Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
08/1994
08/23/1994CA1331614C Substituted acyl derivatives of 1,2,3,4-tetrahydroisoquinoline- 3-carboxylic acids
08/21/1994CA2115967A1 Substituted benzoylguanidines, process for their preparation, their use as a pharmaceutical, as inhibitors of the cellular na+/h+exchange or as a diagnostic, and pharmaceutical containing them
08/16/1994US5338851 Synthesis of cis-decahydroisoquinoline-3-carboxylic acids
08/10/1994EP0609960A1 New N-heteroarylamide derivatives as inhibitors of acyl coenzyme A: cholestrol acyl transferase
08/10/1994EP0609625A1 Inhibitors of HIV protease useful for the treatment of AIDS
08/10/1994EP0609211A1 Adenosine diphosphoribose polymerase binding nitroso aromatic compounds useful as anti-tumor and anti-retroviral agents
08/10/1994CN1025618C Compound having vessel smoth muscle relaxation activity
08/04/1994WO1994017034A1 Substituted amino compounds, their preparation and their use as inhibitors of thrombocyte aggregation
08/03/1994CN1090274A Condensed heterocyclic compounds, their production and use
08/02/1994US5334724 Reacting a pyridine-1-oxide with an aromatic carbonyl chloride in presence of an acid acceptor in solvents
08/02/1994US5334600 Lipoxygenase inhibitors
07/1994
07/26/1994US5332838 Cyclization process utilizing copper aluminum borate as a catalyst
07/26/1994US5332821 Process for preparing isoquinolines
07/21/1994WO1994015959A1 New peptides
07/21/1994WO1994015928A1 Piperazine derivatives as 5-ht antagonists
07/21/1994WO1994015906A1 Hiv protease inhibitors and their preparation
07/21/1994WO1994015608A1 Hiv protease inhibitors
07/21/1994WO1994009625A3 Stabilization of fluorocarbon emulsions
07/21/1994CA2153777A1 Hiv protease inhibitors
07/21/1994CA2152380A1 New peptides
07/19/1994US5330991 Tetrahydroisoquinoline compounds and fungicides containing the same
07/19/1994CA1330798C Benzo- and thieno-3,4-dihydro-pyridine derivatives
07/12/1994US5328915 Insecticides
07/07/1994CA2110337A1 O-aryl ethers of morphinans
07/05/1994US5326870 Substituted sulfonamide derivative and a pharmaceutical composition comprising the same
07/05/1994CA1330560C Di- and tetrahydroisoquinoline derivatives
06/1994
06/29/1994EP0604186A1 Inhibitors of HIV protease useful for the treatment of aids
06/29/1994EP0604185A1 Inhibitors of HIV protease useful for the treatment of aids
06/29/1994EP0604183A1 Inhibitors of HIV protease useful for the treatment of aids
06/28/1994US5324839 Hypotensive agents, gastrointestinal and urogenital disorders
06/23/1994CA2112052A1 Inhibitors of hiv protease useful for the treatment of aids
06/23/1994CA2112042A1 Inhibitors of hiv protease useful for the treatment of aids
06/23/1994CA2112041A1 Inhibitors of hiv protease useful for the treatment of aids
06/23/1994CA2112019A1 Inhibitors of hiv protease useful for the treatment of aids
06/22/1994EP0602523A1 Substituted benzoylguanidines, process for their preparation, their use as medicament or diagnostic agent, as well as a medicament containing them
06/22/1994EP0602306A1 Retroviral protease inhibitors
06/22/1994EP0602028A1 Aromatic sulfonamide derivatives, their use as enzyme inhibitors and pharmaceutical compositions containing them.
