| Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005) |
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| 07/04/2000 | US6083903 Boronic ester and acid compounds, synthesis and uses |
| 06/29/2000 | WO2000037444A1 Compounds useful in the treatment of inflammatory diseases |
| 06/29/2000 | WO2000037429A2 INHIBITORS OF α4β1 MEDIATED CELL ADHESION |
| 06/29/2000 | WO2000002887A3 Ligands for metals and metal-catalyzed processes |
| 06/29/2000 | WO1999064034A9 β2-ADRENERGIC RECEPTOR AGONISTS |
| 06/29/2000 | CA2355630A1 Compounds useful in the treatment of inflammatory diseases |
| 06/28/2000 | EP1012134A1 Quaternary ammonium phosphate compound and method of preparing the same |
| 06/28/2000 | EP1012131A1 Enantioselective reduction of ketones with a silane agent/metal compound/chiral ligand system |
| 06/28/2000 | CN1053895C Substd. sulfonic acid amide, preparation process and pharmaceutical composition of same |
| 06/28/2000 | CN1053886C Naphthyl compounds, intermediates and their preparing method and use |
| 06/27/2000 | US6080865 A polymerization catalysts in the production of polyurethanes; a reaction product of the 2-methylglutaronitrile with hydrogen |
| 06/27/2000 | US6080863 Activating a hydrogenation catalyst in the presence of hydrogen and under activation conditions including heating and pressurization |
| 06/27/2000 | US6080860 Urea compound where one of the urea nitrogens is part of an (un)substituted 5 or 6 membered ring and/or the other urea nitrogen is substituted with a 2-cyano-4,5-dialkoxyphenyl group; reacting with electrophile to form a leaving group |
| 06/27/2000 | CA2017193C N-(aryloxyalkyl)heteroarylpiperidines and-heteroarylpiperazines, a pro cess for their preparation and their use as medicaments |
| 06/22/2000 | WO2000035892A1 Piperazine ethylamide derivatives with 5-ht1a receptor activity |
| 06/22/2000 | WO2000035882A1 1,2,3,4-tetrahydronaphthalenes and their pharmaceutical use |
| 06/22/2000 | WO2000035879A1 3-phenyl-2,6-dioxopiperidin-3-yl propionamide derivatives and method for preparing same |
| 06/22/2000 | WO2000035864A1 New biphenyl and biphenyl-analogous compounds as integrin antagonists |
| 06/22/2000 | WO2000035860A2 Acyl isothiocyanate resins and their use in solid-supported synthesis of guanidines |
| 06/22/2000 | WO2000035859A1 Substituted aryl and heteroaryl derivatives, their production and their use as medicines |
| 06/22/2000 | WO2000035858A1 Phenylglycine derivatives |
| 06/22/2000 | WO2000035855A1 3,4-diamino-3-cyclobutene-1,2-dione derivatives which inhibit leukocyte adhesion mediated by vla-4 |
| 06/22/2000 | WO2000035442A1 Hydroxy diphenyl urea sulfonamides as il-8 receptor antagonists |
| 06/22/2000 | WO2000035436A2 Treatment of arthritis with mek inhibitors |
| 06/22/2000 | WO2000035435A1 Use of a mek inhibitor for preventing transplant rejection |
| 06/22/2000 | WO2000004954A3 Novel urokinase inhibitors |
| 06/22/2000 | CA2369115A1 3-phenyl-2,6-dioxopiperidin-3-yl propionamide derivatives and method for preparing same |
| 06/22/2000 | CA2355890A1 Hydroxy diphenyl urea sulfonamides as il-8 receptor antagonists |
| 06/22/2000 | CA2355161A1 Biphenyl and biphenyl-analogous compounds as integrin antagonists |
| 06/22/2000 | CA2353151A1 Substituted aryl and heteroaryl derivatives, the preparation thereof and their use as medicaments |
| 06/22/2000 | CA2351860A1 Piperazine ethylamide derivatives with 5-ht1a receptor activity |
