Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
09/2003
09/03/2003EP1340749A1 Isoxazole derivatives
09/03/2003EP1070065B1 Azabicyclic 5ht1 receptor ligands
09/03/2003EP0975588B1 Antipicornaviral compouds, compositions containing them, and methods for their use
09/03/2003EP0612318B1 Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics
09/03/2003CN1440383A PPARγ调制剂 PPARγ modulators
09/03/2003CN1120160C Isoxazole and cortonamide derivatives and their use as pharmaceuticals and disgnositics
09/02/2003US6613790 Prodrugs of COX-2 inhibitors
09/02/2003US6613771 Prevent human retroviral reproduction, infections
09/02/2003US6613719 Agricultural herbicides; acylation
08/2003
08/28/2003WO2003070690A2 Novel amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative
08/28/2003US20030162813 Heterocyclic nitrogen comppounds such as 4-(5-methyl-3-phenyl-isoxazol-1-yl)benzenesulfonamide, used as non-steroidal antiinflammatory agents or antiarthritic agents; cyclooxygenase inhibitors
08/28/2003CA2474785A1 Novel amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative
08/27/2003EP1338644A1 Concentrated aqueous solutions of betains or amine oxides
08/27/2003EP1337247A1 Gaba enhancers in the treatment of diseases relating to reduced neurosteroid activity
08/27/2003EP1073672B1 Antipicornaviral compounds, their preparation and use
08/27/2003EP0874809B1 Carbamoyloxy derivatives of mutiline and their use as antibacterials
08/27/2003CN1439002A Muscarinic agonists
08/27/2003CN1438995A Method for producing 4-bromine-aniline derivatives
08/27/2003CN1438887A 水性液体制剂 The aqueous liquid preparation
08/27/2003CN1438221A Isooxazole-azo-diketo metal azo-chelate and preparation method
08/26/2003US6610858 Antagonists of the platelet glycoprotein IIb/IIIa fibrinogen receptor complex; thrombolytic agents
08/26/2003US6610846 Heteroaromatic glucokinase activators
08/26/2003US6610718 And dosage forms for treating rheumatoid arthritis
08/21/2003WO2003068170A2 Enzyme treatment of foodstuffs for celiac sprue
08/21/2003WO2002002512A3 Compounds to treat alzheimer's disease
08/21/2003US20030158252 Especially trypsin-like serine proteases, such as chymotrypsin, trypsin, thrombin, plasmin and factor Xa.
08/21/2003US20030158233 Compositions and methods for treating heart failure
08/21/2003US20030158205 N-benzyl-substituted, e.g., (2S)-1-(p-chlorophenoxy)methyl)-carbonyl-2-methyl-4-(p -fluorobenzyl)piperazine; inhibit the activity of the chemokines, MIP-1 alpha and RANTES
08/21/2003US20030158185 Novel use of phenylheteroakylamine derivatives
08/21/2003CA2475972A1 Enzyme treatment of foodstuffs for celiac sprue
08/20/2003EP1335909A1 3-nitroisoxazoles and their use in the protection of materials
08/20/2003EP1150944B1 N2-phenylamidine derivatives
08/20/2003EP0923542B1 Aryl substituted cyclic amines as selective dopamine d3 ligands
08/19/2003US6608209 Reacting a nitro-o-methylphenyl compound with an organic nitrite in presence of a base to give an oxime, cyclizing the oxime with an alkene in presence of a base to give an intermediate, reducing nitrogroup in presence of catalyst
08/19/2003US6608077 Il-8 receptor antagonists
08/19/2003CA2067404C Benzoisothiazole and benzoisoxazole-3-carboxamides a process for their preparation and their use as medicaments
08/14/2003WO2003066577A1 N-biphenylmethyl aminocycloalkanecarboxamide derivatives with a substiituent on the methyl useful as bradykinin antagonists
08/14/2003WO2003065789A2 N-biphenylmethyl aminocycloalkanecarboxamide derivatives
08/14/2003WO2003024955A3 Small molecule inhibitors of caspases
08/14/2003WO2003013655A3 Carbonic anhydrase inhibitors
08/14/2003US20030153801 Compositions of cyclooxygenase-2 selective inhibitors and radiation for inhibition or prevention of cardiovascular disease
08/14/2003US20030153606 Antiproliferative agents for treating adipocyte differentiation, cancer, osteoarthritis, rheumatoid arthritis, Crohn's Disease or Inflammatory Bowel Disease
08/14/2003CA2473778A1 N-biphenylmethyl aminocycloalkanecarboxamide derivatives
08/13/2003EP1334969A1 Process for preparation of 4-n-substituted amino-2-aza-1-oxabicyclo 3.3.0]oct-2-ene-6-carboxylic acid esters and process for preparation of their intermediates
08/13/2003EP1334083A2 1,4-disubstituted benzenes as insecticides
08/13/2003EP1242427B1 Novel piperidine and piperazine derivatives as p2x7 receptor antagonists
08/13/2003EP1216244B1 Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as D4 antagonists
08/13/2003EP1178987B1 Substituted benzoylisoxazoles and the use thereof as herbicides
08/13/2003EP0946539B1 Sulphonamide derivatives, process for their preparation, and their use as medicaments
08/13/2003CN1436168A Beta-amino acid nitrile derivs.
