Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
07/2005
07/26/2005US6921774 Administering compounds such as N-(3-(5-Cyano-1-(4-fluoro-phenyl)-1,3-dihydroisobenzofuran-1-yl)-1 -propyl)glycine ethyl ester, for prophylaxis of psychological disorders
07/26/2005US6921767 Such as (2-(4-(3-(1,4,5,6-Tetrahydropyrimidin-2-ylamino)prop oxy)phenyl) -cyclopropyl)acetic acid; for treating angiogenesis/osteoporosis/ humoral hypercalcemia/smooth muscle cell migration/atherosclerosis/arthritis
07/26/2005US6921758 Amino acid derivatives
07/26/2005CA2256609C 5-aroylpyrrol-2-ylmethylarene derivatives as inhibitors of prostaglandin g/h synthase
07/26/2005CA2234642C 3,4-diaryl-2-hydroxy-2,5-dihydrofurans as prodrugs to cox-2 inhibitors
07/26/2005CA2112011C Substituted pyridines
07/21/2005WO2005066162A1 Synthetic compounds and derivatives as modulators of smoking or nicotine ingestion and lung cancer
07/21/2005WO2005066161A1 Tricyclic steroid hormone nuclear receptor modulators
07/21/2005WO2005066160A1 Dutpase inhibitors
07/21/2005WO2005066159A1 Cathepsin cysteine protease inhibitors
07/21/2005WO2005066156A1 Selective kinase inhibitors
07/21/2005WO2005066151A2 Histone deacetylase inhibitors
07/21/2005WO2005066139A2 2-(amino-substituted)-4-aryl pyramidines and related compounds useful for treating inflammatory diseases
07/21/2005WO2005066137A1 2,5-diaryl-1h-imidazole-4-carboxamides as neurokinin-3 receptor modulators for the treatment of central nervous system and peripheral diseases
07/21/2005WO2005066131A1 Non-nucleotide reverse transcriptase inhibitors
07/21/2005WO2005066126A1 Cb1 modulator compounds
07/21/2005WO2005065779A1 Calcitonin gene related peptide receptor antagonists
07/21/2005WO2005065689A1 Dutpase inhibitors
07/21/2005WO2005065681A1 N- hydroxy-3-(3-(1h-imidazol-2-yl)-phenyl)-acrylamide derivatives and related compounds as histone deacetylase (hdac) inhibitors for the treatment of cancer
07/21/2005WO2005065150A2 Mutagenic heterocycles
07/21/2005WO2005042497A3 Benzimidazoles useful as modulators of ion channels
07/21/2005WO2005037824A3 Method for the production of amino crotonyl compounds
07/21/2005WO2005013914A3 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain
07/21/2005WO2004087051A3 Ophthalmic compositions for treating ocular hypertension
07/21/2005WO2004055004A8 Carboxylic acid, phosphate or phosphonate substituted quinazolin-4-ylamine analogues as capsaicin receptor modulators
07/21/2005WO2004050609A8 Substituted ureas and carbamates
07/21/2005US20050159475 Making intermediates to alpha-ethyl-2-oxo-1-pyrrolidine acetamide, also referred to as levetiracetam an antihypoxic agent and antiischemic agent; by reduction via catalytic hydrogenation of an alkenyl intermediate
07/21/2005US20050159473 3-Substituted oxindole beta3 agonists
07/21/2005US20050159470 Histone deacetylase inhibitors
07/21/2005US20050159469 HIV protease inhibiting compounds
07/21/2005US20050159467 5-Aryltetrazole compounds and uses thereof
07/21/2005US20050159463 5-methoxy-3-(2-(2-furamido) ethyl)indole; related to melatonin, but pharmacologicaly and pharmacokineticy different; longer duration, selective localization and greater efficacy
