Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397) |
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07/26/2005 | US6921774 Administering compounds such as N-(3-(5-Cyano-1-(4-fluoro-phenyl)-1,3-dihydroisobenzofuran-1-yl)-1 -propyl)glycine ethyl ester, for prophylaxis of psychological disorders |
07/26/2005 | US6921767 Such as (2-(4-(3-(1,4,5,6-Tetrahydropyrimidin-2-ylamino)prop oxy)phenyl) -cyclopropyl)acetic acid; for treating angiogenesis/osteoporosis/ humoral hypercalcemia/smooth muscle cell migration/atherosclerosis/arthritis |
07/26/2005 | US6921758 Amino acid derivatives |
07/26/2005 | CA2256609C 5-aroylpyrrol-2-ylmethylarene derivatives as inhibitors of prostaglandin g/h synthase |
07/26/2005 | CA2234642C 3,4-diaryl-2-hydroxy-2,5-dihydrofurans as prodrugs to cox-2 inhibitors |
07/26/2005 | CA2112011C Substituted pyridines |
07/21/2005 | WO2005066162A1 Synthetic compounds and derivatives as modulators of smoking or nicotine ingestion and lung cancer |
07/21/2005 | WO2005066161A1 Tricyclic steroid hormone nuclear receptor modulators |
07/21/2005 | WO2005066160A1 Dutpase inhibitors |
07/21/2005 | WO2005066159A1 Cathepsin cysteine protease inhibitors |
07/21/2005 | WO2005066156A1 Selective kinase inhibitors |
07/21/2005 | WO2005066151A2 Histone deacetylase inhibitors |
07/21/2005 | WO2005066139A2 2-(amino-substituted)-4-aryl pyramidines and related compounds useful for treating inflammatory diseases |
07/21/2005 | WO2005066137A1 2,5-diaryl-1h-imidazole-4-carboxamides as neurokinin-3 receptor modulators for the treatment of central nervous system and peripheral diseases |
07/21/2005 | WO2005066131A1 Non-nucleotide reverse transcriptase inhibitors |
07/21/2005 | WO2005066126A1 Cb1 modulator compounds |
07/21/2005 | WO2005065779A1 Calcitonin gene related peptide receptor antagonists |
07/21/2005 | WO2005065689A1 Dutpase inhibitors |
07/21/2005 | WO2005065681A1 N- hydroxy-3-(3-(1h-imidazol-2-yl)-phenyl)-acrylamide derivatives and related compounds as histone deacetylase (hdac) inhibitors for the treatment of cancer |
07/21/2005 | WO2005065150A2 Mutagenic heterocycles |
07/21/2005 | WO2005042497A3 Benzimidazoles useful as modulators of ion channels |
07/21/2005 | WO2005037824A3 Method for the production of amino crotonyl compounds |
07/21/2005 | WO2005013914A3 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain |
07/21/2005 | WO2004087051A3 Ophthalmic compositions for treating ocular hypertension |
07/21/2005 | WO2004055004A8 Carboxylic acid, phosphate or phosphonate substituted quinazolin-4-ylamine analogues as capsaicin receptor modulators |
07/21/2005 | WO2004050609A8 Substituted ureas and carbamates |
07/21/2005 | US20050159475 Making intermediates to alpha-ethyl-2-oxo-1-pyrrolidine acetamide, also referred to as levetiracetam an antihypoxic agent and antiischemic agent; by reduction via catalytic hydrogenation of an alkenyl intermediate |
07/21/2005 | US20050159473 3-Substituted oxindole beta3 agonists |
07/21/2005 | US20050159470 Histone deacetylase inhibitors |
07/21/2005 | US20050159469 HIV protease inhibiting compounds |
07/21/2005 | US20050159467 5-Aryltetrazole compounds and uses thereof |
07/21/2005 | US20050159463 5-methoxy-3-(2-(2-furamido) ethyl)indole; related to melatonin, but pharmacologicaly and pharmacokineticy different; longer duration, selective localization and greater efficacy |
