazin-1-yl) aryl (oxylamino) carbonyl/4-aryl-piperidine as selective 5-HTiD beta receptor antagonist
03/31/1999CN1212689A Novel aryl glycinamide derivatives, method of producing said derivatives and pharmaceutical compositions containing these compounds
03/30/1999US5889042 Method of treating diseases and conditions with estrogen agonists and antagonists
03/30/1999US5889007 Chemisensitizing agents; cancer therapy drug resistance
03/30/1999US5889006 Muscarinic antagonists
03/30/1999US5889000 Naphthofluorene compounds, intermediates, compositions and methods
03/30/1999US5888992 Polar substituted hydrocarbons
03/30/1999US5888419 Granular N-alkyl ammonium acetontrile compositions
03/25/1999WO1999014207A1 Substituted indan derivatives
03/25/1999WO1999001427A3 Novel nitric oxide-releasing amidine- and enamine-derived diazeniumdiolates, compositions and uses thereof and method of making same
03/25/1999DE19742014A1 Use of new and known tetracyclene compounds as phospholipase inhibitors
03/25/1999CA2303839A1 Substituted indan derivatives
03/24/1999EP0903349A2 CCR-3 receptor antagonists
03/24/1999CN1211572A Cyclic amine derivatives-CCR-3 receptor antagonists
03/23/1999US5886226 Process for producing amines from olefins on zeolites of types SSZ-33, CIT-1 or mixtures thereof
03/23/1999US5886177 Phosphate linked oligomers
03/23/1999US5886175 Tetracycline antibiotics
03/23/1999US5886043 Antiarthritic agents, antitumor agents, antiinflammatory agents
03/23/1999US5886036 Treating hiv infections