Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397) |
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05/19/2005 | US20050107365 adrenoceptor or G-protein coupled receptors inhibitors such as 3-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-6,7-dimethoxy-2H-benzo[1,2,4]-thiadiazine-1,1-dioxide and carriers, used for prophylaxis of urogenital disorders, or as analgesics |
05/19/2005 | US20050104042 Process for the synthesis of amine ethers from secondary amino oxides |
05/19/2005 | DE10348044A1 Duale Alanyl-Aminopeptidase- und Dipeptidylpeptidase IV-Inhibitoren zur funktionellen Beeinflussung unterschiedlicher Zellen und zur Behandlung immunologischer, entzündlicher, neuronaler und anderer Erkrankungen Dual-alanyl aminopeptidase and dipeptidyl peptidase IV inhibitors for the functional influence of different cells and for the treatment of immunological, inflammatory, neuronal and other diseases |
05/19/2005 | DE10348023A1 Neue Alanyl-Aminopeptidasen-Inhibitoren zur funktionellen Beeinflussung unterschiedlicher Zellen und zur Behandlung immunologischer, entzündlicher, neuronaler und anderer Erkrankungen New alanyl aminopeptidase inhibitors for functional interference of different cells and for the treatment of immunological, inflammatory, neuronal and other diseases |
05/19/2005 | CA2551056A1 Benzo[b][1,4]dioxepine derivatives |
05/19/2005 | CA2544678A1 Modulators of cellular adhesion |
05/19/2005 | CA2543943A1 2-azetidinones as anti-hypercholesterolemic agents |
05/19/2005 | CA2543643A1 Pyridine carboxylic acid derivatives as glucokinase modulators |
05/19/2005 | CA2543602A1 Triazole compounds and uses related thereto |
05/18/2005 | EP1531166A2 Cycloaliphatic epoxy compounds containing styrenic, cinnamyl, or maleimide functionality |
05/18/2005 | EP1530567A1 Pyridinyl substituted (1,2,3,)triazoles as inhibitors of the tgf-beta signalling pathway |
05/18/2005 | EP1530472A1 Isoquinoline derivatives as matrix metalloproteinase inhibitors |
05/18/2005 | EP1467991B1 Prucalopride-n-oxide |
05/18/2005 | EP1301502B1 Compounds and their use as glycine transport inhibitors |
05/18/2005 | EP1250047B9 Herbicidal composition |
05/18/2005 | EP1224195B1 C-aryl glucoside sglt2 inhibitors |
05/18/2005 | EP1098885B9 Imidazole compounds and their use as adenosine deaminase inhibitors |
05/18/2005 | CN1617859A 5-sulfanyl-4h-1, 2, 4-triazole derivatives and their use as a medicament |
05/18/2005 | CN1617858A Pyrimidine derivatives as modulators of insulin-like growth factor-1 receptor (igf-1) |
05/18/2005 | CN1617856A Substituted 4-phenyltetrahydroisoquinolinium, process for their preparation, their use as a medicament, and medicament containing them |
05/18/2005 | CN1617855A Inhibitors of cytosolic phospholipase A2 |
05/18/2005 | CN1617852A Alpha-(n-sulphonamido)acetamide derivatives as beta-amyloid inhibitors |
05/18/2005 | CN1617849A Hiv整合酶抑制剂 Hiv integrase inhibitors |
05/18/2005 | CN1617726A N4-acylcytosine nucleosides for treatment of viral infections |
05/18/2005 | CN1617718A N-aryl-N'-arylcycloalkyl-urea derivatives as MCH antagonists for the treatment of obesity |
05/18/2005 | CN1615853A Enhancement of bone growth and inhibition of bone resorption |
05/18/2005 | CN1202108C Spiro compounds, preparing method and intermediate |
05/18/2005 | CN1202107C 2-(4-methiopnoxy)-5-furfural imidazolone derivative with bactericiding activity |
05/18/2005 | CN1202104C 2-phenylpyran-4-one derivatives |
05/18/2005 | CN1202095C Heteroaromatic ring compounds |
05/18/2005 | CN1202093C Substituted heterocyclic compound |