07/21/2005 | US20050159462 Elevates extracellular adenosine concentration for antiinflammatory and immunosuppressive effects; reaction of imidazole-4-carboxamide with a hydroxyalkylbenzoxazole or benzothiazole compound; 1-[4-hydroxy-1-(2-phenyl-4-benzoxazolyl)-3-pentyl]-imidazole-4-carboxamide |
07/21/2005 | US20050159452 Nociceptin analogs |
07/21/2005 | US20050159451 NMDA (N-methyl-D-aspartate) receptors; eg 6-(4-benzylpiperidin-1-carbonyl)-1,5-dihydro-oxazolo[4,5-f]indole-2-one |
07/21/2005 | US20050159437 Pharmaceutical agents |
07/21/2005 | US20050159436 Bicyclic heterocycles, pharmaceutical compositions containing these compounds, their use and processes for the preparation thereof |
07/21/2005 | US20050159435 [3-Methyl-4-(pyridin-3-yloxy)-phenyl]-(6-piperidin-3-ylethynyl-quinazolin-4-yl)-amine; selective inhibitors of receptor tyrosine kinases and non-receptor tyrosine kinases (eg: Ick, src, abl) or serine/threonine kinases (e.g.: cyclin dependent kinases); carcinoma |
07/21/2005 | US20050159424 pharmaceutically-acceptable salts, prodrugs, solvates, isomers, and/or hydrates thereof, wherein Q is an optionally-substituted phenyl, pyridyl, pyridazinyl, pyrimidinyl, or pyrazinyl ring; R2 is alkyl or an amino group as defined herein; and Z is optionally-substituted oxadiazolyl or C( .dbd. O)NR6, |
07/21/2005 | US20050159418 Nitrogen compounds used as xanthine oxidase inhibitors, for prophylaxis of inflammation, reperfusion injuries, gout or inflammatory bowel disorders |
07/21/2005 | US20050159416 Substituted urea derivatives activate the cardiac sarcomere by potentiating cardiac myosin; systolic heart failure including congestive heart failure; 1-[3-(1-Acetyl-piperidin-3-yloxy)-5-fluoro-phenyl]-3-(6-methoxy-pyridin-3-yl)-urea |
07/21/2005 | US20050159406 Treating impaired fundic relaxation; [1(R),[A-(3 alpha ,4 alpha )]]-1-[1-[(3,4-dihydro-2H-1-benzopyran-2-yl)methyl]-3-methoxy-4-piperidinyl]-2(1H)-pyrimidinone |
07/21/2005 | US20050158785 Non-peptide compounds 2-(5(6)-nitro-2-benzimidazoyl)-5-(4-nitrophenyl)furan; for use in bioassay, fluorescent quantitative analysis; control of gene expression, treatment/prevention of cancer |
07/21/2005 | US20050158708 High thoughput assay; rapid profiling; proteomics |
07/21/2005 | US20050158642 photoreceptors comprising electroconductive substrate, charge generating compounds and photoconductors comprising charge transport compounds such as 9-(3-Chloro-2-hydroxypopyl)-3,3'-bicarbazole on the substrates, used for electrography |
07/21/2005 | US20050156753 Digital sound processing system for a vehicle |
07/21/2005 | CA2559888A1 2-(amino-substituted)-4-aryl pyramidines and related compounds useful for treating inflammatory diseases |
07/21/2005 | CA2552726A1 Cathepsin cysteine protease inhibitors |
07/21/2005 | CA2549396A1 Cb1 modulator compounds |
07/21/2005 | CA2549330A1 Calcitonin gene related peptide receptor antagonists |
07/21/2005 | CA2548283A1 Mutagenic heterocycles |
07/20/2005 | EP1555577A2 Organophotoreceptor with a charge transport material having two epoxidated-carbazolyl groups |
07/20/2005 | EP1555263A1 Process for producing paroxetine hydrochloride hydrate |
07/20/2005 | EP1555262A1 Methods of crystal precipitation |
07/20/2005 | EP1554272A1 Benzimidazoles and benzothiazoles as inhibitors of map kinase |
07/20/2005 | EP1554271A1 Substituted indoles and their use as hcv inhibitors |
07/20/2005 | EP1554269A1 Imidazoles, oxazoles and thiazoles with protein kinase inhibiting activities |
07/20/2005 | EP1554268A1 Pyrazole inhibitors of the transforming growth factor |
