Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
03/2002
03/20/2002EP1187827A1 Antiviral agents
03/20/2002EP0944590B1 Aminoguanidines and alkoxyguanidines as protease inhibitors
03/20/2002CN1341124A Anti-CD3 immunotoxins and therapeutic use thereof
03/20/2002CN1341106A Process crystallising N-(4-trifluoromethylphenyl)-5-methyl-isoxazole-4-carboxamide
03/19/2002US6359143 Heterocycle-bearing thio phenol compounds, intermediates for the preparation of the same and processes for the preparation of both
03/19/2002US6358983 Heterocyclically substituted α-hydroxycarboxylic acid derivatives, method for producing the same and their use as endothelin receptor antagonists
03/19/2002CA2079548C Carbamate derivatives of 4-amino-3- isoxazolidinones, 3-amino-1- hydroxypyrrolidin-2-ones and 1-amino-1- cyclopropanecarboxylic acid analogs, a process for their preparation and their use as medicaments
03/14/2002WO2001070673A3 CYCLIC β-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-$g(a)
03/14/2002US20020032237 Antipicornaviral compounds, compositions containing them, and methods for their use
03/14/2002US20020032227 Oxime derivative and bactericide containing the same as active ingredient
03/14/2002DE10043075A1 Heterocyclyl-substituierte Benzoylcyclohexandione, Verfahren zu ihrer Herstellung und ihre Verwendung als Herbizide Heterocyclyl-substituted benzoylcyclohexanediones, process for their preparation and their use as herbicides
03/12/2002US6355807 Multistep process including cyanomethylation, reduction, cyclization, deprotection, oxidation, olefination and amidation
03/12/2002US6355796 Reacting beta-amino-beta-(perfluoroalkyl)acrylate compound with base and carbamoyl chloride compound to form urea compound, reacting urea compound with phosphorus pentahalide or oxalyl halide
03/12/2002US6355673 Substituted diaminocarboxylic acids
03/12/2002US6355662 Peptide and nonpeptides autoimmune diseases, antiinflammatory agents
03/07/2002WO2002018352A1 Heterocyclically substituted benzoylcyclohexanediones, methods for producing them and their use as herbicides
03/07/2002WO2002017923A1 Pharmaceutical compositions for topical delivery of cyclooxygenase-2 enzyme inhibitors
03/07/2002WO2002017712A2 Disubstituted benzenes as insecticides
03/07/2002WO2001068033A3 Il-8 receptor antagonists
03/07/2002US20020028834 Heterocyclic-cyclic amine derivatives
03/07/2002US20020028774 C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cysteine proteases
03/07/2002CA2420804A1 Pharmaceutical compositions for topical delivery of cyclooxygenase-2 enzyme inhibitors
03/06/2002EP1183233A2 Bradykinin receptor antagonists
03/06/2002EP1183232A2 Monofluoroalkyl derivatives
03/06/2002EP1183019A2 Ace-2 inhibiting compounds and methods of use thereof
03/05/2002CA2206122C Arylacrylamide derivatives
02/2002
02/28/2002WO2002016311A1 Carboxylic acid derivatives, process for producing the same and drugs containing the same as the active ingredient
02/28/2002WO2002016305A1 METHOD FOR PRODUCING β KETOENOL ESTERS
02/28/2002WO2002015884A2 Rapidly disintegrating oral formulation of a cyclooxygenase-2 inhibitor
02/28/2002WO2001046200A8 Novel piperidine and piperazine derivatives
02/28/2002US20020026060 RAR selective retinoid agonists
02/28/2002US20020025963 Novel guanidine mimics as factor Xa inhibitors
02/28/2002US20020025910 3-heterocycly1 - substituted benzoyl derivatives
02/28/2002CA2419592A1 Rapidly disintegrating oral formulation of a cyclooxygenase-2 inhibitor
02/26/2002US6350749 Aminoguanidine hydrazone derivatives, process for producing the same and drugs thereof
02/21/2002WO2002014267A1 Novel aminocyclohexane derivatives
02/21/2002WO2002013822A1 Micronized leflunomide
02/21/2002WO2001081328A3 Thiazolidinedione analogues and their use for the treatment of diabetes
02/21/2002WO2001072960A3 Il-8 receptor antagonists
02/21/2002US20020022724 Organic initiators and their use in the polymerization of unsaturated monomers
02/21/2002US20020022646 Method for systhesizing leflunomide
02/21/2002US20020022623 A substituted hydroxyethylene compound useful for treating Alzheimer's disease, mild cognitive impairment, Down's syndrome, herediatary cerebral hemmorrhage with amyloidosis, degenerative dementia
02/19/2002CA2025939C Carboxamides of isoxazole- and isothiazole-carboxylic acids
02/14/2002US20020019412 Antidiabetic agents
02/14/2002US20020019403 Inhibit amyloid protein deposits
02/13/2002EP1178987A1 Substituted benzoylisoxazoles and the use thereof as herbicides
02/12/2002US6346517 Synergy between low molecular weight heparin and platelet aggregation inhibitors, providing a combination therapy for the prevention and treatment of various thromboembolic disorders
02/07/2002US20020016461 Biphenyl and biphenyl-analogous compounds as integrin antagonists
02/07/2002US20020016361 Beta-amino acid nitrile derivatives as cathepsin K inhibitors
02/07/2002US20020016342 Combination therapy using COX-2 selective inhibitor and thromboxane inhibitor and compositions therefor
02/07/2002US20020016336 Treatment of rheumatoid and osteoarthritis, corneal, epidermal or gastric ulceration, tumor metastasis or invasion, periodontal disease and bone disease
02/07/2002US20020016323 Oxazolidinone antibacterial agents having a thiocarbonyl functionality
02/06/2002EP1177193A1 Process for the preparation of 6-(perfluoroalkyl)uracil compounds
02/06/2002EP1177176A1 Tri-aryl acid derivatives as ppar receptor ligands
02/06/2002CN1334801A Biphenyl and biphenyl-analogous compounds as integrin antagonists
02/06/2002CN1334798A Phenylglycine derivatives
02/06/2002CN1334726A Hydroxy diphenyl urea sulfonamides as IL-8 receptor antagonists
02/05/2002US6344471 Diisopropyl fluorophosphate (dfp), treatment of cognitive disorders, depression, schizophrenia and anxiety.