06/17/1994CA2111454A1 Retroviral protease inhibitors
06/07/1994USRE34630 Antagonist for platelet activating factor
06/01/1994EP0599518A1 Process and intermediates for the preparation of excitatory amino acide receptor antagonists
06/01/1994EP0462148B1 Substituted 2-propenyl derivatives of nitrogen heterocycles
05/1994
05/26/1994WO1994011345A1 Process for optically pure decahydroisoquinolines
05/25/1994EP0598171A1 Nitrogen bridge tetrahydroisoquinolines
05/19/1994CA2102931A1 Process and intermediates for the preparation of excitatory amino acid receptor antagonists
05/18/1994EP0597423A2 Azetidinone compound and process for preparation thereof
05/17/1994CA2088436A1 Nitrogen bridge tetrahydroisoquinolines
05/11/1994WO1994010150A1 1,2,3,5,6,7,8,8a-OCTAHYDRO-5,5,8a-TRIMETHYL-(8aβ)-6-ISOQUINOLINEAMINE DERIVATIVES, PREPARATION METHOD THEREFOR AND THERAPEUTICAL USE THEREOF
05/11/1994WO1994010118A1 Tri-substituted phenyl derivatives and processes for their preparation
05/11/1994WO1994009776A1 Adenosine diphosphoribose polymerase binding nitroso aromatic compounds useful as anti-retroviral agents and anti-tumor agents
05/11/1994WO1994009625A2 Stabilization of fluorocarbon emulsions
05/11/1994CA2148455A1 Adenosine diphosphoribose polymerase binding nitroso aromatic compounds useful as anti-retroviral agents and anti-tumor agents
05/11/1994CA2148002A1 1,2,3,5,6,7,8,8a-octahydro-5,5,8a-trimethyl-(8a.beta.)-6- isoquino lineamine derivatives, preparation method therefor and therapeutical usethereof
05/04/1994EP0594795A1 Michellamines useful as antiviral agents, composition and method of treatment
05/03/1994CA1329209C 2-amino-tetrahydro-isoquinoline derivatives and a process for the preparation thereof and pharmaceutical compositions containing same
04/1994
04/28/1994WO1994009000A1 Quinoxalinedione derivatives as eaa antagonists
04/28/1994WO1994008968A1 Propenoic acid derivatives useful as fungicides
04/26/1994US5306789 Amorphous, soluble, aromatic polymers with high glass transition temperatures
04/19/1994US5304558 Diphenylmethyl piperazine derivatives
04/19/1994US5304552 Renin inhibitors
04/13/1994EP0591937A1 Use of isoquinolinone derivatives for treating hyperlipoproteinemia
04/13/1994CN1085214A Tetrahydro- and perhydroisoquinoline derivatives and therapeutic compositions containing these
04/10/1994CA2108065A1 Antiarteriosclerosis agent and antihyperlipoproteinemics
04/06/1994EP0590789A1 Excitatory amino acid receptor antagonists
04/06/1994EP0590455A1 Antiarrhythmic and cardioprotective substituted -1(2H)Isoquinolines, process for their production, medicament containing them and their use for the production of a medicament for combating heart failures
04/05/1994US5300672 For water systems, plant diseases
04/05/1994US5300646 Heterocyclic amine derivatives, their production and use
03/1994
03/31/1994WO1994006280A1 Inhibitors of metazoan parasite proteases
03/30/1994EP0589484A1 1,2-Ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
03/29/1994US5298657 From a cyanamide and an amine, Lewis acid catalyst
03/23/1994EP0587698A1 Substituted 1-(2h)-isoquinolinones bearing acidic functional groups as angiotensin ii antagonists
03/17/1994WO1994005640A1 Process for producing tetrahydroisoquinoline-3-carboxylic acid derivative
03/17/1994WO1994005290A1 Platelet aggregation inhibitor
03/16/1994EP0587194A1 2-(Heterocycloalkoxy)-1-(subst.-phenyl)-ethanol derivatives as cerebral function improving agents
03/16/1994EP0587193A1 1,2-Ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
03/15/1994US5294621 Thieno tetrahydropyridines useful as class III antiarrhythmic agents
03/09/1994EP0585913A2 Condensed heterocyclic compounds, their production and use
03/08/1994US5292746 Cyclic nitrones, pharmaceutical compositions thereof and their use in treating shock
03/08/1994US5292521 And an organic acid or salt
03/08/1994CA1327577C 6-phenyl-3-(piperazinylalkyl)-2,4(1h,3h)- pyrimidinedione derivatives, their preparation and their application in therapy
03/08/1994CA1327576C Phenoxyacetic acid amide derivatives and their use in the treatment of obesity and related conditions
03/04/1994CA2484248A1 Excitatory amino acid receptor antagonists
03/03/1994WO1994004503A1 Pyridinyl/quinolinyl-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
03/03/1994WO1994004495A1 Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
03/03/1994CA2138518A1 Pyridinyl/quinolinyl-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
03/02/1994EP0584088A1 Substituted guanidines and derivatives thereof as modulators of neurotransmitter release and novel methodology for identifying neurotransmitter release blockers
03/02/1994CN1083054A Tachykinin receptor antagonists, isoquinolones and their production
02/1994
02/23/1994EP0583433A1 Diphosphine ligands
02/23/1994EP0583358A1 Partial liquid breathing of fluorocarbons
02/23/1994EP0583322A1 Antiserotonines, prepartion thereof and medicaments containing them
02/23/1994CN1082535A Carbocyclic and heterocyclic annelleted dihydropyridine and application of same in preparation of pharmaceutical
02/22/1994US5288866 5,6-disubstituted-3-pyridylmethyl ammonium halide compounds useful for the preparation of 5- (substituted methyl)-2,3-pyridinedicarboxylic acids
02/22/1994US5288749 Tertiary and secondary amines as alpha-2 antagonists and serotonin uptake inhibitors
02/17/1994WO1994003432A1 Polyhydroxylated naphthyl 2-carboxylate, and quinolyl and isoquinolyl 3-carboxylate derivatives as protein tyrosine kinase inhibitors
02/17/1994WO1994003171A1 Cardiac protective
02/16/1994EP0582925A1 Acetylenic derivatives and their use as plant-protective agents
02/16/1994CN1082029A Biphenylmethyl-substituted pyridones
02/15/1994US5286732 Nitrogen-containing bicyclic compounds and pharmaceutical compositions thereof
02/12/1994CA2101664A1 Acetylene derivatives and crop protection agents containing them
02/08/1994US5284957 Substituted 1H- or 2H-tetrazoles
02/03/1994WO1993010741A3 Sex steroid activity inhibitors