Patents
Patents for C07D 281 - Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms (1,924)
02/2002
02/21/2002WO2001079187A3 Substituted 1,4-thiazepine and analogs and their use as activators of caspases
02/19/2002CA2024040C Dibenz [b,f] [1,4]oxazepin (and thiazepin)-11 (10h)-ones and-thiones and their use in the prevention or treatment of aids
02/13/2002EP0861250B1 Amidine and isothiourea derivatives as inhibitors of nitric oxide synthase
02/13/2002EP0691961B1 Substituted caprolactams and derivatives thereof useful for treatment of hiv disease
02/12/2002US6346632 Crystallization of esters of methoxyphenylglycidic acid from alcohol solvents
02/07/2002WO2002010174A1 Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo [2,1-b][1,3]benzotiazepines
02/07/2002WO2001051506A3 Oligomers of nonpeptide restricted mimetics of dipeptides or tripeptides and the use thereof in the synthesis of synthetic proteins and polypeptides
02/06/2002EP0882024B1 Retroviral protease inhibiting compounds
02/05/2002US6344556 Thio containing monomers for polymers
01/2002
01/31/2002WO2002008211A2 Benzothiazepines and their use as antihyperlipidemics
01/24/2002US20020010169 Substituted 1, 4-thiazepine and analogs as activators of caspases and inducers of apoptosis and the use thereof
01/10/2002US20020004503 Viricides
01/10/2002US20020004500 Drug mixture for cardiovascular disorders
01/09/2002EP1170289A2 Retroviral protease inhibiting compounds
01/09/2002EP1169313A2 1,4-benzothiazepine-1,1-dioxide derivatives substituted by sugar radicals, methods for the production thereof, medicaments containing these compounds and the use thereof
01/03/2002WO2002000626A1 Fused azepine derivatives and their use as antidiuretic agents
01/03/2002CA2412555A1 Fused azepine derivatives and their use as antidiuretic agents
01/02/2002EP1165532A1 Antibacterial agents
01/02/2002CN1329002A Intermediate product for preparing aralkyl and aryl alkylene heterocyclic lactam and imide
01/01/2002CA2051830C Tricyclic heterocycles
11/2001
11/21/2001EP1155007A2 1,2-benzothiazepines for the treatment of hyperlipidemic diseases
11/21/2001EP0659179B1 Benzo-fused lactams promote release of growth hormone
11/08/2001US20010039272 Compounds activating pharmacological effect of retinoids
11/06/2001US6313296 2-pyrrolidinone-1-acetic acid derivatives; viricides for human immunodeficiency virus (hiv); acquired immune deficiency syndrome (aids) treatment
11/01/2001US20010037021 11-keto-3-chloro-6,11-dihydro-5,5-dioxo-6-methyl-dibenzo(c,f)( 1,2)thiazepine is reacted with sodium borohydride in presence of chlorinated solvent and a catalyst to form alcohol, then chlorinating to form chloride, finally forming a salt
10/2001
10/31/2001CN1319593A Process for prpearing 11-amino-3-chlorine-6,11-dihydrogen-5,5-dioxo-6-methyl-dibenzo [c,f][1,2] thiazine and application of synthetic tianeptine
10/25/2001WO2001079187A2 Substituted 1,4-thiazepine and analogs and their use as activators of caspases
10/25/2001CA2406271A1 Substituted 1,4-thiazepine and analogs and their use as activators of caspases
10/23/2001CA2203310C Compressed matrix for slow release of salt of tianeptine sodium following oral administration
10/18/2001WO2001077089A1 New neurokinin antagonists for use as medicaments
10/17/2001EP1144396A2 Substituted 2-arylimino heterocycles and compositions containing them, for use as progesterone receptor binding agents
10/17/2001EP1144368A2 Acetylenic alpha-amino acid-based sulfonamide hydroxamic acid tace inhibitors
10/11/2001WO2001074348A2 Vasopeptidase inhibitors to treat isolated systolic hypertension
10/11/2001CA2405496A1 Vasopeptidase inhibitors to treat isolated systolic hypertension
10/10/2001EP1140190A1 Combinations of ileal bile acid transport inhibitors and bile acid sequestering agents for cardiovascular indications
10/04/2001EP1138677A1 Process for the preparation of 11-amino-3-chloro-6,11-dihydro-5,5-dioxo-6-methyl-dibenzo[c,f][1,2]-thiazepine and application to the synthesis of tianeptine
09/2001
09/19/2001CN1313855A Inhibitors of alpha4Betal mediated cell adhesion alpha Beta
09/13/2001WO2001066533A1 1,5-benzothiazepines and their use as hypolipidaemics
09/13/2001CA2401055A1 1,5-benzothiazepines and their use as hypolipidaemics
09/05/2001CN1070484C Hypolipidemic 1,4-benzothiazepine-1,1-dioxides
09/04/2001US6284767 Retroviral protease inhibiting compounds
08/2001
08/23/2001WO2001060808A1 Thiazepinyl hydroxamic acid derivatives as matrix metalloproteinase inhibitors
08/23/2001CA2400862A1 Thiazepinyl hydroxamic acid derivatives as matrix metalloproteinase inhibitors
08/21/2001US6277831 1,4-benzothiazepine-1,1-dioxide derivatives substituted by sugar residues, process for their preparation, pharmaceuticals comprising these compounds, and their use
08/16/2001EP1123268A1 New compounds, their preparation and use
08/02/2001WO2001055125A1 A process for the preparation of quetiapine and intermediates therefor
07/2001
07/25/2001EP1117408A1 Use of diltiazem for treating retinal pathologies
07/24/2001CA2030162C Benzothiazepines
