Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
02/2005
02/03/2005WO2003106450A8 Phenylaminopyrimidines and their use as rho-kinase inhibitors
02/03/2005US20050027129 Novel heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them
02/03/2005US20050027121 Heterocyclic carboxy amines such as (2R)-1-[3,5-Bis(trifluoromethyl)benzoyl]-4-[4-((3S)-3-ethylmorpholino)-2-butynyl]-2-[(1H-indol-3-yl)methyl]piperazine, used as substance P and neurokinin antagonist for prophylaxis of diseases
02/03/2005US20050026991 mono-N-substituted amide monohydroxyamide derivatives, e.g., 1-Benzyl-3-(3,4-dichloro-benzyloxy)-1H-pyrrole-2,4-dicarboxylic acid 2-[(1-benzyl-piperidin-4-yl)-amide]4-hydroxyamide, that modulate levels of gene expression in cellular systems, including cancer cells
02/03/2005US20050026988 Cyclopenta'b! indole derivatives as spla inhibitors
02/03/2005US20050026985 Such as N-{5-[1-(4-tert-butylphenyl)-3-pyridin-2-yl-1H-pyrazol-5-yl]pentanoyl}tyrosinamide; useful for the treatment of mammalian infertility
02/03/2005US20050026976 Isoindolinone kinase inhibitors
02/03/2005US20050026971 New effector conjugates, process for their production and their pharmaceutical use
02/03/2005US20050026970 Antiproliferative agents, enzyme inhibitor for treating cancer, restenosis, psoriasis, autoimmune disease, atherosclerosis, osteoarthritis, rheumatoid arthritis, heart failure, chronic pain, and neuropathic pain; chemical synthesis
02/03/2005US20050026969 Heterocyclic compounds useful as malonyl-CoA decarboxylase inhibitors
02/03/2005US20050026965 Pharmaceutical uses and synthesis of nicotinanilide-N-oxides
02/03/2005US20050026959 Ethanol solvate of (-)-cis-2-(2-chloropheny)-5,7-dihydroxy-8-[4R-(3S-hydroxy-1-methyl)piperidinyl]-4H-1benzopyran-4-one
02/03/2005US20050026956 Carbinols for the treatment of neuropathic dysfunction
02/03/2005US20050026954 Muscarinic receptor antagonists; overactive bladder, irritable bowel syndrome, chronic obstructive pulmonary disease, and asthma
02/03/2005US20050026923 For therapy of viral diseases
02/03/2005US20050026916 Heterocyclic compounds as P2X7 ion channel blockers
02/03/2005US20050026915 As melanin concentrating hormone (MCH)receptor antagonists, for prevention or treatment of obesity or eating disorders; (2E)-3-(4-chlorophenyl)-N-[2-(dimethylamino)quinolin-6-yl]prop-2-enamide
02/03/2005US20050026914 Pyrimidine or pyridine carbamate compounds as for example 1,1-dimethylethyl 4-(4-((4-((((2,6-dimethylphenyl)oxy)carbonyl)(4-(methyloxy)phenyl)amino)-2-pyrimidinyl)amino)phenyl)-1-piperazinecarboxylate; for the treatment of protein tyrosine kinase-associated disorders
02/03/2005US20050026913 N-substituted aniline and diphenylamine analogs; exhibit improved PDE4 inhibition; novel rolipram analogs which facilitate entry into cells, especially cells of the nervous system
02/03/2005US20050026911 Benzotriazapinone salts and methods for using same
02/03/2005US20050026905 2-Phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
02/03/2005US20050026903 Pyrazole compound; gastrointestinal disorders; central nervous system disorders
02/03/2005US20050023507 pi-electron donor group bonded to a pi-electron conjugated bridge group bonded to a mono- or dicyanodihydrofuran acceptor; large hyperpolarizability, dipole moment, and electrooptic coefficients; electrooptics
02/03/2005CA2534262A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005CA2532980A1 2-aminopyrimidine and 2-aminopyridine-4-carbamates for use in the treatment of autoimmune diseases
