Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
01/1997
01/01/1997CN1138983A Preparation of drug composition
12/1996
12/27/1996WO1996041796A1 Bicyclolactam compounds, use of the same and intermediate in the production of the same
12/27/1996EP0749421A1 Sulphonamide derivatives as aspartyl protease inhibitors
12/24/1996US5587481 Preparation of (S)-decahydroisoquinoline-3-carboxylic acid t-butylamide
12/24/1996US5587479 Basic derivatives of glutamic acid and aspartic acid as gastrin or cholecystokinin antagonists
12/24/1996US5587385 Tyrosine kinase inhibitor
12/19/1996WO1996040647A1 α-(1,3-DICARBONYLENOL ETHER) METHYL KETONES AS CYSTEINE PROTEASE INHIBITORS
12/19/1996WO1996040640A1 BIPHENYL-2-CARBOXYLIC ACID-TETRAHYDRO-ISOQUINOLIN-6-YL AMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN AND/OR APOLIPOPROTEIN B (Apo B) SECRETION
12/19/1996WO1996040202A1 Synthesis of n-substituted oligomers
12/19/1996CA2223268A1 .alpha.-(1,3-dicarbonylenol ether) methyl ketones as cysteine protease inhibitors
12/18/1996EP0666736B1 Stabilization of fluorocarbon emulsions
12/18/1996CN1138325A Anellated dihydropyridines and their use in the production of pharmaceutical preparations
12/18/1996CN1138324A Anellated dihydropyridines and their use in the production of pharmaceutical preparations
12/18/1996CN1138322A 2,3-diaminopropionic acid derivative
12/17/1996US5585357 Heteroaryloxymethyl ketones as interleukin-1βconverting enzyme inhibitors
12/12/1996WO1996039383A1 Substituted benzene-fused hetero- and carbocyclics as neurokinin antagonists
12/12/1996WO1996039194A1 Novel cathepsin and methods and compositions for inhibition thereof
12/12/1996WO1996039142A1 Pharmaceutical composition comprising a proteinase inhibitor and a monoglyceride
12/12/1996CA2223239A1 Substituted benzene-fused hetero- and carbocyclics as neurokinin antagonists
12/12/1996CA2221684A1 Novel cathepsin and methods and compositions for inhibition thereof
12/10/1996US5583249 Pesticides
12/10/1996US5583238 Method for making intermediates useful in synthesis of retroviral protease inhibitors
12/05/1996WO1996038471A1 Dipeptides which promote release of growth hormone
12/04/1996EP0745066A1 Antimalarial korupensamines and pharmaceutical compositions and medical uses thereof
12/04/1996CN1137268A Amidino derivatives useful as nitric oxide synthase inhibitors
12/03/1996US5580999 Alcohols
12/03/1996US5580881 1,2,3,5,6,7,8,8a-Octahydro-5,5,8a-trimethyl-(8aβ)-6-isoquinolineamine derivatives, preparation method therefor and therapeutical use thereof
11/1996
11/28/1996WO1996037463A1 Process for producing n-methylmethoxyiminoacetamide derivatives and intermediates therefor
11/27/1996CN1136562A Estrogen excitant/antagonist
11/26/1996US5578730 Process for producing β-aminoalcohols compounds
11/26/1996US5578729 Dimeric arylisoquinoline alkaloid compounds
11/26/1996US5578601 Nonpeptide bradykinin antagonists
11/21/1996WO1996036611A1 3,4-disubstituted-phenylsulphonamides and their therapeutic use
11/19/1996US5576435 Process and intermediates for the preparation of excitatory amino acid receptor antagonists
11/19/1996US5576338 Bis (biaryl) compounds as inhibitors of leukotriene biosynthesis
11/19/1996US5576282 Color-safe bleach boosters, compositions and laundry methods employing same
11/14/1996WO1996035676A1 1,8-difluorisoquinoline derivatives and the use thereof in liquid crystalline mixtures
11/14/1996WO1996035675A1 1-fluor-5,6,7,8-tetrahydroisoquinoline derivatives and their use in liquid crystal mixtures
11/14/1996WO1996035674A1 1-fluorisoquinoline derivatives and the use thereof in liquid crystalline mixtures
11/14/1996WO1996035673A1 1-fluor-6,7-dihydro-5h-isoquinoline-8-one-derivatives and the use thereof in liquid crystalline mixtures
11/14/1996WO1996035672A1 Trifluortetrahydro-isoquinoline derivatives and the use thereof in liquid crystalline mixtures
11/14/1996DE19517060A1 1-Fluorisochinolinderivate und ihre Verwendung in flüssigkristallinen Mischungen 1-Fluorisochinolinderivate and their use in liquid crystal mixtures
11/14/1996DE19517056A1 1-Fluor-5,6,7,8-tetrahydroisochinolin-Derivate und ihre Verwendung in flüssigkristallinen Mischungen 1-fluoro-5,6,7,8-tetrahydroisoquinoline derivatives and their use in liquid crystal mixtures
11/14/1996DE19517051A1 1-Fluor-6,7-dihydro-5H-isochinolin-8-on-Derivate und ihre Verwendung in flüssigkristallinen Mischungen 1-fluoro-6,7-dihydro-5H-isoquinolin-8-one derivatives and their use in liquid crystal mixtures
11/14/1996DE19517038A1 1,8-Difluorisochinolinderivate und ihre Verwendung in flüssigkristallinen Mischungen 1,8-Difluorisochinolinderivate and their use in liquid crystal mixtures
11/14/1996DE19517025A1 Trifluortetrahydroisochinolin-Derivate und ihre Verwendung in flüssigkristallinen Mischungen Trifluortetrahydroisochinolin derivatives and their use in liquid crystal mixtures
11/13/1996EP0741720A1 Heterocyclic chemoluminescent derivatives
