| Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459) |
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| 03/26/2003 | EP1025085B1 Heterocycles useful in the treatment of benign prostatic hyperplasia and intermediates thereof |
| 03/26/2003 | CN1406233A Medicine for viral diseases |
| 03/25/2003 | US6537986 Oxazolidinone antibacterial agents having a thiocarbonyl funtionality |
| 03/20/2003 | WO2003022824A1 Oxazolidinone and/or isoxazoline as antibacterial agents |
| 03/20/2003 | WO2002048100A3 Thiosulphonic s-esters as material protective agent |
| 03/20/2003 | US20030055292 Preparation of ketones from aldehydes |
| 03/20/2003 | US20030055286 Il-8 receptor antagonists |
| 03/20/2003 | US20030055093 For therapy of cardiovascular diseases, stable or unstable angina pectoris, coronary heart disease, stable or unstable angina pectoris, coronary heart disease, Prinzmetal angina, acute coronary syndrome, heart failure, myocardial infarction |
| 03/20/2003 | US20030055025 For therapy of bacterial infections and neoplasms, |
| 03/20/2003 | US20030055012 Prodrugs of COX-2 inhibitors |
| 03/20/2003 | US20030054974 Non-oxidatively metabolized compounds and compositions, synthetic pathways therefor, and uses thereof |
| 03/20/2003 | CA2459766A1 Oxazolidinone and/or isoxazoline as antibacterial agents |
| 03/19/2003 | EP1292573A2 Substituted thioacetamides |
| 03/19/2003 | EP0984914B1 Substituted 2-(3-alkenyl-benzoyl)-cyclohexane-1,3-diones |
| 03/18/2003 | US6534509 Derivatives are useful as anti-inflammatory agents. This invention is also directed to pharmacetutical compostions for inflammation |
| 03/18/2003 | CA2268028C 3-alkoxyisoxazol-4-yl-substituted 2-amino carboxylic acid compounds |
| 03/13/2003 | WO2003020708A1 Zonisamide intermediate and synthesis |
| 03/13/2003 | WO2003020269A1 Diaryl cycloalkyl derivatives, method for producing the same and the use thereof as ppar activators |
| 03/13/2003 | WO2002078625A3 Therapeutic combinations for cardiovascular and inflammatory indications |
| 03/13/2003 | US20030050298 A sulfonamide substituted diphenyl thiourea compounds treating a chemokine mediated disease |
| 03/13/2003 | CA2458905A1 Zonisamide intermediate and synthesis |
| 03/12/2003 | CN1402723A 3-(4,5-dihydroisoxazol-3-yl)-substd. benzoylpyrazoles as herbicides |
| 03/12/2003 | CN1402715A Processes for production of oxadiazoline derivs. |
| 03/11/2003 | US6531610 Intermediate acylating carbonate |
| 03/11/2003 | US6531498 Antiallergens, etc |
| 03/11/2003 | US6531452 Peptide-like and peptidomimetic compounds that inhibit enzymatic activity of picornaviral 3C proteases and inhibit picornavirus replication |
| 03/06/2003 | WO2003018551A1 New mandelic acid derivatives and their use as thrombin inhibitors |
| 03/06/2003 | WO2003018008A1 Apo ai expression accelerating agent |
| 03/06/2003 | WO2003017946A2 Non-oxidatively metabolized compounds and compositions, synthetic pathways therefor, and uses thereof |
| 03/06/2003 | US20030045518 Certain bis(thio-hydrazide amide) compounds significantly enhance the anticancer activity of taxol. |
| 03/06/2003 | CA2457532A1 Non-oxidatively metabolized compounds and compositions, synthetic pathways therefor, and uses thereof |
| 03/05/2003 | EP1288206A1 Substituted benzenesulfonamide derivatives as prodrugs of COX-2 inhibitors |
| 03/05/2003 | EP1286991A2 Cyclopropyl-anellated 3-(4,5-dihydroisoxazol-3-yl)-substitued benzoylpyrazoles |
| 03/05/2003 | EP1286974A2 Medicament for viral diseases |