| 06/22/2000 | CA2351464A1 3,4-diamino-3-cyclobutene-1,2-dione derivatives which inhibit leukocyte adhesion mediated by vla-4 |
| 06/22/2000 | CA2346684A1 Use of a mek inhibitor for preventing transplant rejection |
| 06/22/2000 | CA2346448A1 Treatment of arthritis with mek inhibitors |
| 06/21/2000 | EP1009737A2 Sulfonylamino substituted hydroxamic acid derivatives as metalloprotease inhibitors |
| 06/21/2000 | EP1009736A1 Malonic acid based matrix metalloproteinase inhibitors |
| 06/21/2000 | EP1009732A2 1-amino-alkylcyclohexane nmda receptor antagonists |
| 06/21/2000 | EP0638073B1 1-piperazino-1,2-dihydroindene derivatives |
| 06/21/2000 | CN1053666C Benzoheterocylic compounds and process for preparing medicated salt thereof |
| 06/21/2000 | CN1053657C Didepside phthaleins based internal parasite compositions, novel didepside phthaleins and preparation process thereof |
| 06/21/2000 | CN1053571C Application of proliferation in preparation of medicine for inhibiting smooth muscle cell and restinosis |
| 06/20/2000 | US6077698 Nonpolymeric compound including at least two aryl ketones and one or more sulfonate, phosphonate, and carboxylate groups; for surface treatments and immobilization in aqueous systems |
| 06/15/2000 | WO2000034268A1 Thiourea inhibitors of herpes viruses |
| 06/15/2000 | WO2000034238A1 Thiourea inhibitors of herpes viruses |
| 06/15/2000 | WO2000034237A2 Acetamide and substituted acetamide-containing thiourea inhibitors of herpes viruses |
| 06/15/2000 | WO2000034231A1 Molecular scaffolds acting as templates comprising carbamate linkages |
| 06/15/2000 | WO2000012454A9 Novel polycationic lipids |
| 06/15/2000 | WO2000006531A3 Nitric esters and nitrate salts of specific drugs |
| 06/15/2000 | CA2353462A1 Molecular scaffolds acting as templates comprising carbamate linkages |
| 06/15/2000 | CA2351403A1 Thiourea inhibitors of herpes viruses |
| 06/15/2000 | CA2350996A1 Thiourea inhibitors of herpes viruses |
| 06/15/2000 | CA2350899A1 Acetamide and substituted acetamide-containing thiourea inhibitors of herpes viruses |
| 06/14/2000 | EP1008592A2 Cyclic amide derivatives which inhibit cathepsin K |
| 06/14/2000 | EP1008346A1 NF-$g(k)B INHIBITORS CONTAINING AS THE ACTIVE INGREDIENT PHENYLMETHYL BENZOQUINONE |
| 06/14/2000 | EP1007033A1 Lymphocyte function antigen-1 antagonists |
| 06/14/2000 | EP0823892B1 Tetralines bearing a phenyl substituant on the aromatic ring and their use in the treatment of epilepsy, stroke and brain or spinal trauma |
| 06/14/2000 | EP0777645B1 Oxime ethers and their use as pesticides |
| 06/14/2000 | CN1256272A Preparation of N-formyl morpholine, N-formyl piperazine and their homologues |
| 06/14/2000 | CN1053441C Compound with 1-(aryl china olefine)-4-(aryl methyl) piperazine structure, its preparation process and medicine containing the compound thereof |
| 06/13/2000 | US6075146 Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceuticals |
| 06/13/2000 | US6075026 Certain substituted 1-aryl-3-piperazin-1'-yl propanones |
| 06/13/2000 | CA1341024C Benzo-fused cycloalkane and oxa- and thia-, cycloalkane trans-1, 2-diamine derivatives |
| 06/08/2000 | WO2000032583A1 Antitumor dibenzofluorene derivatives |
| 06/08/2000 | WO2000032582A1 Benzamide derivatives and their use as apob-100 secretion inhibitors |
| 06/08/2000 | WO2000032570A1 Hydrazine derivatives |
| 06/08/2000 | WO2000032569A2 Alpha-sulfin- and alpha-sulfonamino acid amides |
