Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
07/2003
07/16/2003EP0832076B1 Novel isoxazoline and isoxazole fibrinogen receptor antagonists
07/16/2003CN1430602A Ary-and heteroaryl sulfonates compounds
07/16/2003CN1430596A New gamma selective retinoids
07/15/2003US6593363 The present invention relates to diterpene derivatives prepared from the components which are extracted from Acanthopanax Koreanum and represented by Chemical Formula (1).
07/10/2003WO2003055847A1 Carboxylic acid derivative
07/10/2003WO2003032908A3 Novel prodrugs of n-h bond-containing compounds and methods of making thereof
07/10/2003US20030130520 Producing substituted 2-nitro-guanidine derivatives.
07/10/2003US20030130236 Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs
07/10/2003US20030130204 Antipicornaviral compounds and compositons, their pharmaceutical uses, and materials for their synthesis
07/10/2003CA2482392A1 Carboxylic acid derivative
07/09/2003CN1429210A Substituted thioacetamides
07/09/2003CN1429198A Novel phenyl-proparylether derivatives
07/09/2003CN1429108A 磷酸盐运输抑制剂 Phosphate transport inhibitor
07/08/2003US6589956 Its enantiomers, diastereoisomers, and addition salts thereof with a pharmaceutically acceptable acid or base, and medicinal products containing the same which are useful as a TXA2 receptor antagonist and 5-HT2 receptor antagonist.
07/08/2003US6589949 3-oxo-2,1-benzisoxazol-1(3H)-carboxamides for treatment of CNS diseases
07/08/2003US6589914 Dihalopropene compounds, insecticidal/acaridcidal agents containing same, and intermediates for their production
07/03/2003WO2003053927A1 Piperazine derivative
07/03/2003WO2003053912A1 α-(N-SULPHONAMIDO)ACETAMIDE DERIVATIVES AS β-AMYLOID INHIBITORS
07/03/2003WO2003053368A2 Chalcone derivatives and their use to treat diseases
07/03/2003WO2003053352A2 Therapeutic compounds for treating dyslipidemic conditions
07/03/2003US20030125383 For treating or preventing emphysema, cancer and dermatological disorders
07/03/2003CA2470931A1 Chalcone derivatives and their use to treat diseases
07/03/2003CA2470808A1 Piperazine derivative
07/03/2003CA2470591A1 Therapeutic compounds for treating dyslipidemic conditions
07/02/2003EP1322598A1 Nitroso diphenylamine derivatives
07/02/2003CN1427718A Pharmaceutical compounds for treating COPD
06/2003
06/26/2003WO2003051842A2 Compositions decreasing activity of hormone-sensitive lipase
06/26/2003WO2003051841A2 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
06/26/2003WO2003002491A3 ENANTIOSELECTIVE TRANSFORMATION OF α, β-UNSATURATED ALDEHYDES USING CHIRAL ORGANIC CATALYSTS
06/26/2003US20030119914 Bis(thio-hydrazide amide) compounds; anticancer agents
06/26/2003US20030119876 Compounds for the treatment of protozoal diseases
06/26/2003US20030119814 Novel prodrugs of N-H bond-containing compounds and methods of making thereof
06/26/2003CA2468413A1 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
06/25/2003EP1025086B1 Benzamidine derivatives as factor xa inhibitors
06/24/2003US6583141 T cell mediated rheumatic diseases
06/24/2003US6583090 Hetaryl-substituted benzyl phenyl ethers, method for the production thereof, and their use for combating harmful fungi and animal pests
06/24/2003CA2126337C 2-amino-1,3-propanediol compound and immunosuppressant
06/19/2003US20030114682 Novel sulfonation method for zonisamide intermediate in zonisamide synthesis and their novel crystal forms