05/18/2005 | CN1202087C Derivatives of acyl-piperazinil-pyrimidins, preparation thereof and application as medicaments |
05/17/2005 | US6894177 Viricides; human immunodeficiency virus |
05/17/2005 | US6894173 Intermediates useful for synthesis of heteroaryl-substituted urea compounds, and processes of making same |
05/17/2005 | US6894164 Process for the preparation of (pyridinylidene)-phthalides |
05/17/2005 | US6894072 Compounds as NS3-serine protease inhibitors of hepatitis C virus |
05/17/2005 | US6894067 5-heteroatom-substituted pyrazoles |
05/17/2005 | US6894065 For therapy of thrombosis, platelet aggregation, coagulation, cancer, inflammatory diseases or respiratory diseases |
05/17/2005 | US6894061 Substituted dihydrophenanthridinesulfonamides |
05/17/2005 | US6894050 3,4,5,6-tetrahydro-2h-(1,2')bipyrazinyl derivatives |
05/17/2005 | US6894047 Triazine compounds useful as sorbitol dehydrogenase inhibitors |
05/17/2005 | US6894042 Azabicyclic compounds for the treatment of disease |
05/17/2005 | US6893859 Antiproliferative agent for treating diseases or conditions characterized by cellular hyperproliferation |
05/17/2005 | CA2306782C Isoquinolines as urokinase inhibitors |
05/17/2005 | CA2301967C Azetidinone derivatives for the treatment of hcmv infections |
05/17/2005 | CA2301543C Azetidinone derivatives for the treatment of hcmv infections |
05/17/2005 | CA2252907C Novel 2,3 disubstituted-4(3h)-quinazolinones |
05/12/2005 | WO2005042533A2 2-cyanopyrrolidinecarboxamides as dipeptidyl peptidase-iv inhibitors |
05/12/2005 | WO2005042524A1 Pyridine carboxamide and methods for inhibiting hiv integrase |
05/12/2005 | WO2005042522A1 Process for the manufacture of the calcium salt of rosuvatatin (e)-7-`4- (4-fluorophenyl) -6-isopropyl-2-`methyl (methylsulfonyl) amino ! pyrimidin -5-yl ! (3r, 5s) -3, 5-dihydroxyhept-6-enoic acid and crystalline intermediates thereof |
05/12/2005 | WO2005042521A2 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors |
05/12/2005 | WO2005042502A1 Amide derivatives |
05/12/2005 | WO2005042500A1 Arylindenopyridines and arylindenopyridines and their use as adenosine a2a receptor antagonist |
05/12/2005 | WO2005042497A2 Benzimidazoles useful as modulators of ion channels |
05/12/2005 | WO2005042496A1 (benzimidazol-2-yl)-phenyl-benzyl-amine derivatives and methods for inhibiting heparanase activity |
05/12/2005 | WO2005042489A1 N-substituted benzene sulfonamides |
05/12/2005 | WO2005042488A1 Pyridine compounds as inhibitors of dipeptidyl peptidase iv |
05/12/2005 | WO2005042487A1 1,4-dihydropyridine compounds, pharmaceutical compositions, and methods for the treatment of cardiovascular disease |
05/12/2005 | WO2005042486A1 1,4-dihydropyridine compounds, pharmaceutical compositions, and methods for the treatment of cardiovascular disease |
05/12/2005 | WO2005042464A1 Androgen receptor modulators |
05/12/2005 | WO2005019209A3 Crystalline anhydrous paroxetine hydrochloride |
05/12/2005 | WO2005018531A3 Pharmaceutical compositions, azo-heterocyclic compounds and method for the production and use thereof |
05/12/2005 | WO2005014539A3 Pyrrole-based hmg-coa reductase inhibitors |
05/12/2005 | WO2005003100A3 4-arylamino-quinazolines as activators of caspases and inducers of apoptosis |
05/12/2005 | WO2005003099A3 Pyrimidines useful as modulators of voltage-gated ion channels |
05/12/2005 | WO2004092145A8 Alpha substituted carboxylic acid as ppar modulators |
05/12/2005 | US20050101781 Eponemycin and epoxomicin analogs and uses thereof |
