Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
10/2001
10/30/2001US6310095 Inhibitors of protein isoprenyl transferases
10/30/2001CA2123101C Nitroxyalkylamide derivative
10/25/2001WO2001079157A1 Hydrazide and alkoxyamide angiogenesis inhibitors
10/25/2001WO2001049288A9 Novel compounds and compositions as protease inhibitors
10/25/2001CA2406442A1 Hydrazide and alkoxyamide angiogenesis inhibitors
10/24/2001EP0840601B1 Thip for treating sleep disorders
10/24/2001CN1319092A Benzamide derivatives and their use as cytokine inhibitors
10/24/2001CN1318535A Dihalopropene compound, insecticide/miticide containing the same and intermediate for producing the same
10/23/2001US6306887 Non-peptidyl inhibitors of VLA-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
10/23/2001US6306886 Solid polymorph anticoagulants
10/23/2001US6306842 Compound of nonsteroid antiinflammatory agent, spacer and cox-2 inhibitor
10/23/2001CA2222657C Intermediates in preparation of new phenylethanolaminomethyltetralins
10/23/2001CA2083179C Isoxazole-4-carboxamides and hydroxyalkylidenecyanoacetamides, pharmaceuticals containing these compounds and their use
10/18/2001US20010031878 Novel processes for making- and a new crystalline form of- leflunomide
10/17/2001EP1144368A2 Acetylenic alpha-amino acid-based sulfonamide hydroxamic acid tace inhibitors
10/17/2001EP1144364A2 Multicyclic compounds which inhibit leukocyte adhesion mediated by vla-4
10/17/2001CN1317965A Compounds having IgE affecting properties
10/16/2001US6303816 N-2-(4-(4-(2-methanesulfonamidoethyl)phenyl)phenyl)-propyl 2-propanesulfonamide or a pharmaceutically acceptable salt thereof.
10/16/2001US6303792 Quantitatively determining amount of by-product in solution of desired compound in water and solvent, adding corresponding amount of base, crystallizing and separating desired compound
10/16/2001US6303609 Used for the inhibition of platelet aggregation, as thrombolytics, and/or for the treatment of thromboembolic disorders
10/11/2001WO2001074763A1 Aryl and heteroaryl sulfonates
10/11/2001WO2001074753A1 Synthetic derivatives of lunularic acid, medicaments containing said compounds, method for producing the lunularic acid derivatives and the use thereof
10/11/2001DE10015866A1 Aryl- und Heteroarylsulfonate Aryl and Heteroarylsulfonate
10/11/2001DE10015525A1 Synthetische Derivate von Lunularsäure, Arzneimittel enthaltend diese Verbindung, Verfahren zur Herstellung der Lunularsäurederivate sowie deren Verwendung Synthetic derivatives of Lunularsäure, to medicaments containing this compound, methods of making them and their use of the Lunularsäurederivate
10/11/2001CA2404545A1 Aryl and heteroaryl sulfonates
10/10/2001EP1141023A2 Anti-cd3 immunotoxins and therapeutic uses therefor
10/10/2001EP1140852A1 1,2,3,4-tetrahydronaphthalenes and their pharamaceutical use
10/10/2001EP1140809A1 New biphenyl and biphenyl-analogous compounds as integrin antagonists
10/10/2001EP1140802A1 Substituted aryl and heteroaryl derivatives, their production and their use as medicines
10/10/2001EP1140784A2 Ion channel modulating agents
10/10/2001EP1140783A1 Ortho-diphenol compounds, methods and pharmaceutical compositions for inhibiting parp
10/10/2001EP1140194A2 Use of cyclooxygenase-2 inhibitor, a matrix metallaproteinase inhibitor, an antineoplastic agent and optionally radiation as a combined treatment of neoplasia
10/10/2001EP1140193A2 Use of an integrin antagonist and one or more antineoplastic agents as a combination therapy in the treatment of neoplasia
10/10/2001EP1140192A2 Use of a cyclooxygenase-2 inhibitor and one or more antineoplastic agents for combination therapy in neoplasia
10/10/2001EP1140183A1 Use of a matrix metalloproteinase inhibitor and an integrin antagonist in the treatment of neoplasia
10/10/2001EP1140182A2 Use of a matrix metalloproteinase inhibitor together with an antineoplastic agent, optionally also together with radiation, in the treatment of neoplasia
10/10/2001EP1140179A2 Use of a cyclooxygenase 2 inhibitor and an integrin antagonist as a combination therapy in the treatment of neoplasia
10/10/2001EP1140178A2 Use of a matrix metallaproteinase inhibitor and radiation as a combined treatment of neoplasia
10/10/2001EP1140177A2 Use of an integrin antagonist and radiation in the treatment of neoplasia
10/10/2001EP1140079A1 Assays for ligands for nuclear receptors
10/09/2001US6300372 3-Cyano-3-(3,4-disubstituted) phenylcyclohexyl-1-carboxylates
10/09/2001CA2018960C Salicylaldehyde derivatives and salicylic acid derivatives and their sulfur analogs, their preparation and their use as herbicides and bioregulators
10/04/2001WO2001072960A2 Il-8 receptor antagonists
10/04/2001WO2001021577A3 Melanin concentrating hormone antagonist
10/04/2001EP1137647A1 Thiourea inhibitors of herpes viruses
10/04/2001EP1137633A2 Acetamide and substituted acetamide-containing thiourea inhibitors of herpes viruses
10/04/2001CA2403787A1 Il-8 receptor antagonists
10/03/2001CN1072221C 3-halo-3-heteroaryl carboxylic acid derivatives, method of preparing them and intermediates
10/02/2001US6297198 Compounds with sulfur groups on isoxazole rings as herbicides
09/2001
09/27/2001WO2001070673A2 CYCLIC β-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-$g(a)
09/27/2001WO2001070672A2 Compounds and methods to treat alzheimer's disease
09/27/2001WO2001014576B1 Process and intermediates for the preparation of isoxazolecaroxamides and analogues
09/27/2001US20010025105 Anticancer agent; Alzheimer's therapy
09/27/2001CA2401870A1 Cyclic .beta.-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-.alpha.
09/27/2001CA2401749A1 Compounds and methods to treat alzheimer's disease
09/26/2001CN1314813A Novel isoxazolinone antibacterial agent
09/25/2001US6294580 For therapy and prophylaxis of type ii or non-insulin dependent diabetes mellitus, hyperglycaemia, dyslipidemia, type ii diabetes, type i diabetes, hypertriglyceridemia, syndrome x, insulin resistance, heart failure
09/20/2001WO2001068585A1 Novel amide compounds
09/20/2001WO2001068568A2 Il-8 receptor antagonists
09/20/2001WO2001068033A2 Il-8 receptor antagonists
09/20/2001CA2402891A1 Il-8 receptor antagonists
09/19/2001CN1313846A C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cystenine proteases
09/18/2001US6291508 Potent ability to bind to retinoic acid receptors thus useful in treating psoriasis and rheumatoid arthritis.
09/18/2001US6291505 Pyrazole estrogen receptor agonist and antagonist
09/18/2001US6291400 Herbicidal compounds
09/13/2001US20010021714 Compounds such as n-(4-bromo-3-methyl-5-isoxazolyl)-2-n-benzylbenzo(b)thiophene-3-sufonamide administered as endothelin peptide receptor antagonists
09/12/2001EP1131307A1 Method of producing 2-alkyl-3-(4,5-dihydroisoxazole-3-yl)-halobenzenes
09/12/2001EP1131306A2 Isoxazoline fibrinogen receptor antagonists
09/12/2001EP0888317B1 Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to ppar-gamma
09/11/2001US6288098 Administering n-(4-trifluoromethyl)-5-methylisoxazole-4-carboxanilide and n-(4-trifluoromethylphenyl)-2-cyano-3-hydroxycrotonamide
09/11/2001US6288071 1-ethylene-2-alkylene-1,4-cyclohexadiene pesticides
09/07/2001WO2001064755A2 Isoxazole gegen virale erkrankungen
09/07/2001WO2000075107A3 Bradykinin receptor antagonists
09/07/2001CA2401405A1 Medicament for viral diseases
09/06/2001US20010020013 Polymerase inhibitors
09/05/2001EP1129082A1 Method and novel intermediate products for producing isoxazolin-3-yl-acylbenzenes
09/05/2001CN1311793A Antipicornaviral compounds, their prepn. and use
09/05/2001CN1311679A Benzimidazole derivatives as modulators of IgE
09/05/2001CN1311675A Compounds having IgE affecting properties
09/04/2001USH1992 Metalloproteinase inhibitors, pharmaceutical compositions containing them, and their pharmaceutical uses
09/04/2001US6284877 Sulfonamide compound and method for its production, metal chelate compound employing the sulfonamide compound, and optical recording medium employing the metal chelate compound
08/2001
08/30/2001WO2001062704A1 Novel use of phenylheteroalkylamine derivatives
08/30/2001WO2001016131A3 Five membered-ring compounds and utilization thereof in liquid crystal mixtures
08/30/2001WO2001014576A3 Process and intermediates for the preparation of isoxazolecaroxamides and analogues
08/30/2001DE10009408A1 Arzneimittel gegen virale Erkrankungen Medicines for viral diseases
08/30/2001CA2397234A1 Novel use of phenylheteroalkylamine derivatives
08/29/2001CN1070022C 3-hydroxy-5-methylisozazole dihydras and its producing process
08/28/2001US6281210 Benzoic acid esters of oxazolidinones having a hydroxyacetylpiperazine substituent
08/28/2001US6281209 Fungicidal alkoximinomethyldioxazine derivatives
08/23/2001WO2001060819A1 Novel isoxazole and thiazole compounds and use thereof as drugs
08/23/2001WO2001060807A1 Aryloxyacetic acids for diabetes and lipid disorders
08/23/2001WO2001060363A1 A method for synthesizing leflunomide
08/23/2001WO2001004116A3 Neurotrophic pyrrolidines and piperidines, and related compositions containing them
08/23/2001CA2400290A1 A method for synthesizing leflunomide
08/23/2001CA2400021A1 Aryloxyacetic acids for diabetes and lipid disorders
08/22/2001EP1124827A1 3-(substituted phenyl)-5-(substituted heterocyclyl)-1,2,4-triazole compounds
08/21/2001US6277849 N-sulphonyl and N-sulphinyl amino acid amides as microbiocides
08/21/2001CA2000362C Methyl .alpha.-arylacrylates substituted by a heterocyclic radical and their use
08/16/2001WO2001058853A1 Dehydroamino acids
08/16/2001EP1123272A1 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
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