Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
04/2005
04/28/2005WO2005037273A1 Substituted benzazoles and use thereof as inhibitors of raf kinase
04/28/2005WO2005037272A1 Benzimidazole derivatives and use thereof as peptide deformylase inhibitors
04/28/2005WO2005037271A2 Large conductance calcium-activated k channel opener
04/28/2005WO2005037257A2 Novel alanyl-amino peptidase inhibitors for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases
04/28/2005WO2005037199A2 Pyrazole derivatives as cannabinoid receptor modulators
04/28/2005WO2005019168A3 Fluorinated lysine derivatives as dipeptidyl peptidase iv inhibitors
04/28/2005WO2005014517A3 Novel dibenzo[b,f]oxepine-10-carboxamides and pharmaceutical uses thereof
04/28/2005WO2004106299A3 Substituted pyrrole derivatives and their use as hmg-co inhibitors
04/28/2005WO2004065548A3 Synthetic molecules for labeling histidine-rich proteins
04/28/2005WO2004065539A3 Androgen receptor antagonists
04/28/2005US20050090669 Aminoalcohol derivatives as beta-3 adrenergic receptor agonists
04/28/2005US20050090667 Dehydrophenylahistins and analogs thereof and the synthesis of dehydrophenylahistins and analogs thereof
04/28/2005US20050090546 Compounds such as N,N-dibenzylphenylalanine benzyl ester, used as enzyme inhibitors; prophylaxis of lymphadenopathy associated virus, cancer and malaria
04/28/2005US20050090542 crystalline polymorphic dosage forms of anticholesterol agents; statins
04/28/2005US20050090541 Indolinone derivatives and their use in treating disease-states such as cancer
04/28/2005US20050090524 Novel adamantane derivatives
04/28/2005US20050090519 1-Alkyl-4-(3-substitutedphenyl)piperidines
04/28/2005US20050090503 5-HT receptor ligands and uses thereof
04/28/2005US20050090501 Heteroaryl-cyclic acetals
04/28/2005US20050090498 3-Quinolin-2(1h)-ylideneindolin-2-one derivative
04/28/2005US20050090485 7-Arylsulfonamido-2,3,4,5-tetrahydro-1h-benzo'diazepine derivatives with 5ht6 receptor affinity for the reatment of cns disorders
04/28/2005US20050089718 Pyran derivative
04/28/2005US20050089713 Organic electroluminescent element
04/28/2005CA2542807A1 Novel dipeptidyl peptidase iv inhibitors used for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases
04/28/2005CA2542723A1 Novel alanyl-amino peptidase inhibitors for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases
04/28/2005CA2542653A1 Substituted benzazoles and use thereof as inhibitors of raf kinase
04/28/2005CA2542076A1 Substituted tricyclic compounds as protein kinase inhibitors
04/28/2005CA2541509A1 Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases
04/28/2005CA2539755A1 Alkanol and cycloalkanol-amine derivatives and methods of their use
04/27/2005EP1525190A1 Cck-1 receptor modulators
04/27/2005EP1525185A1 Acetylamino benzoic acid compounds and their use for nonsense suppression and the treatment of disease
04/27/2005EP1524979A2 New effector conjugates, process for their production and their pharmaceutical use
04/27/2005EP1524974A2 Transcription factor modulating compounds and methods of use thereof
04/27/2005EP1423110A4 Cbi analogues of cc-1065 and the duocarmycins
04/27/2005EP1373202B1 Preparation of non-crystalline atorvastatin calcium
04/27/2005EP1261327B1 Adenosine receptor modulators
04/27/2005EP0964861B1 Process for the production of tetrazolylbenzopyrans
04/27/2005EP0838453B1 Heterocyclic carboxylic acid derivatives and drugs containing the same
04/27/2005CN1610678A Pyrrolidone carboxamides
04/27/2005CN1610671A Quinoline compounds with 5-HT-antagonistic properties for therapy
04/27/2005CN1610547A N-(2-arylethyl)benzylamines as antagonists of the 5-HT6 receptor
04/27/2005CN1610546A 病毒聚合酶抑制剂 Viral polymerase inhibitor
04/27/2005CN1198820C N-substituted nitrogen heterocyclic compound
04/27/2005CN1198813C Benzofuran derivatives their preparation and use
04/27/2005CN1198807C 5-aryl-1H-1,2,4-triazole compounds as inhibitors of cyclooxygenase-2 and pharmaceutical composition containing the same
04/27/2005CN1198806C Oxodiethylenediamine derivative and light stabilized composition
04/27/2005CN1198804C Amide compounds and use thereof
04/27/2005CN1198801C Indole derivatives
04/27/2005CN1198618C Novel use of 1-[4-(5-cyanoindol-3-yl)butyl]-4-(2-carbamoyl-benzofuran-5-yl)-piperazine and its physiologically acceptable salts
04/26/2005US6884895 Using dihydropyran, triethyl orthoformate and alkyl acrylate
04/26/2005US6884892 Production methods of epoxytriazole derivative and intermediate therefor
04/26/2005US6884815 An amino compound containing imidazole and aromatic, or heteroaromatic rings is useful for treating inflammatory and immune system disorders
04/26/2005US6884808 Acids and salts such as 4-(4-(2-(2-(5,6,7,8-Tetrahydro-5,5,8, 8-tetramethylquinoxalyl))pyrrolyl))benzoic acid, used retinoic acid receptor agonists for the prophylaxis of cancer, skin disorders, asthma, alopecia or autoimmune diseases
04/26/2005US6884804 Inhibitors of Src and other protein kinases
