Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
01/2001
01/03/2001CN1060172C Substituted biphenyl sulfonamide endothelin antagonists
01/03/2001CN1060171C Substituted biphenyl isoxazole sulfonamides
01/02/2001US6168776 Alkyl, alkenyl and alkynyl Chrysamine G derivatives for the antemortem diagnosis of Alzheimer's disease and in vivo imaging and prevention of amyloid deposition
01/02/2001CA2026761C Preparation of isoxazole-4,5-dicarboxylic diesters
01/02/2001CA2009604C Diaryl-substituted heterocyclic compounds, their preparation and drugs and cosmetics obtained therefrom
01/02/2001CA1341163C Oxime ether derivatives, their preparation and fungicides containing these derivatives
12/2000
12/30/2000CA2313131A1 Compositions and treatment for diabetic complications
12/28/2000WO2000078746A1 Antiviral agents
12/28/2000CA2375211A1 Antiviral agents
12/27/2000EP1062218A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases)
12/27/2000EP1062208A1 Hetaryl-substituted benzyl phenyl ethers, method for the production thereof, and their use for combating harmful fungi and animal pests
12/27/2000EP1062199A1 Modulators of protein tyrosine phosphatases (ptpases)
12/27/2000CN1278247A Alpha-hydroxy, amino and -fluoro derivatives of beta-sulphenyl hydroxamic acids matrix metalloproteinases inhibitors
12/26/2000US6166055 Antiinflammatory agents
12/26/2000US6166020 Aryl and heteroaryl alkoxynaphthalene derivatives
12/26/2000US6165944 4-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides
12/21/2000WO2000044709A3 ACETYLENIC α-AMINO ACID-BASED SULFONAMIDE HYDROXAMIC ACID TACE INHIBITORS
12/20/2000EP1060179A1 Substituted aminomethyl isoxazoline derivatives useful as antimicrobials
12/14/2000WO2000075107A2 Bradykinin receptor antagonists
12/13/2000CN1276785A N-aroylphenylalanine derivs.
12/12/2000US6160000 Antidiabetic agents based on aryl and heteroarylacetic acids
12/12/2000US6159995 Substituted diaminocarboxylic acids
12/12/2000US6159973 Aromatic amides, their preparation process, the compositions containing them and their use as pesticides
12/12/2000CA2023560C 5-methyl-isoxazole-4-carboxylic acid anilides and 2-hydroxyethylidene-cyano acetic acid anilides for the treatment of ocular diseases
12/07/2000WO2000073287A1 Isoxazoline carboxylate derivatives of mutiline and their use as antibacterials
12/06/2000EP1057812A1 Aminoguanidine hydrazone derivatives, process for producing the same and drugs thereof
12/06/2000EP1056710A1 Diterpene derivatives and anti-inflammatory analgesic agents comprising the same
12/06/2000EP1056341A1 Method and apparatus for the preparation of ketones
12/06/2000CN1275909A In-modulators
12/05/2000US6156896 Fluorous reaction and separation systems
12/05/2000US6156761 Substituted tetralone derivatives for enhancing cognition
12/05/2000US6156702 As herbicides
11/2000
11/29/2000EP1054874A1 Substituted aminophenyl isoxazoline derivatives useful as antimicrobials
11/29/2000CN1275123A Prostaglandin agonists and their use to treat bone disorders
11/28/2000US6153759 Herbicide comprising a 5-membered or 6-membered heterocyclic, saturated or unsaturated radical containing one to three hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen
11/28/2000US6153752 Cyclization for preparing pyrazoles, isoxazoles and pyrimidines
11/23/2000WO2000069800A2 Process for preparing ketones or aldehydes
11/23/2000WO2000043354A3 Multicyclic compounds which inhibit leukocyte adhesion mediated by vla-4
11/23/2000WO2000034237A3 Acetamide and substituted acetamide-containing thiourea inhibitors of herpes viruses
11/23/2000WO1999065871A3 Thiolesters and uses thereof
11/22/2000CN1274350A Efficient method for conversion of nitriles to amidines
11/21/2000US6150530 Amidation of amine with acid
11/21/2000US6150394 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
11/21/2000US6150390 Accelerates bone formation; osteoporosis; (ltb-4(leukotriene-b-4; 5,12-dihydroxyeicosatetra-6,8,10,14-enoic acid) receptor antagonist
11/21/2000US6150303 Herbicides
11/21/2000US6150129 Antimicrobial determination of N-(aminoalkyl) and/or N-(Amidoalkyl) dinitrogen heterocyclic compositions
11/16/2000WO2000068227A1 Substituted benzoylisoxazoles and the use thereof as herbicides
11/16/2000WO2000038665A3 Use of an integrin antagonist and one or more antineoplastic agents as a combination therapy in the treatment of neoplasia
11/16/2000WO2000006525A3 Synthesis of combinatorial libraries of compounds reminiscent of natural products
11/16/2000DE19920247A1 Arzneimittel mit einem Gehalt an Verbindungen mit einem Stickstoff-Sauerstoff-Heterocyclus als Wirkstoff und ihre Verwendung Medicaments with an amount of compounds having a nitrogen-oxygen heterocycle as active ingredient and their use
11/16/2000CA2372963A1 Substituted benzoylisoxazoles and the use thereof as herbicides
11/15/2000EP1052255A1 Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics.
