Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
07/1995
07/05/1995EP0661264A1 Substituted benzenesulfonylureas and -thioureas as antiarrhythmics
07/04/1995US5430191 Assymetric hydrogenation catalysts, enantioselective hydrogen displacement
07/04/1995US5430151 Trifluoromethyl-containing pseudopeptides active against retroviruses
07/04/1995US5430150 N-(1-(((1H-benzimidazol-2-ylmethyl)amino)carbonyl)-2-methyl -butyl)-3-(((1,1-dimethylethyl)amino)-carbonyl)decahydro-gamma-hydroxyalpha -(phenylmethyl)-2-isoquinolinepentanamide compounds; AIDS
07/04/1995US5430062 Combretastatin analogues; inhibition of tubulin polymerization and colchicine binding; antitumor,-mitotic and -neoplastic agents
06/1995
06/29/1995WO1995017389A1 Anellated dihydropyridines and their use in the production of pharmaceutical preparations
06/29/1995WO1995017388A1 Anellated dihydropyridines and their use in the production of pharmaceutical preparations
06/29/1995DE4345266A1 New isoquinolone or phthalazinone carboxylic acid ester and derivs.
06/29/1995DE4343641A1 New fused di:hydro-pyridine derivs.
06/29/1995CA2178209A1 Anellated dihydropyridines and the use thereof for preparing pharmaceutical preparations
06/29/1995CA2178088A1 Anellated dihydropyridines and their use in the production of pharmaceutical preparations
06/28/1995EP0659748A1 Substituted 1-oxo-1,2-dihydro-isoquinolinoyl-and 1,1-dioxo-2H-1,2-benzothiazinoylguanidines, process for their preparation, their use as medicament or diagnostic agent, as well as a medicament containing them
06/27/1995US5428167 Asymmetric synthesis of intermediates for retroviral protease inhibitor compounds
06/25/1995CA2138466A1 Substituted 1-oxo-1,2-dihydroisoquinolinoylguanidines and 1,1-dioxo-2h-1,2-benzothiazinoylguanidines, a process for their preparation, their use as a medicament or diagnostic agent, and also a medicament containing them
06/21/1995EP0658545A1 Decahydro-isoquinoline derivatives
06/14/1995EP0657419A1 Alcohols
06/13/1995US5424313 Bibyclic heteroacrylpiperazine derivatives having psychotropic activity, and pharmaceutical compositions containing these derivatives
06/07/1995EP0656348A2 Aceric acid derivatives as medicaments
06/07/1995EP0616532A4 Use of peripheral-type benzodiazepine sites for treatment of cns trauma or disease.
05/1995
05/31/1995EP0655058A1 Pyridinyl/quinolinyl-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
05/31/1995EP0655056A1 Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
05/31/1995CN1028638C Method for preparation of isoquinoline amides of sulphonic acids derivatives
05/26/1995WO1995014005A1 Diaminocyclobutene-3,4-diones as smooth muscle relaxants
05/26/1995CA2175386A1 Diaminocyclobutene-3,4-diones as smooth muscle relaxants
05/24/1995EP0654266A1 Cardiac protective
05/16/1995US5416218 Photographic silver halide material
05/16/1995US5416094 Antiarrhythmic and cardioprotective substituted -1(2H)isoquinolines, medicament containing them, and their use for combating heart failures
05/11/1995WO1995012611A1 Endothelin receptor antagonists
05/11/1995CA2173875A1 Endothelin receptor antagonists
05/10/1995EP0652208A1 Phenylalkan(en)oic acids with leukotriene B4 antagonistic activity
05/09/1995US5413999 HIV protease inhibitors useful for the treatment of AIDS
05/09/1995US5413997 Triphenylmethane derivatives
05/06/1995CA2135000A1 Isoquinolines
05/04/1995DE4337270A1 Substituted heterocyclic carboxamidoesters, their preparation and their use as medicaments
05/03/1995EP0650961A1 Substituted heterocyclic carboxylic acid amides, their preparation, and their use as medicaments
05/03/1995EP0650960A1 Substituted heterocyclic carboxylic acid amide esters, their preparation and their us as medicaments
05/03/1995CA2134866A1 Substituted heterocyclic carboxamides, their preparation and their use as pharmaceuticals
05/03/1995CA2134865A1 Substituted heterocyclic carboxamide esters, their preparation and their use as pharmaceuticals
04/1995
04/27/1995WO1995011231A1 Amidino derivatives useful as nitric oxide synthase inhibitors
04/27/1995WO1995011228A1 2,3-diaminopropionic acid derivative
04/27/1995CA2174516A1 2,3-diaminopropionic acid derivative
04/27/1995CA2173468A1 Amidino derivatives useful as nitric oxide synthase inhibitors
04/26/1995EP0649839A1 Isoquinolinone-, phthalazinone-, quinazolinone- and benzotriazolinone derivatives, their preparation and their use as anti-thrombotics
04/26/1995EP0634997A4 Preparation of substituted guanidines.
