Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
05/2005
05/11/2005EP1254138B1 Pyridine derivatives inhibiting angiogenesis and/or vegf receptor tyrosine kinase
05/11/2005EP0973752B1 Heterocyclically substituted aromatic amino compounds with a herbicidal effect
05/11/2005CN1615308A Prucalopride-N-oxide
05/11/2005CN1615307A Process and intermediates for pyridazinone antidiabetic agents
05/11/2005CN1615305A Coumarin derivatives, process for their production and use thereof
05/11/2005CN1615300A Benzimidazole derivatives and their use as GNRH antagonists
05/11/2005CN1200940C Triazole pyrimidine compounds
05/11/2005CN1200939C Novel tetrahydropyridines, preparation method and pharmaceutical compositions containing same
05/11/2005CN1200933C Substituted N-benzoyl-N'-(tetrazolylphenyl)-ureas and their use as pest control agents
05/10/2005US6890940 Immoglobulin E (IgE) antibody production inhibitor; treating allergic immune diseases such as asthma, dermatitis, inflammatory bowel disease and allergic opthalmopathy
05/10/2005US6890937 Inhibiting the activity of one or more of MMP-2, MMP-9 and MMP-13, while exhibiting substantially less inhibitory activity against MMP-1
05/10/2005US6890935 Pharmaceutical compositions and methods for use
05/10/2005US6890932 Anthranilic acid derivative
05/10/2005US6890930 Quinazolinones
05/10/2005US6890928 Aromatic sulfone hydroxamic acids and their use as protease inhibitors
05/10/2005US6890924 Substituted bicyclic derivatives for the treatment of abnormal cell growth
05/10/2005US6890915 Hydantoins and related heterocycles as inhibitors of matrix metalloproteinases and/or TNF-α converting enzyme (TACE)
05/10/2005US6890885 Herbicidal composition
05/06/2005WO2005040355A2 Tao kinase modulators and methods of use
05/06/2005WO2005040345A2 4-azole substituted imidazole compositions useful as inhibitors or c-met receptor tyrosine kinase
05/06/2005WO2005040161A1 Biaryl linked hydroxamates: preparation and pharmaceutical applications
05/06/2005WO2005040156A1 Azole derivative useful as antifungal agents with reduced interaction with metabolic cytochromes
05/06/2005WO2005040155A1 Pyrimidin-2-amine derivates and their use as a2b adenosine receptor antagonists
05/06/2005WO2005040151A1 Pyrazine derivatives and pharmaceutical use thereof
05/06/2005WO2005040144A1 Novel compounds
05/06/2005WO2005040136A1 Piperazine derivatives and their use as modulators of nuclear hormone receptor function
05/06/2005WO2005040132A1 Dicationic triaryl analogs as anti-protozoan agents
05/06/2005WO2005040131A1 1,5,7-trisubstituted benzimidazole derivatives and their use for modulating the gabaa receptor complex
05/06/2005WO2005040116A2 Indolinone derivatives and their use in treating disease-states such as cancer
05/06/2005WO2005040110A1 Pyrrole and pyrazole derivatives as potentiators of glutamate receptors
05/06/2005WO2005040109A1 Ligands of melanocortin receptors and compositions and methods related thereto
05/06/2005WO2005039564A1 Phthalimide compounds useful as protein kinase inhibitors
05/06/2005WO2005039496A2 Inhibitors of cathepsin s
05/06/2005WO2005028443A3 Protein tyrosine kinase enzyme inhibitors
05/06/2005WO2005005395A3 Arylamine-substituted quinazolinone compounds
05/06/2005WO2004092116A8 Bicyclic compounds having bradykinin receptors affinity and pharmaceutical compositions thereof
05/06/2005CA2543644A1 Pyrazine derivatives and pharmaceutical use thereof
05/06/2005CA2543079A1 Dicationic triaryl analogs as anti-protozoan agents
05/06/2005CA2542963A1 Inhibitors of cathepsin s
05/06/2005CA2542064A1 Tao kinase modulators and methods of use
05/06/2005CA2541460A1 Indolinone derivatives and their use in treating disease-states such as cancer
05/06/2005CA2540765A1 Pyrimidin-2-amine derivatives and their use as a2b adenosine receptor antagonists
05/06/2005CA2539726A1 4-azole substituted imidazole compositions useful as inhibitors or c-met receptor tyrosine kinase
05/05/2005US20050096478 Derivatives of fluoro(hydro)carbons attached to an -alkylene-oxy-carbonyl-leaving group; reactive with amine-containing compounds to form a fluoro-substituted carbamyl protective group useful for the efficient separation, recovery and purification of synthsized organic compounds; libraries
05/05/2005US20050096468 Inhibitors of histone deacetylase
05/05/2005US20050096378 Fundic relaxation; dyspepsia, early satiety, bloating and anorexia; 1-[3-[[(3,4-dihydro-2H-1-benzopyran-2-yl- )methyl]amino]-2-hydroxypropyl]-2,4-imidazolidinedione
05/05/2005US20050096368 Heterocyclo-substituted imidazoles for the treatment of inflammation
05/05/2005US20050096363 Activator of peroxisome proliferator-activated receptor delta
05/05/2005US20050096359 melanocortin receptor agonist, antagonist; preventing or treating inflammatory diseases, AIDS, obesity, bulimia, anorexia or sexual dysfunction; N-(2-aminoethyl)-3'-[1-{N-(1-benzylpiperidin-4-yl)-N-(2-naphthylacetyl)aminoethyl][1,1'-biphenyl)-2-carboxamide dihydrochloride
