Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
05/1996
05/17/1996WO1996014300A1 N-aryl and n-heteroaryl-1,2-diaminocyclobutene-3,4-diones with smooth muscle relaxing activities
05/17/1996CA2204415A1 N-aryl and n-heteroaryl-1,2-diaminocyclobutene-3,4-diones with smooth muscle relaxing activities
05/15/1996CN1122600A Second messenger cell signaling inhibitors
05/14/1996US5516941 Oxidizing 3-aminobenzamide to 3-nitrosobenzamide; viricides; anticarcinogenic and antitumor agents
05/14/1996US5516930 Ethyl 3-amino-2-hydroxy-4-phenylbutyrate
05/14/1996US5516913 Viricide intermediates
05/08/1996EP0710651A1 Process for the preparation of a decahydroisoquinoline-alpha, alpha' diamino alcohol
05/07/1996US5514802 Intermediates for preparing HIV protease inhibitors
05/07/1996US5514689 Antitumor
05/07/1996US5514683 Bicyclo 2,2,2!octane derivatives
05/01/1996EP0709370A1 Bicyclic compounds useful as platelet aggregation inhibitors
04/1996
04/30/1996US5512688 Sulphonic acid esters which are useful as intermediates in the production of βaminoalcohols
04/30/1996US5512682 Nitrile compounds useful as intermediates in the production of beta amino alcohols
04/30/1996US5512585 Diaminocyclobutene-3,4-diones
04/24/1996EP0707570A1 Isoquinoline derivatives as therapeutic agents
04/23/1996US5510487 Retroviral protease inhibitors
04/23/1996US5510380 Nonpeptide bradykinin antagonists
04/23/1996US5510378 Retroviral protease inhibitors
04/23/1996US5510349 Retroviral protease inhibitors
04/17/1996EP0640073B1 Process for preparing n-allyl compounds
04/17/1996EP0558673B1 Retroviral protease inhibitors
04/17/1996CN1120537A Novel substituted sulphonic acid amide, preparation and pharmaceutical composition of same
04/16/1996US5508430 Azidoalkyl- or phthalimidoalkyl-oxiranes which can be used to make viricides
04/16/1996US5508407 Treating or preventing infection by hiv
04/10/1996EP0705821A1 Oxidation of nitrogen heterocycles and heterocyclic N-oxides produced thereby
04/10/1996EP0705100A1 Therapeutic substituted guanidines
04/10/1996CN1120333A Imino-substituted phenylacetic acid amides, their preparation and fungicides containing them
04/09/1996US5506252 Substituted N-heteroaryl and N-aryl-1,2-diaminocyclobutene-3,4-diones
04/09/1996US5506240 Hypotensive agents
04/09/1996US5506232 High purity antitumor agents with reduced side effects
04/04/1996WO1996010012A1 Novel prostaglandin synthase inhibitors
04/04/1996WO1996009820A1 Inhibitors of farnesyl-protein transferase
04/03/1996EP0703905A1 Inhibitors of farnesyl-protein transferase
03/1996
03/28/1996WO1996009286A1 Isothiourea derivatives as no synthase inhibitors
03/28/1996DE4434288A1 Substd. heterocyclic carboxylic acid amides and their prepn.
03/28/1996DE4433928A1 Substd. heterocyclic carboxylic acid amides and their prepn.
03/27/1996EP0702671A1 Bicyclic fibrinogen antagonists
03/26/1996US5502060 HIV protease inhibitors
03/26/1996US5502027 Algicides
03/21/1996WO1996008228A2 Derivatives of 2-amino-1,2,3,4-tetrahydro-naphthalene active on the cardiovascular system
03/21/1996CA2199484A1 Derivatives of 2-amino-1,2,3,4-tetrahydro-naphthalene active on the cardiovascular system
03/20/1996EP0702004A2 2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amid derivatives
03/19/1996US5500430 Amidic derivatives of glutamic, aspartic and 2-amino adipic acids, a process for preparing same, and anti-gastrin composition containing the derivatives
03/16/1996CA2158227A1 2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amide derivatives
03/14/1996WO1996007642A1 PROCESS FOR PRODUCING A β-AMINO ALCOHOL
03/14/1996DE4431530A1 Verfahren zur Herstellung eines beta-Aminoalkohols A method for producing a beta-aminoalcohol
03/14/1996CA2198460A1 Process for producing a .beta.-amino alcohol
03/13/1996EP0700389A1 Anti-arrhythmic n-substituted 3-benzazepines or isoquinolines
03/13/1996EP0700388A1 Substituted beta-aryl and beta-heteroaryl-alpha-cyanoacrylamide derivatives as tyrosine kinase inhibitors
03/12/1996US5498786 Enzyme inhibitors, cardiovascular disorders
03/12/1996US5498778 By preventing free radical oxygen oxidation
03/12/1996US5498717 6,7-dialkoxy-3,4-diydroisoquinolin-8-yl compounds
