Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
01/2003
01/23/2003WO2003006430A1 Taxol enhancer compounds
01/23/2003WO2003006429A1 Synthesis of taxol enhancers
01/23/2003WO2003006428A1 Taxol enhancer compounds
01/23/2003WO2003006423A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003US20030018200 Preparation of isoxazolin-3-ylacylbenzenes
01/23/2003US20030018013 Cardiovascular disorders; antilipemic agents; Alzheimer's disease
01/23/2003US20030017166 Combination preparation for the therapy of immunological diseases
01/23/2003CA2453503A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003CA2453415A1 Synthesis of taxol enhancers
01/23/2003CA2453175A1 Interaction inhibitors of tcf-4 with beta-catenin
01/22/2003EP1277729A1 Ppar (gamma) modulators
01/22/2003EP1276736A2 Regioselective synthesis of 3,4-di(carbocyclyl or heterocyclyl)thiophenes
01/22/2003EP1276730A2 Thiazolidinedione analogues and their use for the treatment of diabetes
01/22/2003EP0646115B1 Heterocyclic-cyclic amine derivatives
01/16/2003WO2003004147A2 Compound libraries
01/16/2003WO2002072527A3 1-butyric acid derivatives such as carbomethoxypropionyl cyanide or leflunomide derivatives, and the therapeutic use thereof
01/16/2003WO2002070467B1 Derivatives of diphenylurea, diphenyloxalic acid diamide and diphenylsulfuric acid diamide and their use as medicaments
01/16/2003US20030013881 Such as 4-((6-(3,5-difluoro-phenyl)-5-(S)-(3-dipropylcarb-amoyl-benzoyl-amino)-2-(R)-ethyl-4-(S)-hydroxy-hexanoylamino)-methyl)-cyclohexanecarboxylic acid for inhibiting secretase activity and cleavage of amyloid precursor protein
01/16/2003US20030013721 Antiinflammatory agents; immunology; cardiovascular disorders; rheumatic disorders
01/16/2003US20030013713 Compounds as PDE IV and TNF-inhibitors
01/15/2003EP1275644A1 Benzenesulfonamide derivatives, process for their preparation and pharmaceutical compositions containing them
01/15/2003EP1275641A2 Benzenesulfonamide derivatives, process for their preparation and pharmaceutical compositions containing them
01/15/2003EP1275638A1 Combination therapy for the treatment of immunological disorders
01/15/2003EP1275301A1 Trisubstituted heterocyclic compounds and their use as fungicides
01/15/2003EP0862571B1 Herbicidal sulfonamides
01/15/2003CN1391565A Benzophenones as inhibitors of reverse transcriptase
01/15/2003CN1391474A 5-membered heterocycle derivatives, production thereof and use as medicaments
01/15/2003CN1391469A Npyy5拮抗剂 Npyy5 antagonist
01/15/2003CN1098843C Isoxazoles
01/14/2003CA2252543C Benzene derivatives substituted by heterocycles and herbicides
01/09/2003WO2003002540A1 Cyclic diamine compound having five-membered cyclic group
01/09/2003WO2003002519A1 Phenol derivatives and their use in medicaments
01/09/2003WO2003002491A2 ENANTIOSELECTIVE TRANSFORMATION OF α, β-UNSATURATED ALDEHYDES USING CHIRAL ORGANIC CATALYSTS
01/09/2003US20030008915 Acylated 6,7,8,9-tetrahydro-5H-benzocycloheptenyl amines and their use as pharmaceutical agents
01/09/2003US20030008908 Isoxazoline compounds having MIF antagonist activity
01/08/2003EP1273572A1 Thiophene substituted piperazines useful in the treatment of benign prostatic hyperplasia
01/08/2003EP1272456A1 Hydrazide and alkoxyamide angiogenesis inhibitors
01/08/2003EP1272175A2 Il-8 receptor antagonists
01/08/2003EP0934286B1 3-alkoxyisoxazol-4-yl-substituted 2-amino carboxylic acid compounds
01/08/2003EP0889033B1 Alpha-substituted benzyl heterocyclic derivatives, intermediates for producing the same, and pesticides containing the same as active ingredient
01/08/2003CN1390211A Benzoic ester comprising ethoxyl acyl piperazine substituted oxazolidone compound
01/08/2003CN1390204A Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
01/08/2003CN1390193A Novel dicarboxylic acid derivatives with pharmaceutical properties
01/08/2003CN1098256C Substd. benzenesulfonamide derivatives as prodrugs of COX-2 inhibitors
01/06/2003CA2392187A1 Combination preparation for the therapy of immunological diseases
01/03/2003WO2003000249A1 Function regulator for retinoid relative receptor
01/02/2003US20030004212 Cyclohexylamine derivatives as subtype selective N-Methyl-D-Aspartate antagonists
01/02/2003US20030004200 Crystalline form of 4-[5-methyl-3-phenylisoxazol-4-YL] benzenesulfonamide
01/02/2003US20030004196 Antiinflamamtory agents; autoimmune disease
01/02/2003EP0934265B1 Amidinophenyl-pyrrolidines, -pyrrolines, and -isoxazolidines and derivatives thereof
12/2002
12/31/2002US6500863 Interleukin binding inhibitors such as n-(2-hydroxyl-3-amino sulfonyl-4-chlorophenyl)-n'-(2-bromophenyl)urea, used for prophylaxis of chemokine mediated diseases
12/31/2002US6500849 Administering antiinflammatory, antiproliferative, nootropic or antigrowth agents, such as 6-(1-dodecynyl)-2-pyridine-carboxaldehyde and enantiomorphs to mammals; alzheimers disease
12/27/2002WO2002102376A1 ORALLY DELIVERABLE PHARMACEUTICAL COMPOSITION COMPRISING AN ACTIVE COMPOUND HAVING AN AMINOSULFONYL GROUP (cox-2 INHIBITOR), A POLYETHYLENE GLYCOL AND A FREE-RADICAL SCAVENGING ANTIOXIDANT
