Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
10/2002
10/10/2002CA2442328A1 Therapeutic combinations for cardiovascular and inflammatory indications
10/10/2002CA2440164A1 Preparation of ketones from aldehydes
10/09/2002EP1246621A1 Nitrosated and nitrosylated cyclooxygenase-2 inhibitors, compositions and methods of use
10/09/2002CN1373754A Antibacterial agents
10/09/2002CN1373126A Crystallization formed N-(4-trifluoromethylphenyl)-5-methyl isooxazo-4-carboxamide
10/09/2002CN1092189C Substd. isoxazolines, process for producing them, agent contg. them and their use as safeners
10/09/2002CN1092181C Benzyloxy substd, aromatics and their use as fungicides and insecticides
10/08/2002USRE37873 Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
10/08/2002US6462076 Beta-amino acid nitrile derivatives as cathepsin K inhibitors
10/08/2002US6462043 Method for producing substituted-2-nitroguanidine derivatives
10/03/2002WO2002076929A1 Aryl and biaryl compounds having mch modulatory activity
10/03/2002US20020143024 As antihypertensive agents; for therapy of disorders related to renal, glomerular and mesangial cell function; therapy of endotoxemia or endotoxin shock as well as hemorrhagic shock; useful in alleviation of pain associated cancer
10/03/2002US20020143020 Novel piperazine derivatives
10/03/2002US20020142045 Cyclooxygenase-2 inhibitor compositions having rapid onset of therapeutic effect
10/03/2002US20020142000 Genetic engineering
10/01/2002US6458960 Sulfonamide derivatives
10/01/2002US6458805 Antagonists; especially sodium salts
10/01/2002CA2241845C 4,5-dihydronaphth¬1,2-c|isoxazoles and derivatives thereof having cns activity
10/01/2002CA2203850C Novel n-phenyl-n-phenyliminonethylbenzamidines and their analogues as muscarinic receptor agonists
09/2002
09/27/2002CA2378876A1 Cyclohexylamine derivatives as subtype selective n-methyl-d-aspartate antagonists
09/26/2002WO2002032872A8 Nitrogenous aromatic ring compounds
09/26/2002WO2001087343A3 Combination therapy using cox-2 selective inhibitor and thromboxane inhibitor and compositions therefor
09/26/2002US20020137968 Treating with amides, ureas, amidines, carbamates, carboximidamides and other derivatives of given formula, e.g. (+)-N-((2,2-dimethylcyclopentyl)methyl)-4-hexyloxybenzamide
09/25/2002EP1242427A1 Novel piperidine and piperazine derivatives
09/25/2002EP1242416A1 Substituted isoxazolines and their use as antibacterial agents
09/25/2002EP1242412A2 3-(4,5-dihydroisoxazol-3-yl)-substituted benzoylpyrazoles
09/25/2002EP1242395A1 Benzoic acid esters of oxazolidinones having a hydroxyacetylpiperazine substituent
09/25/2002EP1242394A1 Novel 3-oxo-2,1-benzisoxazol-1(3h)-carboxamides for treatment of cns diseases
09/25/2002EP1242393A1 Herbicidal 3-(4,5-dihydroisoxazole-3-yl)-substituted benzoylcyclohexenone derivatives
09/25/2002EP1242077A1 Novel processes for making- and a new crystalline form of- leflunomide
09/25/2002EP0968179B1 N-sulphonyl and n-sulphinyl amino acid amides as microbiocides
09/25/2002CN1371286A Use of cyclooxygenase-2 inhibitor matrix metallappoteinase inhibitor antineoplastic agent and optionally radiation as combination treatment of neoplasia
09/24/2002US6455550 N-alkanoylphenylalanine derivatives
09/24/2002US6455520 Benzamide derivatives and their use as cytokine inhibitors
09/19/2002WO2002072559A1 Process to intermediates for biologically active compounds
09/19/2002WO2002072527A2 1-butyric acid derivatives such as carbomethoxypropionyl cyanide or leflunomide derivatives, and the therapeutic use thereof
09/19/2002WO2002071827A2 Retinoid x receptor modulators
09/19/2002US20020133020 Efficient synthetic routes for the preparation of rhinovirus protease inhibitors and key intermediates
09/19/2002US20020132838 Methods for the preparation of biphenyl isoxazole sulfonamides
09/19/2002DE10109204A1 Use of new and known diphenylurea compounds for the preparation of a medicament for the inhibition of intracellular protein-degradation pathway
09/19/2002CA2441088A1 1-butyric acid derivatives such as carbomethoxypropionyl cyanide or leflunomide derivatives, and the therapeutic use thereof
09/19/2002CA2438586A1 Retinoid x receptor modulators
09/18/2002EP1240163A1 3-(4,5-dihydroisoxazole-5-yl)benzoylpyrazole
09/18/2002EP0917528B1 New amidino derivatives and their use as thrombin inhibitors
09/17/2002US6452011 Process for production of piperidine derivatives
09/17/2002US6451842 Cyclic amine derivatives and their use as drugs
09/17/2002US6451829 Coumarinic compounds having IgE affecting properties
09/17/2002CA2007332C Use of a glycine b partial agonist as an antipsychotic
09/12/2002WO2002070541A2 Peptide deformylase inhibitors
09/12/2002WO2002070495A1 Process for the preparation of 1,2-benzisoxazole-3-acetic acid
09/12/2002WO2002070467A1 Derivatives of diphenylurea, diphenyloxalic acid diamide and diphenylsulfuric acid diamide and their use as medicaments
09/12/2002WO2002069901A2 Cathepsin cysteine protease inhibitors
09/12/2002US20020128267 Especially celecoxib, deracoxib, valdecoxib, a benzopyran COX-2 inhibitor, parecoxib, rofecoxib etoricoxib, or a 2-(3,5-difluorophenyl)-3-(4-(methylsulfonyl)phenyl) -substituted cyclopentenone, or pyridazinone