| 06/08/2000 | CA2353394A1 Benzamide derivatives and their use as apob-100 secretion inhibitors |
| 06/08/2000 | CA2352878A1 Antitumor dibenzofluorene derivatives |
| 06/08/2000 | CA2351321A1 Hydrazine derivatives |
| 06/07/2000 | EP1006153A1 Cationic amino-dianthraquinones, use thereof, dyeing compositions containing them and dyeing processes |
| 06/07/2000 | EP1005448A2 Novel inhibitors of aggrecanase and matrix metalloproteinases for the treatment of arthritis |
| 06/07/2000 | EP1005446A1 N-aroylphenylalanine derivatives |
| 06/07/2000 | EP1005445A1 N-alkanoylphenylalanine derivatives |
| 06/07/2000 | CN1255497A Method for preparing pyrazo [4,3-d] pyrimidine-7-one and its intermediate |
| 06/06/2000 | US6071970 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases |
| 06/06/2000 | US6071920 Bind to 5ht 1a receptors for treating disorders of the lower urinary tract; cns disorders; anxiolytic agents; antidepressants; hypotensive agents; sleep and eating disorders |
| 06/06/2000 | US6071915 Arylsubstituted piperazines useful in the treatment of benign prostatic hyperplasia |
| 06/06/2000 | US6071895 Polar-substituted hydrocarbons |
| 06/06/2000 | US6071510 Modified amino acids and compositions comprising the same for delivering active agents |
| 06/06/2000 | CA2015033C Tertiary alkyl functionalized piperazine derivatives |
| 06/02/2000 | WO2000031030A1 Bifunctional photoinitiators suitable for photopolymerization and photopolymerizable systems containing the same |
| 06/02/2000 | WO2000031021A1 β-AMYLOID PROTEIN PRODUCTION/SECRETION INHIBITORS |
| 06/02/2000 | WO2000030444A1 Cationic liposomes for gene transfer |
| 06/02/2000 | CA2351692A1 Inhibitors of production and/or secretion of amyloid-.beta. protein |
| 05/31/2000 | EP1004306A2 Estrogen agonists/antagonists |
| 05/31/2000 | EP1003728A1 2- 3- 4-(2-t-butyl-6- trifluoromethylpyridin-4-yl) piperazin-1-yl] propylmercapto pyrimidin-4-ol-fumarate |
| 05/31/2000 | EP1003714A1 Aromatic amides, their preparation process and their use as pesticides |
| 05/31/2000 | EP1003540A1 $g(b)2-ADRENERGIC RECEPTOR AGONISTS |
| 05/31/2000 | EP1003514A1 Cyclic amine modulators of chemokine receptor activity |
| 05/31/2000 | EP1003495A1 Pharmaceutical compounds |
| 05/31/2000 | EP1003373A1 Compositions and methods for reducing respiratory depression and attendant side effects of mu opioid compounds |
| 05/31/2000 | EP0882016B1 Alkylated styrenes as prodrugs to cox-2 inhibitors |
| 05/31/2000 | EP0633775B1 Compounds useful for treating inflammatory diseases and for inhibiting production of tumor necrosis factor |
| 05/31/2000 | CN1255119A Protease inhibitors |
| 05/31/2000 | CN1254596A Process for preparing composition to kill internal parasites |
| 05/31/2000 | CN1052977C Method for preparing moclobemide |
| 05/30/2000 | US6069247 Reacting an acetylenecarboxy amide and an aryl or heterocyclyl halide or a group enhancing the electrophilicity of the atom to which it is attached for displacement; using a palladium compound catalyst, a base and an acid |
| 05/30/2000 | US6069176 Phenylethanolamine compounds with a beta-3 adrenergic receptor stimulating effect, use as a therapy for urinary incontinence |
| 05/30/2000 | US6069175 Administering to a mammal in need a therapeutically effective amount of a member selected from the 4-hydroxy tamoxifen, raloxifene, toremifene, centchroman, idoxifene to treat atherosclerosis |
| 05/30/2000 | US6069143 Anticoagulants |