08/13/2003CN1117750C 3-heterocyclyl-substd. benzoyl derivs.
08/13/2003CN1117738C Endothelin antagonists
08/12/2003US6605632 Affinity for melatonin receptors
08/12/2003US6605631 Ortho-substituted 2-methoxyiminophenyl-N-methylacetamides
08/12/2003US6605626 Antithrombotic agents
08/12/2003CA2212836C Substituted isoxazoles for the treatment of inflammation
08/07/2003WO2003063797A2 Cycloalkyl inhibitors of potassium channel function
08/07/2003WO2002002593A3 Modulators of cellular proliferation and angiogenesis, methods for use and identification thereof
08/07/2003US20030149276 Preparation of -4-thioalkybrobenzene derivatives
08/07/2003US20030149078 For therapy of cyclooxygenase-2 mediated disorders, cancer
08/07/2003US20030149020 For therapy or prophylaxis of obesity, type II diabetes, or disorders of the central nervous system
08/07/2003US20030149019 For therapy or prophylaxis of obesity, type II diabetes, or disorders of the central nervous system
08/07/2003US20030146420 Organic dye molecules and nonlinear optical polymeric compounds containing chromophores
08/07/2003CA2474451A1 Cycloalkyl inhibitors of potassium channel function
08/06/2003EP1332131A2 Acid derivatives useful as serine protease inhibitors
08/06/2003CN1434827A 新的哌啶和哌嗪衍生物 The new piperidine and piperazine derivatives
08/06/2003CN1434712A Nitrosated and nitrosylated cyclooxygenase-2 inhibitors compositions and methods of use
08/06/2003CN1117092C Azadicyclic compound, its medicinal composition and medicinal use
08/05/2003US6603017 Preparation of 2-alkyl-3-(4,5-dihydroisoxazol-3-yl) halobenzenes
08/05/2003US6603012 RAR selective retinoid agonists
07/2003
07/31/2003WO2002030863A3 Ether compounds and compositions for cholesterol management and related uses
07/31/2003US20030144527 Novel sulfonation method for zonisamide intermediate in zonisamide synthesis and their novel crystal forms
07/31/2003US20030144332 Diarylcycloalkyl derivatives, processes for their preparation and their use s pharmaceuticals
07/30/2003EP1330233A1 Method of treating stroke
07/30/2003EP1066270B1 Isoxazole derivatives and their use as herbicides
07/29/2003US6600052 With a ring cyclizing reagent to form the compound of Formula V to yield a compound of Formula V: inhibitors of the cyclooxygenase- II enzyme. and antiinflammatory agents and analgesic pharmaceutical agents.
07/29/2003US6599904 Sulphonamide derivatives, process for their preparation, and their use as medicaments
07/29/2003US6599860 Methods for controlling undesirable vegetation using the compounds
07/29/2003CA2076555C Pharmaceuticals for the treatment of rejection reactions in organ transplantations
07/29/2003CA2048959C 3-(1,2-benzisoxazol-3-yl)-4-pyridinamines and derivatives
07/24/2003WO2003059900A1 Coumarin derivatives, process for their production and use thereof
07/24/2003WO2003059346A1 Beta-secretase inhibitors
07/24/2003WO2003059258A2 Compositions and methods for treating heart failure
07/24/2003WO2003059064A1 Insecticides containing hydrazone derivatives as the active ingredient and novel hydrazone derivatives
07/24/2003US20030139606 Process for preparing 5-methylisoxazole-4-carboxylic- (4'-trifluoromethyl)-anilide
07/24/2003US20030139425 Piperazine derivatives and their use as anti-inflammatory agents
07/24/2003US20030139404 N-monoacylated derivatives of o-phenylenediamines, their analogs and their use as pharmaceutical agents
07/24/2003US20030139379 Autoimmune disease, osteoporosis, rheumatic diseases, skin disorders
07/24/2003CA2473441A1 Beta-secretase inhibitors
07/24/2003CA2472419A1 Coumarin derivatives, process for their production and use thereof
07/23/2003EP1329457A2 Antipicornaviral compounds, their preparation and use
07/23/2003EP1328523A2 Methods for the preparation of biphenyl isoxazole sulfonamides
07/23/2003EP0888278B1 Antidiabetic agents
07/23/2003CN1431201A Producing technique for preparing 5-methyl-3-amido isoxazole
07/22/2003US6596716 2-propane-sulphonamide derivatives
07/17/2003WO2003057225A2 Phosphate transport inhibitors
07/17/2003WO2003057215A1 Neurotrophic factor production/secretion accelerator
07/17/2003US20030134874 Multicyclic compounds which inhibit leukocyte adhesion mediated by VLA-4
07/17/2003US20030134859 Substituted 2-chloro-5-nitrobenzamides; treating retrograde osteoporosis and diabetes mellitus
07/16/2003EP1326822A2 Ketone compounds and compositions for cholesterol management and related uses
1 ... 53 54 55 56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 ... 115