Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
02/2005
02/22/2005US6858642 For use in pharmaceutical, skin-protective and cosmetic formulations
02/22/2005US6858638 Substituted indazoles, compositions containing them, method of production and use
02/22/2005US6858630 Administering substituted naphthimidazole derivative for therapy of thrombocytopenia
02/22/2005US6858628 Substituted cyclic amine metalloprotease inhibitors
02/22/2005US6858627 For therapy of inflammatory, allergic, or proliferative conditions
02/22/2005US6858626 Cyclic hydroxamic acid as metalloproteinase inhibitors
02/22/2005US6858623 Amidino and guanidino peptidyl compounds
02/22/2005US6858615 Phenyl guanidine sodium channel blockers
02/22/2005US6858609 Substituted diamino-1,3,5-triazine derivatives
02/22/2005US6858603 Acetindine derivatives, their preparation and medicaments containing them
02/22/2005US6858227 Useful in solubilizing lipophilic and relatively water-insoluble compounds; cosmetics, drugs
02/22/2005CA2218493C Benzimidazole compounds and their use as modulators of the gabaa receptor complex
02/22/2005CA2129039C Tri-substituted phenyl derivatives as phosphodiesterase inhibitors
02/17/2005WO2005014587A1 Novel process for the preparation of 2h-chromenes
02/17/2005WO2005014586A1 Novel process for the preparation of 2h-chromenes
02/17/2005WO2005014585A1 Halogenated quinazolinyl nitrofurans as antibacterial agents
02/17/2005WO2005014579A1 Imidazol derivatives of piperdine as histamine antagonists
02/17/2005WO2005014558A1 Condensed pyramidine compounds as inhibitors of voltage-gated ion channels
02/17/2005WO2005014555A1 4,5-dihydro-imidazole as p2x7 ion channel blockers
02/17/2005WO2005014554A1 1h-indazole-3-carboxamide compounds as mapkap kinase modulators
02/17/2005WO2005014552A1 Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors
02/17/2005WO2005014540A1 Cyclic amine base-1 inhibitors having a heterocyclic substituent
02/17/2005WO2005014539A2 Pyrrole-based hmg-coa reductase inhibitors
02/17/2005WO2005014517A2 Novel dibenzo[b,f]oxepine-10-carboxamides and pharmaceutical uses thereof
02/17/2005WO2005013990A1 2-`4-(hydroxymethyl-phenylamino) -piperidine-1-yl!-n- (9h-carbazol-3-yl) - acetamine derivatives and related compounds as neuropeptide y5 (npy5) ligands for the treatment of obesity
02/17/2005WO2005013988A1 2-`4(phenylamino)-piperidin-1-yl!-n-phenyl-acetamine derivatives and related compounds as neuropeptide y5 (npy5) ligands for the treatement of obesity
02/17/2005WO2005013914A2 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain
02/17/2005WO2004110993A3 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
02/17/2005WO2004094386A8 Isoquinoline-5-sulfonic acid amides as inhibitors of akt (protein kinase b)
02/17/2005WO2004092115A3 Hydroxamates as therapeutic agents
02/17/2005WO2004084813A3 Chemical compounds
02/17/2005WO2004067489A8 Hydroxyl compounds and compositions for cholesterol management and related uses
02/17/2005US20050038247 topoisomerase inhibitors such as [5-(4-Cyclopropylcarbamoyl-imidazol-1-yl)-7-pyrimidin-2-yl-1H-benzoimidazol-2-yl]-carbamic acid ethyl ester, used for prophylaxis of bacterial infections in mammals
02/17/2005US20050038246 PPAR active compounds
02/17/2005US20050038243 2, 4-pyrimidinediamine compounds and their uses
02/17/2005US20050038112 prevention, control and treatment of cancer; leukemia
02/17/2005US20050038107 Substituted 2-phenyl benzofurans as estrogenic agents
02/17/2005US20050038101 Substituted 2 5-diamidoindoles as ece inhibitors for the treatment of cardiovascular diseases
02/17/2005US20050038087 Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
02/17/2005US20050038086 Epothilone derivatives and methods for making and using the same
02/17/2005US20050038085 Substituted benzimidazole antiviral agents
02/17/2005US20050038084 Phenylalanine enamide derivatives
02/17/2005US20050038072 Nitrogeneous cyclic ketone derivative, process for producing the same, and use
02/17/2005US20050038069 Tumor necrosis factor antagonist; antiinflammatory agents; such as 2-Cyclopropyl-4-(3,5-dimethyl-4-pyridylmethoxy)-7-methoxy-3H-benzimidazole
02/17/2005US20050038057 3-[2(R)-{hydroxycarbonylpropyl-amino}-2-phenylethyl]-5-(2-fluoro-3-methoxyphenyl)-1-[2-fluoro-6-(trifluoromethyl)benzyl]-6-methyl-pyrimidine-2,4(1H,3H)-dione; utility in treatment of a variety of sex-hormone related conditions in both men and women
02/17/2005US20050038050 Therapeutic treatment of autoimmune disease, transplant rejection, rheumatoid arthritis, by administering 4-(6-chloro-2,3-methylenedioxyanilino)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-tetrahydropyran-4-yloxyquinazoline
02/17/2005US20050038037 N-(naphth-2-ylaminocarbonylacetyl)- or N-(naphth-2-ylcarbonylamino- acetyl)- piperazine derivatives, e.g., 2-[((4-(ethoxycarbonyl)piperazin-1-yl)carbonylmethyl)carbonyl]aminonaphthalene; useful as antithrombotic agents
02/17/2005US20050038035 Heterocyclic amide compounds as apolipoprotein b inhibitors
02/17/2005US20050038031 Novel bicyclic urea derivatives useful in the treatment of cancer and other disorders
