| Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865) |
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| 02/11/2010 | US20100035923 Vr1 vanilloid receptor antagonists with a iononic substructure |
| 02/10/2010 | EP2150534A1 Isoquinolinone derivatives as nk3 antagonists |
| 02/09/2010 | US7659402 use as pain relievers, gastrointestinal disorders; 2-Amino-3-aryl-1-[3-((hetero)aryl)piperidin-1-yl]-propan-1-one compounds |
| 02/09/2010 | US7659400 Radiolabelled benzamide analogues, their synthesis and use in diagnostic imaging |
| 02/09/2010 | US7659297 improved selectivity and pharmacokinetic properties; 6-Fluoro-1-[(1 H-indazol-4-yl)amino]-4,4-dimethyl-2-(trifluoromethyl)-1,2,3,4-tetrahydronaphthalene-2,5-diol; cyclization of imines |
| 02/09/2010 | CA2268403C Anthranilic acid derivatives as multi drug resistance modulators |
| 02/04/2010 | US20100029658 Heterocyclic derivatives, pharmaceutical compositions and methods of use thereof |
| 02/04/2010 | US20100028936 Detection of cancer cells in vitro using sigma-2 receptor ligands as radiotracers |
| 02/04/2010 | US20100028807 Imide Compound and Chemically Amplified Resist Composition Containing The Same |
| 02/03/2010 | EP2149561A1 Tetrahydroisoquinolin-1-one derivative or salt thereof |
| 02/03/2010 | EP2149560A1 1-substituted tetrahydroisoquinoline compound |
| 02/03/2010 | EP2149559A1 A process for the preparation of hexahydroisoquinolines from 1,2,3,4-Tetrahydroisoquinolines |
| 02/03/2010 | CN101638387A A process for the preparation of hexahydroisoquinolines from 1, 2, 3, 4-tetrahydroisoquinolines |
| 02/03/2010 | CN101638386A Improved preparation of 3, 4-dihydroisoquinolines from an acid and an amine |
| 02/03/2010 | CN100586927C Amide derivatives and their use as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
| 02/02/2010 | CA2442478C Use of group i mglur antagonists in the treatment of fragile x syndrome, autism, mental retardation |
| 01/28/2010 | WO2010011853A2 Beta-and gamma-amino-isoquinoline amide compounds and substituted benzamide compounds |
| 01/28/2010 | WO2010010174A1 1,1'-diadamantyl carboxylic acids, medicaments containing such compounds and their use |
| 01/28/2010 | WO2009124962A3 Sulfonamides |
| 01/28/2010 | US20100022776 Preparation of Hexahydroisoquinolines from Dihydroisoquinolines |
| 01/28/2010 | US20100022775 Process for the preparation of rho-kinase inhibitor compounds |
| 01/28/2010 | US20100022582 Tetrahydroisoquinoline Compound and Medicinal Use Thereof |
| 01/28/2010 | US20100022514 Heterocycle Compounds and Methods of Use Thereof |
| 01/28/2010 | US20100022486 Compounds |
| 01/28/2010 | CA2731869A1 Beta-and gamma-amino-isoquinoline amide compounds and substituted benzamide compounds |
| 01/28/2010 | CA2730208A1 1,1'-diadamantyl carboxylic acids, medicaments containing such compounds and their use |
| 01/26/2010 | US7652141 Immunosuppressants, analgesics, antiinflammatory agents |
| 01/26/2010 | US7652020 novel hydantoin derivatives to inhibit matrix metalloproteinases (MMPs), a disintegrin and metalloproteases (ADAMs) and/or tumor necrosis factor alpha converting enzyme (TACE) and in so doing prevent the release of tumor necrosis factor alpha (TNF- alpha ); autoimmune diseases; side effect reduction |
| 01/26/2010 | CA2481012C Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors |
| 01/21/2010 | US20100016596 Process for the purification of neuromuscular blocking agents |
| 01/21/2010 | US20100016309 1,2,3,4-Tetrahydroisoquinoline Derivatives, Preparation Process therefor and Pharmaceutical Composition Containing the Same |