| 03/05/2003 | EP0892791B1 N-[[4-(5-METHYL-3-PHENYLISOXAZOL-4-YL]PHENYL]SULFONYLPROPYLAMIDE and its SODIUMSALT AS PRODRUGS OF COX-2 INHIBITORS |
| 03/04/2003 | US6528543 Glucokinase activating for treating type II diabetes; acylurea compound, phenylacetyl-substituted; 1-(2-(3-chloro-phenyl)-3cyclopentyl-propionyl)-3-methyl-urea |
| 02/27/2003 | WO2003016280A1 Nr1h4 nuclear receptor binding compounds |
| 02/27/2003 | WO2003015774A1 Compounds effecting glucokinase |
| 02/27/2003 | WO2003015771A1 Fxr nr1h4 nuclear receptor binding compounds |
| 02/27/2003 | WO2002096884A3 Substituted benzoylketones as herbicidal agents for use as plant treatment agent |
| 02/26/2003 | EP1284969A1 3-(4,5-dihydroisoxazole-5-yl)benzoylcyclohexenones and the use thereof as herbicides |
| 02/26/2003 | EP1284730A1 Aralkyl ester soft drugs |
| 02/25/2003 | US6525204 Oximination reaction of nitro-o-methylphenyl compound with organic nitrite; cyclization with alkene in basic catalyst presence; reduction, bromination, oxidation, carboxylation |
| 02/25/2003 | US6525099 N-substituted sulfonamide derivatives |
| 02/25/2003 | US6525072 Prevention and treatment of cellular disorders such as cancer |
| 02/25/2003 | US6525048 Aminomethylphenoxymethyl/benzisoxazole substituted azabicyclic compounds; depression, generalized anxiety disorder, obesity, migraine; 2-(5-Fluoro-benzo(d)isoxazol-3-y)-7-(3-morpholin-4-ylmethylphenoxymethyl) -octahydro-pyrido(1,2-a)pyrazine; |
| 02/25/2003 | US6525036 Compounds and compositions as protease inhibitors |
| 02/20/2003 | WO2003014064A1 Naphthylurea and naphthylacetamide derivatives as vanilloid receptor 1 (vr1) antagonists |
| 02/20/2003 | WO2003013655A2 Carbonic anhydrase inhibitors |
| 02/20/2003 | WO2003013484A2 N-monoacylated derivatives of o-phenylenediamines, their six membered heterocyclic analogues and their use as pharmaceutical agents |
| 02/20/2003 | WO2002096516A8 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease |
| 02/20/2003 | WO2002030882A9 Sulfoxide and bis-sulfoxide compounds and compositions for cholesterol management and related uses |
| 02/20/2003 | WO2002030860A9 Ketone compounds and compositions for cholesterol management and related uses |
| 02/20/2003 | WO2002024635A3 Aminoalcohol derivatives |
| 02/20/2003 | CA2456939A1 Carbonic anhydrase inhibitors |
| 02/20/2003 | CA2455754A1 Amine derivatives |
| 02/19/2003 | EP1283723A2 Combination therapy using cox-2 selective inhibitor and thromboxane inhibitor and compositions therefor |
| 02/19/2003 | CN1398252A Dehydroamino acids compounds |
| 02/19/2003 | CN1398189A Combination therapy of radiation and COX-2 inhibitor for treatment of neoplasia |
| 02/19/2003 | CN1397550A Novel benzene amine compound, its prepn. process and medicinal compsns. contg. them |
| 02/19/2003 | CN1397547A Novel benzene amine compound, its prepn. process and medicinal compsns. contg. them |
| 02/18/2003 | US6521666 Inhibitors of α4 mediated cell adhesion |
| 02/18/2003 | US6521622 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation |
| 02/18/2003 | CA2420042A1 Carboxylic acid derivatives, processes for the preparation thereof and pharmaceutical agents comprising the same as active ingredient |
| 02/13/2003 | WO2003011210A2 Arylheteroalkylamine derivatives and their use as inhibitors of nitric oxide synthase |
| 02/13/2003 | US20030032803 Novel amide derivatives as inhibitors of matrix metalloproteinases, TNF-alpha, and aggrecanase |
