Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
03/2004
03/11/2004US20040049053 Reacting 4-hydroxycoumarin with hydroxylamine in the presence of a base; sulfonating product to form salt of the methanesulfonic acid; forming benzisoxazolemethanesulfonamide from either the acetic acid or methanesulfonic acid
03/11/2004US20040048908 E.g., 3-(5-(3,4-dichlorophenyl)- 4-isoxazolyl)propan-1-ol; prophylaxis or treatment of diabetes, impaired glucose tolerance or diabetic complications
03/11/2004US20040048864 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
03/11/2004US20040048858 Chalcone derivatives and their use to treat diseases
03/11/2004US20040048857 Treatment and/or prevention of diseases or disorders mediated by lymphocyte interactions.
03/11/2004US20040048316 Comprises phosphorescence and fluorescence resonance energy transfer; binding chenodeoxycholic acid to farnesoid X receptors; for regulating cholesterol absorption; for treatment of obesity
03/10/2004EP1395571A1 Compounds and methods for the treatment or prevention of flavivirus infections
03/10/2004EP1395551A2 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer's disease and similar diseases
03/10/2004EP1395548A1 Derivatives of diphenylurea, diphenyloxalic acid diamide and diphenylsulfuric acid diamide and their use as medicaments
03/10/2004CN1481377A Cyclic Beta-amino acid derivatives as inhibitors of matrix metalloproteases and TNF alhpa
03/10/2004CN1141095C Preparation containing combination of N-5-methylisoxazole-4-carboxylic acid-(4-trifluoromethy1)-anilid and N-(4 trifluoromethylphenyl)-2-cyano-3-hyroxycrotonic acid amide
03/09/2004US6703422 For therapy and prophylaxis of cardiovascular disease, dyslipidemia; dyslipoproteinemia; disorder of glucose metabolism; alzheimer's disease; syndrome x; peroxisome proliferator activated receptor-associated disorder
03/09/2004US6703348 Heterocyclyl-substituted benzoylcyclohexandiones, their preparation, and their use as herbicides
03/04/2004WO2004018428A1 Antibacterial benzoic acid derivatives
03/04/2004WO2004018410A1 Substituted benzanilide compound and pest control agent
03/04/2004US20040044062 Method of treatment of viral infection including HIV using water soluble fullerenes - III
03/04/2004US20040044052 N-Aryl-2-oxazolidinone-5-carboxamides and their derivatives
03/03/2004EP1394152A1 2-iminoimidazole derivatives (1)
03/03/2004EP1394147A1 Carboxylic acid derivative and medicine comprising salt or ester of the same
03/03/2004EP1392660A1 Substituted benzoylcyclohexenones and their use as herbicidal agents
03/03/2004EP0929217B1 Sordarin derivatives
03/03/2004CN1479721A Sulfoxide and bis-sulfoxide compounds and compositions for cholesterol management and related uses
03/03/2004CN1479712A Ketone compounds and compositions for cholesterol management and related uses
03/02/2004US6699996 Production method of isoxazolidinedione compound
03/02/2004US6699910 Ketone compounds and compositions for cholesterol management and related uses
03/02/2004US6699891 Npyy5 antagonists
03/02/2004US6699884 Antiinflammatory cyclooxygenase inhibitors.
02/2004
02/26/2004WO2004016596A1 Condensed heterocyclic compounds as pde-iv inhibitors for the treatment of inflammatory and allergic disorders
02/26/2004WO2004016576A1 Fused benzene derivative and use
02/26/2004WO2003039549A8 Selective antibacterial agents
02/26/2004US20040039034 Hydroxypropyl amides for the treatment of Alzheimer's disease
02/26/2004US20040037022 Aminoalcohol derivatives
02/26/2004CA2495383A1 Fused benzene derivative and use
02/25/2004EP1391456A1 2-iminoimidazole derivative (2)
02/25/2004EP1391451A1 2-iminopyrrolidine derivates
02/25/2004EP1005446B1 N-aroylphenylalanine derivatives
02/25/2004CN1478078A Nitrogenous aromatic ring compounds
02/25/2004CN1139580C Substituted benzylamines and their use for treatment of depression
02/25/2004CN1139579C Isoxazolecarboxamide derivatives
02/25/2004CN1139578C Preparation of isoxazoline-3-yl-acyl benzene
02/24/2004US6696494 α-hydroxyarylbutanamine inhibitors of aspartyl protease
02/24/2004CA2065983C Crop-protecting compositions containing isoxazolines or isothiazolines, novel isoxazolines and isothiazolines, and their preparation
02/19/2004WO2004014879A1 New process
02/19/2004WO2004014867A2 Matrix metalloproteinase inhibitors and methods for identification of lead compounds
02/19/2004WO2004014847A1 Mcp-1 receptor antagonists and method of use thereof
02/19/2004WO2004014844A2 Aryl and heteroaryl compounds and methods to modulate coagulation
02/19/2004WO2004014430A1 Compositions of a cyclooxygenase-2 selective inhibitor and a carbonic anhydrase inhibitor for the treatment of neoplasia
02/19/2004WO2004014381A2 Matrix metalloproteinase inhibitors and methods for identification of lead compounds
02/19/2004WO2004014370A2 Oxadiazoles as modulators of metabotropic glutamate receptor-5