02/17/2005US20050038023 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease
02/17/2005US20050038021 2,4,5,-trisubstituted phenylketo-enols for use as pesticides and herbicides
02/17/2005US20050038016 Arylamine-substituted quinazolinone compounds useful as alpha 1A/B adrenergic receptor antagonists
02/17/2005US20050037925 Mixture with other herbicides
02/17/2005US20050037332 Pyridylalkyl-amino-substituted spiro(phthalan-1,9'-xanthene) or xanthene compounds that complex zinc; can measure zinc ions with high sensitivity without damaging cells; can measure fluorescence with a long wavelength excitation light
02/17/2005DE10328533A1 New 6-amino-substituted indolinone derivatives, useful e.g. for treating tumours and angiogenesis, are inhibitors of receptor tyrosine kinases
02/17/2005DE10326918A1 Substituierte Alkylamide Substituted alkyl amides
02/17/2005CA2554566A1 Condensed pyramidine compounds as inhibitors of voltage-gated ion channels
02/17/2005CA2539227A1 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain
02/17/2005CA2534494A1 Pyrrole-based hmg-coa reductase inhibitors
02/17/2005CA2534405A1 Halogenated quinazolinyl nitrofurans as antibacterial agents
02/17/2005CA2534101A1 2-`4-(hydroxymethyl-phenylamino) -piperidine-1-yl!-n- (9h-carbazol-3-yl) - acetamine derivatives and related compounds as neuropeptide y5 (npy5) ligands for the treatment of obesity
02/17/2005CA2534096A1 2-`4(phenylamino)-piperidin-1-yl!-n-phenyl-acetamine derivatives and related compounds as neuropeptide y5 (npy5) ligands for the treatement of obesity
02/17/2005CA2533174A1 Novel dibenzo[b,f]oxepine-10-carboxamides and pharmaceutical uses thereof
02/17/2005CA2532910A1 4,5-dihydro-imidazole as p2x7 ion channel blockers
02/17/2005CA2532452A1 Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors
02/16/2005EP1506967A1 Dipeptidyl peptidase inhibitors
02/16/2005EP1506962A2 Nitrogen-containing aromatic heterocycles
02/16/2005EP1506960A1 Indole compounds as inhibitors of tubulin polymerisation for the treatment of angiogenesis-related disorders
02/16/2005EP1506189A1 Pyrrole derivatives as inhibitors of erk2 and uses thereof
02/16/2005EP1506188A1 Process for the preparation of a hydrate of an anthranilic acid derivative
02/16/2005EP1506187A1 2-thio-substituted imidazole derivatives and their use in pharmaceutics
02/16/2005EP1506185A1 Novel compounds and their use
02/16/2005EP1506176A1 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
02/16/2005EP1506175A1 N-substituted tricyclic 3-aminopyrazoles as pdgf receptor inhibitors
02/16/2005EP1506166A1 Aminotetralin-derived urea modulators of vanilloid vr1 receptor
02/16/2005EP1401832B1 High molecular weight hydroxyphenylbenzotriazole uv-absorbers for thin film applications
02/16/2005EP1281709B1 Novel heterocyclic compounds with anti-inflammatory activity
02/16/2005EP1268463B1 Polycyclic aryl and heteroaryl substituted 4-pyrones useful for selective inhibition of the coagulation cascade
02/16/2005EP1246814B1 Compounds and methods for modulation of estrogen receptors
02/16/2005EP1244617B1 Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone
02/16/2005EP1068200B1 2,4,4-trisubstituted-1,3-dioxolane antifungals
02/16/2005CN1582286A Novel 4-2-furoylaminopiperidines, intermediates in synthesizing the same, process for producing the same and medicinal use of the same
02/16/2005CN1582285A Heteroaryl amines as glycogen synthase kinase 3beta inhibitors (GSK3 inhibitors)
02/16/2005CN1582284A Aminopyrimidines and pyridines
02/16/2005CN1582281A Mch受体拮抗剂 Mch receptor antagonist
02/16/2005CN1582280A 3, 4-di-substituted pyridazinediones as CXC chemokine receptor antagonists
02/16/2005CN1582279A Peroxisome proliferator activated receptor agonists
02/16/2005CN1582277A Amide derivatives as glycogen synthase kinase 3-beta inhibitors
02/16/2005CN1582276A Phenylalanine enamide derivatives
02/16/2005CN1189467C Pharmaceutically active sulfonamide derivatives
02/16/2005CN1189466C New direct chain or cyclic urea, its preparing method and medicinal composition containing them
02/15/2005US6855822 Benzo[b]furan dimers
02/15/2005US6855821 Processes for preparing 1,3-dioxolane nucleosides
02/15/2005US6855730 3-methylidenyl-2-indolinone modulators of protein kinase
02/15/2005US6855726 Heterocyclic amides such as 3-(1-5-((2R,6S)-2,6-dimethyltetra-hydro-1(2H)-pyridinyl)pentyl-2-oxo-1,2 -dihydro-3-quinolinyl) benzenecarboximidamide, administered as anticoagulants or for prophylaxis of cardiovascular disorders
02/15/2005US6855717 A 2(2-(4-benzamido-cyclohexyl)ethyl)-1,2,3,4-tetrahydroisoquinol ine derivatives, for use in psychotherapy
02/15/2005US6855715 Drugs such as 1-(3-Amino-4-chlorobenzoyl-D-phenylglycinyl)-4-(4-fluoro-2 -methylsulphonylphenyl)piperazine, used as anticoagulants
02/15/2005US6855714 For therapy of inflammatory, allergic, infectious or autoimmune diseases
02/15/2005US6855713 Benzimidazole derivatives, a process for their manufacture and use as a medicine
02/10/2005WO2005012320A2 Novel lincomycin derivatives possessing antimicrobial activity