Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
09/2009
09/16/2009EP2099765A2 5, 6, or 7-substituted-3-(hetero)arylisoquinolinamine derivatives as antitumor agents
09/16/2009EP2099764A1 Preparation of substituted morphinan-6-ones and salts and intermediates thereof
09/16/2009EP2099745A2 Preparation of 3,4-dihydroisoquinolines from an acid and an amine
09/16/2009EP2099303A1 Therapeutic tetrahydroisoquinoline-based compositions for cancer therapy
09/16/2009EP1363629B1 Kappa opioid receptor ligands
09/16/2009CN100540537C Glutamine fructose-y-phosphate amidotransferase (GFAT) inhibitors
09/16/2009CN100540534C N-alkynyl-2- (substituted aryloxy) alkylthioamide derivatives as fungicides
09/11/2009WO2009109648A1 Process for preparing compounds containing a hydronaphtalene structure with an unsymmetrically substituted benzene ring
09/11/2009WO2009073545A3 Tetrahydro-isoquinoline ppat inhibitors as antibacterial agents
09/11/2009WO2009015067A3 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
09/11/2009CA2716664A1 Oxadiazoanthracene compounds for the treatment of diabetes
09/10/2009US20090227558 Amino-derivatives as novel inhibitors of histone deacetylase
09/09/2009EP2098511A1 Process for preparing compounds containing a hydronaphtalene structure with an unsymmetrically substituted benzene ring
09/09/2009EP1809284A4 Niacin receptor agonists, compositions containing such compounds and methods of treatment
09/09/2009EP1567477B1 Substituted amino phenylacetic acids, derivatives thereof, their preparation and their use as cyclooxygenase 2 (cox-2) inhibitors
09/09/2009CN101528703A 2-(1-oxo-1H-isoquinolin-2-yl) acetamide derivatives
09/09/2009CN100537534C Aryloxyalkylcarbamate-type derivatives, preparation method thereof and use of same in therapeutics
09/08/2009US7585976 chemical intermediate for Hemiasterlin, first isolated from the sponge Hemiasterella; anticarcinogenic agent for treatment of colon cancer, tumor; prevention of restenosis of blood vessels subject to traumas such as angioplasty and stenting
09/08/2009US7585885 Beta -secretase (BACE); Alzheimer's disease; 2-(R)-[2-(S)-Amino-3-(3,5-difluorophenyl)-1-(S)-hydroxypropyl]-pyrrolidine-1-carboxylic acid tert-butyl ester
09/08/2009US7585878 2-[(2,5-dimethylpyrrolidin-1-yl)methyl]-N-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)biphenyl-4-carboxamide; capsaicin receptor VR1 inhibitory activity; inflammatory pain and neurogenic pain, migraine, cluster headache, bladder diseases including overactive bladder
09/08/2009US7585574 Pyrene derivative and organic electroluminescence device making use of the same
09/08/2009CA2287558C Heterocyclic derivatives and their use as antithrombotic agents
09/08/2009CA2213466C Inhibitors of microsomal triglyceride transfer protein and method
09/03/2009WO2009106547A1 Process for the resolution of isoquinoline derivatives
09/03/2009US20090221829 3,4-Dihydroisoquinolinium Salt Derivatives
09/03/2009US20090221633 Inhibitors of akt (protein kinase b)
09/03/2009US20090221575 Sulfonamide derivatives and use thereof for the modulation of metalloproteinases
09/03/2009US20090220454 Use of the histone deacetylase inhibitor N-hydroxy-4-[2-(3-dimethylaminobenzofuran-2-ylcarbonylamino)ethoxy]benzamide (aka CRA-24781, PCI-24781) for treating myelogenous leukemia (MML) or acute myelogenous leukemia (AML), optionally in combination therapy
09/03/2009CA2708666A1 Process for the resolution of isoquinoline derivatives
09/02/2009EP2096104A1 Organic diamines as mGluR7 modulators
09/02/2009EP1899322B1 Isoquinoline derivatives as inhibitors of rho-kinase
09/02/2009CN101522633A 6-substituted isoquinoline derivatives as ROCK-I inhibitors
