Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397) |
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06/28/2005 | US6911469 For therapy of disease treatable based on a blood sugar level-depressing activity or a disease treatable based on a cGMP-PDE inhibiting activity, smooth muscle relaxing activity, bronchodilating activity, vasodilating activity |
06/28/2005 | US6911463 Capable of increasing lipolysis and energy expenditure in cells and therefore is useful for treating Type 2 diabetes and/or obesity |
06/28/2005 | US6911461 For treating epilepsy, epileptogenesis, seizure disorders, convulsions, bipolar disorders, mania, depression, anxiety, migraine, neuralgia, chronic pain, neuropathic pain, cerebral ischemia, cardiac arrhythmia, myotonia, cocaine abuse |
06/28/2005 | US6911457 Diabetes imaging probes |
06/28/2005 | US6911453 Substituted 4-phenyltetrahydroisoquinolinium, process for their preparation, their use as a medicament, and medicament containing them |
06/28/2005 | US6911439 Alpha 4 beta 1 integrin and CD49d/ CD29 (vla-4); antiinflammatory agents |
06/28/2005 | US6911424 2′-fluoronucleosides |
06/28/2005 | US6911416 Substituted N-benzoyl-n′(tetrazolylphenyl)-ureas and their use as pest control agents |
06/28/2005 | CA2259977C Taxane derivatives and drugs containing the same |
06/23/2005 | WO2005056549A1 Water-soluble etoposide analogs and methods of use thereof |
06/23/2005 | WO2005056548A1 Enantiomerically pure epoxiconazole and its use as crop protection agent |
06/23/2005 | WO2005056544A1 2- ( (2, 3-dihydroxypropyl) aminomethyl) chromane derivatives for use as beta-3 adrenoreceptor agonists in the treatment of urological and inflammatory disorders |
06/23/2005 | WO2005056543A2 Process for use in the preparation of oxiranes from alkenes, and catalysts for use therein |
06/23/2005 | WO2005056535A1 1,2,3-triazole amide derivatives as inhibitors of cytokine production |
06/23/2005 | WO2005056533A1 Novel benzimidazole and imidazopyridine derivatives and use thereof as a medicament |
06/23/2005 | WO2005056532A1 Indazole derivatives which interact with the g-protein coupled receptor family |
06/23/2005 | WO2005056015A1 Substituted piperazines |
06/23/2005 | WO2005056004A1 N-alkyl pyrroles as hmg-coa reductase inhibitors |
06/23/2005 | WO2005055941A2 Novel m3 muscarinic acetylcholine receptor antagonists |
06/23/2005 | WO2005055940A2 Novel m3 muscarinic acetylcholine receptor antagonists |
06/23/2005 | WO2005055715A2 Insecticidal n-(heteroarylalkyl) alkanediamine derivatives |
06/23/2005 | WO2005040156A8 Azole derivative useful as antifungal agents with reduced interaction with metabolic cytochromes |
06/23/2005 | WO2005037272A8 Benzimidazole derivatives and use thereof as peptide deformylase inhibitors |
06/23/2005 | WO2005034870A3 Amide compounds and ion channel ligands and uses thereof |
06/23/2005 | WO2005033105A3 Vanilloid receptor ligands and their use in treatments |
06/23/2005 | WO2004052366A9 2-aminocarbonyl-quinoline compounds as platelet adenosine diphosphate receptor antagonists |
06/23/2005 | WO2004041258A8 Cyclic nucleotide phosphodiesterase inhibitors, preparation and uses |
06/23/2005 | US20050137399 A lithium-free reaction to produce a substituted/unsubstituted 4-amino-3-benzimidazol-2-yl-quinolin-2-one compound by reacting a 2-aminobenzonitrile with a 2-alkyloxycarbonylmethyl-benzimidazole in a solvent in the presence of a sodium or potassium salt of a base; excellent yields |