02/19/2004WO2004014352A2 Methods for treating carbonic anhydrase mediated disorders
02/19/2004WO2003004147A8 Compound libraries
02/19/2004US20040034231 Amidinophenyl-4-aminoacetic acid derivative is useful for treating diseases such as thrombosis, apoplexy, cardiac infarction, inflammation and arteriosclerosis, which are associated with coagulation factors xa, IXa and thrombin
02/19/2004US20040034084 Side effect reduction; for treatment of AIDS, cancer and arthritis
02/19/2004US20040034081 Estrogen receptor modulators
02/19/2004US20040034025 Having a high residual activity, greater activity at lower application rates, curative activity, and a broader spectrum of efficacy; heterocyclic aromatic amides having a hydroxy group adjacent to the amide functionality
02/19/2004US20040033994 Use of compounds comprising a nitrogen-oxygen heterocycle
02/19/2004CA2495516A1 Compositions of a cyclooxygenase-2 selective inhibitor and a carbonic anhydrase inhibitor for the treatment of neoplasia
02/19/2004CA2495502A1 Methods for treating carbonic anhydrase mediated disorders
02/19/2004CA2495120A1 Oxadiazoles as modulators of metabotropic glutamate receptor-5
02/19/2004CA2495067A1 Mcp-1 receptor antagonists and method of use thereof
02/19/2004CA2493008A1 Aryl and heteroaryl compounds and methods to modulate coagulation
02/18/2004EP1389190A1 Diamide invertebrate pest control agents containing a non-aromatic heterocyclic ring
02/18/2004EP1119568B1 4,5-dihydro-isoxazole derivatives and their pharmaceutical use
02/18/2004CN1138765C Oxazolidinone antibacterial agents having thiocarbonyl functionality
02/18/2004CN1138764C Isoxazole derivatives
02/18/2004CN1138760C Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and TACE inhibitors
02/17/2004US6693124 3h-1,2,4-triazol-3-one or 3h-isooxazol-3-one derivatives; efficient fungicidal activity
02/17/2004US6693123 (4-(3-pyridylaminomethylene)-2-phenylbenzoyl)-n -methylmethionine, methyl ester for example; restenosis, hyperplasia
02/12/2004WO2003096979A3 Drug therapy for celiac sprue
02/12/2004WO2002058698A3 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators
02/12/2004US20040030132 Anticancer agents; arterosclerosis; bone disorders; antiarthritic agents; vision defects
02/12/2004US20040029946 Topical applying
02/12/2004US20040029941 Zonisamide use in obesity and eating disorders
02/12/2004US20040029933 Substituted phenylacetic acids
02/12/2004US20040029871 Pharmaceutical compounds for treating copd
02/11/2004EP1387831A1 Substituted arylketones
02/11/2004EP1387825A1 Thyroid hormone receptor antagonists for cardiac & metabolic disorders ii
02/11/2004EP0901479B1 Isoxazole derivatives and their use as herbicides
02/11/2004EP0797567B1 Novel amino acid derivatives with improved multi-drug resistance activity
02/11/2004CN1137888C Inhibitor of cysteninyl aspartic acid proteinase
02/10/2004US6689787 Method of using an integrin antagonist and radiation therapy as combination therapy in the treatment of neoplasia
02/10/2004US6689771 Amide derivatives as inhibitors of matrix metalloproteinases, TNF-α, and aggrecanase
02/05/2004WO2004011448A1 Therapeutic compounds for treating dyslipidemic conditions
02/05/2004WO2004011444A2 Novel method for preparing styryl pyrazole, isoxazole and isothiazole derivatives
02/05/2004WO2004010995A1 Fused heteroaryl derivatives for use as p38 kinase inhibitors in the treatment of i.a. rheumatoid arthristis
02/05/2004WO2003075857A3 Amino-methyl substituted tetracycline compounds
02/05/2004US20040024059 Novel pleuromutilin derivatives
02/05/2004US20040024038 GABA enhancers in the treatment of diseases relating to reduced neurosteroid activity
02/05/2004US20040023999 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
02/05/2004US20040023806 Agrochemicals in agriculture for controlling acarids and insects and for preventing the infestation of crop plants by phytopathogenic fungi.
02/04/2004EP1386912A1 Cyclic amidine derivative
02/04/2004EP0992503B1 Process for producing isooxazolidinedione compound
02/03/2004US6686493 Antiproliferation agent; antiinflammatory agents; side effect reduction
02/03/2004US6686353 Diarylalkyl cyclic diamine derivatives as chemokine receptor antagonists
01/2004
01/29/2004WO2004009552A1 Phosphodiesterase 4 inhibitors, including n-substituted aniline and diphenylamine analogs
01/29/2004WO2004009017A2 Modulators of the glucocorticoid receptor and method
01/29/2004US20040019113 Phosphate transport inhibitors
01/29/2004US20040019059 Drugs such as N-(4-benzoylphenyl)-4,5-dihydro-3-(3-pyridinyl)-5-isoxazolecarboxamide, used as antiinflammatory or antiarthritic agents
01/29/2004CA2492907A1 Phosphodiesterase 4 inhibitors, including n-substituted aniline and diphenylamine analogs
01/28/2004EP1384722A1 Process for the production of 2-(5-methyl-4-oxazolyl)acetates
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