11/13/1996EP0741719A1 Intermediate and process for making
11/13/1996EP0741697A1 Amino acid derivatives and their use as phospholipase a2 inhibitors
11/13/1996EP0741569A1 Naphthylisoquinoline alkaloids, pharmaceutical compositions containing them and their use for the treatment of malaria
11/13/1996EP0489850B1 New bis-platinum complexes as chemotherapeutic agents
11/07/1996WO1996034870A1 Azacycloalcane derivatives, preparation thereof and their applications in therapy
11/07/1996WO1996034853A1 Azocompounds for the antemortem diagnosis of alzheimer's disease and in vivo imaging and prevention of amyloid deposition
11/07/1996CA2220015A1 Azacycloalcane derivatives, preparation thereof and their applications in therapy
11/07/1996CA2219880A1 Azocompounds for the antemortem diagnosis of alzheimer's disease and in vivo imaging and prevention of amyloid deposition
11/05/1996US5571920 Alcohols
11/05/1996US5571919 Dimeric naphthylisoquinoline alkaloids and synthesis methods thereof
10/1996
10/29/1996US5569762 Asymmetric synthesis of intermediates for retroviral protease inhibitor compounds
10/29/1996US5569669 Treating anxiety, depression
10/29/1996US5569659 4-arylpiperazines and 4-arylpiperidines
10/23/1996EP0643699B1 6-(2-hydroxyethylaminoalkyl)-5,11-dioxo-5,6-dihydro-11h- indeno[1,2-c]isoquinolines and their use as antineoplastic agents
10/22/1996CA1338669C Substituted aryl ureas as high potency sweeteners
10/16/1996EP0737671A2 Aromatic hydroxamic acid compounds, their production and use
10/16/1996EP0540673B1 Acetylene derivatives having lipoxygenase inhibitory activity
10/15/1996US5565470 Cycloaminoalkoxyphenyl derivatives, a process for their preparation as well as the compositions containing them
10/15/1996US5565457 For treatment of myocardial ischemias and cerebral vascular disorders
10/15/1996CA2020027C Isoquinoline- or quinoline-sulfonamide derivative and a pharmaceutical composition comprising the same
10/11/1996CA2173806A1 Aromatic hydroxamic acid compounds, their production and use
10/10/1996WO1996031527A1 Protease inhibiting succinic acid derivatives
10/10/1996WO1996031474A1 Novel heterocyclic compounds
10/10/1996WO1996031473A1 Novel heterocyclic compounds
10/10/1996WO1996031461A1 Phenoxyethylamine derivatives having high affinity for the 5-ht1a receptor, preparation thereof, use thereof as drugs, and pharmaceutical compositions containing said derivatives
10/10/1996CA2217194A1 Novel heterocyclic compounds
10/09/1996EP0736530A2 Retinoid-like heterocycles
10/09/1996EP0736036A1 Kininogen inhibitors
10/09/1996EP0736012A1 Anellated dihydropyridines and their use in the production of pharmaceutical preparations
10/09/1996EP0736011A1 Anellated dihydropyridines and their use in the production of pharmaceutical preparations
10/09/1996CN1132745A Substituted henzoylguanidines, process for their preparation, their use as medicament or diagnostic, and medicament containing them
10/08/1996US5563154 Tetrahydro-quinolinyl/isoquinolinyl-terminal alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
10/08/1996US5563144 Antiserotonins, their preparation and pharmaceutical compositions containing them
10/06/1996CA2173047A1 Retinoid-like heterocycles
10/02/1996EP0735026A1 Method for the production of isoquinoline derivatives and their use as intermediates in the preparation of indole derivatives
10/02/1996EP0735019A2 Retroviral protease inhibitors
10/01/1996US5561141 MDR reversal agents
09/1996
09/26/1996WO1996029327A1 Trypsin and thrombin inhibitors
09/26/1996WO1996029309A1 N-ACYLPIPERIDINYLCARBONYLAMINOCARBOXYLIC ACIDS AND THEIR USE AS GLYCOPROTEIN IIB/IIa ANTAGONISTS AND FIBRINOGEN-BLOOD PLATELETS BINDING INHIBITORS
09/26/1996CA2215106A1 N-acylpiperidinylcarbonylaminocarboxylic acids and their use as glycoprotein iib/iiia antagonists and fibrinogen-blood platelets binding inhibitors
09/25/1996CN1131942A HIV protease inhibitors
09/24/1996US5559256 Aminediol protease inhibitors
09/24/1996US5559248 For prevention and treatment of skin disorders
09/24/1996US5559144 Furyl and thienyl alkynyl-N-hydroxy urea derivatives
09/24/1996US5559140 Difluoro statone analogs
09/24/1996US5558974 Photographic material containing a new type of hydrazide
09/19/1996WO1996028445A1 Novel glutamate (ampa/kainate) receptor antagonists: n-substituted fused azacycloalkylquinoxalinediones
09/19/1996WO1996028418A1 Sulfonylalkanoylamino hydroxyethylamino sulfonamide retroviral protease inhibitors
09/18/1996EP0565631B1 Anti-viral compounds
09/18/1996EP0531370B1 Inhibition of viral infection
09/18/1996CN1131150A 3-phenyl isoquinolin-1(2H)-one derivant, its preparation method and medicinal use thereof
09/18/1996CN1131144A Glycinamide derivatives, processes for their preparation and medicines containing them
09/17/1996US5556978 Preparing 1r-cis, 1'r-cis 2',2'-/3,11-dioxo-4,10-dioxatridecylene/-bis/1,2,3,4-tetra-hy dro-6,7-dimethoxy-2-methyl-1-veratrylisoquinolinium salt