04/26/2005US6884802 Phenanthridines substituted in position 6 by a mono, bi- or tricyclic heteroaryl radical; cyclic nucleotidephosphoesterase (PDE4) inhibitor and useful for treating respiratory system disorders
04/26/2005US6884801 Nitrogen compounds such as N-(4,5-dihydro-1H-imidazol-2-yl-methyl)-2-(methylsulfonyl)aniline, used for prophylaxis of incontinence
04/26/2005US6884782 Amino acid containing compounds useful as modulators of the immune system
04/26/2005US6884758 2,4-Diamino-1,3,5-triazines, their preparation, and their use as herbicides and plant growth regulators
04/26/2005CA2213124C Benzoyl derivatives
04/21/2005WO2005035529A1 Substituted phenanthropyrans
04/21/2005WO2005035524A1 Pyrrolidinyl urea derivatives as angiogensis inhibitors
04/21/2005WO2005035522A1 1-‘2-(4-hydroxyphenyl)-2-hydroxyethyl!-piperidin-4-ol compounds as nmda receptor antagonists
04/21/2005WO2005035521A1 Substituted quinolines as mcr modulators
04/21/2005WO2005035510A1 Derivatives of 4-phenylthiazoles and 4-phenylimidazoles and the use thereof as medicaments for treating neurodegenerative diseases, pain and epilepsy
04/21/2005WO2005035508A2 Method for producing acyl urea derivatives, salts of said acyl urea derivatives, and the use thereof as pesticides
04/21/2005WO2005035507A2 4-aminopyrimidine derivatives for treatment of hyperproliferative disorders
04/21/2005WO2005035499A1 Substituted 2-carbonylamino-6-piperidinaminopyridines and substituted 1-carbonylamino-3-piperidinaminobenzenes as 5-ht1f agonists
04/21/2005WO2005034955A1 Substituted quinolines as protein tyrosine kinase enzyme inhibitors
04/21/2005WO2005034940A2 Dual alanyl aminopeptidase and dipeptidyl peptidase iv inhibitors for functionally influencing different cells and for treating immunological, inflammatory, neuronal and other diseases
04/21/2005WO2005034870A2 Amide compounds and ion channel ligands and uses thereof
04/21/2005WO2005034856A2 Targeted drug-formaldehyde conjugates and methods of making and using the same
04/21/2005WO2005020882A3 Compound capable of binding s1p receptor and pharmaceutical use thereof
04/21/2005WO2005005414A3 Pyrazolyl-indole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
04/21/2005WO2005004606A3 Pyridinylanilides
04/21/2005WO2004094375A3 4 - (3,4 - disubstituted phenyl) - pyrrolidin-2-one compounds as phosphodiesterase 4 inhibitors
04/21/2005US20050085638 Process for producing dioxolane nucleoside analogues
04/21/2005US20050085519 Controlling cell differentiation, cell proliferation; anticancer agents
04/21/2005US20050085510 Drug for gastrointestinal disorders
04/21/2005US20050085509 KInase inhibitors; antiarthritic agents; autoimmune diseases; sepsis; cachexia; Alzheimer's disease; antihistamines; thrombosis; glomerulonephritis; inflammatory bowel disorders; crohn's disese; multiple sclerosis; antitumor agents; skin disorders
04/21/2005US20050085508 Gastrointestinal disorders; antiemetic agents; irritable bowel disorders; antipruritic agents
04/21/2005US20050085507 p-phenylethenyl hydroxamates; anticarcinogenic, antitumor, antiproliferative agents; regulating p21 promoter; improved stability
04/21/2005US20050085505 Quinoline derivatives, process for preparing them and use for the treatment of diseases mediated by s-cd23
04/21/2005US20050085496 Microbiocidal n-phenyl-n-{4-(4-pyridyl)-2-pyrimidin-2-yl}-amine derivatives
04/21/2005US20050085495 Reacting with acry bromide compound; activation withphosphonacetic acid compound; antitumor agents
04/21/2005US20050085476 Polymerase inhibitors; antiischemic agents; brain disorders; cardiovascular disorders; antiinflammatory agents; antiarthritic agents; neurodegenerative agents; Alzheimer's disease; muscular disorders; antidiabetic agents; kidney disorders; viricides; anticancer agents; immunosuppressants
04/21/2005US20050085467 Androgen receptor antagonists
04/21/2005US20050085466 such as 1-[4-(2-oxo-4-trifluoromethyl-1,2-dihydroquinolin-6-ylmethyl)benzenesulfonyl]-piperidine-3-carboxylic acid ethyl ester; for treatment of acne, alopecia, and oily skin; kits
04/21/2005US20050085461 Benzenesulfonamide derivatives
04/21/2005US20050085457 Therapeutic quinolone compounds with 5-ht-antagonistic properties
04/21/2005US20050084451 Novel chelating agents and chelates and their use
04/21/2005CA2542031A1 Pyrimidine derivatives for treatment of hyperproliferative disorders
04/21/2005CA2541831A1 1-'2-(4-hydroxyphenyl)-2-hydroxyethyl!-piperidin-4-ol compounds as nmda receptor antagonists
04/21/2005CA2540868A1 Pyrrolidinyl urea derivatives as angiogenesis inhibitors
04/20/2005EP1523473A1 Indoline derivatives substituted in position 6, production and use thereof as medicaments
04/20/2005EP1349847B1 Oxybenzamides derivatives as factor xa inhibitors
04/20/2005EP1140904B1 Farnesyl protein transferase inhibitors
04/20/2005EP1129077B1 Fluorinated 3,4-dihydroquinoline derivatives used as nos inhibitors
04/20/2005EP0766669B1 Tri-substituted phenyl derivatives useful as pde iv inhibitors
04/20/2005CN1608064A Novel compounds
04/20/2005CN1608061A Therapeutic isoquinoline compounds