02/05/2002CA2123403C Acyclic ethylenediamine derivatives as substance p receptor antagonists
01/2002
01/31/2002US20020013357 Valdecoxib compositions
01/30/2002EP1175214A2 Cyclooxygenase-2 inhibitor compositions having rapid onset of therapeutic effect
01/30/2002EP0907634B1 Pesticides
01/30/2002CN1333769A Thiourea inhibitors of herps viruses
01/30/2002CN1333750A Acetamide and substituted acetamide-containing thiourea inhibitors of herpes viruses
01/29/2002US6342610 Compounds such as n-(4-bromo-3-methyl-5-isoxazolyl)-2-n-benzylbenzo(b)thiophene-3-sufonamide administered as endothelin peptide receptor antagonists
01/29/2002US6342513 Oxazolidinone antibacterial agents having a thiocarbonyl functionality
01/24/2002WO2002006276A1 Beta3 adrenergic agonists
01/24/2002WO2002006213A2 Oxygenated esters of 4-iodo phenylamino benzhydroxamic acids
01/24/2002WO2002006211A1 Preparation of 4-thioalkylbromobenzene derivatives
01/24/2002WO2002006189A2 Aniline derivatives
01/24/2002WO2002005848A2 Use of cox-2 inhibitors in the treatment and prevention of ocular cox-2 mediated disorders
01/24/2002WO2002005815A1 Ophthalmic formulation of a selective cyclooxygenase-2 inhibitory drug
01/24/2002WO2000053168A3 Synergy between low molecular weight heparin and platelet aggregation inhibitors, for preventing and treating thromboembolic disorders
01/24/2002WO2000045799A3 Use of substituted isoxazol carboxylic acids and derivatives and novel substances
01/24/2002US20020010343 Compounds having IgE affecting properties
01/24/2002CA2416722A1 Preparation of 4-thioalkylbromobenzene derivatives
01/24/2002CA2415331A1 Beta3 adrenergic agonists
01/24/2002CA2414780A1 Ophthalmic formulation of a selective cyclooxygenase-2 inhibitory drug
01/24/2002CA2414674A1 Use of cox-2 inhibitors in the treatment and prevention of ocular cox-2 mediated disorders
01/23/2002EP1174429A1 Process for the preparation of (e)-3-(1-propenyl)isoxazoline
01/23/2002EP1173183A2 Use of compounds with a nitrogen-oxygen heterocycle
01/23/2002CN1078202C Method of preparing essentially pure isomers of alpha-bis-oximes
01/22/2002CA2024956C Isoxazoles herbicides
01/17/2002WO2002004407A2 7-substituted tetracycline compounds
01/17/2002US20020006951 Solid-state form of celecoxib having enhanced bioavailability
01/17/2002US20020006945 Immunology diseases
01/17/2002DE10032874A1 New 4-substituted 3,5-dialkyl-isoxazole derivatives, useful as antiviral agents having strong activity against hepatitis B virus and low cytotoxicity
01/16/2002EP1171427A1 Process for the preparation of 6-(perfluoroalkyl) uracil compounds from urea compounds
01/16/2002EP0882028B1 New intermediates to pesticides
01/15/2002US6339099 Guanidine mimics as factor Xa inhibitors
01/10/2002WO2002002593A2 Modulators of cellular proliferation and angiogenesis, methods for use and identification thereof
01/10/2002WO2002002555A1 Novel isoxazolinone antibacterial agents
01/10/2002WO2002002537A1 Method for producing 4-bromine-aniline derivatives
01/10/2002WO2002002512A2 Compounds to treat alzheimer's disease
01/10/2002CA2410651A1 Compounds to treat alzheimer's disease
01/09/2002EP1169312A2 Glucokinase activators
01/09/2002EP1169308A1 Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils
01/09/2002CN1330631A Amide derivatives which are useful as cell factor inhibitors
01/09/2002CN1329827A 3-hydroxy-5-methyl-isoxazole pesticide composition and using method
01/03/2002WO2002000651A2 Factor xa inhibitors
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