Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
12/1995
12/19/1995US5476873 Acetylene derivatives having lipoxygenase inhibitory activity
12/14/1995WO1995033731A1 Hydroxamic acid derivatives
12/14/1995WO1995033464A2 Retroviral protease inhibitor combinations
12/14/1995CA2191948A1 Retroviral protease inhibitor combinations
12/13/1995EP0686629A2 Cyclohexyl tachykinine receptor antagonists
12/12/1995US5475027 Retroviral protease inhibitors
12/12/1995US5475013 Inhibit human immunodeficiency virus protease
12/11/1995CA2150992A1 Cyclohexyl tachykinin receptor antagonists
12/07/1995WO1995032949A1 Gastrin and cck antagonists
12/07/1995WO1995032710A1 Compounds for inhibiting osteoclast-mediated bone resorption
12/07/1995CA2190870A1 Compounds for inhibiting osteoclast-mediated bone resorption
12/05/1995US5473074 Adenosine diphosphoribose polymerase binding nitroso aromatic compounds useful as retroviral inactivating agents, anti-retroviral agents and anti-tumor agents-54
12/05/1995US5472984 1,2-ethanediol derivative and salt thereof and cerebral function-improving agent comprising the same
11/1995
11/28/1995US5470979 Enzyme inhibitors of retroviral protease enzymes and antagonist of excitatory amino acid receivers
11/28/1995US5470978 Process and intermediates for the preparation of excitatory amino acid receptor antagonists
11/28/1995US5470878 Cell signaling inhibitors
11/22/1995EP0466933B1 Bicyclolactam derivative
11/22/1995CN1112104A Acetic acid derivatives
11/15/1995EP0682017A1 Substituted bicycle heteroaroylguanidines, their preparation and their application in medicaments and diagnostic agents
11/15/1995CN1111620A New alkylaminoindane compounds, processes for preparing them and pharmaceutical compositions containing them
11/14/1995US5466712 Substituted n-aryl-1,2-diaminocyclobutene-3,4-diones
11/09/1995WO1995029929A1 Novel erythromycin derivatives, method for their preparation and their use as drugs
11/09/1995WO1995029892A1 Hydroxamic acid and amino acid derivatives and their use as anti-arthritic agents
11/08/1995EP0680967A1 Erythromycin derivatives, their process of preparation and their use as medicaments
11/08/1995EP0680953A1 1-[Styryl]- and 1-[2'-(heteroaryl)-ethenyl]-isoquinoline derivatives, a process for preparing them as well as medicaments containing them and the use of them
11/08/1995EP0680951A2 Sulfur-containing benzimides
11/08/1995EP0680468A1 Substituted amino compounds, their preparation and their use as inhibitors of thrombocyte aggregation
11/08/1995CN1111237A Preparation of amides and peptides
11/07/1995US5464871 Aromatic nitro and nitroso compounds and their metabolites useful as anti-viral and anti-tumor agents
11/07/1995US5464867 Smooth muscle relaxants
11/06/1995CA2148666A1 Substituted bicyclic heteroaroylguanidines, a process for their preparation, their use as a medicament or a diagnostic agent, and a medicament containing them
11/04/1995CA2148412A1 1-¬styryl|- and 1-¬2'-(heteroaryl) -ethenyl| -isoquinoline derivatives, a process for preparing them as well as medicaments containing them and the use of them
11/02/1995EP0679642A1 Condensed heterocyclic compounds, their production and use
11/02/1995EP0471841B1 Sulfonamide derivative and pharmaceutical composition containing the same
10/1995
10/31/1995US5463124 Treating with niobium trichloride-dimethoxyethane complex and simultaneously controlling all four corners of chirality
10/29/1995CA2148047A1 Condensed heterocyclic compounds, their production and use
10/25/1995EP0678099A1 New peptides
10/24/1995US5461156 Stereocontrolled synthesis of cis-bicyclic compounds
10/24/1995US5461154 HIV protease inhibitors
10/19/1995WO1995027701A1 Metal-containing steroid mimics and ligands useful in the preparation thereof
10/17/1995CA1337351C Spiro-isoquinoline-pyrrolidine tetrones and analogs thereof useful as aldose reductase inhibitors
10/12/1995DE4410881A1 Substd. heterocyclic carboxylic acid amides and their prepn.