09/02/2009CN101522632A Process for the preparation of substituted-1,2,3,4-tetrahydroisoquinoline derivates
09/02/2009CN100534986C Method for preparing derivative of 1,4 - dichloro isoquinoline category
09/01/2009US7582657 Vanilloid receptor ligands and their use in treatments
08/2009
08/27/2009WO2009105206A1 Modulators of the histamine h3 receptor useful for the treatment of disorders related thereto
08/27/2009US20090215764 Antimicrobial agents
08/27/2009CA2714122A1 Modulators of the histamine h3 receptor useful for the treatment of disorders related thereto
08/26/2009EP2091929A1 Agents that disrupt cellular replication and their use in inhibiting pathological conditions
08/26/2009EP1773817B1 Substituted aryl-amine derivatives and methods of use
08/26/2009EP1590338B1 Modulators of melanocortin receptor
08/26/2009EP1501804B1 Isoquinoline derivatives mao-b inhibitors
08/26/2009CN101516854A Preparation of substituted morphinan-6-ones and salts and intermediates thereof
08/26/2009CN101516839A Compounds which modulate the cb2 receptor
08/26/2009CN101516834A Isoserine derivatives for use as coagulation factor ixa inhibitors
08/26/2009CN101516833A Tartrate derivatives for use as coagulation factor IXa inhibitors
08/26/2009CN100532362C Process for preparing N-methyl quinoline compounds by ester reaction solvent
08/25/2009US7579469 For therapy of disease characterized by inflammatory, allergic, or proliferative processes
08/25/2009US7579347 Vanilloid receptor ligands and their use in treatments
08/20/2009WO2009083899A3 Process for the preparation of an enantiomeric trisubstituted 3,4-dihydro-isoquinoline derivative
08/20/2009WO2009074733A3 Addition salts of angiotensine-converting enzyme inhibitors with no donor acids, method for preparing same and pharmaceutical compositions containing same
08/20/2009US20090209765 Process for production of 4-fluoroisoquinoline-5-sulfonyl halide or salt thereof
08/20/2009US20090209562 Fused ring 4-oxopyrimidine derivative
08/20/2009US20090209528 Substituted tetrahydroisoquinoline compound, their preparation and use in medicaments
08/20/2009US20090206326 Electroluminescent iridium compounds with fluorinated phenylpryidines, phenylpyrimidines, and phenylquinolines and devices made with such compounds
08/19/2009EP2090566A2 Certain phenylacetic acids and derivatives
08/19/2009EP2089417A2 Methods, compounds, compositions and vehicles for delivering 3-amino-1-propanesulfonic acid
08/19/2009EP1999113B1 Substituted 1-amino-4-phenyl-dihydroisoquinolines, method for the production thereof, use thereof as a medicament, and medicaments containing them
08/19/2009CN100528879C S type 4-substituted hydroxy-pyranindolelidinyl compounds and its derivatives and production method
08/18/2009US7576245 Using a fluorinated phenyl compound containing electrophilic and nucleophilic groups; increasing the fluorous nature of an organic compound; 4-(1H,1H,2H,2H-Perfluorodecyl)benzenesulfonamide; N-[4-(1H,1H,2H,2H-perfluorodecyl)benzyloxycarbonyloxy]succinimide
08/18/2009US7575816 Ln( beta -enolate)3(mono-imine) where in mono-imine is selected from 3-cyanopyridine; 2-dimethylaminopyridine; isoquinoline; 4-tertbutyl-pyridine; 4-phenylpyridine; and 2-(2-thienyl)pyridine, Ln is selected from Eu, Tb and Tm; beta -enolate such as 2,4-pentanedionate
08/13/2009WO2009019534A3 Methods, compounds, compositions and vehicles for delivering 3-amino-1-propanesulfonic acid
08/12/2009EP1624868B9 "(2-hydroxy-2-(4-hydroxy-3-hydoxymethylphenyl)-ethylamino)- propyl]phenyl derivatives as beta2 agonists
08/12/2009CN101506171A Isoquinoline derivatives and their use as inhibitors of cytokine mediated diseases
