Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
06/2005
06/09/2005WO2005051919A1 Aminopyrazole derivatives as gsk-3 inhibitors
06/09/2005WO2005051913A1 Cyclic amine derivative having heteroaryl ring
06/09/2005WO2005051911A1 4-phenylpiperidine derivatives as renin inhibitors
06/09/2005WO2005051879A1 Process for producing epoxytriazole compound and intermediate therefor
06/09/2005WO2005051391A1 Quinazolinone compounds with reduced bioaccumulation
06/09/2005WO2005051387A1 Amino substituted pyridinyl methanone compounds useful in treating kinase disorders
06/09/2005WO2005051382A1 Agent enhancing lipid-loewring effect
06/09/2005WO2005051381A1 Substituted urea-octatydroindols as antagonists of melanin concentrating hormone receptor 1 (MCH1R)
06/09/2005WO2005051380A1 Substituted urea-octahydroindols as antagonists of melanin concentrating hormone receptor 1 (mch1r)
06/09/2005WO2005035508A3 Method for producing acyl urea derivatives, salts of said acyl urea derivatives, and the use thereof as pesticides
06/09/2005WO2005016893A3 2,4-pyrimidinediamine compounds for use in the treatment or prevention of autoimmune diseases
06/09/2005WO2003088897A3 Fab i inhibitors
06/09/2005US20050124682 Such as N-{2-[5-(methylthio)-1H-indol-3-yl]ethyl}acetamide for treatment of disorders of the melatoninergic system; hormone replacement therapy
06/09/2005US20050124677 Peptide deformylase inhibitors
06/09/2005US20050124672 Antineoplastic agents, analgesics, antipyretics; prostaglandin E2 receptor antagonists; 3-Methyl-4-[6-[N-isobutyl-N-(2-thiazolylsulfonyl)amino]indan-5-yloxymethyl]benzoic acid, a C1-4 alkyl ester, or a non-toxic salt
06/09/2005US20050124671 Benzylcycloalkyl amines as modulators of chemokine receptor activity
06/09/2005US20050124664 Compounds for treatment of cardiovascular disorders using inhibitors of plasmnogen activator as anticoagulants for blood
06/09/2005US20050124654 Compounds and methods of use
06/09/2005US20050124641 Process for preparing chiral diol sulfones and dihydroxy acid HMG CoA reductase inhibitors
06/09/2005US20050124640 Pyrimidine derivatives useful as inhibitors of PKC-theta
06/09/2005US20050124638 Benzimidazoles and analogs thereof as antivirals
06/09/2005US20050124634 1,4-dihydropyridine compounds, pharmaceutical compositions, and methods for the treatment of cardiovascular disease
06/09/2005US20050124633 For the treatment of myosin heavy chain-mediated diseases, and in particular, heart failure
06/09/2005US20050124625 For example, ((2R,5S)-4-(8-cyano-quinolin-5-yl)-2,5-dimethyl-piperazine-1-carboxylic acid(4-trifluoromethyl-pyridin-3-yl)-amide); use in treatment of nuclear hormone receptor-associated conditions such as cancer and immune disorders
06/09/2005US20050124619 Medical devices employing triazine compounds and compositions thereof
06/09/2005US20050124614 E. g., 3,5-bis-trifluoromethylphenyl)-4-[(furan-2-ylmethyl)-aminocarbonyl]-2-methyl-1-oxo-1,2,3,4-tetrahydroisoquinoline;anticarcinogenic agents; antitumor agents; antiproliferative agents; activators of the caspase cascades; enzyme inhibitors used in combination with radiation or chemotherapy
06/09/2005US20050124610 cyclin dependent kinase (CDK) inhibitors useful in treating or ameliorating a CDK mediated disorder consisting of cervical adenocarcinoma, colon carcinoma and malignant melanoma
06/09/2005US20050124607 5-Substituted quinazolinone compounds useful as alpha 1A/B adrenergic receptor antagonists
06/09/2005US20050124599 Novel benzoimidazole derivatives useful as antiproliferative agents
06/09/2005US20050124577 8-Azaprostaglandin derivative compounds and drugs containing the compounds as the active ingredient
06/09/2005US20050124561 Administering fungicide for mucous membrane; asthma therapy
06/09/2005US20050124532 Using nucleoside, or prodrug thereof
06/09/2005US20050124209 Illuminated electrical cords and outlets
06/09/2005US20050123831 used for ionic conducting materials, electronic conducting materials, colorant, and the catalysis of various chemical reactions
06/09/2005US20050123533 Prodrugs activated by targeted catalytic proteins
06/09/2005CA2547472A1 Cyclic amine derivative having heteroaryl ring
06/09/2005CA2546709A1 Amino substituted pyridinyl methanone compounds useful in treating kinase disorders
06/09/2005CA2546264A1 4-phenylpiperidine derivatives as renin inhibitors
06/09/2005CA2545601A1 Quinazolinone compounds with reduced bioaccumulation
06/09/2005CA2545262A1 Quinazoline derivatives
06/09/2005CA2544857A1 Vitamin d receptor modulators
06/08/2005EP1537870A2 Methods and compositions for treating cancer
06/08/2005EP1537103A1 Antidepressant cycloalkylamine derivates of 2,3-dihydro-1,4-benzodioxan
06/08/2005EP1537102A1 Inhibition of phsphoinostide 3-dinase beta
06/08/2005EP1537100A1 Pyrrolidinedione substituted piperidine-phthalazones as pde4 inhibitors
06/08/2005EP1537099A1 Pyrrole based inhibitors of glycogen synthase kinase 3
06/08/2005EP1537096A2 Derivatives of dioxane-2-alkyl carbamates, preparation method thereof and application of same in therapeutics
06/08/2005EP1537087A1 Novel aminoindazole derivatives as medicines and pharmaceutical compositions containing same