07/21/2005US20050159462 Elevates extracellular adenosine concentration for antiinflammatory and immunosuppressive effects; reaction of imidazole-4-carboxamide with a hydroxyalkylbenzoxazole or benzothiazole compound; 1-[4-hydroxy-1-(2-phenyl-4-benzoxazolyl)-3-pentyl]-imidazole-4-carboxamide
07/21/2005US20050159452 Nociceptin analogs
07/21/2005US20050159451 NMDA (N-methyl-D-aspartate) receptors; eg 6-(4-benzylpiperidin-1-carbonyl)-1,5-dihydro-oxazolo[4,5-f]indole-2-one
07/21/2005US20050159437 Pharmaceutical agents
07/21/2005US20050159436 Bicyclic heterocycles, pharmaceutical compositions containing these compounds, their use and processes for the preparation thereof
07/21/2005US20050159435 [3-Methyl-4-(pyridin-3-yloxy)-phenyl]-(6-piperidin-3-ylethynyl-quinazolin-4-yl)-amine; selective inhibitors of receptor tyrosine kinases and non-receptor tyrosine kinases (eg: Ick, src, abl) or serine/threonine kinases (e.g.: cyclin dependent kinases); carcinoma
07/21/2005US20050159424 pharmaceutically-acceptable salts, prodrugs, solvates, isomers, and/or hydrates thereof, wherein Q is an optionally-substituted phenyl, pyridyl, pyridazinyl, pyrimidinyl, or pyrazinyl ring; R2 is alkyl or an amino group as defined herein; and Z is optionally-substituted oxadiazolyl or C( .dbd. O)NR6,
07/21/2005US20050159418 Nitrogen compounds used as xanthine oxidase inhibitors, for prophylaxis of inflammation, reperfusion injuries, gout or inflammatory bowel disorders
07/21/2005US20050159416 Substituted urea derivatives activate the cardiac sarcomere by potentiating cardiac myosin; systolic heart failure including congestive heart failure; 1-[3-(1-Acetyl-piperidin-3-yloxy)-5-fluoro-phenyl]-3-(6-methoxy-pyridin-3-yl)-urea
07/21/2005US20050159406 Treating impaired fundic relaxation; [1(R),[A-(3 alpha ,4 alpha )]]-1-[1-[(3,4-dihydro-2H-1-benzopyran-2-yl)methyl]-3-methoxy-4-piperidinyl]-2(1H)-pyrimidinone
07/21/2005US20050158785 Non-peptide compounds 2-(5(6)-nitro-2-benzimidazoyl)-5-(4-nitrophenyl)furan; for use in bioassay, fluorescent quantitative analysis; control of gene expression, treatment/prevention of cancer
07/21/2005US20050158708 High thoughput assay; rapid profiling; proteomics
07/21/2005US20050158642 photoreceptors comprising electroconductive substrate, charge generating compounds and photoconductors comprising charge transport compounds such as 9-(3-Chloro-2-hydroxypopyl)-3,3'-bicarbazole on the substrates, used for electrography
07/21/2005US20050156753 Digital sound processing system for a vehicle
07/21/2005CA2559888A1 2-(amino-substituted)-4-aryl pyramidines and related compounds useful for treating inflammatory diseases
07/21/2005CA2552726A1 Cathepsin cysteine protease inhibitors
07/21/2005CA2549396A1 Cb1 modulator compounds
07/21/2005CA2549330A1 Calcitonin gene related peptide receptor antagonists
07/21/2005CA2548283A1 Mutagenic heterocycles
07/20/2005EP1555577A2 Organophotoreceptor with a charge transport material having two epoxidated-carbazolyl groups
07/20/2005EP1555263A1 Process for producing paroxetine hydrochloride hydrate
07/20/2005EP1555262A1 Methods of crystal precipitation
07/20/2005EP1554272A1 Benzimidazoles and benzothiazoles as inhibitors of map kinase
07/20/2005EP1554271A1 Substituted indoles and their use as hcv inhibitors
07/20/2005EP1554269A1 Imidazoles, oxazoles and thiazoles with protein kinase inhibiting activities
