Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
09/1996
09/17/1996US5556862 Pharmaceutical compositions containing isoquinoline derivatives
09/11/1996EP0731088A2 Retroviral protease inhibitors
09/10/1996US5554756 Amino acid derivatives
09/10/1996US5554735 Azo oxime ethers and their use as fungicides
09/05/1996DE19507522A1 Prodn. of 3,4-di:hydro-isoquinoline or deriv.
09/04/1996EP0729457A1 Diaminocyclobutene-3,4-diones as smooth muscle relaxants
09/03/1996US5552550 Monomeric Naphthylisoquinoline alkaloids and synthesis methods thereof
09/03/1996US5552549 Process for the dechlorination of chlorinated aromatic compounds
09/03/1996US5552412 5-substitued-6-cyclic-5,6,7,8-tetrahydronaphthalen2-ol compounds which are useful for treating osteoporosis
08/1996
08/29/1996WO1996026205A1 Inhibitors of microsomal triglyceride transfer protein and method
08/29/1996WO1996026201A1 Benzopyran-containing compounds and method for their use
08/29/1996WO1996026187A1 Fibrinogen receptor antagonists
08/29/1996CA2211890A1 Fibrinogen receptor antagonists
08/28/1996EP0728744A2 Process for the preparation of carboxylic acids of nitrogen-containing heterocycles
08/28/1996EP0728145A1 Endothelin receptor antagonists
08/27/1996US5550229 Alkylation process for preparing azetidinone compound and starting compound therefor
08/27/1996US5550162 N-(-3-aminopropyl)-N-phenyl-5,6,7,8-tetrahydro-naphthalene-2-carboxamide derivatives, their preparation and their therapeutic use
08/27/1996US5550149 Sulfur-containing compounds that are effective in potentiating the activity of chemotherapeutic anti-cancer agents by increasing sensitivity of multi-drug resistant cells
08/27/1996US5550124 Use of peripheral-type benzodiazpine sites for treatment of CNS trauma or disease
08/22/1996WO1996025157A1 Il-8 receptor antagonists
08/20/1996US5547984 N-Acetonyl-substituted-amides
08/20/1996US5547953 Antiarrhythmia agents, antiischemic agents, antigrowth agents
08/16/1996CA2169231A1 Bis(biaryl) compounds as inhibitors of leukotriene biosynthesis
08/15/1996WO1996024588A1 Bicyclic isothiourea derivatives useful in therapy
08/15/1996CA2211299A1 Bicyclic isothiourea derivatives useful in therapy
08/14/1996CN1128992A Therapeutic agents
08/13/1996US5545835 Chemical intermediates for preparation of substituted 2,3-pyridinedicarboxylic acids
08/13/1996US5545750 Retroviral protease inhibiting compounds
08/13/1996US5545640 Viricides, hiv; aids
08/13/1996CA2100066C Michellamines useful as antiviral agents, composition and method of treatment
08/07/1996EP0725059A1 2,3-diaminopropionic acid derivative
08/07/1996EP0724908A1 Noble metal raney catalysts and preparation of hydrogenated compounds using such catalysts
08/07/1996EP0724570A1 Amidino derivatives useful as nitric oxide synthase inhibitors
08/07/1996EP0476156B1 Solid oral preparation containing catechol compound
08/06/1996US5543523 Method and intermediates for the synthesis of korupensamines
08/01/1996WO1996022791A1 Novel synergistic compositions useful as anti-tumor or anti-retroviral agents
07/1996
07/30/1996US5541334 Treating hiv
07/25/1996WO1996022288A1 GLYCOPROTEIN IIb/IIIa ANTAGONISTS
07/25/1996WO1996008228A3 Derivatives of 2-amino-1,2,3,4-tetrahydro-naphthalene active on the cardiovascular system
07/25/1996CA2210682A1 Glycoprotein iib/iiia antagonists
07/24/1996EP0722439A1 Hiv protease inhibitors
07/24/1996CN1127251A Process for the preparation of a alpha, alpha'-diaminoalcohol
07/23/1996US5539119 Multistage formation by oxidation, reducing a carbamate to form an enamine, forming an oxide
07/18/1996WO1996021656A1 Estrogen agonists/antagonists
07/18/1996WO1996021456A1 Inhibitors of prenyl transferases
07/18/1996CA2207252A1 Inhibitors of prenyl transferases
07/17/1996EP0721451A1 Acylated sulphonamides as insecticides and acaricides
07/16/1996US5536816 Process for producing amides using catalytic amounts of an N-hydroxy compound
07/16/1996US5536741 Diaminocyclobutene-3,4-diones
07/16/1996US5536731 Smooth muscle relaxants
07/11/1996WO1996020710A1 Compounds for inhibition of ceramide-mediated signal transduction