06/19/2003US20030114505 Novel isoxazole and thiazole compounds and use thereof as drugs
06/19/2003US20030114499 Antiarrhythmic agents for the treatment and prophylaxis of atrial arrhythmias, atrial fibrillation (AF) or atrial flutter; potassium channel modulators, beta-blocker
06/19/2003US20030114447 Controlling apoptosis; central nervous system disorders
06/19/2003US20030114441 Heterocyclic anti-epileptogenic agents and methods of use thereof
06/18/2003EP1318976A2 Substituted aminopropoxyaryl derivatives useful as agonists for lxr
06/18/2003EP0819125B1 Thienyl-, furyl-, pyrrolyl- and biphenylsulfonamides and derivatives thereof that modulate the activity of endothelin
06/17/2003US6579880 Isoxazoles and oxadiazoles as anti-inflammatory inhibitors of IL-8
06/12/2003WO2002064094A3 2-aryloxy-2-arylalkanoic acids for diabetes and lipid disorders
06/12/2003WO2002017712A3 Disubstituted benzenes as insecticides
06/12/2003US20030109718 Enantioselective transformation of alpha, beta-unsaturated aldehydes using chiral organic catalysts
06/12/2003US20030109715 3,4-Dihydro-1H-naphthalene derivatives as a highly selective cyclooxygenase-2 inhibitor
06/12/2003US20030109559 N-(3-amino-2-hydroxy-propyl)substituted alkylamide compounds
06/12/2003US20030109533 New benzenesulphonamide compounds
06/12/2003US20030109527 Novel hydroxy diphenylurea sulfonamides, compositions and intermediates thereof. The hydroxy
06/12/2003US20030109459 Activity as inhibitors of binding between VCAM-1 and cells expressing VLA-4. Such compounds are useful for treating diseases whose symptoms and/or damage are related to the binding of VCAM-1 to cells expressing VLA-4.
06/11/2003EP1317424A2 Polyamine analogues as therapeutic and diagnostic agents
06/11/2003EP1021413B1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
06/11/2003EP0996614B1 Acrylonitrile compounds, process for their production and pesticides containing them
06/10/2003US6576786 Reacting an n-protected carboxy-amine-cyclopentane derivative with a nitrile oxide followed by salt formation, desalting, decyclization, deprotecting and amidation
06/10/2003US6576780 Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors
06/10/2003US6576730 For the polymerization of unsaturated vinyl and/or vinylidene monomers
06/10/2003CA2055670C Retroviral protease inhibiting compounds
06/05/2003WO2003045382A1 Therapeutic compounds for treating dyslipidemic conditions
06/05/2003WO2002048124A3 Piperazine derivatives
06/05/2003US20030105334 Such as valdecoxib, parecoxib (sodium), and 4-(5-methyl-3-phenylisoxazol-4-yl)benzenesulfonyl chloride; reacting 3,4-diphenyl- 5-methyl-isoxazole compound with halosulfonic acid and trifluoroacetic acid, and then reacting with ammonia
06/05/2003US20030105144 Celecoxib dissolving in polyethylene glycol; antiinflammatory agents, osteoporosis, respiratory system disorders, antitumor agents, analgesics
06/05/2003US20030105142 Amide derivatives useful as inhibitors of the production of cytokines
06/05/2003US20030105141 Mixture containing fatty acid and aromatic amine; administering by mouth; cyclooxygenase enzyme inhibitor
06/05/2003US20030105066 For use in producing antiviral, antifungal and antibacterial medicaments
06/05/2003CA2467165A1 Therapeutic compounds for treating dyslipidemic conditions
06/04/2003EP1315706A1 Heterocyclically substituted benzoylcyclohexanediones, methods for producing them and their use as herbicides
06/04/2003EP1315500A1 Pharmaceutical compositions for topical delivery of cyclooxygenase-2 enzyme inhibitors
