Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
01/2004
01/27/2004US6683215 N-(4-carbamimidoyl-phenyl)-glycine derivatives
01/27/2004US6683211 Fungicides for crops
01/27/2004US6683201 Analine derivatives as OSC inhibitors
01/27/2004US6683104 Cholesterol and triglyceride-modulating drugs and methods
01/27/2004US6683103 Sulfonamides containing oxazole and substituted thiophene rings, useful for treating hypertension, cardiovascular disease, asthma, pulmonary hypertension, inflammatory diseases, vision defects, menstrual disorders, renal failure
01/22/2004WO2004006834A2 Leflunomide analogs for treating rheumatoid arthritis
01/22/2004WO2003080545A3 Substituted phenylacetic acids
01/22/2004US20040014983 Chlorinating benzisoxazole methane sulfonic acid with thionyl chloride to form an intermediate of benzisoxazole methane sulfonamide
01/22/2004US20040014968 Such as 2-(3-chloro-phenyl)-3-cyclopentyl-N-thiazol-2-yl-propionamide which increases insulin secretion in treatment of type II diabetes
01/22/2004US20040014796 Antiinflammatory agents; rheumatic diseases; antitumor agents
01/21/2004EP1381590A1 3,4-di-substituted cyclobutene-1,2-diones as cxc-chemokine receptor ligands
01/21/2004EP1381369A1 Use of selective cox-2 inhibitors for the treatment of urinary incontinence
01/21/2004CN1469748A Pharmaceutical compositions for topical delivery of cyclooxygenase-2 enzyme inhibitors
01/20/2004US6680387 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis
01/20/2004US6680319 Treatment of obstructive syndromes of the lower urinary tract, including benign prostatic hyperplasia, treatment of lower urinary tract symptoms
01/20/2004US6680317 N-(phenyl)-n*-(2-hydroxy-3-aminosulfonylphenyl)guanidine derivatives; chemokine inhibitors; respiratory, cardiovascular, rheumatic, brain, and nervous system disorders
01/15/2004US20040009979 Use of compounds for the elevation of pyruvate dehydrogenase activity
01/14/2004EP1379513A1 Prodrugs of cox-2 inhibitors
01/14/2004EP1379279A1 Orally deliverable pharmaceutical composition comprising a drug of low water solubility (cox-2 inhibitor), a solvent, a fatty acid and an organic amine
01/14/2004EP1379136A1 Preparation of ketones from aldehydes
01/14/2004EP1155004B1 Method crystallising n-(4-trifluoromethylphenyl)-5-methyl-isoxazole-4-carboxamide
01/14/2004CN1468214A Novel derivatives of aminocyclohexane
01/14/2004CN1468211A Nitroso diphenylamine derivatives
01/14/2004CN1134411C Bicyclic amino derivatives and PGD2 antagonist containing same
01/13/2004US6677458 Process for the preparation of 1,2-benzisoxazole-3-acetic acid
01/13/2004US6677369 Antithrombotic agents
01/13/2004US6677360 Biphenyl and biphenyl-analogous compounds as integrin antagonists
01/08/2004WO2004002965A1 Arylcarbonylpiperazines and heteroarylcarbonylpiperazines and the use thereof for treating benign and malignant tumour diseases
01/08/2004WO2004002530A1 Remedy for chronic disease
01/08/2004WO2004002409A2 Cyclooxygenase-2 selective inhibitors, compositions and methods of use
01/08/2004WO2003077828A3 Novel florfenicol-type antibiotics
01/08/2004US20040006236 Diaminopropionic acid derivatives
01/08/2004US20040006100 Administering phenylacetic acid derivative for therapy of Parkinson's disease
01/08/2004US20040005637 Intermediate products coupled to solid polymeric support suitable for synthesis of heterocyclic compounds in simple and fast methods on solid phase; for synthesis of heterocycles with large structural diversity in high yields
01/08/2004CA2489428A1 Cyclooxygenase-2 selective inhibitors, compositions and methods of use
01/07/2004EP1377291A2 1-butyric acid derivatives such as carbomethoxypropionyl cyanide or leflunomide derivatives, and the therapeutic use thereof
01/07/2004EP1377290A2 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators
01/07/2004EP1377288A1 2,1-oxazoline and 1,2-pyrazoline-based inhibitors of dipeptidyl peptidase iv and method
01/06/2004US6673824 Phenyl sulfonamide endothelin antagonists
01/06/2004US6673818 Fluoro-substituted benzenesulfonyl compounds for the treatment of inflammation
01/06/2004US6673800 4,5,-dihydroisoxazolylakylpiperazine derivatives having selective biological activity at dopamine D3 or D4 receptor, and preparation thereof
01/06/2004US6673780 Such as 4-(4-(3-hydroxy-3-methyl-butane-1-sulfinylmethyl)-phenylmethanesulfinyl)-2 -methyl-butan1-ol for treating and preventing cardiovascular diseases, dyslipidemias, dysproteinemias, and glucose metabolism disorders
01/02/2004EP1375499A1 Process for the production of 2-(5-methyl-4-oxazolyl)ethanol derivatives
01/02/2004EP1375472A1 Benzene compound and salt thereof
01/02/2004EP1374871A1 Crystalline isoxazole derivative and medical preparation thereof
01/02/2004EP1373240A2 Retinoid x receptor modulators