12/27/2002CA2444356A1 Orally deliverable pharmaceutical composition comprising an active compound having an aminosulfonyl group (cox-2 inhibitor), a polyethylene glycol and a free-radical scavenging antioxidant
12/25/2002CN1387518A Heterocyclic substd, diphenyl leukotriene antagonists
12/25/2002CN1097049C Processes for preparing intermediate product used in method of diastereoselective synthesis of nucleosides
12/24/2002US6498275 Use of compounds for the elevation of pyruvate dehydrogenase activity
12/24/2002US6498255 Cholinesterase inhibitors; cognition activators; alzheimer's disease; e.g., 3-(2-(1-(phenylmethyl)-4-piperidinyl)ethyl)-1,2-benzisoxazole
12/24/2002US6498190 Bicyclic amino derivatives and PGD2 antagonist containing the same
12/24/2002US6498172 Prostaglandin agonists and their use to treat bone disorders
12/19/2002WO2002100846A1 Compounds and methods for the treatment or prevention of flavivirus infections
12/19/2002WO2002100825A2 Anthranilic acid amides with a heteroarylsulfonyl side chain, and use thereof as antiarrhythmic active substances
12/19/2002WO2002100332A2 Isoxazoline compounds having mif antagonist activity
12/19/2002WO2002070541A3 Peptide deformylase inhibitors
12/19/2002US20020193638 Method and apparatus for the preparation of ketones
12/19/2002US20020193596 Inhibitors of protein isoprenyl transferases
12/19/2002DE10128331A1 New 2-(heteroarylsulfonyl-amino)-benzamide derivatives, which are potassium ion channel blocking antiarrhythmic agents, useful for e.g. treating atrial fibrillation or flutter
12/18/2002EP1265849A2 Compounds and methods to treat alzheimer's disease
12/18/2002CN1096446C N-(ortho-substd-benzyloxy)imine derivs, and their use as fungicides, acaricides or insecticides
12/17/2002US6495696 First carboxylic acid or aldehyde or derivatives and a second carboxylic acid in the ratio of 1:2 to 1:20, passing through acatalytic bed at a temperature of 350-500 degrees c at weight hourly space velocity of > 2
12/17/2002US6495581 Drug for treating diabetes mellitus, hyperlipemia, impaired glucose tolerance, arterial sclerosis and improving insulin resistance, inflammatory disease
12/17/2002US6495580 Compounds, compositions and methods for treating or preventing pneumovirus infection and associated diseases
12/12/2002WO2002098849A2 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer’s disease and similar diseases
12/12/2002WO2002098840A1 Carboxylic acid derivative and medicine comprising salt or ester of the same
12/12/2002WO2002081398A3 Additives for building industry obtained from by-products and process for their production
12/12/2002US20020188133 Producing an isoxazolidinedione compound from beta - methyl L-aspartate via an important intermediate oxazolylethanol derivative
12/12/2002CA2448834A1 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer's disease and similar diseases
12/11/2002EP1264820A1 Novel amide compounds
12/11/2002EP1263755A2 Cyclic beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha
12/11/2002EP1263743A1 Heterocycle substituted diphenyl leukotriene antagonists
12/11/2002EP1263711A1 Novel use of phenylheteroalkylamine derivatives
12/11/2002EP0624155B2 Carbamates and plant-protecting agents containing them
12/11/2002CN1384825A Benzylidene thiazolidiones and analogues and their use in treatment of inflammation
12/11/2002CN1384744A Isoxazole derivatives to be used as phosphodiestesterase VII inhibitors
12/10/2002US6492423 Hepatitis c and b viricides
12/10/2002US6492396 Substituted thioacetamides
12/10/2002US6492368 Benzamidine derivatives as factor XA inhibitors
12/10/2002US6492362 Compounds and compositions as cathepsin S inhibitors
12/05/2002WO2002096884A2 Substituted benzoylketones as herbicidal agents for use as plant treatment agent
12/05/2002WO2002096882A1 Substituted anilide derivatives, intermediates thereof, agricultural and horticultural chemicals, and their usage
12/05/2002WO2002096516A1 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
12/05/2002WO2002096424A1 Hetereocyclic beta-aminoacids and their use as anti-epileptogenic agents
12/05/2002US20020183525 Process for the preparation of 1,2-benzisoxazole-3-acetic acid
12/05/2002US20020183367 2,1-Oxazoline and 1,2-pyrazoline-based inhibitors of dipeptidyl peptidase IV and method
12/05/2002US20020183362 2-Fluorobenzenesulfonyl compounds for the treatment of inflammation
12/05/2002US20020183342 For use as insecticides against a variety of insects, including larvae, such as tobacco budworm
12/05/2002US20020183334 For therapy of sleepiness, promotion of wakefulness, treatment of Parkinson's disease, cerebral ischemia, stroke, sleep apneas, eating disorders, stimulation of appetite and weight gain, treatment of attention deficit hyperactivity disorder
12/05/2002CA2448160A1 Heterocyclic beta-amino acids and their use as anti-epileptogenic agents
12/05/2002CA2447657A1 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
12/04/2002EP1261579A1 Dehydroamino acids
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