| 01/20/2010 | EP2144881A1 Isoquinolinone derivatives, processes for their preparation and their use in the treatment of chronic obstructive pulmonary disease ( copd ) and asthma |
| 01/20/2010 | CN100581543C Tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents |
| 01/19/2010 | US7649085 Saquinavir conjugates and antibodies useful in immunoassay |
| 01/19/2010 | CA2402751C Decahydro-isoquinolines |
| 01/14/2010 | WO2010005087A1 Amidine derivative |
| 01/14/2010 | WO2009121872A3 Tetrahydroisoquinolines, pharmaceutical compositions containing them, and their use in therapy |
| 01/14/2010 | US20100010226 Trisubstituted 3,4-dihydro-1h-isoquinolin compound, process for its preparation, and its use |
| 01/14/2010 | US20100010004 Inhibitors of histone deacetylase |
| 01/14/2010 | US20100009988 Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase |
| 01/14/2010 | US20100009960 Pyridone/hydroxypyridine 11-beta hydroxysteroid dehydrogenase type i inhibitors |
| 01/13/2010 | EP2143714A1 Tetrahydroisoquinoline compound |
| 01/13/2010 | EP2142510A1 Novel isoquinolinium compounds useful in the preparation of cisatracurium and associated intermediates |
| 01/13/2010 | EP2035385B1 Inhibitors of akt (protein kinase b) |
| 01/13/2010 | EP1910298B1 Phenylglycinamide and pyridylglycinamide derivatives useful as anticoagulants |
| 01/12/2010 | US7645757 Derivatives of heteroaryl-alkylcarbamates, methods for their preparation and use thereof as fatty acid amido hydrolase enzyme inhibitors |
| 01/12/2010 | CA2387675C Novel hydronaphtalene compounds, prepared by a rhodium catalyzed ring opening reaction in the presence of phosphine ligand |
| 01/07/2010 | US20100004241 Non-imidazole aryloxyalkylamines |
| 01/07/2010 | US20100004222 Amide Derivatives as Ion-Channel Ligands and Pharmaceutical Compositions and Methods of Using the Same |
| 01/06/2010 | CN101619038A Isoquinoline compound or salt thereof, medicinal composition, preparation method and application thereof |
| 01/05/2010 | CA2465723C Process for reacting alkaloids and use of the reaction products in the preparation of medicaments |
| 12/31/2009 | US20090325962 Tyrosine derivative |
| 12/31/2009 | US20090325228 Fungal cell wall synthesis gene |
| 12/30/2009 | WO2009156100A1 Substituted isoquinolines and isoquinolinones as rho kinase inhibitors |
| 12/30/2009 | WO2009156099A1 6-substituted isoquinolines and isoquinolinones |
| 12/30/2009 | WO2009156092A2 Bi- and polycyclic substituted isoquinoline and isoquinolinone derivatives |
| 12/30/2009 | EP2138482A1 Bicyclic heterocyclic compound |
| 12/30/2009 | CN100575345C Pyridone derivative having affinity for cannabinoid 2-type receptor |
| 12/30/2009 | CA2728137A1 Substituted isoquinolines and isoquinolinones as rho kinase inhibitors |
| 12/30/2009 | CA2728128A1 6-substituted isoquinolines and isoquinolinones |
| 12/30/2009 | CA2728123A1 Bi- and polycyclic substituted isoquinoline and isoquinolinone derivatives |
| 12/29/2009 | US7638635 Using alkylmetal reagents for directed metalation of azaaromatics |
| 12/29/2009 | US7638513 inhibitors of matrix metalloproteinases, aggrecanases, tumor necrosis factor-alpha converting enzyme, and tumor necrosis factors |
| 12/29/2009 | CA2370250C Di-aryl acid derivatives as ppar receptor ligands |
| 12/29/2009 | CA2348993C Substituted phenethylsulfones and method of reducing tnf.alpha. levels |
| 12/24/2009 | US20090318423 Ion Channel Modulators & Uses Thereof |
| 12/24/2009 | US20090314990 Novel triphenylamine derivatives useful as fluorophores in biology, in particular for two-photon microscopy |
| 12/23/2009 | EP2134693A2 Metalloprotease inhibitors containing a heterocyclic moiety |
| 12/23/2009 | CN101611012A Cycloalkylamine substituted isoquinoline derivatives |