06/03/2003US6573287 2,1-oxazoline and 1,2-pyrazoline-based inhibitors of dipeptidyl peptidase IV and method
06/03/2003US6573266 Piperazine derivatives and their use as anti-inflammatory agents
06/03/2003CA2053954C Process for the preparation of nitroguanidine derivatives
05/2003
05/29/2003US20030100594 Carbonic anhydrase inhibitor
05/29/2003US20030100590 3-(4,5-dihydroisoxazol-5-yl)benzoylpyrazole
05/29/2003US20030100585 For example 3-(2-(1-(2-(3-Methoxy-4-(3-o-tolyl-ureido)-phenyl)-acetylamino )- 3-methyl-butyl)-4,5-dihydro-oxazol-5-yl)-2-methyl-propionic acid
05/27/2003US6569897 Alkenyldiarylmethane non-nucleoside HIV-1 reverse transcriptase inhibitors
05/27/2003US6569879 Agonists of peroxisome proliferator activated receptor (PPAR) alpha and/or gamma; benzisoxazole compounds; e.g. ((5,7-dipropyl-3-trifluoromethyl-1,2-benzisoxazol-6-yl)oxy)acetic acid, methyl ester
05/27/2003US6569874 Such as 2-acetylamino-4-(3-amidinophenyl)-5-((2'-amino-sulfonyl-(1,1')-biphen-4 -yl)aminocarbonyl)thiazole; for treatment of thromboembolic disorders
05/22/2003WO2003042193A1 Process for preparing 5-methylisoxazole-4-carboxylic-(4'-trifluoromethyl)-anilide
05/22/2003WO2003042168A1 NOVEL α-OXYGENATED OR α-THIOLATED CARBOXYLIC ACID PHENETHYLAMIDE DERIVATIVES
05/22/2003WO2003042167A1 NOVEL α-OXYGENATED OR α-THIOLATED CARBOXYLIC ACID PENETHYLAMIDE DERIVATIVES
05/22/2003WO2003041728A1 Novel phenyl-propargylether derivatives
05/22/2003WO2003024943A3 Aryl derivatives for the treatment of diabetes, hyperlipidemia, hypercholesterolemia and atherosclerosis
05/22/2003US20030096858 The parent drug compound is modified by forming one or more of predetermined chemical arrangement within parent drug structure for programming specific course and rate of metabolism for drug that leads to inactive nontoxic metabolite
05/22/2003US20030096844 Cannabinoid receptor ligands
05/22/2003US20030095992 Altering a drug's distribution, metabolism and elimination properties, especially by modifying with aralkyl ester moieties to increase rate of metabolism to inactive and nontoxic metabolites when exposure is halted; surgery, riots
05/22/2003CA2464775A1 Novel alpha-oxygenated or alpha-thiolated carboxylic acid phenethylamide derivatives
05/21/2003EP1312601A1 Carboxylic acid derivatives, process for producing the same and drugs containing the same as the active ingredient
05/21/2003EP1311475A1 Novel aminocyclohexane derivatives
05/21/2003EP1311469A1 Method for producing beta- ketoenol esters
05/21/2003CN1419450A Nitrite salts of antimicrobial agents
05/21/2003CN1418870A 3,4-dibidro-1H-anphthalene derivatives used as high selectivity inhibitor of cyclooxygenase-2
05/21/2003CN1109030C Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
05/20/2003US6565997 Superior in vibration transmittability between ceramic substrate and piezoelectric
05/20/2003CA2110693C Amino acid derivative anticonvulsant
05/15/2003WO2003040113A1 3-amido-1,2-benzoisoxazole derivatives, process for preparation, and use thereof
05/15/2003WO2003040112A1 Substituted diphenyl heterocycles useful for treating hcv infection
05/15/2003WO2003040096A2 N, n'-substituted-1,3-diamino-2-hydroxypropane derivatives
05/15/2003WO2003040086A1 5-amidino-2-hydroxybenzenesulfonamide derivatives, medicinal compositions containing the same, medicinal use thereof and intermediates in the production thereof
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