03/07/1996WO1996006855A1 NEW PEPTIDE DERIVATIVES WITH δ OPIOID RECEPTOR ANTAGONIST OR MIXED ν AGONIST/δ ANTAGONIST EFFECTS
03/07/1996CA2197566A1 New peptide derivatives with .delta. opioid receptor antagonist or mixed.mu. agonist/.delta. antagonist effects
02/1996
02/29/1996WO1996006072A1 Oxime ethers and their use as pesticides
02/29/1996CA2194231A1 Oxime ethers and their use as pesticides
02/28/1996EP0698019A1 Novel aromatic nitro compounds and their metabolites useful as anti-viral and anti-tumor agents
02/27/1996US5495025 Isoindole compounds which are useful as intermediates
02/27/1996US5494909 Antiischemic agents
02/22/1996WO1996004913A1 Hiv protease inhibitor combination
02/21/1996EP0697403A1 Derivatives of glycinamides as cholecystokinin receptor agonists
02/21/1996CN1117045A Substituted bicyclic heteroaroylguanidines, a process for their preparation, their use as a medicament or a diagnostic agent, and a medicament containing them
02/20/1996CA2065271C New bis-platinum complexes as chemotherapeutic agents
02/15/1996WO1996004241A2 Benzoylguanidine derivatives as medicaments
02/15/1996WO1996004231A1 Novel amine derivative, process for producing the same, and use thereof as antiarrhythmic
02/15/1996CA2196763A1 Benzoylguanidine derivatives as medicaments
02/15/1996CA2196672A1 Amine derivatives, processes for producing same, and use thereof as antiarrhythmic drugs
02/14/1996EP0696277A1 Hiv protease inhibitors useful for the treatment of aids
02/13/1996US5491232 Sulfur compounds useful for preparation of dyes
02/13/1996US5491166 Inhibitors of HIV protease useful for the treatment of AIDS
02/13/1996US5491164 Inhibitors of farnesyl-protein transferase
02/13/1996US5491149 Viricides
02/13/1996US5491147 Tri-substituted phenyl derivatives and their use in pharmaceutical compositions and methods of treatment
02/13/1996US5491132 Amino acid derivatives, a process for the preparation thereof and pharmaceutical composition comprising the same
02/13/1996US5490498 Adding fluorocarbon along with breathing gas which oxygenates the fluorocarbon; treatment of respiratory distress syndrome
02/08/1996WO1996003382A1 Monomeric and dimeric naphthylisoquinoline alkaloids and synthesis methods thereof
02/08/1996WO1996003381A1 Dimeric arylisoquinoline alkaloids and synthesis methods thereof
02/08/1996CA2195647A1 Monomeric and dimeric naphthylisoquinoline alkaloids and synthesis methods thereof
02/08/1996CA2195646A1 Dimeric arylisoquinoline alkaloids and synthesis methods thereof
02/07/1996EP0695294A1 Michellamines useful as antiviral agents
02/07/1996EP0695184A1 Hiv protease inhibitors
02/07/1996CN1030922C Process for preparation of new amino acid derivatives
02/06/1996US5489709 Reacting mono-substituteed cyanamide with a secondary amine
02/06/1996US5489686 Substituted 1,2,3,4-tetrahydroisoquinolines with angiotensin II receptor antagonist properties
01/1996
01/30/1996US5488115 Alcohols
01/17/1996EP0691950A1 Imino-substituted phenylacetic acid amides, their preparation and fungicides containing them
01/17/1996EP0602028B1 Aromatic sulfonamide derivatives, their use as enzyme inhibitors and pharmaceutical compositions containing them
01/16/1996US5484926 HIV protease inhibitors
01/10/1996EP0691345A2 HIV protease inhibitor combinations
01/10/1996EP0690851A1 Guanidine derivatives useful in therapy
01/10/1996CN1114650A MDR reversal agents
01/10/1996CN1114649A Sulfur compounds
01/09/1996US5482975 Adenosine diphosphoribose polymerase binding nitroso aromatic compounds useful as retroviral inactivating agents, anti-retroviral agents and anti-tumor agents
01/09/1996US5482967 Condensed heterocyclic compounds, their production and use
01/09/1996US5482947 Retroviral protease inhibitors
01/06/1996CA2153270A1 Hiv protease inhibitor combinations
01/04/1996WO1995033464A3 Retroviral protease inhibitor combinations
12/1995
12/27/1995EP0688312A1 New derivatives of glutamic acid, a method of preparing them, and their use as drugs for enhancing memory and learning
12/26/1995US5478938 Antagonists for angiotensin II receptors; hypotensive, cardiotonic agents; cognitive activators
12/19/1995US5476875 Catechol derivatives