| 12/23/2009 | CN101607938A Novel isoquinoline anti-tumor compound and preparation method thereof |
| 12/23/2009 | CN100572360C Isoquinoline compound and its salt preparation method and application |
| 12/22/2009 | US7635703 as tyrosine, serine/threonine, cyclin-dependent kinases, HER protein; 5-{2-[3-[4-trifluoromethyl-1-(2-trimethylsilanyl-ethoxymethyl)-1H-imidazol-2-yl]-1-(2-trimethylsilanyl-ethoxymethyl)-1H-pyrazol-4-yl]-vinyl}-pyridine-3-carbaldehyde; antiproliferative, antiinflammatory agent, neurodegenerative diseases |
| 12/22/2009 | CA2346563C Novel 2-[3-phenyl-2-propenyl]-1,2,3,4-tetrahydroxyisoquinoline derivatives, preparation method and use as fungicides |
| 12/22/2009 | CA2330976C Preparation of fused polycyclic alkaloids by ring closure of azomethine ylides, novel compounds thereof and their use as chemotherapeutic agents |
| 12/17/2009 | US20090312324 Compositions and Methods Related to RAD51 Inactivation in the Treatment of Neoplastic Diseases, and Especially CML |
| 12/16/2009 | EP2132181A1 (1r,1'r)-atracurium salts separation process |
| 12/16/2009 | CN101602725A Hexahydroisoquinoline-1-keto compound and synthetic method thereof |
| 12/15/2009 | US7632850 2-amino-2-oxoethyl 1-(4'-fluoro-1,1'-biphenyl-4-yl)cyclopropylmethylcarbamate and 2-(methylamino)-2-oxoethyl 1-(4'-fluoro-1,1'-biphenyl-4-yl)cyclopropylmethylcarbamate; fatty acid amide (FAAH) hyrdrolase inhibitors; analgesics; neuropathic pain;psychological disorders; anticarcinogenic agents; AIDS |
| 12/15/2009 | CA2393437C Exo-s-mecamylamine formulation and use in treatment |
| 12/10/2009 | US20090306390 Chiral ligands, their preparation and uses thereof in asymmetric reactions |
| 12/10/2009 | US20090306130 Novel tetrahydro-isoquinolines |
| 12/10/2009 | US20090306079 3,4-di-substituted cyclobutene-1,2-diones as cxc-chemokine receptor ligands |
| 12/09/2009 | EP2130820A1 Antipruritics |
| 12/09/2009 | EP2130534A1 Use of ritonavir for improving the pharmacokinetics of drugs metabolized by cytochrome P450 |
| 12/09/2009 | CN101600730A Methods, compounds, compositions and vehicles for delivering 3-amino-1-propanesulfonic acid |
| 12/09/2009 | CN101600698A Quinazolinone and isoquinolinone acetamide derivatives |
| 12/09/2009 | CN101597259A Organic material and application thereof in organic electroluminescence device (OELD) |
| 12/09/2009 | CN100567268C Process for synthesis of amine ethers from secondary amino oxides |
| 12/08/2009 | US7629358 For therapy of inflammatory, allergic and respiratory diseases |
| 12/08/2009 | US7629357 Antihypoxic agents; adjust concentration of erythropoietin concentration in blood; strokes; antiepileptic agents; neurodegenerative disease ; liver disorders; antiischemic agents |
| 12/08/2009 | CA2388475C Preparation of chiral 1,2,3,4-tetrahydro-6,7-dialkoxy-3-isoquinolinecarboxylic acid and derivatives |
| 12/03/2009 | US20090298825 Bicycloheteroaryl Compounds as P2x7 Modulators and Uses Thereof |
| 12/02/2009 | EP2125745A1 Cycloalkylamine substituted isoquinolone derivatives |
| 12/02/2009 | EP2125744A1 Cycloalkylamine substituted isoquinolone and isoquinolinone derivatives |
| 12/02/2009 | EP2125743A1 (1r,1'r)-atracurium salts separation process |
| 12/02/2009 | EP2125742A2 (1r,1'r)-atracurium salts separation process |
| 12/02/2009 | EP2124562A1 Bicycloheteroaryl compounds as p2x7 modulators and uses thereof |
| 12/02/2009 | EP1965805B1 Urea derivatives useful as calcium receptor modulators |
| 12/02/2009 | EP1812399B1 Opiate intermediates and methods of synthesis |
| 12/02/2009 | CN101595094A Cycloalkylamine substituted isoquinolone derivatives |