09/12/2002US20020128255 Substituted hydroxyl amine derivatives; inhibitors of beta-secretase, inhibit beta-secretase-mediated cleavage, inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques
09/12/2002CA2440030A1 Process for the preparation of 1,2-benzisoxazole-3-acetic acid
09/12/2002CA2439827A1 Peptide deformylase inhibitors
09/11/2002EP1237888A2 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
09/11/2002EP1237881A1 Herbicidal halogenalkyl-substituted 3-(4,5-dihydroisoxazol-3-yl)-benzoyl-cyclohexenones
09/11/2002EP1237852A1 N-phenylcarbamates having a microbicide, insecticide and acaricide effect
09/11/2002CN1368965A Isoxazoline derivatives and herbicides containing same as active ingredient
09/10/2002US6448443 Synthesis of combinatorial libraries of compounds reminiscent of natural products
09/10/2002US6448406 Improved process for preparation of terfenadine carboxylic acid metabolite and carebastine derivatives; histamine h1 receptor blocking and calcium antagonists; respiratory, allergic, and cardiovascular disease states
09/10/2002US6448201 Benzoylcyclohexanediones and benzoylpyrazoles, their preparation, and their use as herbicides and plant growth regulators
09/10/2002CA2240946C Isoxazoline, isothiazoline and pyrazoline factor xa inhibitors
09/10/2002CA2195129C Substituted piperidine intermediates for producing heterocyclic-cyclic amine derivatives capable of inhibiting cholinesterase
09/05/2002DE10109856A1 Use of N-phenyl arylamide for treating or preventing chronic or acute hepatitis B viral infections in humans or animals, including co-infections with hepatitis D virus
09/04/2002EP1235816A1 Benzoylcyclohexandione and benzoylpyrazols, method for the production and use thereof as herbicides and plant growth regulators
09/04/2002EP0809636B1 Substituted isoxazoles for the treatment of inflammation
09/04/2002CN1367776A Process for preparing substituted cyclopentane derivatives and novel crystalline structures
09/04/2002CN1367730A Homogenization enhancing thermoplastic foam extrusion screw
09/03/2002US6444827 From beta-methyl l-aspartate via chemical intermediate; efficiency; antidiabetic agents
08/2002
08/29/2002WO2002066484A1 Isoxazoline derivatives as anti-depressants
08/29/2002WO2002066446A1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands
08/29/2002WO2002066431A1 Substituted heterocyclo-norbornylamine derivatives, method for producing the same, their use as medicament or diagnostic agent and medicament containing the same
08/29/2002WO2002042273A3 Acid derivatives useful as serine protease inhibitors
08/29/2002WO2001087845A3 N-containing heterocyclic compounds and their use as 5-ht antagonists
08/29/2002WO2000066104A9 Ace-2 inhibiting compounds and methods of use thereof
08/29/2002US20020120007 Benzamide inhibitors of factor Xa
08/29/2002US20020119983 Novel isoxazolylalkylpiperazine derivatives having selective biological activity at dopamine D3 or D4 receptor, and preparation thereof
08/29/2002CA2438264A1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands
08/29/2002CA2432208A1 Substituted heterocyclo-norbornylamine derivatives, method for producing the same, their use as medicament or diagnostic agent and medicament containing the same
08/28/2002EP1234819A1 Processes for production of oxadiazoline derivatives
08/28/2002EP1054874B1 Substituted aminophenyl isoxazoline derivatives useful as antimicrobials
08/28/2002CN1089759C Crystal form of N-(4-trifluoromethylphenyl)-5-methylisoxazole-4-carboxamide
08/27/2002US6441021 Type-iv collagenase inhibitors
08/27/2002US6441014 Antiinflammatory agent, useful for treating cylcoocygenase-2 associated disorders
08/27/2002US6440963 Use of selective COX-2 inhibitors for the treatment of urinary incontinence
08/22/2002WO2002064565A1 Acylated 1,2,3,4-tetrahydronaphthyl amines and their use as pharmaceutical
08/22/2002WO2002064546A2 Acylated 6,7,8,9-tetrahydro-5h-benzocycloheptenyl amines and their use as pharmaceutical
08/22/2002WO2002064545A1 Acylated indanyl amines and their use as pharmaceuticals
08/22/2002WO2002064136A2 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators
08/22/2002WO2002064094A2 2-aryloxy-2-arylalkanoic acids for diabetes and lipid disorders
08/22/2002CA2437118A1 2-aryloxy-2-arylalkanoic acids for diabetes and lipid disorders
08/21/2002EP1231939A2 Oncolytic combinations for the treatment of cancer
08/20/2002US6437177 α-hydroxy, -amino, and halo derivatives of β-sulfonyl hydroxamic acids as matrix metallopropteinases inhibitors
08/20/2002US6436967 Process for preparing prodrugs of benzenesulfonamide-containing cox-2 inhibitors
08/20/2002US6436930 Thio derivatives of sordarin as antifungal agents
08/15/2002WO2002062770A1 Isoxazoline derivative and herbicide comprising the same as active ingredient
08/15/2002WO2002062750A1 Cannabinoid receptor ligands
08/15/2002WO2002062389A1 Remedies for urinary diseases comprising lpa receptor controlling agents
1 ... 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 79 ... 115