06/08/2005EP1537085A1 Oxytocin inhibitors
06/08/2005EP1537084A1 Substituted 2-alkylamine nicotinic amide derivatives and use there of
06/08/2005EP1537081A1 Dihydropyridine derivatives for use as human neutrophil elastase inhibitors
06/08/2005EP1537078A1 Indoles having anti-diabetic activity
06/08/2005EP1536799A1 Novel 2-amino-4-oxoquinazolones as lxr nuclear receptor binding compounds with partial agonistic properties
06/08/2005EP1536797A1 1-amido-4-phenyl-4-benzyloxymethyl-piperidine derivatives and related comounds as neurokinin-1 (nk-1) antagonsists for the treatment of emesis, depression, anxiety and cough
06/08/2005EP1536784A1 Hetero biaryl derivatives as matrix metalloproteinase inhibitors
06/08/2005EP1370528B1 Mch antagonists and their use in the treatment of obesity
06/08/2005EP1268306A4 Inverted aerosol dispenser
06/08/2005EP1089735B1 4-benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective nmda receptor antagonists
06/08/2005EP0922029B1 Ether muscarinic antagonists
06/08/2005CN1625559A Novel compounds that inhibit factor Xa activity
06/08/2005CN1625554A Amides of aminoalkyl substituted azetidines, pyrrolidines, piperidines and azepanes
06/08/2005CN1625550A Process for the manufacture of organic compounds
06/08/2005CN1625410A 2, 4, 6-triamino-1, 3, 5-triazine derivative
06/08/2005CN1625400A 2, 4-pyrimidinediamine compounds and their uses
06/08/2005CN1623984A Fused-ring compounds and use thereof as drugs
06/08/2005CN1623537A Biaryl sulfonamides and its using method
06/08/2005CN1205245C Epoxy resins, process for production thereof, epoxy resin compositions and crured articles
06/08/2005CN1205213C Method for the production of imidazol-[1,2-c][2,3]-benzodiazepines and intermediates in production thereof
06/08/2005CN1205198C Cyclic ketone derivative and pharmaceutical use thereof
06/08/2005CN1205187C New amidino derivatives and their use as thrombin inhibitors
06/08/2005CN1205185C Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
06/07/2005US6903224 Substituted with purine or pyrimidine bases
06/07/2005US6903219 Process to produce derivatives from UK-2A derivatives
06/07/2005US6903218 Substituted or unsubstituted aryl-1-hydroxyethylaminocarbonylalkyl-chroman-sulfonamide compounds are useful in the treatment of beta-3 receptor mediated conditions
06/07/2005US6903216 Antiarrhythmic agents for the treatment and prophylaxis of atrial arrhythmias, atrial fibrillation (AF) or atrial flutter; potassium channel modulators, beta-blocker
06/07/2005US6903215 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
06/07/2005US6903212 Reacting cyanuric acid with epichlorohydrin to form an addition product; removing epichlorohydrin; dissolving the triglycidyl isocyanurate in a solvent; gradually cooling at a rate within 20 degrees C./hr followed by filtration
06/07/2005US6903180 Epoxy resins, process for preparation thereof, epoxy resin compositions and cured articles
06/07/2005US6903132 Non-peptide GnRH agents, pharmaceutical compositions and methods for their use
06/07/2005US6903131 Administering to a patient an antiangiogenesis or anticancer agent (N,N-disubstituted-3,4-diamino-2,4-dione-pyrroline derivatives for the treatment of chemokine-mediated diseases such as acute and chronic inflammatory disorders and cancer
06/07/2005US6903123 Antitussive agents, anxiolytic agents, analgesics for treating cough, anxiety and pain
06/07/2005US6903120 Modulators of dopamine neurotransmission
06/07/2005US6903116 For therapy and prophylaxis of cancer and stress diseases such as depression
06/07/2005US6903115 Bipiperidine compounds
06/07/2005US6903109 Arylindenopyridines and related therapeutic and prophylactic methods
06/07/2005US6903105 Nitrogen compounds such as 4-(4-(N-(3,5-diamino-6-chloro-pyrazine-2-carbonyl)guanidino)butyl)-N-(2 -aminoethyl)benzamide hydrochloride, administered for prophylaxis of respiratory system disorders; pharmocokinetics
06/07/2005US6903103 Linear cyclic ureas
06/07/2005US6903102 17β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
06/07/2005US6903097 Heterocycle carboxamides as antiviral agents
06/07/2005US6903095 Phthalimido derivatives and a process for their preparation
06/07/2005US6903094 As analgesic
06/07/2005US6903088 Compounds which inhibit leukocyte adhesion mediated by VLA-4
06/07/2005US6903086 Alkoxycarbonylamino benzoic acid or alkoxycarbonylamino tetrazolyl phenyl derivatives as IP antagonists
06/07/2005US6903085 Substituted piperidine compounds useful as modulators of chemokine receptor activity
06/07/2005US6902936 Analyzing protein mixturea, obtain protein mixture, in cubate withblocking agent, digent protein, reduce disulfides, incubate with thiol specific substrates, detect and measure signal from sample
06/07/2005CA2299036C 4-phenyl-4-heteroarylpiperidine derivatives
06/02/2005WO2005049610A1 Process for preparing thiazolidinediones
06/02/2005WO2005049608A1 Quinolonecarboxylic acid compounds having 5-ht4 receptor agonistic activity
06/02/2005WO2005049604A2 Antithrombotic aromatic ethers
06/02/2005WO2005049589A2 Heterocyclic compounds for the treatment of hyperlipidemia, diabetes, obesity and similar diseases