02/03/2005CA2532443A1 Tyrosine kinase inhibitors
02/03/2005CA2532403A1 Ppar active compounds
02/03/2005CA2532400A1 Tyrosine kinase inhibitors
02/03/2005CA2532248A1 Novel compounds
02/03/2005CA2530352A1 Quinolone derivative or salt thereof
02/03/2005CA2530302A1 Novel aminobenzophenone compounds
02/02/2005EP1502916A1 Piperidine derivatives having ccr3 antagonism
02/02/2005EP1502915A1 Compounds with a sulfamate group
02/02/2005EP1501827A2 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acid and their use as protease inhibitors
02/02/2005EP1501817A1 Imidazolinylmethyl aralkylsulfonamides
02/02/2005EP1501815A1 Substituted phenylacetamides and their use as glucokinase activators
02/02/2005EP1501812A1 Pna monomer and precursor
02/02/2005EP1501808A1 Tachykinin receptor antagonists
02/02/2005EP1501807A1 Sulfonylquinoxalone acetamide derivatives and related compounds as bradykinin antagonists
02/02/2005EP1501805A1 Substituted pyrazolyl compounds for the treatment of inflammation
02/02/2005EP1501804A1 Isoquinoline derivatives mao-b inhibitors
02/02/2005EP1501803A2 Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity
02/02/2005EP1501801A1 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as vla-4 inhibitors
02/02/2005EP1501800A1 Bombesin antagonists
02/02/2005EP1501797A1 3-substituted amino-1h-indole-2-carboxylic acid and 3-substituted amino-benzo[b]thiophene-2-carboxylic acid derivatives as interleukin-4 gene expression inhibitors
02/02/2005EP1501796A1 3-substituted amino-1h-indole-2-carboxylic acid and 3-substituted amino-benzo[b]thiophene-2-carboxylic acid derivatives as interleukin-4 gene expression inhibitors
02/02/2005EP1501795A1 Cinnamic acid amides
02/02/2005EP1501786A1 Biphenyl carboxamides
02/02/2005EP1501516A1 A process for the preparation of benazepril hydrochloride
02/02/2005EP1501514A2 Protein kinase modulators and methods of use
02/02/2005EP1501508A1 Inhibitors of histone deacetylase
02/02/2005EP1501504A1 1-substituted imidazole derivatives as nos inhibitors
02/02/2005EP1501467A2 Heterocyclo inhibitors of potassium channel function
02/02/2005EP1414814B1 6-aryl-4-aminopicolinates and their use as herbicides
02/02/2005EP1303506B1 6-heteroarylphenanthridines
02/02/2005EP1292591B1 Substituted bicyclic derivatives for the treatment of abnormal cell growth
02/02/2005EP1286955B1 Aryl and heteroarylcyclopropyl oxime ethers and their use as fungicides
02/02/2005CN1575290A Pyrimidine derivatives and pharmaceutical compositions containing that compounds
02/02/2005CN1575284A Substituted triazole diamine derivatives as kinase inhibitors
02/02/2005CN1575283A Piperazine derivatives with CCRI receptor antagonist activity
02/02/2005CN1575273A 3, 4-di-substituted cyclobutene-1, 2-diones as CXC-chemokine receptor antagonists
02/02/2005CN1575177A Cxcr3 antagonists
02/02/2005CN1575174A Pharmaceutically active isoindoline derivatives
02/02/2005CN1187342C Substituted 1-aminoalkyl-lactams compound and their use as muscarinic receptor antagonists
02/02/2005CN1187336C New imidazole derivatives
02/02/2005CN1187331C Esters of 3-hydroxy-piperidinemethanol derivatives, pharmaceutical composition containing same and their preparation method and uses
02/01/2005US6849739 N-heterocyclic derivatives as NOS inhibitors
02/01/2005US6849660 Antimicrobial biaryl compounds
02/01/2005US6849658 Biaromatic compounds and pharmaceutical and cosmetic compositions comprising them
02/01/2005US6849657 Osteoporosis; increase bone density
02/01/2005US6849653 Substituted pyrazolyl benzenesulfamide compounds for the treatment of inflammation
02/01/2005US6849646 Chromenone and chromanone derivatives as integrin inhibitors
02/01/2005US6849643 Indazolyl-substituted pyrroline compounds as kinase inhibitors
02/01/2005US6849639 Anticancer agents, antiinflamatory agents, osteoporosis, atherosclerosis
02/01/2005US6849636 Useful for treatment of noninsulin-dependent diabetes, hyperglycemia, obesity, insulin resistance, dyslipidemia, hyperlipidemia, hypertension, Metabolic Syndrome
02/01/2005US6849634 Potassium channel inhibitors
02/01/2005US6849631 Semicarbazides and their uses
02/01/2005US6849629 Heteroaromatic substituted sulfonyl or sulfoxide or thio-pyridazinone derivatives, useful for treating diabetic complications and cardiovascular disorders
02/01/2005US6849625 Use in manufacture of a medicament for use as an anti-invasive agent in containment and/or treatment of solid tumor disease
02/01/2005US6849622 May be useful for the prophylaxis and treatment of diabetes, particularly type 2 diabetes, and for prophylaxis and treatment of other diseases induced or exacerbated by impaired glucose tolerance
02/01/2005US6849621 Treating: allergy, allergy-induced airway responses, congestion, hypotension, cardiovascular disease, hypotension, diseases of the GI tract, hyper and hypo motility and acidic secretion of the gastrointestinal tract, obesity, sleep
01/2005
01/27/2005WO2005007650A1 Chemical compounds containing tocopherol and at least one additional pharmaceutical active substance
01/27/2005WO2005007647A1 Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
01/27/2005WO2005007645A1 Substituted 4-amino-1-benzylpiperidine compounds
01/27/2005WO2005007643A1 Novel acridine derivatives and use thereof as medicaments
01/27/2005WO2005007632A1 Substituted pyridazinones as inhibitors of p38
01/27/2005WO2005007628A1 Tetrahydroquinoline derivatives as cannabinoid receptor modulators
01/27/2005WO2005007165A1 Pyrimidine-2, 4-dione derivatives as gonadotropin-releasing hormone receptor antagonists
01/27/2005WO2005007163A1 Antipruritic agent containing chroman compound as active ingredient
01/27/2005WO2005007157A1 Pyrazolines as par-1 antagonists for treatment of cardiovascular diseases
01/27/2005WO2005007111A2 Tetrahydroquinoline derivatives as cannabinoid receptor modulators
01/27/2005WO2004098518A3 Pyrazole-amide compounds useful as kinase inhibitors
01/27/2005WO2004085418A3 Xanthones, thioxanthones and acridinones as dna-pk inhibitors
01/27/2005WO2004064972A3 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions
01/27/2005US20050020661 Antidiabetic agents
01/27/2005US20050020652 For example, 2-(4-{2-[1-(4-tert-Butyl-benzyl)-3-methyl-2-oxo-imidazolidin-4-yl]-ethoxy}-2-methyl-phenoxy)-2-methyl-propionic acid, 2-(4-{3-[1-(4-tert-Butyl-benzyl)-3-methyl-2-oxo-imidazolidin-4-yl]-propyl}-2-methyl-phenoky)-2-methyl-propionic acid; for treating diabetes mellitus
01/27/2005US20050020648 "PGI2-preferring" (IP) receptors; p-(imidazolin-2-ylamino-optional alkyl)phenyl p'-substituted ethers or sulfides, e.g., 4,5-Dihydro-1H-imidazol-2-yl)-[4-(4-isopropoxy-phenylsulfanyl)-phenyl]-amine, used to induce hyperalgesia
01/27/2005US20050020635 C7 carbamoyloxy substituted taxane compositions
01/27/2005US20050020634 Acat inhibitors; cardiovascular disorders; restenosis; Alzheimer's disease
01/27/2005US20050020631 3-Substituted benzofurans as therapeutic agents