07/19/2001WO2001051506A2 Oligomers of nonpeptide restricted mimetics of dipeptides or tripeptides and the use thereof in the synthesis of synthetic proteins and polypeptides
07/18/2001EP1115881A1 Process for the enzymatic kinetic resolution of 3-phenylglycidates by transesterification with aminoalcohols
06/2001
06/27/2001CN1301265A Novel substituted arylhydroxamic acids as metalloproteinase inhibitors
06/27/2001CN1067550C Calcium receptor active molecules
06/21/2001WO2000061568A8 1,4-benzothiazepine-1,1-dioxide derivatives substituted by sugar radicals, methods for the production thereof, medicaments containing these compounds and the use thereof
05/2001
05/15/2001CA2238978C Retroviral protease inhibiting compounds
05/10/2001WO2001032639A1 Nonpeptide substituted benzothiazepines as vasopressin antagonists
05/10/2001CA2389439A1 Nonpeptide substituted benzothiazepines as vasopressin antagonists
05/08/2001US6228955 Catalytic epoxidation of a corresponding prochiralm, non-enolizable a/b-unsaturated ketone
05/08/2001US6228395 Sustained-release microgranules containing Diltiazem as the active principle
04/2001
04/25/2001EP1093372A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING $g(b)-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS
04/25/2001CN1292785A Hypolipidemic benzothiazepine compounds
04/19/2001WO2000061568A3 1,4-benzothiazepine-1,1-dioxide derivatives substituted by sugar radicals, methods for the production thereof, medicaments containing these compounds and the use thereof
04/11/2001EP1089989A1 Inhibitors of alpha4beta1 mediated cell adhesion
04/11/2001EP1089977A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
04/11/2001CN1064354C Trilcyclic benzazepine vasopressin antagnonists
04/04/2001CN1064043C Process for preparing 1,5-benzothiazepine derivative
04/03/2001US6211174 Osteoporosis; milk production and carcass quality in livestock; short stature; metabolic disorders
03/2001
03/28/2001EP1085863A1 Cross-reference to related applications
03/13/2001CA2030866C Process for the preparation of an intermediate of diltiazem
03/06/2001US6197953 Process for preparing optically active trans-3-substituted glycidic acid ester
02/2001
02/28/2001EP1077978A1 Novel substituted aryl hydroxamic acids as metalloproteinase inhibitors
02/22/2001WO1999063992A8 Novel calcium channel drugs and uses
02/13/2001US6187936 Transesterification of mixture of trans enantiomers catalysed by enzymes in organic solvent with aminoalcohols to give mixture of trans esters, non transesterified and transesterified, having opposite configuration, separating
02/08/2001WO2001055118A1 Benzene-fused heterocycle derivatives and drugs containing the same as the active ingredient
01/2001
01/30/2001US6180785 Process for preparing diltiazem
01/18/2001WO2001004106A1 Process for producing dibenzothiazepine derivatives
01/11/2001DE19916108C1 Mit Zuckerresten substituierte 1,4-Benzothiazepin-1,1-dioxidderivate, Verfahren zu deren Herstellung und deren Verwendung With sugar residues substituted 1,4-benzothiazepine-1,1-dioxide derivatives, processes for their preparation and their use
01/04/2001WO2001000185A2 1,4-denzothiazepines to treat obesity related disorders
01/04/2001CA2376023A1 Therapeutic agents
12/2000
12/26/2000US6166005 Heterocyclic metalloprotease inhibitors
12/21/2000WO2000044709A3 ACETYLENIC α-AMINO ACID-BASED SULFONAMIDE HYDROXAMIC ACID TACE INHIBITORS
12/20/2000CN1059674C Hypolipidemic benzothiazepines
12/20/2000CN1059673C Hypolipidemic 1,4-benzothiazepine-1,1-dioxides
12/14/2000WO2000047568A3 1,2-benzothiazepines for the treatment of hyperlipidemic diseases
12/13/2000CN1059436C Benzoazepine-benzooxaazepine-benzothiaazepin-N-acetate deriv.
12/12/2000CA2041305C Process for the resolution of 3-(4-substituted-phenyl)-glycidic acid derivatives
12/06/2000CN1275912A Novel amide derivatives
11/2000
11/30/2000WO2000071106A2 Method of treating weight gain
11/30/2000CA2363784A1 Method of treatment
11/15/2000CN1273608A Process for preparing (2R, 3S)-3-(4-lower alkoxyphenyl) glycidic acid esters
11/09/2000WO2000042031A3 Substituted 2-arylimino heterocycles and compositions containing them, for use as progesterone receptor binding agents
10/2000
10/25/2000EP1045840A1 Hypolipidemic benzothiazepine compounds
10/25/2000CN1271340A Process for recycle of waste product of diltiazem synthesis
10/19/2000WO2000061568A2 1,4-benzothiazepine-1,1-dioxide derivatives substituted by sugar radicals, methods for the production thereof, medicaments containing these compounds and the use thereof
10/05/2000WO2000058294A1 Antibacterial agents
10/03/2000US6127359 Bicyclic fibrinogen antagonists
09/2000
09/27/2000EP0848703B1 Derivatives of benzosulphonamides as inhibitors of the enzyme cyclo-oxygenase ii
09/19/2000US6121258 For treatment of arthritis, cancer, cardiovascular disorders, skin disorders, ocular disorders, inflammation, gum disease
09/19/2000US6121256 4-(2,3-(2,5-dimethyl-2,5-hexano)dibenzo(b,f)(1,4)thiazepine-11 -yl)benzoic acid or salt
09/13/2000CN1266430A Process for preparing optically active phenyloxirane compounds
09/12/2000CA2030076C 2-aromatic-3-halobenzothiazepines
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