05/05/2005US20050096354 Process for the preparation of substituted aryl pyrazoles
05/05/2005US20050096347 Beta3-Adrenoreceptor agonists, agonist compositions and methods of using
05/05/2005US20050096344 controlling signal transduction; anticancer agents; antitumor agents; angiogenesis inhibitors; atherosclerosis; vision defects; antidiabetic agents; antiinflammatory agents; antiischemic agents
05/05/2005US20050096325 use of specified inhibitors of chemokine receptors to treat inflammatory diseases such as asthma, allergic rhinitis, atopic dermatitis, inflammatory bowel diseases, idiopathic pulmonary fibrosis, bullous pemphigoid, allergic colitis, eczema, conjunctivitis, familial eosinophilia
05/05/2005US20050096316 Quinoline derivatives(2)
05/05/2005US20050096312 Antiserotonine agents; antidepressants; eating disorders; anxiolytic agents; sleep disorders; gastrointestinal disorders; cardiovascular disorders; muscular disorders; endocrine system diseases; muscular disorders; psychological disorders
05/05/2005US20050096309 For use as anticoagulant agents for therapy of thromboembolic disorders
05/05/2005US20050096278 Antibacterial agents
05/04/2005EP1528061A1 Heterocyclic derivatives which inhibit factor Xa
05/04/2005EP1527067A1 4-trifluoromethylpyrazolyl substituted pyridines and pyrimidines
05/04/2005EP1527062A1 Tetrahydropyran derivatives and their use as therapeutic agents
05/04/2005EP1527053A1 Process for preparing rizatriptan
05/04/2005EP1527051A1 Pyrimidyl sulphone amide derivatives as chemokine receptor modulators
05/04/2005EP1527050A1 Quinoline derivatives and their use as mycobacterial inhibitors
05/04/2005EP1527049A2 Fused heterocyclic compounds as peptidase inhibitors
05/04/2005EP1527046A1 Indoline derivatives substituted in position 6, production and use thereof as medicaments
05/04/2005EP1526895A2 Methods for treating carbonic anhydrase mediated disorders
05/04/2005EP1526869A1 Compositions of a cyclooxygenase-2 selective inhibitor and a carbonic anhydrase inhibitor for the treatment of neoplasia
05/04/2005EP1446399B1 Piperazine derivatives having sst1 antagonistic activity
05/04/2005EP1317448B1 Pyrazole compounds useful as protein kinase inhibitors
05/04/2005EP1159254B1 Oxyalkylene-substituted aminophenol intermediate
05/04/2005EP1119567B1 Quinazoline derivatives
05/04/2005EP0946537B1 Process for the stereoselective production of nitro-enamine compounds
05/04/2005EP0886637B9 Inhibitors of microsomal triglyceride transfer protein and method
05/04/2005EP0755923B1 Ameliorant or remedy for symptoms caused by Ischemic diseases and Phenylpiperidine compounds useful therefor
05/04/2005CN1612856A 1, 3-diarylprop-2-en-1-ones, compositions containing same and use thereof
05/04/2005CN1612733A Benzimidazoles useful as protein kinase inhibitors
05/04/2005CN1199971C Quaternary ammonium compounds as tachykinin antagonists
05/04/2005CN1199963C Coumarin derivatives with COMT inhibiting activity
05/04/2005CN1199954C Benzodiazepine derivatives
05/04/2005CN1199947C Process for production of pyridine derive
05/03/2005US6887998 Process for 8-carboxamido-2,6-methano-3-benzazocines
05/03/2005US6887893 Methods and compositions for treatment and prevention of tumors, tumor-related disorders and cachexia
05/03/2005US6887889 Aryl and biaryl piperdines with MCH modulatory activity
05/03/2005US6887877 Viricide for hepatitis virus
05/03/2005US6887875 2,5-diarypyrimidine compounds
05/03/2005US6887873 Nitrogen heteroaromatic ring connected with the same or another aromatic ring through a triazine distribution agent; anticancer agents
05/03/2005US6887870 Useful as antianginal and cardioprotective agents; for therapy and prophylaxis of angina pectoris, cardiac dysfunction, myocardial necrosis, and arrhythmia
05/03/2005US6887865 N-heterocyclic derivatives as NOS inhibitors
05/03/2005US6887864 Anticancer agents, a benzoylamino-azepan-3-yl-isonicotinamide compounds
05/03/2005US6887854 Absorption, fluorescence; using light for optical medical diagnosis
05/03/2005CA2236208C Substituted sulphonylamino (thio)carbonyl compounds as herbicides
05/03/2005CA2149886C Process for preparing tetrazolyl-benzopyranones
04/2005
04/28/2005WO2005037830A1 Piperidinylchromen-6-ylsulfonamide compounds as 5-hydroxytryptamine-6 ligands
04/28/2005WO2005037826A1 Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases
04/28/2005WO2005037825A2 Protein kinase inhibitors
04/28/2005WO2005037824A2 Method for the production of amino crotonyl compounds
04/28/2005WO2005037797A1 Substituted pyrazole urea compounds for the treatment of inflammation
04/28/2005WO2005037796A1 Compounds and methods for treating dyslipidemia
04/28/2005WO2005037791A1 Compositions and methods for viral inhibition
04/28/2005WO2005037779A2 Novel dipeptidyl peptidase iv inhibitors used for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases