| Patents for C07D 281 - Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms (1,924) |
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| 10/12/2005 | CN1681768A Process for production of high-purity enamines |
| 10/06/2005 | US20050222121 Atypical antipsychotic agents having low affinity for the D2 receptor |
| 10/05/2005 | CN1678597A Novel quaternary ammonium compounds |
| 09/28/2005 | EP1578198A1 Pesticidal dibenzo(hetero)azepine derivatives |
| 09/20/2005 | CA2285119C Retroviral protease inhibiting compounds |
| 09/15/2005 | DE102004010830A1 Neue 1,4-Benzooxazepane oder 1,4-Benzothiazepane und Derivate New 1.4-Benzooxazepane or 1,4-Benzothiazepane and derivatives |
| 09/09/2005 | WO2005082874A1 Novel benzothiazepine and benzothiepine compounds |
| 09/09/2005 | WO2005082873A2 1,4-benzothiazepans and derivatives thereof |
| 09/06/2005 | US6939895 Renalosteodystrophy comprising a compound, or a pharmaceutically acceptable salt or hydrate thereof, having the formula: Ar5-(CHR16)t-W-(CH2)u-CHR17)-NH-CH(R18)-Ar6 wherein: Ar5 is phenyl, indole, carbazole, pyridine, |
| 09/01/2005 | WO2005080976A1 Method of in vivo screening of therapeutic agent for memory/learning dysfunction by schizophrenia |
| 08/31/2005 | EP1567524A1 Thia-epothilone derivatives for the treatment of cancer |
| 08/24/2005 | EP1565448A2 METHOD OF PREPARING 10H-DIBENZO b,f 1,4 THIAZEPIN-11-ONE |
| 08/03/2005 | CN1213036C Novel amide derivatives |
| 07/26/2005 | US6921760 Psychotherapeutic agents. |
| 07/21/2005 | WO2005066146A1 Method for the production of a thiazolo[3,4,5-de][4,1]benzothiazepine-type product |
| 07/21/2005 | WO2004047722A8 METHOD OF PREPARING 10H-DIBENZO[b,f][1,4]THIAZEPIN-11-ONE |
| 07/20/2005 | EP1554250A1 Novel lactams and uses thereof |
| 07/13/2005 | EP1553077A1 Process for production of high-purity enamines |
| 07/13/2005 | CN1639140A Benzothiazepine derivatives for the treatment of hyperlipidemia |
| 06/30/2005 | US20050143576 Process for production of high-purity enamines |
| 06/30/2005 | CA2549072A1 Tricyclic indole hydroxyethylamine derivatives and their use in the treatment of alzheimer's disease |
| 06/22/2005 | CN1207288C Retroviral protease inhibiting compounds |
| 06/14/2005 | US6906058 Prevent bile acid transportation; anticholesterol agents |
| 06/02/2005 | WO2005049585A1 Macrocyclic lactams and pharmaceutical use thereof |
| 06/02/2005 | CA2544751A1 Macrocyclic lactams and pharmaceutical use thereof |
| 06/01/2005 | EP1535913A1 Novel quaternary ammonium compounds |
| 05/25/2005 | EP1532115A2 Protease inhibitors |
| 05/18/2005 | CN1616432A Compound, its use and pharmaceutical compositions comprising same |
| 05/10/2005 | US6890919 Atypical antipsychotic agents having low affinity for the D2 receptor |
| 05/10/2005 | CA2001515C Process for preparing optically active glycidate esters |
| 05/06/2005 | WO2005014590A3 Procedure for preparing 11-(4`2-(2-hydroxyethoxy )ethyl!-1-piperazinyl!-dibenzo`b,f!`1,4!thiazepine |
| 04/19/2005 | US6881839 Process for preparing diltiazem using a heterogeneous trifunctional catalyst |
| 04/14/2005 | US20050080265 Sleep disorders; side effect reduction |
| 04/06/2005 | CN1195748C 1, 2-benzothiazepines for the treatment of hyperlipidemic diseases |
| 03/31/2005 | WO2005028459A1 Preparation method for quetiapine |
| 03/31/2005 | WO2005028458A1 Preparation of quetiapine |
| 03/31/2005 | WO2005028457A1 Preparation of quetiapine |
| 03/31/2005 | CA2538866A1 Preparation of quetiapine |
| 03/31/2005 | CA2538745A1 Preparation of quetiapine |
| 03/30/2005 | EP1326616B1 Use of quetiapine for attention deficit hyperactivity disorder or conduct disorder |
| 03/30/2005 | EP1115881B1 Process for the enzymatic kinetic resolution of 3-phenylglycidates by transesterification with aminoalcohols |
| 03/23/2005 | CN1599731A Benzothiazepine derivatives |
| 03/17/2005 | WO2004073642A3 2-aminoethyl substituted pyrimidin-2-ones, cyclopropanes, pyrazolines, pyrimidines and benzothiazepines and their use as urotensin ii and somatostatin 5 receptor ligands |
| 03/17/2005 | US20050059699 N-acylated lipophilic amino acid derivatives |
| 03/08/2005 | US6864250 N-acylated lipophilic amino acid derivatives |
| 03/01/2005 | US6861419 Substituted 1, 4-thiazepine and analogs as activators of caspases and inducers of apoptosis and the use thereof |
| 02/17/2005 | WO2005014590A2 Procedure for preparing 11-(4`2-(2-hydroxyethoxy )ethyl!-1-piperazinyl!-dibenzo`b,f!`1,4!thiazepine |
| 02/17/2005 | WO2004080391A3 Novel antibacterial agents |
| 02/17/2005 | US20050038009 1,1-dioxo-3,3-dibutyl-5-phenyl-7-methylthio-8-(N-{(R)- alpha -[N-((S)-1-carboxypropyl) carbamoyl]-4-hydroxybenzyl}carbamoylmethoxy)-2,3,4,5-tetrahydro-1,2,5-benzothiadiazepine |
| 02/16/2005 | CN1582151A Benzothiazepine and benzothiazepine derivatives with ileal bile acid transport (IBAT) inhibitory activity for the treatment hyperlipidaemia |
| 02/10/2005 | WO2005012274A1 Process for the preparation of 11-(1-piperazinyl)dibenzo `b, f! `1 ,4!-thiazepine, an intermediate in the synthesis of the antipsychotic drug quetiapine |
| 02/10/2005 | US20050032776 Benzothiazepine derivatives for the treatment of hyperlipidemia |
| 02/09/2005 | CN1188404C Cyclic compound |
| 01/27/2005 | US20050020571 Antiserotonine agents; psycholgical disorders; headaches |
| 01/13/2005 | US20050009805 Quaternary ammonium 1,4-benzothiazepinedione derivatives useful for treatment and prevention of hyperlipidemia, cholestasis-accompanying hepatopathy, particularly primary biliary cirrhosis and primary sclerosing cholangitis, and obesity and fatty liver. |
| 01/13/2005 | US20050009755 (74)(3S)-3-amino-1-(1-benzyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-4-yl)-5-methyl-2-heptanone for example; cysteine protease inhibitors; treating bone resorption diseases such as osteoporosis |
| 01/12/2005 | EP1495008A1 Synthesis of quetiapine and pharmaceutically acceptable salts thereof |
| 01/12/2005 | EP1165532B1 Antibacterial agents |
| 12/23/2004 | WO2004078735A9 Novel polymorphs of quetiapine fumarate |
| 12/16/2004 | US20040254160 Benzothiazepine derivatives |
| 12/08/2004 | EP1482945A1 Crystalline forms of quetiapine hemifumarate |
| 12/02/2004 | WO2004047722A3 METHOD OF PREPARING 10H-DIBENZO[b,f][1,4]THIAZEPIN-11-ONE |
| 12/02/2004 | US20040242562 stable, reproducible two crystalline forms; prepared by dissolving quetiapine free base and fumaric acid in suitable solvent and crystallizing fumarate salt; suitable solvents are ketones like acetone, methyl iso butyl ketone; esters like ethyl acetate, ethyl formate, methyl acetate; and mixture |
| 12/01/2004 | CN1550496A Acetylenic alpha-amino acid-based sulfamide hydroxamic acid TACE inhibitors |
| 12/01/2004 | CN1177839C Process for preparation of quetiapine and intermediates therefor |
| 11/24/2004 | EP1263747B1 1,5-benzothiazepines and their use as hypolipidaemics |
| 11/10/2004 | EP1117408B9 Use of diltiazem for treating retinal pathologies |
| 11/04/2004 | US20040220400 Using phase transfer catalyst and base in solvent; refluxing |
| 10/26/2004 | US6809092 1,3,4,5-tetrahydro-2h-2-benzazepin-2-yl derivatives; cysteine protease inhibitors |
| 10/20/2004 | CN1537847A Internediate for preparing quetiapin and preparation method of the intermediate |
| 10/14/2004 | US20040204500 Preventives/remedies for organ functional disorders and organ dysfunction |
| 10/07/2004 | US20040198974 applying deemed racemates to continuos enantioselective liquid chromatography like SMB (simulated moving bed); for industrial scale production of pure enantiomers of amino acids useful as intermediates in organic synthesis such as N-benzyloxycarbonyl-tert-leucine |
| 09/23/2004 | WO2004080391A2 Novel antibacterial agents |
| 09/23/2004 | US20040186154 treating or preventing a hypercholesterolemia-related or an inflammation-related condition ; apical sodium co-dependent bile acid transport inhibitor and an amount of a cyclooxygenase-2 (COX-2) selective inhibitor or its prodrug; kits |
| 09/23/2004 | US20040186093 Cyclizing a sulfamide acyclic compound with a deprotonating agent in an aprotic solvent; forming an intermediates for the preparation of naphthyridine carboxamide compounds which are HIV integrase enzyme inhibitors; commercial available starting materials alkanesulfonyl halides, haloalkylamine |
| 09/23/2004 | CA2801100A1 Novel antibacterial agents |
| 09/16/2004 | WO2004078735A1 Novel polymorphs of quetiapine fumarate |
| 09/16/2004 | WO2003104257A3 Protease inhibitors |
| 09/10/2004 | WO2004076431A1 Synthesis of quetiapine and pharmaceutically acceptable salts thereof |
| 09/10/2004 | WO2004076430A1 Benzothiazepine and benzothiepine derivatives |
| 09/10/2004 | CA2516646A1 Synthesis of quetiapine and pharmaceutically acceptable salts thereof |
| 09/08/2004 | CN1527709A Therapeutic combinations for cardiovascular and inflammatory indications |
| 09/02/2004 | WO2004073642A2 2-aminoethyl substituted pyrimidin-2-ones, cyclopropanes, pyrazolines, pyrimidines and benzothiazepines and their use as urotensin ii and somatostatin 5 receptor ligands |
| 09/02/2004 | CA2515706A1 2-aminoethyl substituted pyrimidin-2-ones, cyclopropanes, pyrazolines, pyrimidines and benzothiazepines and their use as urotensin ii and somatostatin 5 receptor ligands |
| 08/03/2004 | US6770668 Pharmaceutically active compounds and methods of use |
| 07/27/2004 | CA2124136C Method for producing benzylidene derivatives |
| 07/15/2004 | WO2004058734A1 Process for preparing diltiazem using a heterogeneous trifunctional catalyst |
| 07/14/2004 | EP1435956A2 Therapeutic combinations for cardiovascular and inflammatory indications |
| 07/14/2004 | EP1144368B1 Acetylenic alpha-amino acid-based sulfonamide hydroxamic acid tace inhibitors |
| 07/14/2004 | CN1157387C Process for preparing 11-amino-3-chlorine-6, 11-dihydrogen-5, 5-dioxo-6-methyl-dibenzo [c,f][1,2] thiazine and application of synthetic tianeptine |
| 07/08/2004 | WO2004056182A1 Pesticidal dibenzo(hetero)azepine derivatives |
| 07/01/2004 | US20040127704 Process for preparing diltiazem using a heterogeneous trifunctional catalyst |
| 06/23/2004 | EP1430040A1 Benzothiazepine derivatives |
| 06/16/2004 | EP1427713A1 Benzothiazepine derivatives for the treatment of hyperlipidemia |
| 06/16/2004 | EP1427423A1 Benzothiazepine and benzothiadiazepine derivatives with ileal bile acid transport (ibat) inhibitory activity for the treatment hyperlipidaemia |
| 06/16/2004 | EP1117408B1 Use of diltiazem for treating retinal pathologies |
| 06/15/2004 | US6750255 Calcium receptor-active compounds |
| 06/10/2004 | WO2004047722A2 METHOD OF PREPARING 10H-DIBENZO[b,f][1,4]THIAZEPIN-11-ONE |
| 06/02/2004 | EP1423112A1 A combination of quetiapine and zolmitriptan |
| 05/12/2004 | EP1417162A1 Chromatographic separation of enantiomers of protected amino acids via smb-method |