05/12/2005 | US20050101779 Antagonistic activity to alpha 4 integrin; antiinflammatory agents treating asthma, rheumatoid arthritis, inflammatory bowel diseases, lupus, diabetes; 1-[[(cyclohexyloxy)carbonyl]oxy]ethyl(2S)-2-[(2,6-dichlorobenzoyl)amino]-3-[4-[1-methyl-2,4-dioxo-1,4-tetrahydro-3-(2H)quinazolinyl]phenyl]Propionate |
05/12/2005 | US20050101776 2' or 3' -deoxy and 2' , 3' -dideoxy-beta-L-pentofuranonucleo-side compounds, method of preparation and application in therapy, especially as anti-viral agents |
05/12/2005 | US20050101657 Pyrrole derivatives for preventing or treating cancer sensitive to hormones; administered with luteininzing hormone releasing hormone derivative |
05/12/2005 | US20050101651 Viricides; protease inbhibitors; useful for inhibiting the activity of picornaviral 3C proteases; for example, 6-carbamoyl-4S-{2S-[(5-naphthalen-1-yl-1H-pyrrole-2-carbonyl)-amino-3-phenyl-propionylamino}-hex-2(trans)-enoic acid ethyl ester |
05/12/2005 | US20050101650 (4-(4-(2,3-difluorophenyl)-4H-1,2,4-triazol-3-yl)-1H-pyrrol-2-yl)(2H-pyrrol-1(5H)-yl)methanone; anticarcinogenic, antiproliferative and antimetastasis agent; inhibitors of c-Met protein kinase |
05/12/2005 | US20050101644 Benzylether amine compounds useful as CCR-5 antagonists |
05/12/2005 | US20050101641 Aromatic sulfone hydroxamic acids and their use as protease inhibitors |
05/12/2005 | US20050101634 Bis(5-aeyl-2-pyridyl) derivatives |
05/12/2005 | US20050101630 4-Anilino-, phenoxy-, or phenylthio-substituted; inhibitors of specific kinase enzymes, such as MEK enzymes |
05/12/2005 | US20050101617 Cyanoguanidines and cyanoamidines as ErbB2 and EGFR inhibitors |
05/12/2005 | US20050101614 Heterocyclic GABAA subtype selective receptor modulators |
05/12/2005 | US20050101590 Cannabinoid receptor agonists |
05/12/2005 | US20050101584 Selective estrogen receptor-beta ligands |
05/12/2005 | US20050101568 Methods and compositions for selectin inhibition |
05/12/2005 | US20050101567 Using a sulfonamide containing compound |
05/12/2005 | US20050101540 STAT modulators |
05/12/2005 | US20050100978 Nitropyrimidine derivative for detection and evaluation of kinase inhibitors |
05/12/2005 | CA2544772A1 1,4-dihydropyridine compounds, pharmaceutical compositions, and methods for the treatment of cardiovascular disease |
05/12/2005 | CA2544763A1 1,4-dihydropyridine compounds, pharmaceutical compositions, and methods for the treatment of cardiovascular disease |
05/12/2005 | CA2544350A1 N-substituted benzene sulfonamides |
05/12/2005 | CA2543918A1 Benzimidazoles useful as modulators of ion channels |
05/12/2005 | CA2543715A1 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors |
05/12/2005 | CA2543533A1 2-cyanopyrrolidinecarboxamide compound |
05/12/2005 | CA2543529A1 Pyridine compounds as inhibitors of dipeptidyl peptidase iv |
05/12/2005 | CA2543358A1 Process for the manufacture of the calcium salt of rosuvastatin(e)-7-[4-(4-fluorophenyl)-6-isopropyl-2-[methyl(methylsulfonyl)amino]pyrimidin-5-yl](3r,5s)-3,5-dihydroxyhept-6-enoic acid and crystalline intermediates thereof |
05/12/2005 | CA2543345A1 Androgen receptor modulators |
05/12/2005 | CA2540686A1 Arylindenopyridines and arylindenopyridines and their use as adenosine a2a receptor antagonist |
05/11/2005 | EP1529530A1 Compounds affecting glucokinase |
05/11/2005 | EP1529044A2 Dehydrophenylahistins and analogs thereof and the synthesis of dehydrophenylahistins and analogs thereof |
05/11/2005 | EP1529042A1 Arylamides |
05/11/2005 | EP1528925A1 Quinazoline derivatives for use in the treatment of cancer |
05/11/2005 | EP1528924A1 Mch1r antagonists |
05/11/2005 | EP1363899B1 Quinazolone derivatives as alpha 1a/b adrenergic receptor antagonists |