07/20/2005EP1554268A1 Pyrazole inhibitors of the transforming growth factor
07/20/2005EP1554264A2 Medicinal arylethanolamine compounds
07/20/2005EP1554263A1 N-benzodioxolyl, n-benzodioxanyl and n-benzodioxepinyl arylcarbonxamide derivatives, and pharmaceutical compositions comprising them
07/20/2005EP1554262A1 Novel tricyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them
07/20/2005EP1554260A1 Aryloxyalkylamine derivatives as h3 receptor ligands
07/20/2005EP1554257A1 Quinazolinone derivatives useful as anti-hyperalgesic agents
07/20/2005EP1554254A1 Novel compounds
07/20/2005EP1554250A1 Novel lactams and uses thereof
07/20/2005EP1554246A2 Dihydropyridinone derivatives as hne inhibitors
07/20/2005EP1554245A1 Piperidinetriol derivatives as inhibitors of glycosylceramidsynthase
07/20/2005EP1553949A2 Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors
07/20/2005EP1553947A2 Quinazolinones and derivatives thereof as factor xa inhibitors
07/20/2005EP1553931A1 Compounds, compositions, and methods
07/20/2005EP1272484B1 Benzoamide piperidine compounds as substance p antagonists
07/20/2005EP1189583B1 Indole derivatives
07/20/2005EP1175402B1 Piperidine derivatives useful as ccr5 antagonists
07/20/2005EP1175401B1 Piperazine derivatives useful as ccr5 antagonists
07/20/2005EP1129077B9 Fluorinated 3,4-dihydroquinoline derivatives used as nos inhibitors
07/20/2005EP1122251B1 Chromene compounds
07/20/2005EP1056717B1 Arylphenyl-substituted cyclic keto-enols
07/20/2005EP1044974B1 N-hydroxyurea derivative and pharmaceutical composition containing the same
07/20/2005CN1642948A Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase
07/20/2005CN1642945A Stable hydrate of a muscarinic receptor antagonist
07/20/2005CN1642944A (3Z) -3-(2, 3-dihydro-1H-ylidene)-1, 3-dihydro-2H-indol-2-ones as kinase inhibitors
07/20/2005CN1642939A Pyridinoylpiperidines as 5-HTLF agonists
07/20/2005CN1642938A New compounds
07/20/2005CN1642937A Process for making chiral 1, 4-disubstituted piperazines
07/20/2005CN1642936A Process for synthesizing chiral N-aryl piperazines
07/20/2005CN1642932A Anomeric derivatives of monosaccharides
07/20/2005CN1642931A Sulfonylamino-derivatives as novel inhibitors of histone deacetylase
07/20/2005CN1642922A Substituted indazoles with anti-cancer activity
07/20/2005CN1642921A 5-substituted-alkylaminopyrazole derivatives as pesticides
07/20/2005CN1642920A 5-substituted-alkylaminopyrazole derivatives as pesticides
07/20/2005CN1642917A Non-peptide GnRH antagonists
07/20/2005CN1642916A Preparation of N1-(2'-pyridyl)-1, 2-propanediamine sulfamic acid and its use in the synthesis of biologically active piperazines
07/20/2005CN1642915A Benzamide derivatives useful as histone deacetylase inhibitors
07/20/2005CN1642912A Sulfonylamino-derivatives as novel inhibitors of histone deacetylase
07/20/2005CN1642911A Phthalimido derivatives as inhibitors of monoamine oxidase B
07/20/2005CN1642907A Carbonylamino-derivatives as novel inhibitors of histone deacetylase
07/20/2005CN1642600A 1, 2-dihydropyrazol-3-ones which controls inflammatory cytokines
07/20/2005CN1642580A Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands
07/20/2005CN1642552A 4-(N-phenylamino)-quinazolines / quinolines as tyrosine kinase inhibitors
07/20/2005CN1642551A Inhibitors of histone deacetylase