11/15/2000EP1052238A1 Novel tricyclic compound
11/15/2000EP1051169A1 Compounds, compositions and methods for treating or preventing pneumovirus infection and associated diseases
11/15/2000CN1273585A Substituted 3-(1,2-benzisothiazol or isoxazel-5-yl)-substituted pyrimidine as heribicides
11/09/2000WO2000066546A2 Monofluoroalkyl derivatives
11/09/2000WO2000066104A2 Ace-2 inhibiting compounds and methods of use thereof
11/09/2000WO2000066094A2 Use of compounds with a nitrogen-oxygen heterocycle as anti-infectious agents
11/09/2000WO2000038718A3 Use of matrix metalloproteinase inhibitor together with an antineoplastic agents, optionally also together with radiation, in the treatment of neoplasia
11/09/2000DE19920791A1 Substituierte Benzoylisoxazole Substituted benzoylisoxazoles
11/09/2000CA2372490A1 Monofluoroalkyl derivatives
11/09/2000CA2372387A1 Ace-2 inhibiting compounds and methods of use thereof
11/09/2000CA2369526A1 Use of compounds with a nitrogen-oxygen heterocycle as anti-infectious agents
11/08/2000EP1049662A1 Inhibitors of alpha4 mediated cell adhesion
11/02/2000WO2000064876A1 Tri-aryl acid derivatives as ppar receptor ligands
11/02/2000WO2000038730A3 Use of a cyclooxygenase-2 inhibitor and one or more antineoplastic agents for combination therapy in neoplasia
11/02/2000EP1048657A1 Thienyl-, furyl-, pyrrolyl- and biphenylsulfonamides and derivatives thereof that modulate the activity of endothelin
11/02/2000EP1047656A1 Alkenyldiarylmethane non-nucleoside hiv-1 reverse transcriptase inhibitors
11/02/2000EP1047418A1 Inhibition of raf kinase using substituted heterocyclic ureas
11/02/2000CA2371308A1 Tri-aryl acid derivatives as ppar receptor ligands
11/01/2000CN1272109A Process for producing isooxazolidinedione compound
11/01/2000CN1272107A Benzamidine derivatives as factor Xa inhibitors
10/2000
10/31/2000US6140528 Alkyl pentafluorosulfanyl-substituted-benzoates
10/31/2000US6140345 For treating psychoses and pain
10/31/2000US6140270 By reacting them with an amine compound and an acid or base; herbicides
10/25/2000CN1271346A Method for producing substituted 2-nitroguanidine derivative
10/25/2000CN1271345A Method for producing substituted 2-nitroguanideine derivatives
10/24/2000US6136837 α-substituted benzyl heterocyclic derivatives, intermediates for producing the same and agrochemical composition containing the same as active ingredient
10/24/2000US6136833 Pharmaceutical formulations and process for their preparation
10/19/2000WO2000007996A8 Pyrazoles as estrogen receptor modulators
10/18/2000CN1057524C Benzoyl isocarboxazid derivatives, their preparing methods and uses
10/17/2000US6133283 Mono- or polyenic carboxylic acid derivatives
10/17/2000US6133265 Treating physiological disorders associated with an excess of neuropeptide y, such as eating disorders, e.g., obesity, bulimia, and certain cardiovascular diseases, e.g., hypertension
10/17/2000US6133259 Diagnosis of alzheimer's disease
10/12/2000WO2000059874A1 NOVEL AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES, TNF-α, AND AGGRECANASE
10/12/2000CA2366264A1 Novel amide derivatives as inhibitors of matrix metalloproteinases, tnf-.alpha., and aggrecanase
10/11/2000EP1042002A1 Pharmaceutical formulations and processes for their preparation
10/11/2000EP1041982A1 INHIBITION OF p38 KINASE ACTIVITY USING SUBSTITUTED HETEROCYCLIC UREAS
10/05/2000WO2000058293A2 Glucokinase activators
10/05/2000WO2000058290A1 Process for the preparation of (e)-3-(1-propenyl)isoxazoline
10/04/2000EP1040094A1 Substituted cyclopentane and cyclopentene compounds useful as neuraminidase inhibitors
10/04/2000EP0766672B1 Arylsulfonamido-substituted hydroxamic acids as matrix metalloproteinase inhibitors
10/03/2000US6127568 Phenylacetic acid derivatives, preparation thereof and intermediates thereof, and compositions containing them
10/03/2000US6127372 Sulfonamide inhibitors of aspartyl protease
09/2000
09/28/2000WO2000056685A1 Methods for the preparation of biphenyl isoxazole sulfonamides
09/28/2000CA2367916A1 Methods for the preparation of biphenyl isoxazole sulfonamides
09/27/2000EP1037883A1 NOVEL HETEROCYCLICALLY SUBSTITUTED $g(a)-HYDROXYCARBOXLIC ACID DERIVATIVES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS
09/27/2000EP1037868A2 $g(a)-HYDROXY, -AMINO, AND HALO DERIVATIVES OF $g(b)-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS
09/27/2000EP0885188B1 Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors
09/27/2000CN1056837C 5-arylisoxazol-4-yl-substituted 2-aminocarboxylic acid compound, its medical composition and use
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