| 02/13/2003 | US20030032662 Micronized leflunomide |
| 02/13/2003 | US20030032657 Fluoro-substituted benzenesulfonyl compounds for the treatment of inflammation |
| 02/13/2003 | US20030032635 Heterocyclic esters and amides |
| 02/12/2003 | EP1283203A1 Crystalline form of 4-(5-methyl-3-phenylisoxazol-4-yl) benzene-sulfonamide |
| 02/12/2003 | EP1283042A1 Aqueous liquid preparation |
| 02/12/2003 | EP1282595A1 Novel phenyl-propargylether derivatives |
| 02/12/2003 | EP1282415A2 Compounds and methods for regulating bacterial growth and pathogenesis |
| 02/12/2003 | EP0988292B1 Piperazine derivatives and their use as anti-inflammatory agents |
| 02/12/2003 | EP0669920B1 Substituted 3-(aminoalkylamino)-1,2-benzisoxazoles and related compounds |
| 02/11/2003 | US6518310 Non-peptidic; inhibits trypsin-like protease, thrombin and embolus formation; anticoagulant |
| 02/11/2003 | CA2250391C Butadiene derivatives and process for their preparation |
| 02/11/2003 | CA2022691C 1,2,4-oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents |
| 02/06/2003 | WO2003010165A1 Isoxazoline derivatives and herbicides for agricultural and horticultural use |
| 02/06/2003 | WO2003010143A1 Dialkylhydroxybenzoic acid derivatives containing metal chelating groups and their therapeutic uses |
| 02/06/2003 | US20030028033 Which are used as herbicides, by forming a 2-(isoxazol-3-yl)-aniline compound of given formula and then halogenation, thioalkylation, oxidation and acylation; fewer steps, efficiency |
| 02/06/2003 | US20030027851 Readily soluble crystal modification; specific X-ray diffraction pattern obtained with a focusing Debye-Scherrer beam and Cu-K alpha 1-radiation |
| 02/06/2003 | US20030027798 For therapy |
| 02/05/2003 | EP1280757A2 New gamma selective retinoids |
| 02/05/2003 | EP1037868B1 $g(a)-HYDROXY, -AMINO, AND HALO DERIVATIVES OF $g(b)-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS |
| 02/05/2003 | CN1395562A Nitrogenous cyclic compounds and pharmaceutical compositions containing the same |
| 02/05/2003 | CN1100761C Benzyloxy substituted aryl copounds and their use as fungicides and insecticides |
| 02/04/2003 | US6515136 To the novel intermediates prepared by these methods. The biphenyl isoxazole sulfonamides prepared by the present methods are endothelin antagonists useful, inter alia, for the treatment of hypertension. |
| 02/04/2003 | US6515124 Dehydroamino acids |
| 02/04/2003 | US6515003 Useful in the treatment of diseases related to lipid and carbohydrate metabolism |
| 01/30/2003 | WO2003008395A1 Substituted isoxazoles and the use thereof as antibiotics |
| 01/30/2003 | US20030022935 Acylated 1,2,3,4-tetrahydronaphthyl amines and their use as pharmaceutical agents |
| 01/30/2003 | US20030022865 Sulfoxide and bis-sulfoxide compounds and compositions for cholesterol management and related uses |
| 01/30/2003 | CA2453846A1 Substituted isoxazoles and the use thereof as antibiotics |
| 01/29/2003 | EP1278741A1 Muscarinic agonists |
| 01/29/2003 | EP1278722A1 Aryl and heteroaryl sulfonates |
| 01/29/2003 | CN1100047C N3-(5-methyl-iso-oxazole) group-3,4-dihydroxy cinnamide and producing process thereof |
| 01/28/2003 | US6511981 Benzyl isooxazole and benzyl pyrazole derivatives as aldose reductase and cyclooxygenase-2 inhibitors |
| 01/23/2003 | WO2003006454A2 Heterocyclic carboxamides and their use as fungicides |
| 01/23/2003 | WO2003006447A2 Interaction inhibitors of tcf-4 with beta-catenin |