07/20/2005 | EP1554264A2 Medicinal arylethanolamine compounds |
07/20/2005 | EP1554263A1 N-benzodioxolyl, n-benzodioxanyl and n-benzodioxepinyl arylcarbonxamide derivatives, and pharmaceutical compositions comprising them |
07/20/2005 | EP1554262A1 Novel tricyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them |
07/20/2005 | EP1554260A1 Aryloxyalkylamine derivatives as h3 receptor ligands |
07/20/2005 | EP1554257A1 Quinazolinone derivatives useful as anti-hyperalgesic agents |
07/20/2005 | EP1554254A1 Novel compounds |
07/20/2005 | EP1554250A1 Novel lactams and uses thereof |
07/20/2005 | EP1554246A2 Dihydropyridinone derivatives as hne inhibitors |
07/20/2005 | EP1554245A1 Piperidinetriol derivatives as inhibitors of glycosylceramidsynthase |
07/20/2005 | EP1553949A2 Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors |
07/20/2005 | EP1553947A2 Quinazolinones and derivatives thereof as factor xa inhibitors |
07/20/2005 | EP1553931A1 Compounds, compositions, and methods |
07/20/2005 | EP1272484B1 Benzoamide piperidine compounds as substance p antagonists |
07/20/2005 | EP1189583B1 Indole derivatives |
07/20/2005 | EP1175402B1 Piperidine derivatives useful as ccr5 antagonists |
07/20/2005 | EP1175401B1 Piperazine derivatives useful as ccr5 antagonists |
07/20/2005 | EP1129077B9 Fluorinated 3,4-dihydroquinoline derivatives used as nos inhibitors |
07/20/2005 | EP1122251B1 Chromene compounds |
07/20/2005 | EP1056717B1 Arylphenyl-substituted cyclic keto-enols |
07/20/2005 | EP1044974B1 N-hydroxyurea derivative and pharmaceutical composition containing the same |
07/20/2005 | CN1642948A Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase |
07/20/2005 | CN1642945A Stable hydrate of a muscarinic receptor antagonist |
07/20/2005 | CN1642944A (3Z) -3-(2, 3-dihydro-1H-ylidene)-1, 3-dihydro-2H-indol-2-ones as kinase inhibitors |
07/20/2005 | CN1642939A Pyridinoylpiperidines as 5-HTLF agonists |
07/20/2005 | CN1642938A New compounds |
07/20/2005 | CN1642937A Process for making chiral 1, 4-disubstituted piperazines |
07/20/2005 | CN1642936A Process for synthesizing chiral N-aryl piperazines |
07/20/2005 | CN1642932A Anomeric derivatives of monosaccharides |
07/20/2005 | CN1642931A Sulfonylamino-derivatives as novel inhibitors of histone deacetylase |
07/20/2005 | CN1642922A Substituted indazoles with anti-cancer activity |
07/20/2005 | CN1642921A 5-substituted-alkylaminopyrazole derivatives as pesticides |
07/20/2005 | CN1642920A 5-substituted-alkylaminopyrazole derivatives as pesticides |
07/20/2005 | CN1642917A Non-peptide GnRH antagonists |
07/20/2005 | CN1642916A Preparation of N1-(2'-pyridyl)-1, 2-propanediamine sulfamic acid and its use in the synthesis of biologically active piperazines |
07/20/2005 | CN1642915A Benzamide derivatives useful as histone deacetylase inhibitors |
07/20/2005 | CN1642912A Sulfonylamino-derivatives as novel inhibitors of histone deacetylase |
07/20/2005 | CN1642911A Phthalimido derivatives as inhibitors of monoamine oxidase B |
07/20/2005 | CN1642907A Carbonylamino-derivatives as novel inhibitors of histone deacetylase |
07/20/2005 | CN1642600A 1, 2-dihydropyrazol-3-ones which controls inflammatory cytokines |
07/20/2005 | CN1642580A Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands |
07/20/2005 | CN1642552A 4-(N-phenylamino)-quinazolines / quinolines as tyrosine kinase inhibitors |
07/20/2005 | CN1642551A Inhibitors of histone deacetylase |