01/02/2004EP1373229A1 Process for the preparation of 1,2-benzisoxazole-3-acetic acid
01/02/2004EP1373191A1 Acylated indanyl amines and their use as pharmaceuticals
01/02/2004EP1373158A2 Additives for building industry obtained from by-products and process for their production
01/02/2004EP1372655A2 Cathepsin cysteine protease inhibitors
01/02/2004EP1372645A1 Reconstitutable parenteral composition containing a cox-2 inhibitor
01/02/2004EP0836595B1 Triazoline and isoxazoline bis-oxime derivatives and their use as pesticides
01/01/2004US20040002539 Enzyme inhibitors; anticoagulants; blood collecting device
01/01/2004US20040002524 Cardiovascular disorders; osteoporosis; central nervous system disorders
01/01/2004US20040002522 Antiinflammatory agents; analgesics
01/01/2004US20040002491 Melatonergic receptors
01/01/2004US20040002490 Melatonergic receptors
12/2003
12/31/2003WO2004000817A2 Benzimidazole compounds and their use as estrogen agonists/antagonists
12/31/2003WO2003088959A3 Treatment of parkinson's disease with cyclooxygenase-2 (cox 2) inhibitor(s)
12/31/2003CA2487266A1 Benzimidazole compounds and their use as estrogen agonists/antagonists
12/31/2003CA2445515A1 Transcription factor modulating compounds and methods of use thereof
12/30/2003US6670482 Process and novel intermediates for preparing isoxazolin-3-ylacyl benzenes
12/30/2003US6670358 Substituted thioacetamides
12/30/2003US6668527 Non-peptidyl inhibitors of VLA-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
12/30/2003CA2088840C 4-benzoyl isoxazole herbicides
12/29/2003CA2433983A1 Aryl- and heteroarylcarbonylpiperazines and their use for the treatment of benign and malignant oncoses
12/25/2003US20030236438 Enantioselective 1,4-addition of aromatic nucleophiles to alpha,beta-unsaturated aldehydes using chiral organic catalysts
12/25/2003US20030236403 Certain substituted 1-aryl-3-piperazine-1'-yl propanones
12/25/2003US20030236294 Anticancer agents
12/25/2003US20030236287 Central nervous system disorders; analgesics; antiinflammatory agents; cognition activators; anticancer agents; antidiabetic agents
12/25/2003US20030236227 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis
12/24/2003WO2003084916A3 Compounds that modulate ppar activity and methods for their preparation
12/23/2003US6667404 Retroviral protease inhibiting compounds
12/23/2003US6667342 Benzenesulfonamide-derivatives and their use as medicaments
12/23/2003US6667333 Herbicidal 3-(4,5 dihydroisoxazole- 3 yl) substituted benzoycyclohexenone derivatives
12/23/2003US6667331 Non-peptidyl inhibitors of VLA-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
12/18/2003US20030232871 Crystalline parecoxib sodium
12/18/2003US20030232867 Comprises (2Z)-2-cyano-3-hydroxy-N-(4-(trifluoromethyl) phenyl)-2-hepten-6-ynamide for preventing/treating chronic rejection in a transplanted organ or tissue
12/18/2003US20030232863 Cathepsin cysteine protease inhibitors
12/18/2003US20030232802 Aryl and heteroaryl sulfonates
12/17/2003EP1370530A1 Acylated 1,2,3,4-tetrahydronaphthyl amines and their use as pharmaceutical
12/17/2003EP1370520A1 Aryl and biaryl compounds having mch modulatory activity
12/17/2003EP1226131B1 Isoxazolecarboxamide derivatives
12/16/2003CA2122633C 2-heterocyclicethylamine derivatives and their use as pharmaceuticals
12/11/2003WO2003101933A1 Intermediate products, methods for their preparation and use thereof
12/11/2003WO2003078392A3 Process for preparing crystalline form i of cabergoline
12/11/2003WO2002100825A3 Anthranilic acid amides with a heteroarylsulfonyl side chain, and use thereof as antiarrhythmic active substances
12/11/2003US20030229232 Herbicides
12/11/2003US20030229065 Measuring drug resistance, calibration; reducing antibiotic resistance
12/11/2003US20030229053 Compounds and methods for the treatment or prevention of flavivirus infections
12/11/2003CA2487659A1 Intermediate products, methods for their preparation and use thereof
12/10/2003EP1368358A1 Isoxazoline derivatives as anti-depressants
12/10/2003EP1368308A1 Cannabinoid receptor ligands
12/10/2003EP1056710B1 Diterpene derivatives and anti-inflammatory analgesic agents comprising the same
12/10/2003CN1461294A Method for producing beta ketoenol esters
12/10/2003CN1130361C Process for producing isooxazolidinedione compound
12/10/2003CN1130355C Thienyl-, furyl-, pyrrolyl-and biphenylsulfonamides and derivatives thereof modulate activity of endothelin
12/09/2003US6660466 Reacting reactive appendage compounds such as meta benzylic compounds or alpha-amide compounds with scaffold molecules having reactive functionalities and contacting the intermediate library with a reducing agent
12/09/2003CA2123697C Novel substituted salicylic acids
12/09/2003CA2022425C 1,3,4-oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents
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