07/11/1996CA2208580A1 Compounds for inhibition of ceramide-mediated signal transduction
07/10/1996EP0720601A1 Gastrin and cck receptor ligands
07/10/1996CN1126469A HIV protease inhibitors useful for the treatment of aids
07/10/1996CN1126434A Therapeutic substituted guanidines
07/09/1996US5535048 Electrooptics; polarizable compound
07/04/1996WO1996020190A1 Piperazine 2,5 dione derivatives as modulators of multi-drug resistance
07/04/1996CA2207500A1 Piperazine 2,5 dione derivatives as modulators of multi-drug resistance
07/03/1996EP0719764A1 3-Phenylisoquinolin-1 (2H)-one derivatives as GABA receptor ligands
07/03/1996EP0719267A1 Second messenger cell signaling inhibitors
07/03/1996CN1125942A Substituted beta-aryl and beta-heteroaryl-alpha-cyanoacrylamide derivatives as tyrosine kinase inhibitors
07/02/1996US5532266 Treatment of hypoxia, antiedemic agents or antiinflammatory agents
07/02/1996US5532252 For the treatment of tissue damage associated with physical trauma
07/02/1996US5532245 To reduce smooth muscle contractions; treatment for urinary incontinence, iritable bowel syndrome
07/02/1996US5532243 Antipsychotic nitrogen-containing bicyclic compounds
06/1996
06/30/1996CA2166234A1 3-phenylisoquinol-1(2h)-one derivatives, their preparation and their therapeutic application
06/27/1996WO1996019440A1 Acetamidine derivatives and their use as inhibitors for the nitric oxide synthase
06/26/1996EP0718292A1 Acetylenic derivatives and their use as plant-protective agents
06/26/1996EP0718281A1 Cyclohexanediurea derivative and process for producing the same
06/25/1996US5530125 Reacting arylacetamide with strong base in inert aprotic solvent, then with specified reactant in presence of transition metal catalyst to add alpha-substituent,reducing to amine
06/25/1996US5530025 Smooth muscle relaxants
06/25/1996US5529978 Fungicide
06/20/1996WO1996018616A1 Substituted 2-aminopyridines as inhibitors of nitric oxide synthase
06/20/1996WO1996018602A1 Bicyclic fibrinogen antagonists
06/20/1996WO1996004241A3 Benzoylguanidine derivatives as medicaments
06/18/1996US5527812 Cyclic nitrones
06/18/1996US5527811 Isoquinolinyl compounds which are useful in treating cerebral vascular disorders
06/18/1996US5527799 HIV protease inhibitors useful for the treatment of AIDS
06/13/1996DE4042595C2 New aryl hydrazide cpds. contg. quat. nitrogen substit.
06/12/1996EP0716082A1 Oxy-phenyl-(phenyl)glycinolamides substituted with a heterocycle having antiatherosclerotic activity
06/11/1996US5525615 Cardiovascular disorders
06/11/1996US5525614 Substituted 1,2,3,4-tetrahydroisoquinolines with angiotensin II receptor antagonist properties
06/06/1996WO1996016943A1 Iminooxybenzylcrotonic acid esters, process for their preparation and use thereof
06/06/1996CA2207381A1 Iminooxybenzylcrotonic acid esters, process for their preparation and use thereof
06/05/1996DE4442560A1 Iminooxybenzylcrotonsäureester, Verfahren zu ihrer Herstellung und ihre Verwendung Iminooxybenzylcrotonsäureester, processes for their preparation and their use
06/04/1996US5523305 Analgesics
05/1996
05/29/1996EP0713864A1 Substituted benzoylguanidines, process for their preparation, their use as medicament of diagnostic agent as well as medicaments containing them
05/25/1996CA2163598A1 Substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them
05/23/1996WO1996015111A1 Method and intermediates for the synthesis of korupensamines
05/23/1996WO1996015103A1 Diaminocyclobutene-3,4-diones
05/23/1996WO1996014842A1 Substituted heterocycles as inhibitors of nitric oxide synthase
05/23/1996CA2205307A1 Diaminocyclobutene-3,4-diones
05/22/1996EP0712628A2 Methods of inhibiting bone loss
05/22/1996EP0712627A2 Methods for lowering serum cholesterol
05/22/1996EP0539470B1 Neuromuscular blocking agents
05/21/1996US5519113 Process for the diastereoselective reductive pinacol coupling of homochiral α-aminoaldehydes
05/21/1996US5519034 Analgesics
05/21/1996US5518735 Anticoagulants administered by mouth
05/19/1996CA2163158A1 Methods for inhibiting bone loss
05/19/1996CA2163156A1 Methods for lowering serum cholesterol