06/23/2005 | US20050137395 E.g., 6-[(7-iodoquinolin-4-yl)oxy]-N,2-dimethyl-1-benzofuran-3-carboxamide; antiproliferative agent for hyperproliferative disorders being either cancerous or noncancerous; vasculogenesis or angiogenesis inhibitors; adminstered with hypotensive agent, antitumor agents, mitotic inhibitors and others |
06/23/2005 | US20050137243 Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor |
06/23/2005 | US20050137234 Histone deacetylase inhibitors |
06/23/2005 | US20050137230 Factor Xa-inhibitors; preventing thromboembolic illnesses and tumors; 2-amino-N-(2'-methylsulfonylbiphenyl-4-yl)-3-phenylpropionamide |
06/23/2005 | US20050137228 Benzyl sulfonamide derivatives |
06/23/2005 | US20050137224 2-Cyanopyrrolidinecarboxamide compound |
06/23/2005 | US20050137216 Heterocyclic sodium/proton exchange inhibitors and method |
06/23/2005 | US20050137213 4-arylamino-quinazolines and analogs as activators of caspases and inducers of apoptosis; antiproliferative, anticarcinogenic, antimetabolic agents; tubulin and topoisomerase II inhibitors; fungicides; synergistic administration with other anticarcinogenic agents |
06/23/2005 | US20050137212 Hppars activators |
06/23/2005 | US20050137202 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors |
06/23/2005 | US20050137200 Potassium channel modulators; antiarrhythmia agents |
06/23/2005 | US20050137196 Medical devices employing triazine compounds and compositions thereof |
06/23/2005 | US20050137193 Antagonists of the chemokine receptor 9 (CCR9); inhibit TECK ligand; antiinflammatory agents and immunoregulators; inflammatory bowel disease; (2-phenylsulfonamidophenyl)-pyridinyl-methanones; N-[4-chloro-2(pyridine4-carbonyl)-phenyl]4-morpholin-4-yl-benzenesulfonamide |
06/23/2005 | US20050137190 Compositions useful as inhibitors of voltage-gated sodium channels |
06/23/2005 | US20050137187 Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor |
06/23/2005 | US20050137161 Methods and compositions for treating hepatitis C virus |
06/23/2005 | US20050135737 Optical interleaver |
06/23/2005 | DE10353657A1 New quinolonyl- or benzopyranonyl-substituted indole derivatives are 5HT(1A)- and/or 5HT(1D)-agonists useful e.g. as anxiolytic, antidepressant, neuroleptic and/or antihypertensive agents |
06/23/2005 | CA2549273A1 Novel m3 muscarinic acetylcholine receptor antagonists |
06/23/2005 | CA2549272A1 Novel m3 muscarinic acetylcholine receptor antagonists |
06/23/2005 | CA2548922A1 2- ( (2, 3-dihydroxypropyl) aminomethyl) chromane derivatives for use as beta-3 adrenoreceptor agonists in the treatment of urological and inflammatory disorders |
06/23/2005 | CA2548426A1 Substituted piperazines |
06/23/2005 | CA2547573A1 N-alkyl pyrroles as hmg-coa reductase inhibitors |
06/23/2005 | CA2547410A1 1,2,3-triazole amide derivatives as inhibitors of cytokie production |
06/23/2005 | CA2547391A1 Novel benzimidazole and imidazopyridine derivatives and use thereof as a medicament |
06/22/2005 | EP1542992A2 Process for preparing quinazoline rho-kinase inhibitors and intermediates thereof |
06/22/2005 | EP1542990A1 Novel imidazole compounds as transforming growth factor (tgf) inhibitors |
06/22/2005 | EP1542987A1 Piperidine-n-oxide-derivatives |
06/22/2005 | EP1542980A1 5-aryltetrazole compounds, compositions thereof, and uses therefor |
06/22/2005 | EP1542977A1 2,5-dioxoimidazolidin-4-yl acetamides and analogues as inhibitors of metalloproteinase mmp12. |
06/22/2005 | EP1542692A1 Amino-pyridine, -pyridine and pyridazine derivatives for use as vanilloid receptor ligands for the treatment of pain |