04/25/1995US5409938 A plant extracts having a naphthyl-tetrahydroisoquinolines group; a new drug treating malarial, parasiticides
04/25/1995US5409930 Inhibits abnoramal cell proliferation; dimethoxyquinoline/ dimethylquinoline/ quinolineoxide/ and quinoxaline derivatives
04/25/1995US5409929 Hydroisoindolines and hydroisoquinolines as psychotropic drugs
04/20/1995WO1995010505A1 Functionalization of acyl pyridinium salts
04/19/1995EP0550635B1 Fused ring analogs of nitrogen containing nonaromatic heterocycles
04/18/1995US5407942 Biphenylmethyl-substituted pyridones
04/13/1995WO1995009843A1 Hiv protease inhibitors
04/13/1995WO1995009842A1 Isoquinolinone-, phthalazinone-, quinazolinone- and benzotriazolinone derivatives, their preparation and their use as anti-thrombotics
04/13/1995CA2148361A1 Isoquinolinone-, phthalazinone-, quinazolinone- and benzotriazolinone derivatives, their preparation and their use as anti-thrombotics
04/12/1995EP0647459A1 Method of dechlorination of chlorinated aromatic compounds
04/12/1995EP0647220A1 Ring-closed dihydropyridines and their use in the preparation of pharmaceutical compositions
04/12/1995EP0647136A1 Use of condensed bis-(3,4-dihydro-pyridinyl)methane for treating crohn's disease, colitis ulcerosa, chronic inflamatory processes and as an antiproliferative.
04/11/1995US5405843 Quinoline derivatives
04/06/1995WO1995009151A1 Acylated sulphonamides as insecticides and acaricides
04/05/1995EP0646115A1 Heterocyclic-cyclic amine derivatives
04/05/1995EP0646112A1 Tertiary and secondary amines as alpha-2 antagonists and serotonin uptake inhibitors
04/04/1995US5403861 Treating or preventing nerve cell death
04/04/1995US5403854 Substituted N-heteroaryl -1,2-diaminocyclobutene-3,4-diones
04/04/1995US5403853 Substituted N-aryl-1,2-diaminocyclobutene-3,4-diones
03/1995
03/28/1995US5401766 Aminoacid derivatives, a process for their preparation, agents containing these compounds, and the use thereof
03/28/1995US5401753 Substituted n-heteroaryl-1, 2-diaminocyclobutene-3, 3-diones
03/28/1995US5401752 Effective against drug resistant fungi
03/28/1995CA1334969C Substituted dihydroisoquinoline and phthalazine derivatives as potentiators of the lethal effects of radiation and certain chemotherapeutic agents, selected compounds, analogs andprocess
03/22/1995EP0644198A1 Alpha-heteroaryloxymethyl ketones as interleukin-1beta converting enzyme inhibitors
03/21/1995US5399748 Derivatives of aspartic acid and glutamic acid having anticholecystokinin activity
03/21/1995US5399696 Excitatory amino acid receptor antagonists; nervous system disorders
03/16/1995WO1995007291A1 Kininogen inhibitors
03/16/1995WO1995007260A1 Tetrahydroisoquinolines as alpha-2 antagonists and biogenic amine uptake inhibitors
03/16/1995WO1995007258A1 Cyclohexanediurea derivative and process for producing the same
03/16/1995CA2171295A1 Cyclohexanediurea derivative and process for producing the same
03/16/1995CA2170896A1 Kininogen inhibitors
03/14/1995US5397790 Substituted isoquinolinyl-1-2-diaminocyclobutene-3,4,-diones
03/14/1995US5397789 Cyclic nitrones
03/08/1995EP0641326A1 Substituted 1,2,3,4-tetrahydroisoquinolines with angiotensin ii receptor antagonist properties
03/08/1995EP0641325A1 Retroviral protease inhibitors
03/08/1995EP0641324A1 Tetrahydro and perhydro isoquinolin derivatives and therapeutic agents containing them
03/08/1995EP0641301A1 Stilbene derivatives as anticancer agents
03/07/1995US5395842 Inhibitors of sex steroids
03/01/1995EP0640073A1 Process for preparing n-allyl compounds.
03/01/1995CN1099387A Process for the manufacture of a beta-aminoalcohol
02/1995
02/28/1995US5393735 N-(halo-oxy-)phenyl substituted cyclic imides
02/28/1995US5393606 Charge-transfer complexes with N-aromatic compounds, the preparation thereof and the use thereof
02/21/1995US5391761 Preparation of novel amido-alcohol derivatives and their therapeutic uses
02/16/1995WO1995004720A2 Gastrin and cck receptor ligands
02/16/1995CA2167154A1 Gastrin and cck receptor ligands
02/14/1995US5389653 Inhibitors of the enzyme catechol-O-methyltransferase; useful as co-medication in treatment of Parkinson's disease
02/14/1995US5389638 Nervous system disorders
02/14/1995US5389610 Carboxyalkylcarbonyl aminoacid endopeptidase inhibitors
02/14/1995CA1334417C Process for preparing pyridine-2,3-dicarboxylic acid compounds
02/08/1995CN1098408A Heterocyclic inhibitors of farnesyl protein transferase
02/08/1995CN1098407A Inhibitors of HIV protease useful for the treatment of aids
02/07/1995US5387685 Bicyclic amines; resensitize multiple drug resistant cells to chemotherapeutic agents
02/01/1995EP0636612A1 Process for producing tetrahydroisoquinoline-3-carboxylic acid derivative
02/01/1995EP0636125A1 Basic derivatives of glutamic acid and aspartic acid as gastrin or cholecystokinin antagonists
02/01/1995EP0556308B1 Oxysulfonyl urea acat inhibitors
02/01/1995CN1098098A 哌嗪衍生物 Piperazine derivatives