08/12/2009CN101506168A Positively charged water-soluble prodrugs of n-arylanthranilic acids with very fast skin penetration rate
08/12/2009CN101503391A 1,2-dihydroisoquinoline derivative and preparation thereof
08/12/2009CN100526277C Method for the treatment or prevention of lower urinary tract symptoms
08/11/2009US7572913 Inhibitors of Rho kinase; N-Benzyloxycarbonyl-4-[N''-(tert-butyloxycarbonyl)hydrazino]piperidine; 4-{[N''-(tert-butyloxycarbonyl)-N'-(1'-propyl)]hydrazino}piperidine
08/11/2009US7572817 Carboxypeptidase U inhibitors; thrombosis, atherosclerosis, adhesions, dermal scarring, cancer, fibrotic conditions, inflammatory diseases; e.g. 2-[(6-Aminopyridin-3-yl)methyl]-3-mercapto-5-[3-(pyrrolidin-1-ylcarbonyl)phenyl]pentanoic acid
08/11/2009US7572787 Substituted naphthalene sulfonamides
08/11/2009US7572783 Obesity; N-(1-benzyl-piperidin-4-yl)-2-(2,5-dioxo-7-phenoxy-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl)-3-methyl-butyramide; modulators of ghrelin receptor (GHSR)
08/11/2009CA2449402C Substituted tetrahydroisoquinolines for use in the treatment of inflammatory diseases
08/06/2009WO2009097433A1 Novel dyes and use thereof in imaging members and methods
08/06/2009WO2009096526A1 Carboxylic acid compound or salt thereof
08/06/2009WO2008103354A3 Modulators of acetyl-coenzyme a carboxylase and methods of use thereof
08/05/2009EP1357111B1 2-pyridone derivatives having affinity for cannabinoid type 2 receptor
08/05/2009EP1249233B9 Npyy5 antagonists
08/05/2009CN101501001A Processes for optical resolution of 1-phenyl-1,2,3,4-tetrahydroisoquinoline
08/05/2009CN101500997A PARP inhibitors
08/05/2009CN101497584A Isoquinoline-3-formyl amino acid formyl amino acid benzyl ester, as well as preparation and use thereof
08/05/2009CN100522946C Stabilization of hypoxia inducible factor (HIF) alpha
08/04/2009US7569678 Protease inhibitor conjugates and antibodies useful in immunoassay
07/2009
07/30/2009US20090192188 Tetrahydroisoquinoline derivatives
07/29/2009EP2081905A2 Sulfonyl compounds which modulate the cb2 receptor
07/29/2009CN100519527C Inhibitors of histone deacetylase
07/28/2009US7566726 3-Trifluoromethyl,6-((3-(methyl,4-hydroxytetrahydropyran-4-yl)-amino-(3-isopropyl-cyclopent-1,3-ylene))-carbonyl-)-5,6,7,8-tetrahydro-1,6-naphthyridine; antiinflammatory agents; immunomodulators; antiallergens; rhintis; dermatitis; conjunctivits, asthma; autoimmune diseases; antiarthritis agents
07/23/2009WO2009091898A2 6-and 7-amino isoquinoline compounds and methods for making and using the same
07/23/2009WO2008076427A3 Naphthalenone compounds exhibiting prolyl hydroxylase inhibitory activity, compositions, and uses thereof
07/23/2009US20090186917 6-And 7-amino isoquinoline compounds and methods for making and using the same
07/23/2009CA2712443A1 6- and 7-amino isoquinoline compounds and methods for making and using the same
07/22/2009CN101490007A VR1 vanilloid receptor antagonists with a iononic substructure
07/22/2009CN101490006A Biarylcarboxyarylamides as vanilloid-1 receptor modulators
07/16/2009WO2009089083A1 Trpa1 antagonists
07/16/2009WO2009088990A1 Certain chemical entities, compositions and methods
07/16/2009WO2009088986A1 Certain chemical entities, compositions and methods
07/16/2009WO2009087649A1 Renin inhibitors
07/16/2009CA2711558A1 Certain chemical entities, compositions and methods
07/16/2009CA2711446A1 Certain chemical entities, compositions and methods
07/16/2009CA2711159A1 Trpa1 antagonists
07/14/2009US7560463 Diaryl ethers as opioid receptor antagonists
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