06/22/2005 | EP1542685A1 Triazole derivatives as transforming growth factor (tgf) inhibitors |
06/22/2005 | EP1542684A2 Novel pyrazole compounds as transforming growth factor (tgf) inhibitors |
06/22/2005 | EP1542675A1 Compounds useful for the inhibition of aldh |
06/22/2005 | EP1542667A2 Ureido substituted benzoic acid compounds and their use for nonsense suppression and the treatment of disease |
06/22/2005 | EP1268466B1 Decahydro-isoquinolines |
06/22/2005 | EP1154774B1 Quinazoline derivatives as angiogenesis inhibitors |
06/22/2005 | EP1082127B1 Succinamide inhibitors of interleukin-1beta converting enzyme |
06/22/2005 | CN1630653A Pyrazolyl-substituted heterocycles and their use as phytosanitary products |
06/22/2005 | CN1630651A Novel gamma secretase inhibitors |
06/22/2005 | CN1630650A Nitrogenous heterocyclic compound and medicine thereof |
06/22/2005 | CN1630645A 5-HT receptor ligands and uses thereof |
06/22/2005 | CN1630644A Pyridine and pyrimidine derivatives |
06/22/2005 | CN1630642A Benzenesulfonamide derivatives |
06/22/2005 | CN1630555A Hydroxylation of beta-dicarbonyls with zirconium catalysts |
06/22/2005 | CN1630517A CXCR4-antagonistic drugs composed of nitrogen-containing compound |
06/22/2005 | CN1629158A Pyran derivative |
06/22/2005 | CN1207288C Retroviral protease inhibiting compounds |
06/22/2005 | CN1207283C 4-aminopiperidine derivatives and their use as medicine |
06/21/2005 | US6908938 Heterocyclic aromatic compounds useful as growth hormone secretagogues |
06/21/2005 | US6908936 Respiratory syncytial virus |
06/21/2005 | US6908935 Calcium receptor modulating agents |
06/21/2005 | US6908931 1-(2,2-diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinoline- 2-carbaldehyde; for treating sleep disorders |
06/21/2005 | US6908924 N4-acylcytosine-1,3-dioxolane nucleosides for treatment of viral infections |
06/21/2005 | US6908922 Linear cyclic ureas |
06/21/2005 | US6908921 Quinoxalinone derivatives as bradykinin B1 antagonists |
06/21/2005 | US6908920 Pyrimidine derivatives |
06/21/2005 | US6908919 Substituted polycyclic aryl and heteroaryl pyrazinones useful for selective inhibition of the coagulation cascade |
06/21/2005 | US6908915 Tricyclic compounds and their uses as antiarrhythmic antifibrillatory and defibrillatory agents |
06/21/2005 | CA2309473C New 4-arylpiperidine derivatives for the treatment of pruritus |
06/21/2005 | CA2250372C 6-phenylpyridyl-2-amine derivatives |
06/16/2005 | WO2005054430A2 Hepatitis c virus inhibitors |
06/16/2005 | WO2005054233A1 Benzoyl amino pyridil carboxylic acid derivatives as gluokinase activators |
06/16/2005 | WO2005054229A1 4-[(arylmethyl)aminomethyl]piperidine derivatives, preparation thereof and application of same in therapeutics |
06/16/2005 | WO2005054227A1 (4-phenylpiperazin-1-yl)acylpiperidine derivatives, preparation thereof and application of same in therapeutics |
06/16/2005 | WO2005054212A2 Electroluminescent device |
06/16/2005 | WO2005054201A1 6-alkenyl and 6-phenylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(adp-ribose) polymerase inhibitors |
06/16/2005 | WO2005054192A1 Cosmetic process for preventing or treating the signs of skin ageing or the orange-peel appearance |
06/16/2005 | WO2005054179A2 Hydroxamic acid esters and pharmaceutical use thereof |
06/16/2005 | WO2005053686A1 Indolinone based protein kinase inhibitors |
06/16/2005 | WO2005053663A2 Norepinephrine reuptake inhibitors useful for treatment of cognitive failure |
06/16/2005 | WO2005053614A2 Advanced indolinone based protein kinase inhibitors |