10/11/1995CN1109872A Substituted benzenesulfonylureas and -thioureas, preparation processes and possible uses of pharmaceutical preparations b ased on these compounds
10/11/1995CN1109870A N-(3-aminopropyl)-N-phenyl-5,6,7,8-tetrahydronaphtalene-2-carboxamide derivative, preparation and application of same
10/10/1995US5457219 Phosphorus compounds
10/05/1995WO1995026341A1 Substituted beta-aryl and beta-heteroaryl-alpha-cyanoacrylamide derivatives as tyrosine kinase inhibitors
10/05/1995WO1995026189A1 AN IMPROVED METHOD OF SYNTHESIS FOR 6,9-BIS[(2-AMINOETHYL)AMINO]BENZO[g]ISOQUINOLINE-5,10-DIONE AND ITS DIMALEATE SALT
10/03/1995US5455353 4-(benzyl-2-oxo-oxazolidin-5 ylmethyl)N tertbutyl-decahydroisoquinoline-3-carboxamides
10/03/1995US5455251 Michellamine antiviral agents, compositions, and treatment methods
09/1995
09/26/1995US5453510 Neuromuscular blocking agents
09/26/1995US5453509 Functionalization of acyl pyridinium salts
09/21/1995WO1995025092A1 Inhibitors of farnesyl-protein transferase
09/21/1995CA2185553A1 Inhibitors of farnesyl-protein transferase
09/20/1995EP0610236B1 Process for making nickel-plated castings
09/19/1995US5451678 Alcohols
09/14/1995WO1995024385A1 Sulphonamide derivatives as aspartyl protease inhibitors
09/14/1995CA2183653A1 Sulphonamide derivatives as aspartyl protease inhibitors
09/13/1995EP0671654A1 Photographic material containing a new type of hydrazide
09/13/1995EP0671397A1 Alkylaminoindanes compounds, processes for their preparation and pharmaceutical compositions containing them
09/13/1995CN1108248A Glycoprotein IIB/IIIA antagonists
09/12/1995US5449809 Acetylene derivatives and crop protection agents containing them
09/12/1995CA2144288A1 Alkylaminoindans compounds; process for preparing the same and pharmaceutical compositions containing them
09/06/1995CN1107840A Substituted 1-oxo-1,2-dihydro-isochinolinoly-and 1,1-dioro-2H-1,2-benothiazinoylguanidine, preparation, application of same and pharmaceutical containing same
08/1995
08/30/1995EP0669322A1 Substituted sulfonamides, process for their preparation and pharmaceutical compositions containing them
08/29/1995US5446164 Process for preparing 6,7-dialkoxy-3,4-dihydroisoquinolin-8-ol
08/29/1995US5446161 Amino acid derivatives
08/29/1995US5446071 Administering anticholesterol agents
08/29/1995US5446051 Nervous system disorder and brain disorder
08/23/1995EP0668268A2 Bicyclolactam derivatives for improving cerebral functions
08/23/1995CN1107144A Substituted heterocyclic carboxamide esters, their preparation and their use as pharmaceuticals
08/17/1995WO1995021826A1 Antimalarial korupensamines and pharmaceutical compositions and medical uses thereof
08/17/1995WO1995021815A1 Cyclobutane derivatives and their use as inhibitors of protein farnesyltransferase and squalene synthase
08/17/1995WO1995021616A1 Naphthylisoquinoline alkaloids, pharmaceutical compositions containing them and their use for the treatment of malaria
08/16/1995EP0666850A1 1,2,3,5,6,7,8,8a-OCTAHYDRO-5,5,8a-TRIMETHYL-(8a-g(b))-6-ISOQUINOLINEAMINE DERIVATIVES, PREPARATION METHOD THEREFOR AND THERAPEUTICAL USE THEREOF.
08/16/1995EP0666742A1 Adenosine diphosphoribose polymerase binding nitroso aromatic compounds useful as anti-retroviral agents and anti-tumor agents
08/16/1995EP0666736A1 Stabilization of fluorocarbon emulsions.
08/16/1995CN1106801A Isoquinolines
08/15/1995US5442055 Azetidinone compound and process for preparation thereof
08/15/1995US5441962 Administering isoquinolinone derivatives
08/10/1995WO1995021164A1 Intermediate and process for making
08/10/1995WO1995020950A1 Therapeutic guanidines
08/10/1995CA2182302A1 Therapeutic guanidines
08/10/1995CA2180860A1 Intermediate and process for making
08/09/1995EP0666250A1 Derivatives of N-(3-aminopropyl)-N-phenyl-5,6,7,8-tetrahydronaphthalene-2-carboxamide having neuroprotective and anti-ischemic properties, their preparation and their use, in therapy
08/08/1995US5439918 Inhibitors of farnesyl-protein transferase
08/08/1995US5439908 Diazinyl butyric acid amides and esters
08/04/1995CA2141729A1 N-(3-aminopropyl)-n-phenyl-5,6,7,8-tetrahydro-naphthalene -2-carboxamide derivatives, their preparation and their therapeutic use
08/03/1995WO1995004720A3 Gastrin and cck receptor ligands
08/02/1995EP0664795A1 Propenoic acid derivatives useful as fungicides
08/02/1995EP0569482B1 Synthesis of intermediates in the preparation of acat inhibitors
08/01/1995US5438140 Using cyclic ammonium compounds as brighteners
08/01/1995US5438059 Certain acrylates having fungicidal activity
07/1995
07/27/1995WO1995019976A1 Heterocyclic chemoluminescent derivatives
07/27/1995WO1995019959A1 Amino acid derivatives and their use as phospholipase a2 inhibitors
07/27/1995DE4337271A1 ubstd. heterocyclic carboxylic acid amides and their prepn.
07/26/1995EP0664289A2 Isoquinolines
07/26/1995EP0664127A2 Pharmaceutical compositions containing isoquinoline derivatives
07/18/1995US5434265 Inhibitors of HIV protease
07/18/1995US5434162 Quinolinyl/isoquinolinyl-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
07/11/1995US5432189 Bis-aryl amide and urea antagonists of platelet activating factor